Trial Outcomes & Findings for Efficacy of Guanfacine and Lidocaine Combination in Trigeminal Nerve Block for Pain Management in Trigeminal Neuropathy (NCT NCT03865940)

NCT ID: NCT03865940

Last Updated: 2025-03-30

Results Overview

Time (hours) until pain returns to baseline number.

Recruitment status

COMPLETED

Study phase

PHASE2

Target enrollment

37 participants

Primary outcome timeframe

up to 2 weeks

Results posted on

2025-03-30

Participant Flow

Participant milestones

Participant milestones
Measure
Lidocaine Then Lidocaine + Guanfacine
Trigeminal nerve block will be performed with injection of 6 mL of 1% lidocaine (Day 1). Patient will return between Day 15-28 and trigeminal nerve block will be performed with injection of 6 mL of 1% lidocaine + 250 mcg guanfacine. Lidocaine: 6 mL of 1% lidocaine Guanfacine: 250 mcg
Lidocaine + Guanfacine Then Lidocaine
Trigeminal nerve block will be performed with injection of 6 mL of 1% lidocaine + 250 mcg guanfacine (Day 1). Patient will return between Day 15-28 and trigeminal nerve block will be performed with injection of 6 mL of 1% lidocaine. Lidocaine: 6 mL of 1% lidocaine Guanfacine: 250 mcg
First Intervention (14 Days)
STARTED
18
19
First Intervention (14 Days)
COMPLETED
18
19
First Intervention (14 Days)
NOT COMPLETED
0
0
Washout Period (14 Days)
STARTED
18
19
Washout Period (14 Days)
COMPLETED
18
19
Washout Period (14 Days)
NOT COMPLETED
0
0
Second Intervention (14 Days)
STARTED
18
19
Second Intervention (14 Days)
COMPLETED
10
18
Second Intervention (14 Days)
NOT COMPLETED
8
1

Reasons for withdrawal

Withdrawal data not reported

Baseline Characteristics

Efficacy of Guanfacine and Lidocaine Combination in Trigeminal Nerve Block for Pain Management in Trigeminal Neuropathy

Baseline characteristics by cohort

Baseline characteristics by cohort
Measure
Lidocaine Then Lidocaine + Guanfacine
n=18 Participants
Trigeminal nerve block will be performed with injection of 6 mL of 1% lidocaine (Day 1). Patient will return between Day 15-28 and trigeminal nerve block will be performed with injection of 6 mL of 1% lidocaine + 250 mcg guanfacine. Lidocaine: 6 mL of 1% lidocaine Guanfacine: 250 mcg
Lidocaine + Guanfacine Then Lidocaine
n=19 Participants
Trigeminal nerve block will be performed with injection of 6 mL of 1% lidocaine + 250 mcg guanfacine (Day 1). Patient will return between Day 15-28 and trigeminal nerve block will be performed with injection of 6 mL of 1% lidocaine. Lidocaine: 6 mL of 1% lidocaine Guanfacine: 250 mcg
Total
n=37 Participants
Total of all reporting groups
Age, Continuous
51.5 years
n=93 Participants
60.1 years
n=4 Participants
60.0 years
n=27 Participants
Sex: Female, Male
Female
16 Participants
n=93 Participants
16 Participants
n=4 Participants
32 Participants
n=27 Participants
Sex: Female, Male
Male
2 Participants
n=93 Participants
3 Participants
n=4 Participants
5 Participants
n=27 Participants
Ethnicity (NIH/OMB)
Hispanic or Latino
1 Participants
n=93 Participants
0 Participants
n=4 Participants
1 Participants
n=27 Participants
Ethnicity (NIH/OMB)
Not Hispanic or Latino
16 Participants
n=93 Participants
19 Participants
n=4 Participants
35 Participants
n=27 Participants
Ethnicity (NIH/OMB)
Unknown or Not Reported
1 Participants
n=93 Participants
0 Participants
n=4 Participants
1 Participants
n=27 Participants
Race (NIH/OMB)
American Indian or Alaska Native
0 Participants
n=93 Participants
0 Participants
n=4 Participants
0 Participants
n=27 Participants
Race (NIH/OMB)
Asian
0 Participants
n=93 Participants
0 Participants
n=4 Participants
0 Participants
n=27 Participants
Race (NIH/OMB)
Native Hawaiian or Other Pacific Islander
0 Participants
n=93 Participants
0 Participants
n=4 Participants
0 Participants
n=27 Participants
Race (NIH/OMB)
Black or African American
1 Participants
n=93 Participants
1 Participants
n=4 Participants
2 Participants
n=27 Participants
Race (NIH/OMB)
White
17 Participants
n=93 Participants
18 Participants
n=4 Participants
35 Participants
n=27 Participants
Race (NIH/OMB)
More than one race
0 Participants
n=93 Participants
0 Participants
n=4 Participants
0 Participants
n=27 Participants
Race (NIH/OMB)
Unknown or Not Reported
0 Participants
n=93 Participants
0 Participants
n=4 Participants
0 Participants
n=27 Participants
Region of Enrollment
United States
18 participants
n=93 Participants
19 participants
n=4 Participants
37 participants
n=27 Participants

PRIMARY outcome

Timeframe: up to 2 weeks

Time (hours) until pain returns to baseline number.

Outcome measures

Outcome measures
Measure
Lidocaine Alone
n=36 Participants
Data from injection where participants received an injection of lidocaine ALONE.
Lidocaine + Guanfacine
n=28 Participants
Data from injection where participants received lidocaine + guanfacine.
Time to Return to Baseline Pain After Injection.
8 hours
Interval 4.0 to 120.0
5 hours
Interval 5.0 to 168.0

SECONDARY outcome

Timeframe: 8 hours

Population: The overall number of participants analyzed corresponds with how many participants were injected; however, not every participant responded at every timepoint. Therefore, only recorded responses at each timeline were analyzed.

Pain Intensity after treatment measured throughout the 8-hour follow-up period on a visual analog scale (VAS) from 0 to 10, where 0 is the least pain and 10 is the most pain.

Outcome measures

Outcome measures
Measure
Lidocaine Alone
n=36 Participants
Data from injection where participants received an injection of lidocaine ALONE.
Lidocaine + Guanfacine
n=28 Participants
Data from injection where participants received lidocaine + guanfacine.
Pain Intensity in Follow-Up
6.5 hours
3.42 score on a scale
Standard Deviation 2.17
2.81 score on a scale
Standard Deviation 2.23
Pain Intensity in Follow-Up
0 hours
6.75 score on a scale
Standard Deviation 1.56
6.63 score on a scale
Standard Deviation 1.43
Pain Intensity in Follow-Up
0.5 hours
1.91 score on a scale
Standard Deviation 2.31
1.88 score on a scale
Standard Deviation 2.72
Pain Intensity in Follow-Up
1 hour
2.24 score on a scale
Standard Deviation 2.2
1.54 score on a scale
Standard Deviation 2.25
Pain Intensity in Follow-Up
1.5 hours
2.83 score on a scale
Standard Deviation 2.6
1.42 score on a scale
Standard Deviation 1.98
Pain Intensity in Follow-Up
2 hours
2.47 score on a scale
Standard Deviation 2.26
1.81 score on a scale
Standard Deviation 2.11
Pain Intensity in Follow-Up
2.5 hours
2.7 score on a scale
Standard Deviation 2.53
2.21 score on a scale
Standard Deviation 2.45
Pain Intensity in Follow-Up
3 hours
2.84 score on a scale
Standard Deviation 2.38
2.4 score on a scale
Standard Deviation 2.61
Pain Intensity in Follow-Up
3.5 hours
3.03 score on a scale
Standard Deviation 2.37
2.38 score on a scale
Standard Deviation 2.45
Pain Intensity in Follow-Up
4 hours
2.74 score on a scale
Standard Deviation 2.18
2.04 score on a scale
Standard Deviation 2.49
Pain Intensity in Follow-Up
4.5 hours
2.79 score on a scale
Standard Deviation 2.18
2.29 score on a scale
Standard Deviation 2.41
Pain Intensity in Follow-Up
5 hours
3.65 score on a scale
Standard Deviation 2.12
2.58 score on a scale
Standard Deviation 2.44
Pain Intensity in Follow-Up
5.5 hours
3.69 score on a scale
Standard Deviation 2.14
3.0 score on a scale
Standard Deviation 2.81
Pain Intensity in Follow-Up
6 hours
3.31 score on a scale
Standard Deviation 2.24
2.67 score on a scale
Standard Deviation 2.45
Pain Intensity in Follow-Up
7 hours
3.76 score on a scale
Standard Deviation 2.4
2.79 score on a scale
Standard Deviation 2.17
Pain Intensity in Follow-Up
7.5 hours
3.52 score on a scale
Standard Deviation 2.65
2.85 score on a scale
Standard Deviation 2.19
Pain Intensity in Follow-Up
8 hours
3.56 score on a scale
Standard Deviation 2.53
2.68 score on a scale
Standard Deviation 2.25

SECONDARY outcome

Timeframe: 14 days

Population: The overall number of participants analyzed corresponds with how many participants were injected; however, not every participant responded at every timepoint. Therefore, only recorded responses at each timeline were analyzed.

Participant Quality of Life as measured by the PROMIS Global Health -10 SF during the 14-day follow-up. The scores reported are T-scores. The T-score rescales the raw sum score into a standardized score with a mean of 50 and a standard deviation (SD) of 10. Therefore a person with a T-score of 40 is one SD below the mean and a person with a T-score of 60 is one SD above the mean. For the Physical Health subscale, raw scores are converted into t-scores ranging from 16.2 to 67.7 and higher t-scores are indicative of better overall physical health.

Outcome measures

Outcome measures
Measure
Lidocaine Alone
n=36 Participants
Data from injection where participants received an injection of lidocaine ALONE.
Lidocaine + Guanfacine
n=28 Participants
Data from injection where participants received lidocaine + guanfacine.
Quality of Life, Physical Health
Day 0
40.35 T-score
Standard Deviation 6.66
39.86 T-score
Standard Deviation 6.07
Quality of Life, Physical Health
Day 7
42.88 T-score
Standard Deviation 6.47
43.2 T-score
Standard Deviation 6.3
Quality of Life, Physical Health
Day 14
42.83 T-score
Standard Deviation 7.89
41.67 T-score
Standard Deviation 7.16

SECONDARY outcome

Timeframe: 14 days

Population: The overall number of participants analyzed corresponds with how many participants were injected; however, not every participant responded at every timepoint. Therefore, only recorded responses at each timeline were analyzed.

Participant Quality of Life as measured by the PROMIS Global Health -10 SF during the 14-day follow-up. The scores reported are T-scores. The T-score rescales the raw sum score into a standardized score with a mean of 50 and a standard deviation (SD) of 10. Therefore a person with a T-score of 40 is one SD below the mean and a person with a T-score of 60 is one SD above the mean. In this Mental Health subscale, raw scores are converted into t-scores ranging from 21.2 to 67.6, where higher t-scores are indicative of better overall physical health.

Outcome measures

Outcome measures
Measure
Lidocaine Alone
n=36 Participants
Data from injection where participants received an injection of lidocaine ALONE.
Lidocaine + Guanfacine
n=28 Participants
Data from injection where participants received lidocaine + guanfacine.
Quality of Life, Mental Health
Day 0
44.98 T-score
Standard Deviation 10.47
44.4 T-score
Standard Deviation 8.93
Quality of Life, Mental Health
Day 7
44.34 T-score
Standard Deviation 8.42
46.07 T-score
Standard Deviation 8.42
Quality of Life, Mental Health
Day 14
43.78 T-score
Standard Deviation 7.91
45.72 T-score
Standard Deviation 9.91

SECONDARY outcome

Timeframe: 14 days

Population: The overall number of participants analyzed corresponds with how many participants were injected; however, not every participant responded at every timepoint. Therefore, only recorded responses at each timeline were analyzed.

Frequency of nerve pain attacks during the 14-day follow-up period. Pain frequency was recorded numerically as 0 - None (no pain), 1 - Weekly, 2 - Daily, 3 - Hourly, and 4 - Constant pain. Data was not collected at baseline, only at Day 7 and Day 14.

Outcome measures

Outcome measures
Measure
Lidocaine Alone
n=36 Participants
Data from injection where participants received an injection of lidocaine ALONE.
Lidocaine + Guanfacine
n=28 Participants
Data from injection where participants received lidocaine + guanfacine.
Frequency of Nerve Pain Attacks
Day 7
3.64 units on a scale
Standard Deviation 1.11
3.70 units on a scale
Standard Deviation 1.17
Frequency of Nerve Pain Attacks
Day 14
3.61 units on a scale
Standard Deviation 1.15
3.81 units on a scale
Standard Deviation 0.83

SECONDARY outcome

Timeframe: 8 hours

Population: The overall number of participants analyzed corresponds with how many participants were injected; however, not every participant responded at every timepoint. Therefore, only recorded responses at each timeline were analyzed.

Number of participants using rescue medication during the 8-hour follow-up period

Outcome measures

Outcome measures
Measure
Lidocaine Alone
n=36 Participants
Data from injection where participants received an injection of lidocaine ALONE.
Lidocaine + Guanfacine
n=28 Participants
Data from injection where participants received lidocaine + guanfacine.
Rescue Medication Use
2.5 hours
1 Participants
2 Participants
Rescue Medication Use
0 hours
16 Participants
12 Participants
Rescue Medication Use
0.5 hours
2 Participants
0 Participants
Rescue Medication Use
1 hour
0 Participants
1 Participants
Rescue Medication Use
1.5 hours
3 Participants
1 Participants
Rescue Medication Use
2 hours
3 Participants
0 Participants
Rescue Medication Use
3 hours
4 Participants
3 Participants
Rescue Medication Use
3.5 hours
1 Participants
1 Participants
Rescue Medication Use
4 hours
1 Participants
1 Participants
Rescue Medication Use
4.5 hours
3 Participants
2 Participants
Rescue Medication Use
5 hours
3 Participants
2 Participants
Rescue Medication Use
5.5 hours
2 Participants
1 Participants
Rescue Medication Use
6 hours
2 Participants
1 Participants
Rescue Medication Use
6.5 hours
1 Participants
3 Participants
Rescue Medication Use
7 hours
3 Participants
2 Participants
Rescue Medication Use
7.5 hours
5 Participants
2 Participants
Rescue Medication Use
8 hours
7 Participants
1 Participants

SECONDARY outcome

Timeframe: 14 days

Population: Not all participants reported using rescue medication, so this analysis only includes participants that reported rescue medication use.

Time, in hours, to use of first rescue medication in the follow-up period following the injection.

Outcome measures

Outcome measures
Measure
Lidocaine Alone
n=30 Participants
Data from injection where participants received an injection of lidocaine ALONE.
Lidocaine + Guanfacine
n=23 Participants
Data from injection where participants received lidocaine + guanfacine.
Time to First Rescue Medication
10.28 hours
Standard Deviation 23.54
23.76 hours
Standard Deviation 60.89

Adverse Events

Lidocaine Alone

Serious events: 0 serious events
Other events: 2 other events
Deaths: 0 deaths

Lidocaine + Guanfacine

Serious events: 0 serious events
Other events: 1 other events
Deaths: 0 deaths

Serious adverse events

Adverse event data not reported

Other adverse events

Other adverse events
Measure
Lidocaine Alone
n=36 participants at risk
Data from injection where participants received an injection of lidocaine ALONE.
Lidocaine + Guanfacine
n=28 participants at risk
Data from injection where participants received lidocaine + guanfacine.
Vascular disorders
Hypertension
0.00%
0/36 • Up to 2 weeks after injection
3.6%
1/28 • Number of events 1 • Up to 2 weeks after injection
Ear and labyrinth disorders
Left ear pressure after procedure
2.8%
1/36 • Number of events 1 • Up to 2 weeks after injection
0.00%
0/28 • Up to 2 weeks after injection
Injury, poisoning and procedural complications
Facial brusing and sensitivity
2.8%
1/36 • Number of events 1 • Up to 2 weeks after injection
0.00%
0/28 • Up to 2 weeks after injection

Additional Information

Shelby Meier, PhD - Senior Scientific Project Manager

Vanderbilt University Medical Center

Phone: 6159369228

Results disclosure agreements

  • Principal investigator is a sponsor employee
  • Publication restrictions are in place