Trial Outcomes & Findings for Safety and Efficacy Study of Cefepime/VNRX-5133 in Patients With Complicated Urinary Tract Infections (NCT NCT03840148)

NCT ID: NCT03840148

Last Updated: 2025-06-06

Results Overview

Microbiologic success is eradication defined as demonstration that any gram-negative bacterial pathogen found at study entry (≥10\^5 CFU/mL) is eradicated to \<10\^3 CFU/mL. Clinical success is defined as symptomatic resolution or return to pre-morbid baseline of all UTI-core symptoms and patient is alive, and patient has not received additional antibacterial therapy for cUTI.

Recruitment status

COMPLETED

Study phase

PHASE3

Target enrollment

661 participants

Primary outcome timeframe

Assessed at Test of Cure visit (occurred once per participant between Study Days 19 to 23)

Results posted on

2025-06-06

Participant Flow

Six-hundred sixty-one (661) male and female patients with complicated urinary tract infection (cUTI) including acute pyelonephritis (AP), were randomized into 2 groups (cefepime - VNRX-5133, and meropenem) at 68 hospital sites in North and South America, Eastern Europe, and China, from August 2019 until the last patient's final visit in December 2021. Of these 661 patients in the intent-to-treat (ITT) population, 436 were in the MicroITT population (293 cefepime - VNRX-5133, 143 meropenem).

Of the 697 patients screened, 36 patients did not qualify for randomization, and 661 patients were randomized into the trial.

Participant milestones

Participant milestones
Measure
Cefepime/VNRX-5133 (Taniborbactam)
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Study Drug Disposition
STARTED
441
220
Study Drug Disposition
COMPLETED
414
212
Study Drug Disposition
NOT COMPLETED
27
8
Study Completion Disposition
STARTED
441
220
Study Completion Disposition
COMPLETED
426
214
Study Completion Disposition
NOT COMPLETED
15
6

Reasons for withdrawal

Reasons for withdrawal
Measure
Cefepime/VNRX-5133 (Taniborbactam)
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Study Drug Disposition
Adverse Event
13
2
Study Drug Disposition
Withdrawal by Subject
8
2
Study Drug Disposition
Lack of Efficacy
3
0
Study Drug Disposition
Physician Decision
2
0
Study Drug Disposition
Randomized but not treated, IWRS issue, lack of IMP supplies.
1
4
Study Completion Disposition
Withdrawal by Subject
6
2
Study Completion Disposition
Physician Decision
2
0
Study Completion Disposition
Covid-19 related
2
0
Study Completion Disposition
Lost to Follow-up
1
1
Study Completion Disposition
Death
1
0
Study Completion Disposition
IWRS issue, patient refused, SAE, randomized in error, patient did not take IMP or attend visits.
3
3

Baseline Characteristics

Safety and Efficacy Study of Cefepime/VNRX-5133 in Patients With Complicated Urinary Tract Infections

Baseline characteristics by cohort

Baseline characteristics by cohort
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=441 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=220 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Total
n=661 Participants
Total of all reporting groups
Age, Continuous
56.2 years
STANDARD_DEVIATION 17.43 • n=5 Participants
55.8 years
STANDARD_DEVIATION 18.15 • n=7 Participants
56.1 years
STANDARD_DEVIATION 17.66 • n=5 Participants
Age, Customized
Age Categories (years) · <65
275 Participants
n=5 Participants
137 Participants
n=7 Participants
412 Participants
n=5 Participants
Age, Customized
Age Categories (years) · 65 - 75
111 Participants
n=5 Participants
56 Participants
n=7 Participants
167 Participants
n=5 Participants
Age, Customized
Age Categories (years) · >75
55 Participants
n=5 Participants
27 Participants
n=7 Participants
82 Participants
n=5 Participants
Sex: Female, Male
Female
248 Participants
n=5 Participants
115 Participants
n=7 Participants
363 Participants
n=5 Participants
Sex: Female, Male
Male
193 Participants
n=5 Participants
105 Participants
n=7 Participants
298 Participants
n=5 Participants
Ethnicity (NIH/OMB)
Hispanic or Latino
47 Participants
n=5 Participants
20 Participants
n=7 Participants
67 Participants
n=5 Participants
Ethnicity (NIH/OMB)
Not Hispanic or Latino
393 Participants
n=5 Participants
199 Participants
n=7 Participants
592 Participants
n=5 Participants
Ethnicity (NIH/OMB)
Unknown or Not Reported
1 Participants
n=5 Participants
1 Participants
n=7 Participants
2 Participants
n=5 Participants
Race (NIH/OMB)
American Indian or Alaska Native
4 Participants
n=5 Participants
1 Participants
n=7 Participants
5 Participants
n=5 Participants
Race (NIH/OMB)
Asian
36 Participants
n=5 Participants
17 Participants
n=7 Participants
53 Participants
n=5 Participants
Race (NIH/OMB)
Native Hawaiian or Other Pacific Islander
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
Race (NIH/OMB)
Black or African American
3 Participants
n=5 Participants
3 Participants
n=7 Participants
6 Participants
n=5 Participants
Race (NIH/OMB)
White
386 Participants
n=5 Participants
191 Participants
n=7 Participants
577 Participants
n=5 Participants
Race (NIH/OMB)
More than one race
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
Race (NIH/OMB)
Unknown or Not Reported
12 Participants
n=5 Participants
8 Participants
n=7 Participants
20 Participants
n=5 Participants

PRIMARY outcome

Timeframe: Assessed at Test of Cure visit (occurred once per participant between Study Days 19 to 23)

Population: The microITT analysis population consists of all patients in the ITT analysis population who had a positive study entry urine culture defined as ≥10\^5 CFU/mL of a gram-negative pathogen(s) against which both cefepime/VNRX-5133 and meropenem have antibacterial activity AND those patients who had no more than 2 microorganisms identified in the study entry culture regardless of colony count.

Microbiologic success is eradication defined as demonstration that any gram-negative bacterial pathogen found at study entry (≥10\^5 CFU/mL) is eradicated to \<10\^3 CFU/mL. Clinical success is defined as symptomatic resolution or return to pre-morbid baseline of all UTI-core symptoms and patient is alive, and patient has not received additional antibacterial therapy for cUTI.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=293 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=143 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Composite Success at Test of Cure (TOC) in the Microbiological Intent-to-treat (microITT) Population
207 Participants
83 Participants

SECONDARY outcome

Timeframe: Assessed at Test of Cure visit (occurred once per participant between Study Days 19 to 23)

Population: The microITT analysis population consists of all patients in the ITT analysis population who had a positive study entry urine culture defined as ≥10\^5 CFU/mL of a gram-negative pathogen(s) against which both cefepime/VNRX-5133 and meropenem have antibacterial activity AND those patients who had no more than 2 microorganisms identified in the study entry culture regardless of colony count.

Microbiologic success is eradication defined as demonstration that any gram-negative bacterial pathogen found at study entry (≥10\^5 CFU/mL) is eradicated to \<10\^3 CFU/mL.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=293 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=143 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Microbiologic Success at Test of Cure (TOC) in the microITT Population
229 Participants
95 Participants

SECONDARY outcome

Timeframe: Assessed at Test of Cure visit (occurred once per participant between Study Days 19 to 23)

Population: The microITT analysis population consists of all patients in the ITT analysis population who had a positive study entry urine culture defined as ≥10\^5 CFU/mL of a gram-negative pathogen(s) against which both cefepime/VNRX-5133 and meropenem have antibacterial activity AND those patients who had no more than 2 microorganisms identified in the study entry culture regardless of colony count.

Symptomatic resolution or return to pre-morbid baseline of all UTI-core symptoms and patient is alive, and patient has not received additional antibacterial therapy for cUTI.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=293 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=143 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Clinical Success at Test of Cure (TOC) in the microITT Population
251 Participants
116 Participants

SECONDARY outcome

Timeframe: Assessed at Test of Cure visit (occurred once per participant between Study Days 19 to 23)

Population: The extended microITT analysis population consists of all patients in the ITT analysis population who had a positive study entry urine culture defined as ≥10\^5 CFU/mL of a gram-negative pathogen(s) against which at least 1 study drug (cefepime/VNRX-5133 and/or meropenem) have antibacterial activity AND those patients who had no more than 2 microorganisms identified in the study entry culture regardless of colony count.

Microbiologic success is eradication defined as demonstration that any gram-negative bacterial pathogen found at study entry (≥10\^5 CFU/mL) is eradicated to \<10\^3 CFU/mL. Symptomatic clinical success is defined as symptomatic resolution or return to pre-morbid baseline of all UTI-core symptoms and patient is alive, and patient has not received additional antibacterial therapy for cUTI.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=305 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=147 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Composite Success at Test of Cure (TOC) in the Extended Microbiological Intent-to-treat (emicroITT) Population
216 Participants
86 Participants

SECONDARY outcome

Timeframe: Assessed within 24 hours after last IV dose (up to 15 days from start of treatment)

Population: The microITT analysis population consists of all patients in the ITT analysis population who had a positive study entry urine culture defined as ≥10\^5 CFU/mL of a gram-negative pathogen(s) against which both cefepime/VNRX-5133 and meropenem have antibacterial activity AND those patients who had no more than 2 microorganisms identified in the study entry culture regardless of colony count.

Microbiologic success is eradication defined as demonstration that any gram-negative bacterial pathogen found at study entry (≥10\^5 CFU/mL) is eradicated to \<10\^3 CFU/mL. Clinical success is defined as symptomatic resolution or return to pre-morbid baseline of all UTI-core symptoms and patient is alive, and patient has not received additional antibacterial therapy for cUTI.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=293 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=143 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Composite Success at End of Treatment (EOT) in the microITT Population
261 Participants
123 Participants

SECONDARY outcome

Timeframe: Assessed within 24 hours after last IV dose (up to 15 days from start of treatment)

Population: The microITT analysis population consists of all patients in the ITT analysis population who had a positive study entry urine culture defined as ≥10\^5 CFU/mL of a gram-negative pathogen(s) against which both cefepime/VNRX-5133 and meropenem have antibacterial activity AND those patients who had no more than 2 microorganisms identified in the study entry culture regardless of colony count.

Microbiologic success is eradication defined as demonstration that any gram-negative bacterial pathogen found at study entry (≥10\^5 CFU/mL) is eradicated to \<10\^3 CFU/mL.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=293 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=143 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Microbiological Success at End of Treatment (EOT) in the microITT Population
284 Participants
139 Participants

SECONDARY outcome

Timeframe: Assessed within 24 hours after last IV dose (up to 15 days from start of treatment)

Population: The microITT analysis population consists of all patients in the ITT analysis population who had a positive study entry urine culture defined as ≥10\^5 CFU/mL of a gram-negative pathogen(s) against which both cefepime/VNRX-5133 and meropenem have antibacterial activity AND those patients who had no more than 2 microorganisms identified in the study entry culture regardless of colony count.

Clinical success is defined as symptomatic resolution or return to pre-morbid baseline of all UTI-core symptoms and patient is alive, and patient has not received additional antibacterial therapy for cUTI.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=293 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=143 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Clinical Success at End of Treatment (EOT) in the microITT Population
265 Participants
127 Participants

SECONDARY outcome

Timeframe: Assessed at Late Follow Up visit (occurred once per participant between Study Days 28 to 35)

Population: The microITT analysis population consists of all patients in the ITT analysis population who had a positive study entry urine culture defined as ≥10\^5 CFU/mL of a gram-negative pathogen(s) against which both cefepime/VNRX-5133 and meropenem have antibacterial activity AND those patients who had no more than 2 microorganisms identified in the study entry culture regardless of colony count.

Microbiologic success is eradication defined as demonstration that any gram-negative bacterial pathogen found at study entry (≥10\^5 CFU/mL) is eradicated to \<10\^3 CFU/mL. Clinical success is defined as symptomatic resolution or return to pre-morbid baseline of all UTI-core symptoms and patient is alive, and patient has not received additional antibacterial therapy for cUTI.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=293 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=143 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Composite Success at Late Follow Up (LFU) in the microITT Population
187 Participants
74 Participants

SECONDARY outcome

Timeframe: Assessed at Late Follow Up visit (occurred once per participant between Study Days 28 to 35)

Population: The microITT analysis population consists of all patients in the ITT analysis population who had a positive study entry urine culture defined as ≥10\^5 CFU/mL of a gram-negative pathogen(s) against which both cefepime/VNRX-5133 and meropenem have antibacterial activity AND those patients who had no more than 2 microorganisms identified in the study entry culture regardless of colony count.

Microbiologic success is eradication defined as demonstration that any gram-negative bacterial pathogen found at study entry (≥10\^5 CFU/mL) is eradicated to \<10\^3 CFU/mL.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=293 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=143 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Microbiological Success at Late Follow Up (LFU) in the microITT Population
207 Participants
90 Participants

SECONDARY outcome

Timeframe: Assessed at Late Follow Up visit (occurred once per participant between Study Days 28 to 35)

Population: The microITT analysis population consists of all patients in the ITT analysis population who had a positive study entry urine culture defined as ≥10\^5 CFU/mL of a gram-negative pathogen(s) against which both cefepime/VNRX-5133 and meropenem have antibacterial activity AND those patients who had no more than 2 microorganisms identified in the study entry culture regardless of colony count.

Clinical success is defined as symptomatic resolution or return to pre-morbid baseline of all UTI-core symptoms and patient is alive, and patient has not received additional antibacterial therapy for cUTI.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=293 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=143 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Clinical Success at Late Follow Up (LFU) in the microITT Population
238 Participants
102 Participants

SECONDARY outcome

Timeframe: Assessed at Test of Cure visit (occurred once per participant between Study Days 19 to 23)

Population: The microITT analysis population consists of all patients in the ITT analysis population who had a positive study entry urine culture defined as ≥10\^5 CFU/mL of a gram-negative pathogen(s) against which both cefepime/VNRX-5133 and meropenem have antibacterial activity AND those patients who had no more than 2 microorganisms identified in the study entry culture regardless of colony count.

The proportion of patients with clinical success based on investigator opinion at TOC.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=293 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=143 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Investigator Opinion of Clinical Success at Test of Cure (TOC) in the microITT Population
271 Participants
128 Participants

SECONDARY outcome

Timeframe: Assessed within 24 hours after last IV dose (up to 15 days from start of treatment)

Population: The microITT analysis population consists of all patients in the ITT analysis population who had a positive study entry urine culture defined as ≥10\^5 CFU/mL of a gram-negative pathogen(s) against which both cefepime/VNRX-5133 and meropenem have antibacterial activity AND those patients who had no more than 2 microorganisms identified in the study entry culture regardless of colony count.

Microbiologic success is eradication defined as demonstration that any gram-negative bacterial pathogen found at study entry (≥10\^5 CFU/mL) is eradicated to \<10\^3 CFU/mL. Clinical success is defined as symptomatic resolution or return to pre-morbid baseline of all UTI-core symptoms and patient is alive, and patient has not received additional antibacterial therapy for cUTI.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=67 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=30 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Composite Success in Patients With Cefepime-Resistant Pathogens at End of Treatment (EOT) in the microITT Population
Cefepime-resistant Enterobacterales
57 Participants
26 Participants
Composite Success in Patients With Cefepime-Resistant Pathogens at End of Treatment (EOT) in the microITT Population
Cefepime-resistant Pseudomonas aeruginosa
1 Participants

SECONDARY outcome

Timeframe: Assessed within 24 hours after last IV dose (up to 15 days from start of treatment)

Population: The microITT analysis population consists of all patients in the ITT analysis population who had a positive study entry urine culture defined as ≥10\^5 CFU/mL of a gram-negative pathogen(s) against which both cefepime/VNRX-5133 and meropenem have antibacterial activity AND those patients who had no more than 2 microorganisms identified in the study entry culture regardless of colony count.

Microbiologic success is eradication defined as demonstration that any gram-negative bacterial pathogen found at study entry (≥10\^5 CFU/mL) is eradicated to \<10\^3 CFU/mL.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=67 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=30 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Microbiologic Success in Patients With Cefepime-Resistant Pathogens at End of Treatment (EOT) in the microITT Population
Cefepime-resistant Enterobacterales
65 Participants
28 Participants
Microbiologic Success in Patients With Cefepime-Resistant Pathogens at End of Treatment (EOT) in the microITT Population
Cefepime-resistant Pseudomonas aeruginosa
1 Participants

SECONDARY outcome

Timeframe: Assessed within 24 hours after last IV dose (up to 15 days from start of treatment)

Population: The microITT analysis population consists of all patients in the ITT analysis population who had a positive study entry urine culture defined as ≥10\^5 CFU/mL of a gram-negative pathogen(s) against which both cefepime/VNRX-5133 and meropenem have antibacterial activity AND those patients who had no more than 2 microorganisms identified in the study entry culture regardless of colony count.

Clinical success is defined as symptomatic resolution or return to pre-morbid baseline of all UTI-core symptoms and patient is alive, and patient has not received additional antibacterial therapy for cUTI.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=67 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=30 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Clinical Success in Patients With Cefepime-Resistant Pathogens at End of Treatment (EOT) in the microITT Population
Enterobacterales
57 Participants
28 Participants
Clinical Success in Patients With Cefepime-Resistant Pathogens at End of Treatment (EOT) in the microITT Population
Pseudomonas aeruginosa
1 Participants

SECONDARY outcome

Timeframe: Assessed at Test of Cure visit (occurred once per participant between Study Days 19 to 23)

Population: The microITT analysis population consists of all patients in the ITT analysis population who had a positive study entry urine culture defined as ≥10\^5 CFU/mL of a gram-negative pathogen(s) against which both cefepime/VNRX-5133 and meropenem have antibacterial activity AND those patients who had no more than 2 microorganisms identified in the study entry culture regardless of colony count.

Microbiologic success is eradication defined as demonstration that any gram-negative bacterial pathogen found at study entry (≥10\^5 CFU/mL) is eradicated to \<10\^3 CFU/mL. Clinical success is defined as symptomatic resolution or return to pre-morbid baseline of all UTI-core symptoms and patient is alive, and patient has not received additional antibacterial therapy for cUTI.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=67 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=30 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Composite Success in Patients With Cefepime-Resistant Pathogens at Test of Cure (TOC) in the microITT Population
Cefepime-resistant Enterobacterales
47 Participants
16 Participants
Composite Success in Patients With Cefepime-Resistant Pathogens at Test of Cure (TOC) in the microITT Population
Cefepime-resistant Pseudomonas aeruginosa
0 Participants

SECONDARY outcome

Timeframe: Assessed at Test of Cure visit (occurred once per participant between Study Days 19 to 23)

Population: The microITT analysis population consists of all patients in the ITT analysis population who had a positive study entry urine culture defined as ≥10\^5 CFU/mL of a gram-negative pathogen(s) against which both cefepime/VNRX-5133 and meropenem have antibacterial activity AND those patients who had no more than 2 microorganisms identified in the study entry culture regardless of colony count.

Microbiologic success is eradication defined as demonstration that any gram-negative bacterial pathogen found at study entry (≥10\^5 CFU/mL) is eradicated to \<10\^3 CFU/mL.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=67 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=30 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Microbiologic Success in Patients With Cefepime-Resistant Pathogens at Test of Cure (TOC) in the microITT Population
Cefepime-resistant Enterobacterales
50 Participants
18 Participants
Microbiologic Success in Patients With Cefepime-Resistant Pathogens at Test of Cure (TOC) in the microITT Population
Cefepime-resistant Pseudomonas aeruginosa
0 Participants

SECONDARY outcome

Timeframe: Assessed at Test of Cure visit (occurred once per participant between Study Days 19 to 23)

Population: The microITT analysis population consists of all patients in the ITT analysis population who had a positive study entry urine culture defined as ≥10\^5 CFU/mL of a gram-negative pathogen(s) against which both cefepime/VNRX-5133 and meropenem have antibacterial activity AND those patients who had no more than 2 microorganisms identified in the study entry culture regardless of colony count.

Clinical success is defined as symptomatic resolution or return to pre-morbid baseline of all UTI-core symptoms and patient is alive, and patient has not received additional antibacterial therapy for cUTI.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=67 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=30 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Clinical Success in Patients With Cefepime-Resistant Pathogens at Test of Cure (TOC) in the microITT Population
Enterbacterales
54 Participants
25 Participants
Clinical Success in Patients With Cefepime-Resistant Pathogens at Test of Cure (TOC) in the microITT Population
Pseudomonas aeruginosa
0 Participants

SECONDARY outcome

Timeframe: Assessed at Late Follow Up visit (occurred once per participant between Study Days 28 to 35)

Population: The microITT analysis population consists of all patients in the ITT analysis population who had a positive study entry urine culture defined as ≥10\^5 CFU/mL of a gram-negative pathogen(s) against which both cefepime/VNRX-5133 and meropenem have antibacterial activity AND those patients who had no more than 2 microorganisms identified in the study entry culture regardless of colony count.

Microbiologic success is eradication defined as demonstration that any gram-negative bacterial pathogen found at study entry (≥10\^5 CFU/mL) is eradicated to \<10\^3 CFU/mL. Clinical success is defined as symptomatic resolution or return to pre-morbid baseline of all UTI-core symptoms and patient is alive, and patient has not received additional antibacterial therapy for cUTI.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=67 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=30 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Composite Success in Patients With Cefepime-Resistant Pathogens at Late Follow Up (LFU) in the microITT Population
Cefepime-resistant Enterobacterales
45 Participants
13 Participants
Composite Success in Patients With Cefepime-Resistant Pathogens at Late Follow Up (LFU) in the microITT Population
Cefepime-resistant Pseudomonas aeruginosa
0 Participants

SECONDARY outcome

Timeframe: Assessed at Late Follow Up visit (occurred once per participant between Study Days 28 to 35)

Population: The microITT analysis population consists of all patients in the ITT analysis population who had a positive study entry urine culture defined as ≥10\^5 CFU/mL of a gram-negative pathogen(s) against which both cefepime/VNRX-5133 and meropenem have antibacterial activity AND those patients who had no more than 2 microorganisms identified in the study entry culture regardless of colony count.

Microbiologic success is eradication defined as demonstration that any gram-negative bacterial pathogen found at study entry (≥10\^5 CFU/mL) is eradicated to \<10\^3 CFU/mL.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=67 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=30 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Microbiologic Success in Patients With Cefepime-Resistant Pathogens at Late Follow Up (LFU) in the microITT Population
Cefepime-resistant Enterobacterales
48 Participants
16 Participants
Microbiologic Success in Patients With Cefepime-Resistant Pathogens at Late Follow Up (LFU) in the microITT Population
Cefepime-resistant Pseudomonas aeruginosa
0 Participants

SECONDARY outcome

Timeframe: Assessed at Late Follow Up visit (occurred once per participant between Study Days 28 to 35)

Population: The microITT analysis population consists of all patients in the ITT analysis population who had a positive study entry urine culture defined as ≥10\^5 CFU/mL of a gram-negative pathogen(s) against which both cefepime/VNRX-5133 and meropenem have antibacterial activity AND those patients who had no more than 2 microorganisms identified in the study entry culture regardless of colony count.

Clinical success is defined as symptomatic resolution or return to pre-morbid baseline of all UTI-core symptoms and patient is alive, and patient has not received additional antibacterial therapy for cUTI.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=67 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=30 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Clinical Success in Patients With Cefepime-Resistant Pathogens at Late Follow Up (LFU) in the microITT Population
Enterobacterales
49 Participants
20 Participants
Clinical Success in Patients With Cefepime-Resistant Pathogens at Late Follow Up (LFU) in the microITT Population
Pseudomonas aeruginosa
0 Participants

SECONDARY outcome

Timeframe: Assessed within 24 hours after last IV dose (up to 15 days from start of treatment)

Population: All patients who meet the criteria for the microITT population AND had a diagnosis of cUTI; received treatment for ≥48 hours; were evaluated at EOT with a response that was not indeterminate; did not violate prior antibacterials exclusion or received concomitant antibiotic therapy with activity against baseline pathogens except for patients failing study drug; or had other confounding factors that interfered with the assessment of outcome including unblinding.

Microbiologic success is eradication defined as demonstration that any gram-negative bacterial pathogen found at study entry (≥10\^5 CFU/mL) is eradicated to \<10\^3 CFU/mL. Clinical success is defined as symptomatic resolution or return to pre-morbid baseline of all UTI-core symptoms and patient is alive, and patient has not received additional antibacterial therapy for cUTI.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=282 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=137 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Composite Success at End of Treatment (EOT) in the Microbiologically-Evaluable (ME) Population
259 Participants
121 Participants

SECONDARY outcome

Timeframe: Assessed within 24 hours after last IV dose (up to 15 days from start of treatment)

Population: All patients who meet the criteria for the microITT population AND had a diagnosis of cUTI; received treatment for ≥48 hours; were evaluated at EOT with a response that was not indeterminate; did not violate prior antibacterials exclusion or received concomitant antibiotic therapy with activity against baseline pathogens except for patients failing study drug; or had other confounding factors that interfered with the assessment of outcome including unblinding.

Microbiologic success is eradication defined as demonstration that any gram-negative bacterial pathogen found at study entry (≥10\^5 CFU/mL) is eradicated to \<10\^3 CFU/mL.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=282 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=137 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Microbiologic Success at End of Treatment (EOT) in the ME Population
279 Participants
137 Participants

SECONDARY outcome

Timeframe: Assessed at Test of Cure visit (occurred once per participant between Study Days 19 to 23)

Population: All patients who meet the criteria for the microITT population AND had a diagnosis of cUTI; received treatment for ≥48 hours; were evaluated at TOC with a response that was not indeterminate; did not violate prior antibacterials exclusion or received concomitant antibiotic therapy with activity against baseline pathogens except for patients failing study drug; or had other confounding factors that interfered with the assessment of outcome including unblinding.

Microbiologic success is eradication defined as demonstration that any gram-negative bacterial pathogen found at study entry (≥10\^5 CFU/mL) is eradicated to \<10\^3 CFU/mL. Symptomatic clinical success is defined as symptomatic resolution or return to pre-morbid baseline of all UTI-core symptoms and patient is alive, and patient has not received additional antibacterial therapy for cUTI.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=261 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=127 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Composite Success at Test of Cure (TOC) in the ME Population
195 Participants
76 Participants

SECONDARY outcome

Timeframe: Assessed at Test of Cure visit (occurred once per participant between Study Days 19 to 23)

Population: All patients who meet the criteria for the microITT population AND had a diagnosis of cUTI; received treatment for ≥48 hours; were evaluated at TOC with a response that was not indeterminate; did not violate prior antibacterials exclusion or received concomitant antibiotic therapy with activity against baseline pathogens except for patients failing study drug; or had other confounding factors that interfered with the assessment of outcome including unblinding.

Microbiologic success is eradication defined as demonstration that any gram-negative bacterial pathogen found at study entry (≥10\^5 CFU/mL) is eradicated to \<10\^3 CFU/mL.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=261 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=127 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Microbiologic Success at Test of Cure (TOC) in the ME Population
214 Participants
88 Participants

SECONDARY outcome

Timeframe: Assessed at Late Follow Up visit (occurred once per participant between Study Days 28 to 35)

Population: All patients who meet the criteria for the microITT population AND had a diagnosis of cUTI; received treatment for ≥48 hours; were evaluated at LFU with a response that was not indeterminate; did not violate prior antibacterials exclusion or received concomitant antibiotic therapy with activity against baseline pathogens except for patients failing study drug; or had other confounding factors that interfered with the assessment of outcome including unblinding.

Microbiologic success is eradication defined as demonstration that any gram-negative bacterial pathogen found at study entry (≥10\^5 CFU/mL) is eradicated to \<10\^3 CFU/mL. Symptomatic clinical success is defined as symptomatic resolution or return to pre-morbid baseline of all UTI-core symptoms and patient is alive, and patient has not received additional antibacterial therapy for cUTI.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=262 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=128 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Composite Success at Late Follow Up (LFU) in the ME Population
178 Participants
69 Participants

SECONDARY outcome

Timeframe: Assessed at Late Follow Up visit (occurred once per participant between Study Days 28 to 35)

Population: All patients who meet the criteria for the microITT population AND had a diagnosis of cUTI; received treatment for ≥48 hours; were evaluated at LFU with a response that was not indeterminate; did not violate prior antibacterials exclusion or received concomitant antibiotic therapy with activity against baseline pathogens except for patients failing study drug; or had other confounding factors that interfered with the assessment of outcome including unblinding.

Microbiologic success is eradication defined as demonstration that any gram-negative bacterial pathogen found at study entry (≥10\^5 CFU/mL) is eradicated to \<10\^3 CFU/mL.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=262 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=128 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Microbiologic Success at Late Follow Up (LFU) in the ME Population
192 Participants
84 Participants

SECONDARY outcome

Timeframe: Assessed within 24 hours after last IV dose (up to 15 days from start of treatment)

Population: All patients who meet the criteria for the microITT population AND had a diagnosis of cUTI; received treatment for ≥48 hours; were evaluated at EOT with a response that was not indeterminate; did not violate prior antibacterials exclusion or received concomitant antibiotic therapy with activity against baseline pathogens except for patients failing study drug; or had other confounding factors that interfered with the assessment of outcome including unblinding.

Microbiologic success is eradication defined as demonstration that any gram-negative bacterial pathogen found at study entry (≥10\^5 CFU/mL) is eradicated to \<10\^3 CFU/mL. Symptomatic clinical success is defined as symptomatic resolution or return to pre-morbid baseline of all UTI-core symptoms and patient is alive, and patient has not received additional antibacterial therapy for cUTI.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=64 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=28 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Composite Success in Patients With Cefepime-Resistant Pathogens at the End of Treatment (EOT) in the ME Population
Cefepime-resistant Enterobacterales
56 Participants
26 Participants
Composite Success in Patients With Cefepime-Resistant Pathogens at the End of Treatment (EOT) in the ME Population
Cefepime-resistant Pseudomonas aeruginosa
1 Participants

SECONDARY outcome

Timeframe: Assessed within 24 hours after last IV dose (up to 15 days from start of treatment)

Population: All patients who meet the criteria for the microITT population AND had a diagnosis of cUTI; received treatment for ≥48 hours; were evaluated at EOT with a response that was not indeterminate; did not violate prior antibacterials exclusion or received concomitant antibiotic therapy with activity against baseline pathogens except for patients failing study drug; or had other confounding factors that interfered with the assessment of outcome including unblinding.

Microbiologic success is eradication defined as demonstration that any gram-negative bacterial pathogen found at study entry (≥10\^5 CFU/mL) is eradicated to \<10\^3 CFU/mL.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=64 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=28 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Microbiologic Success in Patients With Cefepime-Resistant Pathogens at the End of Treatment (EOT) in the ME Population
Cefepime-resistant Enterobacterales
62 Participants
28 Participants
Microbiologic Success in Patients With Cefepime-Resistant Pathogens at the End of Treatment (EOT) in the ME Population
Cefepime-resistant Pseudomonas aeruginosa
1 Participants

SECONDARY outcome

Timeframe: Assessed at Test of Cure visit (occurred once per participant between Study Days 19 to 23)

Population: All patients who meet the criteria for the microITT population AND had a diagnosis of cUTI; received treatment for ≥48 hours; were evaluated at TOC with a response that was not indeterminate; did not violate prior antibacterials exclusion or received concomitant antibiotic therapy with activity against baseline pathogens except for patients failing study drug; or had other confounding factors that interfered with the assessment of outcome including unblinding.

Microbiologic success is eradication defined as demonstration that any gram-negative bacterial pathogen found at study entry (≥10\^5 CFU/mL) is eradicated to \<10\^3 CFU/mL. Symptomatic clinical success is defined as symptomatic resolution or return to pre-morbid baseline of all UTI-core symptoms and patient is alive, and patient has not received additional antibacterial therapy for cUTI.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=58 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=24 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Composite Success in Patients With Cefepime-Resistant Pathogens at Test of Cure (TOC) in the ME Population
Cefepime-resistant Enterobacterales
44 Participants
12 Participants
Composite Success in Patients With Cefepime-Resistant Pathogens at Test of Cure (TOC) in the ME Population
Cefepime-resistant Pseudomonas aeruginosa
0 Participants

SECONDARY outcome

Timeframe: Assessed at Test of Cure visit (occurred once per participant between Study Days 19 to 23)

Population: All patients who meet the criteria for the microITT population AND had a diagnosis of cUTI; received treatment for ≥48 hours; were evaluated at TOC with a response that was not indeterminate; did not violate prior antibacterials exclusion or received concomitant antibiotic therapy with activity against baseline pathogens except for patients failing study drug; or had other confounding factors that interfered with the assessment of outcome including unblinding.

Microbiologic success is eradication defined as demonstration that any gram-negative bacterial pathogen found at study entry (≥10\^5 CFU/mL) is eradicated to \<10\^3 CFU/mL.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=58 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=24 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Microbiologic Success in Patients With Cefepime-Resistant Pathogens at Test of Cure (TOC) in the ME Population
Cefepime-resistant Enterobacterales
46 Participants
14 Participants
Microbiologic Success in Patients With Cefepime-Resistant Pathogens at Test of Cure (TOC) in the ME Population
Cefepime-resistant Pseudomonas aeruginosa
0 Participants

SECONDARY outcome

Timeframe: Assessed at Late Follow Up visit (occurred once per participant between Study Days 28 to 35)

Population: All patients who meet the criteria for the microITT population AND had a diagnosis of cUTI; received treatment for ≥48 hours; were evaluated at LFU with a response that was not indeterminate; did not violate prior antibacterials exclusion or received concomitant antibiotic therapy with activity against baseline pathogens except for patients failing study drug; or had other confounding factors that interfered with the assessment of outcome including unblinding.

Microbiologic success is eradication defined as demonstration that any gram-negative bacterial pathogen found at study entry (≥10\^5 CFU/mL) is eradicated to \<10\^3 CFU/mL. Symptomatic clinical success is defined as symptomatic resolution or return to pre-morbid baseline of all UTI-core symptoms and patient is alive, and patient has not received additional antibacterial therapy for cUTI.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=60 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=26 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Composite Success in Cefepime-Resistant Pathogens at Late Follow Up (LFU) in the ME Population
Cefepime-resistant Enterobacterales
44 Participants
11 Participants
Composite Success in Cefepime-Resistant Pathogens at Late Follow Up (LFU) in the ME Population
Cefepime-resistant Pseudomonas aeruginosa
0 Participants

SECONDARY outcome

Timeframe: Assessed at Late Follow Up visit (occurred once per participant between Study Days 28 to 35)

Population: All patients who meet the criteria for the microITT population AND had a diagnosis of cUTI; received treatment for ≥48 hours; were evaluated at LFU with a response that was not indeterminate; did not violate prior antibacterials exclusion or received concomitant antibiotic therapy with activity against baseline pathogens except for patients failing study drug; or had other confounding factors that interfered with the assessment of outcome including unblinding.

Microbiologic success is eradication defined as demonstration that any gram-negative bacterial pathogen found at study entry (≥10\^5 CFU/mL) is eradicated to \<10\^3 CFU/mL.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=60 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=26 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Microbiologic Success in Cefepime-Resistant Pathogens at Late Follow Up (LFU) in the ME Population
Cefepime-resistant Enterobacterales
45 Participants
14 Participants
Microbiologic Success in Cefepime-Resistant Pathogens at Late Follow Up (LFU) in the ME Population
Cefepime-resistant Pseudomonas aeruginosa
0 Participants

SECONDARY outcome

Timeframe: Assessed within 24 hours after last IV dose (up to 15 days from start of treatment)

Population: The CE analysis population consists of all patients in the ITT analysis population who had a diagnosis of cUTI; received treatment for ≥48 hours; were evaluated at EOT with a response that was not indeterminate; did not violate prior antibacterials exclusion or received concomitant antibiotic therapy with activity against baseline pathogens except for patients failing study drug; or had other confounding factors that interfered with the assessment of outcome including unblinding.

Symptomatic clinical success is defined as symptomatic resolution or return to pre-morbid baseline of all UTI-core symptoms and patient is alive, and patient has not received additional antibacterial therapy for cUTI.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=425 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=211 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Clinical Success at End of Treatment (EOT) in the Clinically Evaluable (CE) Population
384 Participants
187 Participants

SECONDARY outcome

Timeframe: Assessed at Test of Cure visit (occurred once per participant between Study Days 19 to 23)

Population: The CE analysis population consists of all patients in the ITT analysis population who had a diagnosis of cUTI; received treatment for ≥48 hours; were evaluated at EOT with a response that was not indeterminate; did not violate prior antibacterials exclusion or received concomitant antibiotic therapy with activity against baseline pathogens except for patients failing study drug; or had other confounding factors that interfered with the assessment of outcome including unblinding.

Symptomatic clinical success is defined as symptomatic resolution or return to pre-morbid baseline of all UTI-core symptoms and patient is alive, and patient has not received additional antibacterial therapy for cUTI.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=392 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=196 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Clinical Success at Test of Cure (TOC) in the CE Population
343 Participants
162 Participants

SECONDARY outcome

Timeframe: Assessed at Late Follow Up visit (occurred once per participant between Study Days 28 to 35)

Population: The CE analysis population consists of all patients in the ITT analysis population who had a diagnosis of cUTI; received treatment for ≥48 hours; were evaluated at EOT with a response that was not indeterminate; did not violate prior antibacterials exclusion or received concomitant antibiotic therapy with activity against baseline pathogens except for patients failing study drug; or had other confounding factors that interfered with the assessment of outcome including unblinding.

Symptomatic clinical success is defined as symptomatic resolution or return to pre-morbid baseline of all UTI-core symptoms and patient is alive, and patient has not received additional antibacterial therapy for cUTI.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=387 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=190 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Clinical Success at Late Follow Up (LFU) in the CE Population
321 Participants
142 Participants

SECONDARY outcome

Timeframe: Assessed within 24 hours after last IV dose (up to 15 days from start of treatment)

Population: The CE analysis population consists of all patients in the ITT analysis population who had a diagnosis of cUTI; received treatment for ≥48 hours; were evaluated at EOT with a response that was not indeterminate; did not violate prior antibacterials exclusion or received concomitant antibiotic therapy with activity against baseline pathogens except for patients failing study drug; or had other confounding factors that interfered with the assessment of outcome including unblinding.

Symptomatic clinical success is defined as symptomatic resolution or return to pre-morbid baseline of all UTI-core symptoms and patient is alive, and patient has not received additional antibacterial therapy for cUTI.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=76 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=35 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Clinical Success in Patients With Cefepime-Resistant Pathogens at End of Treatment (EOT) in the CE Population
Enterobacterales
63 Participants
31 Participants
Clinical Success in Patients With Cefepime-Resistant Pathogens at End of Treatment (EOT) in the CE Population
Pseudomonas aeruginosa
6 Participants
2 Participants

SECONDARY outcome

Timeframe: Assessed at Test of Cure visit (occurred once per participant between Study Days 19 to 23)

Population: The CE analysis population consists of all patients in the ITT analysis population who had a diagnosis of cUTI; received treatment for ≥48 hours; were evaluated at EOT with a response that was not indeterminate; did not violate prior antibacterials exclusion or received concomitant antibiotic therapy with activity against baseline pathogens except for patients failing study drug; or had other confounding factors that interfered with the assessment of outcome including unblinding.

Symptomatic clinical success is defined as symptomatic resolution or return to pre-morbid baseline of all UTI-core symptoms and patient is alive, and patient has not received additional antibacterial therapy for cUTI.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=70 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=30 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Clinical Success in Patients With Cefepime-Resistant Pathogens at Test of Cure (TOC) in the CE Population
Enterobacterales
56 Participants
23 Participants
Clinical Success in Patients With Cefepime-Resistant Pathogens at Test of Cure (TOC) in the CE Population
Pseudomonas aeruginosa
4 Participants
2 Participants

SECONDARY outcome

Timeframe: Assessed at Late Follow Up visit (occurred once per participant between Study Days 28 to 35)

Population: The CE analysis population consists of all patients in the ITT analysis population who had a diagnosis of cUTI; received treatment for ≥48 hours; were evaluated at EOT with a response that was not indeterminate; did not violate prior antibacterials exclusion or received concomitant antibiotic therapy with activity against baseline pathogens except for patients failing study drug; or had other confounding factors that interfered with the assessment of outcome including unblinding.

Symptomatic clinical success is defined as symptomatic resolution or return to pre-morbid baseline of all UTI-core symptoms and patient is alive, and patient has not received additional antibacterial therapy for cUTI.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=70 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=30 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Clinical Success in Patients With Cefepime-Resistant Pathogens at Late Follow Up (LFU) in the CE Population
Enterobacterales
52 Participants
19 Participants
Clinical Success in Patients With Cefepime-Resistant Pathogens at Late Follow Up (LFU) in the CE Population
Pseudomonas aeruginosa
3 Participants
1 Participants

SECONDARY outcome

Timeframe: Assessed within 24 hours after last IV dose (up to 15 days from start of treatment)

Population: The microITT analysis population consists of all patients in the ITT analysis population who had a positive study entry urine culture defined as ≥10\^5 CFU/mL of a gram-negative pathogen(s) against which both cefepime/VNRX-5133 and meropenem have antibacterial activity AND those patients who had no more than 2 microorganisms identified in the study entry culture regardless of colony count.

Per-pathogen eradication by baseline gram-negative pathogens. The number analyzed corresponds to the number of specified pathogens. The number is the percent of the specified pathogen identified at baseline in each treatment group that had been eradicated.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=297 pathogens
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=147 pathogens
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Per-Pathogen Microbiologic Eradication at End of Treatment (EOT) in the microITT Population
Citrobacter koseri
1 pathogens
1 pathogens
Per-Pathogen Microbiologic Eradication at End of Treatment (EOT) in the microITT Population
Enterobacter cloacae complex
14 pathogens
3 pathogens
Per-Pathogen Microbiologic Eradication at End of Treatment (EOT) in the microITT Population
Providencia rettgeri
1 pathogens
Per-Pathogen Microbiologic Eradication at End of Treatment (EOT) in the microITT Population
Pseudomonas aeruginosa
11 pathogens
6 pathogens
Per-Pathogen Microbiologic Eradication at End of Treatment (EOT) in the microITT Population
Citrobacter freundii complex
2 pathogens
2 pathogens
Per-Pathogen Microbiologic Eradication at End of Treatment (EOT) in the microITT Population
Escherichia coli
197 pathogens
95 pathogens
Per-Pathogen Microbiologic Eradication at End of Treatment (EOT) in the microITT Population
Klebsiella aerogenes
1 pathogens
1 pathogens
Per-Pathogen Microbiologic Eradication at End of Treatment (EOT) in the microITT Population
Klebsiella oxytoca
5 pathogens
1 pathogens
Per-Pathogen Microbiologic Eradication at End of Treatment (EOT) in the microITT Population
Klebsiella pneumoniae
37 pathogens
20 pathogens
Per-Pathogen Microbiologic Eradication at End of Treatment (EOT) in the microITT Population
Klebsiella variicola
1 pathogens
1 pathogens
Per-Pathogen Microbiologic Eradication at End of Treatment (EOT) in the microITT Population
Kluyvera ascorbata
1 pathogens
Per-Pathogen Microbiologic Eradication at End of Treatment (EOT) in the microITT Population
Morganella morganii
2 pathogens
2 pathogens
Per-Pathogen Microbiologic Eradication at End of Treatment (EOT) in the microITT Population
Proteus hauseri
1 pathogens
Per-Pathogen Microbiologic Eradication at End of Treatment (EOT) in the microITT Population
Proteus mirabilis
10 pathogens
10 pathogens
Per-Pathogen Microbiologic Eradication at End of Treatment (EOT) in the microITT Population
Proteus penneri
1 pathogens
Per-Pathogen Microbiologic Eradication at End of Treatment (EOT) in the microITT Population
Proteus vulgaris
2 pathogens
Per-Pathogen Microbiologic Eradication at End of Treatment (EOT) in the microITT Population
Serratia marcescens
2 pathogens

SECONDARY outcome

Timeframe: Assessed at Test of Cure visit (occurred once per participant between Study Days 19 to 23)

Population: The microITT analysis population consists of all patients in the ITT analysis population who had a positive study entry urine culture defined as ≥10\^5 CFU/mL of a gram-negative pathogen(s) against which both cefepime/VNRX-5133 and meropenem have antibacterial activity AND those patients who had no more than 2 microorganisms identified in the study entry culture regardless of colony count.

Per-pathogen eradication by baseline gram-negative pathogens. The number analyzed corresponds to the number of specified pathogens. The number is the percent of the specified pathogen identified at baseline in each treatment group that had been eradicated.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=297 pathogens
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=147 pathogens
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Per-Pathogen Microbiologic Eradication at Test of Cure (TOC) in the microITT Population
Citrobacter freundii complex
2 pathogens
2 pathogens
Per-Pathogen Microbiologic Eradication at Test of Cure (TOC) in the microITT Population
Citrobacter koseri
0 pathogens
1 pathogens
Per-Pathogen Microbiologic Eradication at Test of Cure (TOC) in the microITT Population
Enterobacter cloacae complex
12 pathogens
1 pathogens
Per-Pathogen Microbiologic Eradication at Test of Cure (TOC) in the microITT Population
Escherichia coli
165 pathogens
67 pathogens
Per-Pathogen Microbiologic Eradication at Test of Cure (TOC) in the microITT Population
Klebsiella aerogenes
0 pathogens
0 pathogens
Per-Pathogen Microbiologic Eradication at Test of Cure (TOC) in the microITT Population
Klebsiella oxytoca
5 pathogens
1 pathogens
Per-Pathogen Microbiologic Eradication at Test of Cure (TOC) in the microITT Population
Klebsiella pneumoniae
27 pathogens
14 pathogens
Per-Pathogen Microbiologic Eradication at Test of Cure (TOC) in the microITT Population
Klebsiella varricola
1 pathogens
1 pathogens
Per-Pathogen Microbiologic Eradication at Test of Cure (TOC) in the microITT Population
Kluyvera ascorbata
1 pathogens
Per-Pathogen Microbiologic Eradication at Test of Cure (TOC) in the microITT Population
Morganella morganii
2 pathogens
2 pathogens
Per-Pathogen Microbiologic Eradication at Test of Cure (TOC) in the microITT Population
Proteus hauseri
0 pathogens
Per-Pathogen Microbiologic Eradication at Test of Cure (TOC) in the microITT Population
Proteus mirabilis
9 pathogens
5 pathogens
Per-Pathogen Microbiologic Eradication at Test of Cure (TOC) in the microITT Population
Proteus penneri
1 pathogens
Per-Pathogen Microbiologic Eradication at Test of Cure (TOC) in the microITT Population
Proteus vulgaris
1 pathogens
Per-Pathogen Microbiologic Eradication at Test of Cure (TOC) in the microITT Population
Providencia rettgeri
1 pathogens
Per-Pathogen Microbiologic Eradication at Test of Cure (TOC) in the microITT Population
Serratia marcescens
2 pathogens
Per-Pathogen Microbiologic Eradication at Test of Cure (TOC) in the microITT Population
Pseudomonas aeruginosa
5 pathogens
4 pathogens

SECONDARY outcome

Timeframe: Assessed at Late Follow Up visit (occurred once per participant between Study Days 28 to 35)

Population: The microITT analysis population consists of all patients in the ITT analysis population who had a positive study entry urine culture defined as ≥10\^5 CFU/mL of a gram-negative pathogen(s) against which both cefepime/VNRX-5133 and meropenem have antibacterial activity AND those patients who had no more than 2 microorganisms identified in the study entry culture regardless of colony count.

Per-pathogen eradication by baseline gram-negative pathogens. The number analyzed corresponds to the number of specified pathogens. The number is the percent of the specified pathogen identified at baseline in each treatment group that had been eradicated.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=297 pathogens
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=147 pathogens
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Per-Pathogen Microbiologic Eradication at Late Follow Up (LFU) in the microITT Population
Enterobacter cloacae complex
12 pathogens
1 pathogens
Per-Pathogen Microbiologic Eradication at Late Follow Up (LFU) in the microITT Population
Escherichia coli
141 pathogens
61 pathogens
Per-Pathogen Microbiologic Eradication at Late Follow Up (LFU) in the microITT Population
Klebsiella aerogenes
0 pathogens
0 pathogens
Per-Pathogen Microbiologic Eradication at Late Follow Up (LFU) in the microITT Population
Klebsiella oxytoca
4 pathogens
1 pathogens
Per-Pathogen Microbiologic Eradication at Late Follow Up (LFU) in the microITT Population
Kluyvera ascorbata
1 pathogens
Per-Pathogen Microbiologic Eradication at Late Follow Up (LFU) in the microITT Population
Morganella morganii
2 pathogens
2 pathogens
Per-Pathogen Microbiologic Eradication at Late Follow Up (LFU) in the microITT Population
Proteus hauseri
0 pathogens
Per-Pathogen Microbiologic Eradication at Late Follow Up (LFU) in the microITT Population
Pseudomonas aeruginosa
5 pathogens
4 pathogens
Per-Pathogen Microbiologic Eradication at Late Follow Up (LFU) in the microITT Population
Citrobacter koseri
0 pathogens
1 pathogens
Per-Pathogen Microbiologic Eradication at Late Follow Up (LFU) in the microITT Population
Klebsiella pneumoniae
30 pathogens
14 pathogens
Per-Pathogen Microbiologic Eradication at Late Follow Up (LFU) in the microITT Population
Klebsiella variicola
1 pathogens
1 pathogens
Per-Pathogen Microbiologic Eradication at Late Follow Up (LFU) in the microITT Population
Proteus mirabilis
8 pathogens
6 pathogens
Per-Pathogen Microbiologic Eradication at Late Follow Up (LFU) in the microITT Population
Proteus penneri
1 pathogens
Per-Pathogen Microbiologic Eradication at Late Follow Up (LFU) in the microITT Population
Proteus vulgaris
2 pathogens
Per-Pathogen Microbiologic Eradication at Late Follow Up (LFU) in the microITT Population
Providencia rettgeri
1 pathogens
Per-Pathogen Microbiologic Eradication at Late Follow Up (LFU) in the microITT Population
Serratia marcescens
2 pathogens
Per-Pathogen Microbiologic Eradication at Late Follow Up (LFU) in the microITT Population
Citrobacter freundii complex
1 pathogens
2 pathogens

SECONDARY outcome

Timeframe: Assessed within 24 hours after last IV dose (up to 15 days from start of treatment)

Population: The microITT analysis population consists of all patients in the ITT analysis population who had a positive study entry urine culture defined as ≥10\^5 CFU/mL of a gram-negative pathogen(s) against which both cefepime/VNRX-5133 and meropenem have antibacterial activity AND those patients who had no more than 2 microorganisms identified in the study entry culture regardless of colony count.

Per-pathogen eradication by baseline gram-negative pathogens (only pathogens identified 10 or more times are reported). The number analyzed corresponds to the number of specified pathogens. The number is the percent of the specified pathogen identified at baseline in each treatment group that had been eradicated.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=67 Pathogens
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=30 Pathogens
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at End of Treatment (EOT) in the microITT Population
Escherichia coli
100 percentage of pathogen eradication
88.9 percentage of pathogen eradication
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at End of Treatment (EOT) in the microITT Population
Enterobacter cloacae complex
100 percentage of pathogen eradication
100 percentage of pathogen eradication
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at End of Treatment (EOT) in the microITT Population
Klebsiella oxytoca
100 percentage of pathogen eradication
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at End of Treatment (EOT) in the microITT Population
Klebsiella pneumoniae
95.0 percentage of pathogen eradication
100 percentage of pathogen eradication
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at End of Treatment (EOT) in the microITT Population
Morganella morganii
100 percentage of pathogen eradication
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at End of Treatment (EOT) in the microITT Population
Proteus mirabilis
100 percentage of pathogen eradication
100 percentage of pathogen eradication
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at End of Treatment (EOT) in the microITT Population
Pseudomonas aeruginosa
100 percentage of pathogen eradication

SECONDARY outcome

Timeframe: Assessed at Test of Cure visit (occurred once per participant between Study Days 19 to 23)

Population: The microITT analysis population consists of all patients in the ITT analysis population who had a positive study entry urine culture defined as ≥10\^5 CFU/mL of a gram-negative pathogen(s) against which both cefepime/VNRX-5133 and meropenem have antibacterial activity AND those patients who had no more than 2 microorganisms identified in the study entry culture regardless of colony count.

Per-pathogen eradication by baseline gram-negative pathogens (only pathogens identified 10 or more times are reported). The number analyzed corresponds to the number of specified pathogens. The number is the percent of the specified pathogen identified at baseline in each treatment group that had been eradicated.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=67 pathogens
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=30 pathogens
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at Test of Cure (TOC) in the microITT Population
Enterobacter cloacae complex
100 percentage of eradicated pathogens
50.0 percentage of eradicated pathogens
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at Test of Cure (TOC) in the microITT Population
Escherichia coli
81.1 percentage of eradicated pathogens
61.1 percentage of eradicated pathogens
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at Test of Cure (TOC) in the microITT Population
Klebsiella oxytoca
100 percentage of eradicated pathogens
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at Test of Cure (TOC) in the microITT Population
Klebsiella pneumoniae
60.0 percentage of eradicated pathogens
71.4 percentage of eradicated pathogens
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at Test of Cure (TOC) in the microITT Population
Morganella morganii
100 percentage of eradicated pathogens
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at Test of Cure (TOC) in the microITT Population
Proteus mirabilis
50.0 percentage of eradicated pathogens
0 percentage of eradicated pathogens
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at Test of Cure (TOC) in the microITT Population
Pseudomonas aeruginosa
0 percentage of eradicated pathogens

SECONDARY outcome

Timeframe: Assessed at Late Follow Up visit (occurred once per participant between Study Days 28 to 35)

Population: The microITT analysis population consists of all patients in the ITT analysis population who had a positive study entry urine culture defined as ≥10\^5 CFU/mL of a gram-negative pathogen(s) against which both cefepime/VNRX-5133 and meropenem have antibacterial activity AND those patients who had no more than 2 microorganisms identified in the study entry culture regardless of colony count.

Per-pathogen eradication by baseline gram-negative pathogens (only pathogens identified 10 or more times are reported). The number analyzed corresponds to the number of specified pathogens. The number is the percent of the specified pathogen identified at baseline in each treatment group that had been eradicated.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=67 pathogens
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=30 pathogens
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at Late Follow Up (LFU) in the microITT Population
Enterobacter cloacae complex
100 percentage of pathogen eradication
50.0 percentage of pathogen eradication
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at Late Follow Up (LFU) in the microITT Population
Escherichia coli
73.0 percentage of pathogen eradication
50.0 percentage of pathogen eradication
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at Late Follow Up (LFU) in the microITT Population
Klebsiella oxytoca
100 percentage of pathogen eradication
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at Late Follow Up (LFU) in the microITT Population
Klebsiella pneumoniae
65.0 percentage of pathogen eradication
71.4 percentage of pathogen eradication
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at Late Follow Up (LFU) in the microITT Population
Morganella morganii
100 percentage of pathogen eradication
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at Late Follow Up (LFU) in the microITT Population
Proteus mirabilis
50.0 percentage of pathogen eradication
0 percentage of pathogen eradication
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at Late Follow Up (LFU) in the microITT Population
Pseudomonas aeruginosa
0 percentage of pathogen eradication

SECONDARY outcome

Timeframe: Assessed within 24 hours after last IV dose (up to 15 days from start of treatment)

Population: All patients who meet the criteria for the microITT population AND had a diagnosis of cUTI; received treatment for ≥48 hours; were evaluated at EOT with a response that was not indeterminate; did not violate prior antibacterials exclusion or received concomitant antibiotic therapy with activity against baseline pathogens except for patients failing study drug; or had other confounding factors that interfered with the assessment of outcome including unblinding.

Per-pathogen eradication by baseline gram-negative pathogens. The number analyzed corresponds to the number of specified pathogens. The number is the percent of the specified pathogen identified at baseline in each treatment group that had been eradicated.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=286 pathogens
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=141 pathogens
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Per-Pathogen Microbiologic Eradication at End of Treatment (EOT) in the ME Population
Citrobacter freundii complex
2 pathogens
2 pathogens
Per-Pathogen Microbiologic Eradication at End of Treatment (EOT) in the ME Population
Citrobacter koseri
1 pathogens
1 pathogens
Per-Pathogen Microbiologic Eradication at End of Treatment (EOT) in the ME Population
Enterobacter cloacae complex
14 pathogens
3 pathogens
Per-Pathogen Microbiologic Eradication at End of Treatment (EOT) in the ME Population
Escherichia coli
193 pathogens
94 pathogens
Per-Pathogen Microbiologic Eradication at End of Treatment (EOT) in the ME Population
Klebsiella aerogenes
1 pathogens
1 pathogens
Per-Pathogen Microbiologic Eradication at End of Treatment (EOT) in the ME Population
Klebsiella oxytoca
5 pathogens
1 pathogens
Per-Pathogen Microbiologic Eradication at End of Treatment (EOT) in the ME Population
Klebsiella pneumoniae
37 pathogens
20 pathogens
Per-Pathogen Microbiologic Eradication at End of Treatment (EOT) in the ME Population
Klebsiella variicola
1 pathogens
1 pathogens
Per-Pathogen Microbiologic Eradication at End of Treatment (EOT) in the ME Population
Kluyvera ascorbata
1 pathogens
Per-Pathogen Microbiologic Eradication at End of Treatment (EOT) in the ME Population
Morganella morganii
2 pathogens
2 pathogens
Per-Pathogen Microbiologic Eradication at End of Treatment (EOT) in the ME Population
Proteus hauseri
1 pathogens
Per-Pathogen Microbiologic Eradication at End of Treatment (EOT) in the ME Population
Proteus mirabilis
9 pathogens
9 pathogens
Per-Pathogen Microbiologic Eradication at End of Treatment (EOT) in the ME Population
Proteus penneri
1 pathogens
Per-Pathogen Microbiologic Eradication at End of Treatment (EOT) in the ME Population
Proteus vulgaris
2 pathogens
Per-Pathogen Microbiologic Eradication at End of Treatment (EOT) in the ME Population
Providencia rettgeri
1 pathogens
Per-Pathogen Microbiologic Eradication at End of Treatment (EOT) in the ME Population
Serratia marcescens
2 pathogens
Per-Pathogen Microbiologic Eradication at End of Treatment (EOT) in the ME Population
Pseudomonas aeruginosa
11 pathogens
6 pathogens

SECONDARY outcome

Timeframe: Assessed at Test of Cure visit (occurred once per participant between Study Days 19 to 23)

Population: All patients who meet the criteria for the microITT population AND had a diagnosis of cUTI; received treatment for ≥48 hours; were evaluated at TOC with a response that was not indeterminate; did not violate prior antibacterials exclusion or received concomitant antibiotic therapy with activity against baseline pathogens except for patients failing study drug; or had other confounding factors that interfered with the assessment of outcome including unblinding.

Per-pathogen eradication by baseline gram-negative pathogens. The number analyzed corresponds to the number of specified pathogens. The number is the percent of the specified pathogen identified at baseline in each treatment group that had been eradicated.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=265 pathogens
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=131 pathogens
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Per-Pathogen Microbiologic Eradication at Test of Cure (TOC) in the ME Population
Citrobacter freundii complex
2 pathogens
2 pathogens
Per-Pathogen Microbiologic Eradication at Test of Cure (TOC) in the ME Population
Citrobacter koseri
0 pathogens
1 pathogens
Per-Pathogen Microbiologic Eradication at Test of Cure (TOC) in the ME Population
Enterobacter cloacae complex
11 pathogens
0 pathogens
Per-Pathogen Microbiologic Eradication at Test of Cure (TOC) in the ME Population
Escherichia coli
154 pathogens
64 pathogens
Per-Pathogen Microbiologic Eradication at Test of Cure (TOC) in the ME Population
Klebsiella aerogenes
0 pathogens
0 pathogens
Per-Pathogen Microbiologic Eradication at Test of Cure (TOC) in the ME Population
Klebsiella oxytoca
5 pathogens
1 pathogens
Per-Pathogen Microbiologic Eradication at Test of Cure (TOC) in the ME Population
Klebsiella pneumoniae
26 pathogens
12 pathogens
Per-Pathogen Microbiologic Eradication at Test of Cure (TOC) in the ME Population
Klebsiella variicola
1 pathogens
1 pathogens
Per-Pathogen Microbiologic Eradication at Test of Cure (TOC) in the ME Population
Kluyvera ascorbata
1 pathogens
Per-Pathogen Microbiologic Eradication at Test of Cure (TOC) in the ME Population
Morganella morganii
2 pathogens
1 pathogens
Per-Pathogen Microbiologic Eradication at Test of Cure (TOC) in the ME Population
Proteus hauseri
0 pathogens
Per-Pathogen Microbiologic Eradication at Test of Cure (TOC) in the ME Population
Proteus mirabilis
8 pathogens
5 pathogens
Per-Pathogen Microbiologic Eradication at Test of Cure (TOC) in the ME Population
Proteus penneri
1 pathogens
Per-Pathogen Microbiologic Eradication at Test of Cure (TOC) in the ME Population
Proteus vulgaris
1 pathogens
Per-Pathogen Microbiologic Eradication at Test of Cure (TOC) in the ME Population
Providencia rettgeri
1 pathogens
Per-Pathogen Microbiologic Eradication at Test of Cure (TOC) in the ME Population
Serratia marcescens
1 pathogens
Per-Pathogen Microbiologic Eradication at Test of Cure (TOC) in the ME Population
Pseudomonas aeruginosa
5 pathogens
4 pathogens

SECONDARY outcome

Timeframe: Assessed at Late Follow Up visit (occurred once per participant between Study Days 28 to 35)

Population: All patients who meet the criteria for the microITT population AND had a diagnosis of cUTI; received treatment for ≥48 hours; were evaluated at LFU with a response that was not indeterminate; did not violate prior antibacterials exclusion or received concomitant antibiotic therapy with activity against baseline pathogens except for patients failing study drug; or had other confounding factors that interfered with the assessment of outcome including unblinding.

Per-pathogen eradication by baseline gram-negative pathogens. The number analyzed corresponds to the number of specified pathogens. The number is the percent of the specified pathogen identified at baseline in each treatment group that had been eradicated.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=266 pathogens
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=132 pathogens
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Per-Pathogen Microbiologic Eradication at Late Follow Up (LFU) in the ME Population
Citrobacter freundii complex
1 pathogens
2 pathogens
Per-Pathogen Microbiologic Eradication at Late Follow Up (LFU) in the ME Population
Citrobacter koseri
1 pathogens
Per-Pathogen Microbiologic Eradication at Late Follow Up (LFU) in the ME Population
Enterobacter cloacae complex
12 pathogens
1 pathogens
Per-Pathogen Microbiologic Eradication at Late Follow Up (LFU) in the ME Population
Escherichia coli
130 pathogens
56 pathogens
Per-Pathogen Microbiologic Eradication at Late Follow Up (LFU) in the ME Population
Klebsiella aerogenes
0 pathogens
0 pathogens
Per-Pathogen Microbiologic Eradication at Late Follow Up (LFU) in the ME Population
Klebsiella oxytoca
3 pathogens
1 pathogens
Per-Pathogen Microbiologic Eradication at Late Follow Up (LFU) in the ME Population
Klebsiella pneumoniae
29 pathogens
14 pathogens
Per-Pathogen Microbiologic Eradication at Late Follow Up (LFU) in the ME Population
Klebsiella variicola
1 pathogens
1 pathogens
Per-Pathogen Microbiologic Eradication at Late Follow Up (LFU) in the ME Population
Kluyvera ascorbata
1 pathogens
Per-Pathogen Microbiologic Eradication at Late Follow Up (LFU) in the ME Population
Morganella morganii
2 pathogens
1 pathogens
Per-Pathogen Microbiologic Eradication at Late Follow Up (LFU) in the ME Population
Proteus hauseri
0 pathogens
Per-Pathogen Microbiologic Eradication at Late Follow Up (LFU) in the ME Population
Proteus mirabilis
6 pathogens
6 pathogens
Per-Pathogen Microbiologic Eradication at Late Follow Up (LFU) in the ME Population
Proteus penneri
1 pathogens
Per-Pathogen Microbiologic Eradication at Late Follow Up (LFU) in the ME Population
Proteus vulgaris
2 pathogens
Per-Pathogen Microbiologic Eradication at Late Follow Up (LFU) in the ME Population
Providencia rettgeri
1 pathogens
Per-Pathogen Microbiologic Eradication at Late Follow Up (LFU) in the ME Population
Serratia marcescens
2 pathogens
Per-Pathogen Microbiologic Eradication at Late Follow Up (LFU) in the ME Population
Pseudomonas aeruginosa
5 pathogens
4 pathogens

SECONDARY outcome

Timeframe: Assessed within 24 hours after last IV dose (up to 15 days from start of treatment)

Population: All patients who meet the criteria for the microITT population AND had a diagnosis of cUTI; received treatment for ≥48 hours; were evaluated at EOT with a response that was not indeterminate; did not violate prior antibacterials exclusion or received concomitant antibiotic therapy with activity against baseline pathogens except for patients failing study drug; or had other confounding factors that interfered with the assessment of outcome including unblinding.

Per-pathogen eradication by baseline gram-negative pathogens (only pathogens identified 10 or more times are reported). The number analyzed corresponds to the number of specified pathogens. The number is the percent of the specified pathogen identified at baseline in each treatment group that had been eradicated.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=64 pathogens
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=28 pathogens
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at End of Treatment (EOT) in the ME Population
Enterobacter cloacae complex
100 percentage of pathogen eradication
100 percentage of pathogen eradication
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at End of Treatment (EOT) in the ME Population
Escherichia coli
100 percentage of pathogen eradication
100 percentage of pathogen eradication
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at End of Treatment (EOT) in the ME Population
Klebsiella oxytoca
100 percentage of pathogen eradication
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at End of Treatment (EOT) in the ME Population
Klebsiella pneumoniae
95.0 percentage of pathogen eradication
100 percentage of pathogen eradication
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at End of Treatment (EOT) in the ME Population
Morganella morganii
100 percentage of pathogen eradication
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at End of Treatment (EOT) in the ME Population
Proteus mirabilis
100 percentage of pathogen eradication
100 percentage of pathogen eradication
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at End of Treatment (EOT) in the ME Population
Pseudomonas aeruginosa
100 percentage of pathogen eradication

SECONDARY outcome

Timeframe: Assessed at Test of Cure visit (occurred once per participant between Study Days 19 to 23)

Population: All patients who meet the criteria for the microITT population AND had a diagnosis of cUTI; received treatment for ≥48 hours; were evaluated at TOC with a response that was not indeterminate; did not violate prior antibacterials exclusion or received concomitant antibiotic therapy with activity against baseline pathogens except for patients failing study drug; or had other confounding factors that interfered with the assessment of outcome including unblinding.

Per-pathogen eradication by baseline gram-negative pathogens (only pathogens identified 10 or more times are reported). The number analyzed corresponds to the number of specified pathogens. The number is the percent of the specified pathogen identified at baseline in each treatment group that had been eradicated.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=58 Pathogens
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=24 Pathogens
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at Test of Cure TOC in the ME Population
Enterobacter cloacae complex
100 percentage of pathogen eradication
0 percentage of pathogen eradication
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at Test of Cure TOC in the ME Population
Escherichia coli
87.5 percentage of pathogen eradication
66.7 percentage of pathogen eradication
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at Test of Cure TOC in the ME Population
Klebsiella oxytoca
100 percentage of pathogen eradication
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at Test of Cure TOC in the ME Population
Klebsiella pneumoniae
64.7 percentage of pathogen eradication
66.7 percentage of pathogen eradication
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at Test of Cure TOC in the ME Population
Proteus mirabilis
50.0 percentage of pathogen eradication
0 percentage of pathogen eradication
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at Test of Cure TOC in the ME Population
Pseudomonas aeruginosa
0 percentage of pathogen eradication

SECONDARY outcome

Timeframe: Assessed at Late Follow Up visit (occurred once per participant between Study Days 28 to 35)

Population: All patients who meet the criteria for the microITT population AND had a diagnosis of cUTI; received treatment for ≥48 hours; were evaluated at LFU with a response that was not indeterminate; did not violate prior antibacterials exclusion or received concomitant antibiotic therapy with activity against baseline pathogens except for patients failing study drug; or had other confounding factors that interfered with the assessment of outcome including unblinding.

Per-pathogen eradication by baseline gram-negative pathogens (only pathogens identified 10 or more times are reported). The number analyzed corresponds to the number of specified pathogens. The number is the percent of the specified pathogen identified at baseline in each treatment group that had been eradicated.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=60 pathogens
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=26 pathogens
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at Late Follow Up (LFU) in the ME Population
Proteus mirabilis
50.0 percentage of pathogen eradication
0 percentage of pathogen eradication
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at Late Follow Up (LFU) in the ME Population
Enterobacter cloacae complex
100 percentage of pathogen eradication
50.0 percentage of pathogen eradication
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at Late Follow Up (LFU) in the ME Population
Escherichia coli
78.1 percentage of pathogen eradication
53.3 percentage of pathogen eradication
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at Late Follow Up (LFU) in the ME Population
Klebsiella pneumoniae
68.4 percentage of pathogen eradication
71.4 percentage of pathogen eradication
Per-Pathogen Microbiologic Eradication in Patients With Cefepime-Resistant Pathogens at Late Follow Up (LFU) in the ME Population
Pseudomonas aeruginosa
0 percentage of pathogen eradication

OTHER_PRE_SPECIFIED outcome

Timeframe: Study Days 1 to 35

Population: Patients with at least one TEAE.

Percent of participants experiencing Treatment Emergent Adverse Events (TEAE). Treatment emergent is defined as any event that starts or worsens during or after treatment.

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=440 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=217 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Number of Patients With Treatment-Emergent Adverse Events
156 Participants
63 Participants

OTHER_PRE_SPECIFIED outcome

Timeframe: Study Days 1 to 35

Population: Patients with at least one treatment-emergent SAE.

Percent of participants experiencing treatment emergent Serious Adverse Events (SAE).

Outcome measures

Outcome measures
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=440 Participants
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period. Cefepime/VNRX-5133 (taniborbactam): Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients will also receive meropenem placebo administered via IV over 30 minutes.
Meropenem
n=217 Participants
Meropenem will be administered q8h IV over 30 minutes. Meropenem: Meropenem will be administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients will also receive cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Number of Patients With Serious Adverse Events
9 Participants
4 Participants

Adverse Events

Cefepime/VNRX-5133 (Taniborbactam)

Serious events: 9 serious events
Other events: 93 other events
Deaths: 1 deaths

Meropenem

Serious events: 4 serious events
Other events: 37 other events
Deaths: 0 deaths

Serious adverse events

Serious adverse events
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=440 participants at risk
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients also received meropenem placebo administered via IV over a 2-hour period.
Meropenem
n=217 participants at risk
Meropenem administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients also received cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Infections and infestations
COVID-19
0.45%
2/440 • Number of events 2 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
0.00%
0/217 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
Infections and infestations
Appendicitis
0.23%
1/440 • Number of events 1 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
0.00%
0/217 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
Infections and infestations
Endocarditis
0.23%
1/440 • Number of events 1 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
0.00%
0/217 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
Infections and infestations
Gastrointestinal candidiasis
0.23%
1/440 • Number of events 1 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
0.00%
0/217 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
Infections and infestations
Renal abscess
0.23%
1/440 • Number of events 1 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
0.00%
0/217 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
Infections and infestations
Urinary tract infection
0.23%
1/440 • Number of events 1 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
0.00%
0/217 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
Infections and infestations
Pyelonephritis
0.00%
0/440 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
0.92%
2/217 • Number of events 2 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
Infections and infestations
Pyelonephritis acute
0.00%
0/440 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
0.46%
1/217 • Number of events 1 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
Infections and infestations
Tubo-ovarian abscess
0.00%
0/440 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
0.46%
1/217 • Number of events 1 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
Blood and lymphatic system disorders
Anaemia
0.23%
1/440 • Number of events 1 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
0.00%
0/217 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
Endocrine disorders
Inappropriate antidiuretic hormone secretion
0.23%
1/440 • Number of events 1 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
0.00%
0/217 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
General disorders
Death
0.23%
1/440 • Number of events 1 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
0.00%
0/217 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
Metabolism and nutrition disorders
Hypoglycemia
0.23%
1/440 • Number of events 1 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
0.00%
0/217 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
Renal and urinary disorders
Ureterolithiasis
0.00%
0/440 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
0.46%
1/217 • Number of events 1 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
Skin and subcutaneous tissue disorders
Angioedema
0.23%
1/440 • Number of events 1 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
0.00%
0/217 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
Vascular disorders
Hypertension
0.23%
1/440 • Number of events 1 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
0.00%
0/217 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).

Other adverse events

Other adverse events
Measure
Cefepime/VNRX-5133 (Taniborbactam)
n=440 participants at risk
Cefepime/VNRX-5133 administered q8h intravenously (IV) over a 2-hour period for 7 days (up to 14 days for patients with bacteremia). Patients also received meropenem placebo administered via IV over a 2-hour period.
Meropenem
n=217 participants at risk
Meropenem administered q8h IV over 30 minutes for 7 days (up to 14 days for patients with bacteremia). Patients also received cefepime/VNRX-5133 placebo administered via IV over a 2-hour period.
Nervous system disorders
Headache
6.1%
27/440 • Number of events 27 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
3.7%
8/217 • Number of events 8 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
Gastrointestinal disorders
Diarrhoea
4.1%
18/440 • Number of events 18 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
2.3%
5/217 • Number of events 5 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
Gastrointestinal disorders
Constipation
3.2%
14/440 • Number of events 14 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
1.4%
3/217 • Number of events 3 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
Vascular disorders
Hypertension
2.0%
9/440 • Number of events 10 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
0.92%
2/217 • Number of events 2 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
Gastrointestinal disorders
Nausea
2.0%
9/440 • Number of events 9 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
0.92%
2/217 • Number of events 2 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
Gastrointestinal disorders
Abdominal distension
1.6%
7/440 • Number of events 7 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
1.4%
3/217 • Number of events 3 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
Blood and lymphatic system disorders
Anaemia
1.4%
6/440 • Number of events 7 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
1.4%
3/217 • Number of events 3 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
Nervous system disorders
Dizziness
1.6%
7/440 • Number of events 7 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
0.46%
1/217 • Number of events 1 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
Metabolism and nutrition disorders
Hypokalaemia
1.6%
7/440 • Number of events 7 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
0.46%
1/217 • Number of events 1 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
Vascular disorders
Phlebitis
1.4%
6/440 • Number of events 6 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
0.46%
1/217 • Number of events 1 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
Gastrointestinal disorders
Vomiting
1.4%
6/440 • Number of events 6 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
0.46%
1/217 • Number of events 1 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
Respiratory, thoracic and mediastinal disorders
Cough
1.1%
5/440 • Number of events 5 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
0.92%
2/217 • Number of events 2 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
General disorders
Pyrexia
1.1%
5/440 • Number of events 5 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
1.4%
3/217 • Number of events 3 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
Investigations
Alanine aminotransferase increased
0.91%
4/440 • Number of events 4 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).
2.3%
5/217 • Number of events 5 • From first dose to last follow-up visit (Day 28-35).
Treatment-Emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) in patients who received at least one dose of study drug (Safety Population).

Additional Information

Paul McGovern, MD

Venatorx Pharmaceuticals, Inc.

Phone: 484-329-8615

Results disclosure agreements

  • Principal investigator is a sponsor employee Certain PIs are not allowed to present or publish data from the Study without Sponsor's prior written consent.
  • Publication restrictions are in place

Restriction type: OTHER