Safety and Pharmacokinetic of Donepezil Pamoate in Healthy Subjects

NCT ID: NCT03932916

Last Updated: 2020-09-29

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

38 participants

Study Classification

INTERVENTIONAL

Study Start Date

2019-07-02

Study Completion Date

2020-09-11

Brief Summary

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The objective of this study is to evaluate the safety and pharmacokinetic profiles of HHT201 in healthy subjects.

Detailed Description

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The study aims to evaluate the safety, pharmacokinetics and to determine the potential dose limiting toxicity of HHT201 in healthy subjects between the ages of 20-59, 6 in 17mg dose group and 20 in 34mg dose group. Another 12 subjects will be administered a tablet of 5mg Donepezil Hydrochloride to get the PK profile of Donepezil as reference. Eligible subjects will be accepted into the protocol after review and providing voluntary written informed consent forms and completion of a comprehensive medical, physical examination, and routine laboratory assessment.

Conditions

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AD

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

SEQUENTIAL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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experimental group 1

HHT201 17mg injection

Group Type EXPERIMENTAL

Donepezil Pamoate for Injection 17mg

Intervention Type DRUG

A dosage of 17mg HHT201 will be injected into the muscle in the gluteus once.

experimental group 2

HHT201 34mg injection

Group Type EXPERIMENTAL

Donepezil Pamoate for Injection 34mg

Intervention Type DRUG

A dosage of 34mg HHT201 will be injected into the muscle in the gluteus once.

experimental group 3

Donepezil Hydrochloride oral tablet 5mg

Group Type ACTIVE_COMPARATOR

Donepezil Hydrochloride 5mg

Intervention Type DRUG

A tablet of 5mg Donepezil Hydrochloride will be administered once.

Interventions

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Donepezil Pamoate for Injection 17mg

A dosage of 17mg HHT201 will be injected into the muscle in the gluteus once.

Intervention Type DRUG

Donepezil Pamoate for Injection 34mg

A dosage of 34mg HHT201 will be injected into the muscle in the gluteus once.

Intervention Type DRUG

Donepezil Hydrochloride 5mg

A tablet of 5mg Donepezil Hydrochloride will be administered once.

Intervention Type DRUG

Other Intervention Names

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HHT201 HHT201 Aricept

Eligibility Criteria

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Inclusion Criteria

* Chinese healthy subjects, male or female
* between the ages of 20 and 60 years
* A body mass index (BMI), calculated as weight in kg/(height in m)², from 19 to 28 kg/m², and female weight≥45kg, male weight≥50kg
* Able to provide written informed consent forms

Exclusion Criteria

1. Clinically significant history of gastrointestinal, cardiovascular, musculoskeletal, endocrine, hematologic, psychiatric, renal, hepatic, bronchopulmonary, neurologic, immunologic, lipid metabolism disorders
2. Resting pulse rate \<55/min or \>100/min; Sitting systolic blood pressure \<90mmHg or \>140mmHg, diastolic blood pressure \<60mmHg or \>90mmHg
3. ALT or Cr, BUN exceeding the upper limit of normal value; test results of urine protein was "++"
4. Clinically significant ECG abnormalities in screening or baseline, such as male QTc interval ≥450ms and female QTc interval ≥470ms, and were considered inappropriate for inclusion by the researchers
5. Positive blood screen for human immunodeficiency virus (HIV), hepatitis B surface antigen (HBsAg), or hepatitis C antibody
6. History or presence of drug or alcohol abuse
7. Positive pregnancy test result, or plan to be pregnant if female
8. An unwillingness or inability to comply with food and beverage restrictions within 24 hours prior to dosing
9. Participation in any other investigational drug trial within 30 days prior to screening.
Minimum Eligible Age

20 Years

Maximum Eligible Age

59 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

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Shanghai Synergy Pharmaceutical Sciences Co., Ltd.

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Huafang Li, PhD

Role: PRINCIPAL_INVESTIGATOR

Shanghai Mental Health Center

Locations

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Shanghai mental health center

Shanghai, Shanghai Municipality, China

Site Status

Countries

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China

Other Identifiers

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DON101-CTP

Identifier Type: -

Identifier Source: org_study_id

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