Trial Outcomes & Findings for Safety and Efficacy of Emixustat in Stargardt Disease (NCT NCT03772665)

NCT ID: NCT03772665

Last Updated: 2024-05-30

Results Overview

Mean rate of change in total area of macular atrophy, as measured by fundus autofluorescence (FAF)

Recruitment status

COMPLETED

Study phase

PHASE3

Target enrollment

194 participants

Primary outcome timeframe

24 months

Results posted on

2024-05-30

Participant Flow

Participant milestones

Participant milestones
Measure
Emixustat
10 mg Emixustat: Once daily oral tablet taken for 24 months
Placebo
Includes identical tablets with only inactive ingredients (0 mg). Placebo: Once daily oral tablet taken for 24 months
Overall Study
STARTED
128
66
Overall Study
COMPLETED
127
66
Overall Study
NOT COMPLETED
1
0

Reasons for withdrawal

Reasons for withdrawal
Measure
Emixustat
10 mg Emixustat: Once daily oral tablet taken for 24 months
Placebo
Includes identical tablets with only inactive ingredients (0 mg). Placebo: Once daily oral tablet taken for 24 months
Overall Study
Protocol Violation
1
0

Baseline Characteristics

Race and Ethnicity were not collected from any participant.

Baseline characteristics by cohort

Baseline characteristics by cohort
Measure
Emixustat
n=128 Participants
10 mg Emixustat: Once daily oral tablet taken for 24 months
Placebo
n=66 Participants
Includes identical tablets with only inactive ingredients (0 mg). Placebo: Once daily oral tablet taken for 24 months
Total
n=194 Participants
Total of all reporting groups
Age, Categorical
<=18 years
5 Participants
n=128 Participants
2 Participants
n=66 Participants
7 Participants
n=194 Participants
Age, Categorical
Between 18 and 65 years
122 Participants
n=128 Participants
64 Participants
n=66 Participants
186 Participants
n=194 Participants
Age, Categorical
>=65 years
1 Participants
n=128 Participants
0 Participants
n=66 Participants
1 Participants
n=194 Participants
Age, Continuous
43.9 years
STANDARD_DEVIATION 15.03 • n=128 Participants
43.0 years
STANDARD_DEVIATION 14.07 • n=66 Participants
43.6 years
STANDARD_DEVIATION 14.75 • n=194 Participants
Sex: Female, Male
Female
59 Participants
n=128 Participants
29 Participants
n=66 Participants
88 Participants
n=194 Participants
Sex: Female, Male
Male
69 Participants
n=128 Participants
37 Participants
n=66 Participants
106 Participants
n=194 Participants
Race and Ethnicity Not Collected
0 Participants
Race and Ethnicity were not collected from any participant.
Region of Enrollment
Canada
3 participants
n=128 Participants
2 participants
n=66 Participants
5 participants
n=194 Participants
Region of Enrollment
Netherlands
3 participants
n=128 Participants
2 participants
n=66 Participants
5 participants
n=194 Participants
Region of Enrollment
United States
34 participants
n=128 Participants
19 participants
n=66 Participants
53 participants
n=194 Participants
Region of Enrollment
Brazil
20 participants
n=128 Participants
9 participants
n=66 Participants
29 participants
n=194 Participants
Region of Enrollment
Denmark
6 participants
n=128 Participants
4 participants
n=66 Participants
10 participants
n=194 Participants
Region of Enrollment
Italy
24 participants
n=128 Participants
9 participants
n=66 Participants
33 participants
n=194 Participants
Region of Enrollment
South Africa
11 participants
n=128 Participants
7 participants
n=66 Participants
18 participants
n=194 Participants
Region of Enrollment
United Kingdom
6 participants
n=128 Participants
3 participants
n=66 Participants
9 participants
n=194 Participants
Region of Enrollment
France
8 participants
n=128 Participants
4 participants
n=66 Participants
12 participants
n=194 Participants
Region of Enrollment
Germany
8 participants
n=128 Participants
5 participants
n=66 Participants
13 participants
n=194 Participants
Region of Enrollment
Spain
5 participants
n=128 Participants
2 participants
n=66 Participants
7 participants
n=194 Participants

PRIMARY outcome

Timeframe: 24 months

Population: ITT

Mean rate of change in total area of macular atrophy, as measured by fundus autofluorescence (FAF)

Outcome measures

Outcome measures
Measure
Emixustat
n=128 Participants
10 mg Emixustat: Once daily oral tablet taken for 24 months
Placebo
n=66 Participants
Includes identical tablets with only inactive ingredients (0 mg). Placebo: Once daily oral tablet taken for 24 months
Mean Rate of Change in Total Area of Macular Atrophy, as Measured by Fundus Autofluorescence (FAF)
1.280 Rate of change from BL (mm^2/yr)
Standard Error 0.0783
1.309 Rate of change from BL (mm^2/yr)
Standard Error 0.1002

Adverse Events

Emixustat

Serious events: 9 serious events
Other events: 1 other events
Deaths: 0 deaths

Placebo

Serious events: 2 serious events
Other events: 0 other events
Deaths: 0 deaths

Serious adverse events

Serious adverse events
Measure
Emixustat
n=127 participants at risk
10 mg Emixustat: Once daily oral tablet taken for 24 months
Placebo
n=66 participants at risk
Includes identical tablets with only inactive ingredients (0 mg). Placebo: Once daily oral tablet taken for 24 months
Cardiac disorders
agina pectoris
0.79%
1/127 • Number of events 1 • 24 months
MedDRA version 25.0
1.5%
1/66 • Number of events 1 • 24 months
MedDRA version 25.0
Cardiac disorders
atrial fibrillation
0.79%
1/127 • Number of events 1 • 24 months
MedDRA version 25.0
0.00%
0/66 • 24 months
MedDRA version 25.0
Neoplasms benign, malignant and unspecified (incl cysts and polyps)
neoplasm
1.6%
2/127 • Number of events 2 • 24 months
MedDRA version 25.0
1.5%
1/66 • Number of events 1 • 24 months
MedDRA version 25.0
Infections and infestations
Infections and infestations
0.79%
1/127 • Number of events 1 • 24 months
MedDRA version 25.0
1.5%
1/66 • Number of events 1 • 24 months
MedDRA version 25.0
Eye disorders
Visual disorder
0.79%
1/127 • Number of events 1 • 24 months
MedDRA version 25.0
0.00%
0/66 • 24 months
MedDRA version 25.0
Injury, poisoning and procedural complications
Injury, posioning and procedural
0.79%
1/127 • Number of events 1 • 24 months
MedDRA version 25.0
0.00%
0/66 • 24 months
MedDRA version 25.0
Nervous system disorders
Nervous system disorder
0.79%
1/127 • Number of events 1 • 24 months
MedDRA version 25.0
0.00%
0/66 • 24 months
MedDRA version 25.0
Vascular disorders
Vascular disorder
0.79%
1/127 • Number of events 1 • 24 months
MedDRA version 25.0
0.00%
0/66 • 24 months
MedDRA version 25.0

Other adverse events

Other adverse events
Measure
Emixustat
n=127 participants at risk
10 mg Emixustat: Once daily oral tablet taken for 24 months
Placebo
n=66 participants at risk
Includes identical tablets with only inactive ingredients (0 mg). Placebo: Once daily oral tablet taken for 24 months
Eye disorders
Visual acuity reduced
0.79%
1/127 • Number of events 1 • 24 months
MedDRA version 25.0
0.00%
0/66 • 24 months
MedDRA version 25.0

Additional Information

Dr. Jeff Gregory

Acucela, dba Kubota Vision

Phone: 2068058310

Results disclosure agreements

  • Principal investigator is a sponsor employee
  • Publication restrictions are in place