A Renal Impairment Study for PF-06651600

NCT ID: NCT04037865

Last Updated: 2021-05-18

Study Results

Results available

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Basic Information

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Recruitment Status

TERMINATED

Clinical Phase

PHASE1

Total Enrollment

8 participants

Study Classification

INTERVENTIONAL

Study Start Date

2019-08-19

Study Completion Date

2020-03-31

Brief Summary

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This is a Phase 1 non-randomized, open-label, parallel cohort study of PF-06651600 in subjects with severe renal impairment and subjects without renal impairment (Part 1) and in subjects with mild and moderate renal impairment (Part 2).

Detailed Description

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This is a Phase 1 non-randomized, open-label, parallel cohort, multi-site study to investigate the effect of renal impairment on the pharmacokinetics, safety and tolerability of PF-06651600 after multiple oral doses of 50 mg daily. Subjects will be selected and categorized into normal renal function or renal impairment groups based on their estimated glomerular filtration rate. Part 1: A total of approximately 16 subjects will be enrolled; approximately 8 subjects with severe renal impairment and approximately 8 with normal renal function. After statistical evaluation of results from Part 1, Part 2 may be conducted with approximately 8 subjects each with moderate and mild renal impairment. The total duration of participation from Screening visit to Day 11 will be a maximum of 39 days and from Screening visit to Follow-up/Contact Visit will a maximum of 73 days.

Conditions

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Renal Impairment

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

BASIC_SCIENCE

Blinding Strategy

NONE

Study Groups

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PF-06651600 Severe Renal Impairment

This arm includes participants with severe renal impairment who will receive oral doses of PF-06651600 50 mg on Day 1 through Day 10

Group Type EXPERIMENTAL

PF-06651600

Intervention Type DRUG

PF-06651600 50 mg oral tablets will be administered on Days 1 to 10

PF-06651600 Normal Renal Function

This arm includes participants with normal renal function who will receive oral doses of PF-06651600 50 mg on Day 1 through Day 10

Group Type EXPERIMENTAL

PF-06651600

Intervention Type DRUG

PF-06651600 50 mg oral tablets will be administered on Days 1 to 10

PF-06651600 Moderate Renal Impairment

This arm is in Part 2 which will be conducted if decision criterion to proceed to Part 2 is met. This arm includes participants with moderate renal impairment who will receive oral doses of PF-06651600 50 mg on Day 1 through Day 10

Group Type EXPERIMENTAL

PF-06651600

Intervention Type DRUG

PF-06651600 50 mg oral tablets will be administered on Days 1 to 10

PF-06651600 Mild Renal Impairment

This arm is in Part 2 which will be conducted if the decision criterion to proceed to Part 2 is met. The arm includes participants with mild renal impairment who will receive oral doses of PF-06651600 50 mg on Day 1 through Day 10.

Group Type EXPERIMENTAL

PF-06651600

Intervention Type DRUG

PF-06651600 50 mg oral tablets will be administered on Days 1 to 10

Interventions

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PF-06651600

PF-06651600 50 mg oral tablets will be administered on Days 1 to 10

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Body mass index (BMI) of \>/= 17.5 to \</= 40.0 kg/m2; and a total body weight \> 50 kg (110 lb)


* Meet the following eGFR criteria during the screening period based upon MDRD equation:
* Severe renal impairment: eGFR \<30 mL/min but not requiring hemodialysis
* Moderate renal impairment (Part 2 only): eGFR \>/=30 mL/min and \<60 mL/min
* Mild renal impairment (Part 2 only): eGFR between 60 and 89 mL/min
* Any form of renal impairment except acute nephritic syndrome (subjects with history of previous nephritic syndrome but in remission can be included)
* Stable drug regimen

Exclusion Criteria

* Females of child-bearing potential must use an accepted, highly effective contraceptive method
* Renal transplant recipients
* Urinary incontinence without catheterization
* Subjects with clinically significant infections within the past 6 months prior to first dose of study drug, evidence of active or chronic infection requiring oral treatment within 4 weeks prior, history of disseminated herpes simplex or recurrent or disseminated herpes zoster
* Subjects with malignancy or with a history of malignancy, with the exception of adequately treated or excised non-metastatic basal cell or squamous cell cancer of skin or cervical carcinoma in situ
* HIV, Hepatitis B, or Hepatitis C infection


* Subjects requiring hemodialysis and peritoneal dialysis
* Screening BP \>/=180 mmHg (systolic) or \>/=110 mmHg (diastolic)
* Screening 12-lead ECG demonstrating QTcF \>470 msec
Minimum Eligible Age

18 Years

Maximum Eligible Age

75 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

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Pfizer

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Pfizer CT.gov Call Center

Role: STUDY_DIRECTOR

Pfizer

Locations

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Investigational Drug Services (IDS) University of Miami Hospitals and Clinics

Miami, Florida, United States

Site Status

University of Miami Division of Clinical Pharmacology

Miami, Florida, United States

Site Status

Prism Clinical Research, LLC

Saint Paul, Minnesota, United States

Site Status

Countries

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United States

References

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Wojciechowski J, S Purohit V, Huh Y, Banfield C, Nicholas T. Evolution of Ritlecitinib Population Pharmacokinetic Models During Clinical Drug Development. Clin Pharmacokinet. 2023 Dec;62(12):1765-1779. doi: 10.1007/s40262-023-01318-3. Epub 2023 Nov 2.

Reference Type DERIVED
PMID: 37917289 (View on PubMed)

Purohit V, Huh Y, Wojciechowski J, Plotka A, Salts S, Antinew J, Dimitrova A, Nicholas T. Leveraging Prior Healthy Participant Pharmacokinetic Data to Evaluate the Impact of Renal and Hepatic Impairment on Ritlecitinib Pharmacokinetics. AAPS J. 2023 Mar 28;25(3):32. doi: 10.1208/s12248-023-00792-8.

Reference Type DERIVED
PMID: 36977960 (View on PubMed)

Provided Documents

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Document Type: Study Protocol

View Document

Document Type: Statistical Analysis Plan

View Document

Related Links

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https://pmiform.com/clinical-trial-info-request?StudyID=B7981020

To obtain contact information for a study center near you, click here.

Other Identifiers

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B7981020

Identifier Type: -

Identifier Source: org_study_id

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