A Dose Escalation Study Of PF-06939999 In Participants With Advanced Or Metastatic Solid Tumors

NCT ID: NCT03854227

Last Updated: 2025-01-13

Study Results

Results available

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Basic Information

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Recruitment Status

TERMINATED

Clinical Phase

PHASE1

Total Enrollment

54 participants

Study Classification

INTERVENTIONAL

Study Start Date

2019-03-14

Study Completion Date

2022-04-27

Brief Summary

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This is a Phase 1, open label, multi center, dose escalation and expansion, safety, tolerability, PK, and pharmacodynamics study of PF 06939999 in previously treated patients with advanced or metastatic cancer.

Detailed Description

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Conditions

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Advanced Solid Tumors Metastatic Solid Tumors

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

PARALLEL

Dose Escalation and Dose expansion
Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Dose Escalation

Participants will receive PF-06939999 orally at escalating doses in 28 day cycles on a continuous basis

Group Type EXPERIMENTAL

PF-06939999 dose escalation

Intervention Type DRUG

PF-06939999 orally at escalating doses on a continuous basis

Non small cell lung cancer monotherapy

Participants will receive PF-06939999 at the recommended Phase 2 dose in 28 day cycles on a continuous basis

Group Type EXPERIMENTAL

PF-06939999 monotherapy

Intervention Type DRUG

PF-06939999 at the recommended Phase 2 dose orally on a continuous basis

Urothelial carcinoma

Participants will receive PF-06939999 at the recommended Phase 2 dose in 28 day cycles on a continuous basis

Group Type EXPERIMENTAL

PF-06939999 monotherapy

Intervention Type DRUG

PF-06939999 at the recommended Phase 2 dose orally on a continuous basis

Head and neck squamous cell carcinoma

Participants will receive PF-06939999 at the recommended Phase 2 dose in 28 day cycles on a continuous basis

Group Type EXPERIMENTAL

PF-06939999 monotherapy

Intervention Type DRUG

PF-06939999 at the recommended Phase 2 dose orally on a continuous basis

Non small cell lung cancer PF-06939999 plus docetaxel

Participants will receive PF-06939999 on a continuous basis in combination with docetaxel

Group Type EXPERIMENTAL

PF-06939999 in combination with docetaxel

Intervention Type DRUG

PF-06939999 orally on a continuous basis in combination with docetaxel

Non small cell lung cancer dose finding

Participants will receive PF-06939999 on a continuous basis at escalating doses in combination with docetaxel

Group Type EXPERIMENTAL

PF-06939999 in combination with docetaxel

Intervention Type DRUG

PF-06939999 orally on a continuous basis in combination with docetaxel

Interventions

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PF-06939999 dose escalation

PF-06939999 orally at escalating doses on a continuous basis

Intervention Type DRUG

PF-06939999 monotherapy

PF-06939999 at the recommended Phase 2 dose orally on a continuous basis

Intervention Type DRUG

PF-06939999 in combination with docetaxel

PF-06939999 orally on a continuous basis in combination with docetaxel

Intervention Type DRUG

Other Intervention Names

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PRMT5 inhibitor PRMT5 inhibitor PRMT5 inhibitor

Eligibility Criteria

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Inclusion Criteria

* Histologically or cytologically confirmed locally advanced or metastatic NSCLC, urothelial carcinoma or HNSCC
* Progressed after at least 1 line of treatment and no more than 3 lines of treatment
* At least one measurable lesion as defined by RECIST version 1.1
* ECOG Performance Status 0 or 1
* Adequate Bone Marrow Function
* Adequate Renal Function
* Adequate Liver Function
* Resolved acute effects of any prior therapy

Exclusion Criteria

* Known active uncontrolled or symptomatic CNS metastases.
* Major surgery, radiation therapy, systemic anti-cancer therapy or investigational drug(s) within 4 weeks prior to study entry.
* Active, uncontrolled infection, including COVID-19
* Known or suspected hypersensitivity to PF-06939999
* Inability to consume or absorb study drug
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Pfizer

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Pfizer CT.gov Call Center

Role: STUDY_DIRECTOR

Pfizer

Locations

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Scottsdale Healthcare Hospitals d/b/a HonorHealth

Scottsdale, Arizona, United States

Site Status

Virginia G. Piper Cancer Pharmacy

Scottsdale, Arizona, United States

Site Status

Keck Hospital of USC

Los Angeles, California, United States

Site Status

LAC + USC Medical Center

Los Angeles, California, United States

Site Status

USC Norris Comprehensive Cancer Center

Los Angeles, California, United States

Site Status

USC/Norris Comprehensive Cancer Center

Los Angeles, California, United States

Site Status

Keck Medical Center of USC Pasadena

Pasadena, California, United States

Site Status

AdventHealth Celebration Infusion Center

Celebration, Florida, United States

Site Status

AdventHealth Medical Group Oncology Research at Celebration

Celebration, Florida, United States

Site Status

University Of Miami Hospital and Clinics/Sylvester Comprehensive Cancer Center

Miami, Florida, United States

Site Status

AdventHealth Orlando - Investigational Drug Services

Orlando, Florida, United States

Site Status

AdventHealth Orlando Infusion Center

Orlando, Florida, United States

Site Status

AdventHealth Orlando

Orlando, Florida, United States

Site Status

St. Joseph Mercy Hospital

Ann Arbor, Michigan, United States

Site Status

St. Joseph Mercy Brighton

Brighton, Michigan, United States

Site Status

Henry-Joyce Cancer Clinic

Nashville, Tennessee, United States

Site Status

Oncology IDS Pharmacy

Nashville, Tennessee, United States

Site Status

The University of Texas

Houston, Texas, United States

Site Status

NEXT Oncology

San Antonio, Texas, United States

Site Status

Inova Schar Cancer Institute

Fairfax, Virginia, United States

Site Status

Seattle Cancer Care Alliance

Seattle, Washington, United States

Site Status

University of Washington Medical Center

Seattle, Washington, United States

Site Status

Countries

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United States

References

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Guo C, Liao KH, Li M, Wang IM, Shaik N, Yin D. PK/PD model-informed dose selection for oncology phase I expansion: Case study based on PF-06939999, a PRMT5 inhibitor. CPT Pharmacometrics Syst Pharmacol. 2023 Nov;12(11):1619-1625. doi: 10.1002/psp4.12882. Epub 2022 Nov 16.

Reference Type DERIVED
PMID: 36394153 (View on PubMed)

Provided Documents

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Document Type: Study Protocol

View Document

Document Type: Statistical Analysis Plan

View Document

Related Links

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https://pmiform.com/clinical-trial-info-request?StudyID=C3851001

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Other Identifiers

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C3851001

Identifier Type: -

Identifier Source: org_study_id

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