Safety, Tolerability, PK and PD of SAD or MAD of APX-115 in Healthy Male Volunteers

NCT ID: NCT03694041

Last Updated: 2019-03-11

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

88 participants

Study Classification

INTERVENTIONAL

Study Start Date

2018-05-28

Study Completion Date

2019-03-06

Brief Summary

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This study aims to evaluate the safety, tolerabilty, pharmacokinetics and pharmacodynamics of single ascending doses and multiple ascending doses of APX-115 in healthy males. This study also aims to evaluate the effect of food consumption on the pharmacokinetics of APX-115 and potential interaction between caffeine and APX-115 in healthy males.

Detailed Description

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Conditions

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Healthy Safety

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Parallel design for SAD and MAD studies Crossover design for Food and Drug interaction studies
Primary Study Purpose

TREATMENT

Blinding Strategy

DOUBLE

Participants Investigators

Study Groups

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SAD: APX-115

Experimental: APX-115 SAD group

Group Type EXPERIMENTAL

SAD: APX-115

Intervention Type DRUG

Drug: APX-115 SAD APX-115 SAD for 1day

SAD: Placebo

Experimental: Placebo group

Group Type PLACEBO_COMPARATOR

SAD: Placebo

Intervention Type DRUG

Drug: Placebo Placebo for 1day

MAD: APX-115

Experimental: APX-115 MAD group

Group Type EXPERIMENTAL

MAD: APX-115

Intervention Type DRUG

Drug: APX-115 MAD APX-115 MAD repeatedly administered.

MAD: Placebo

Experimental: Placebo group

Group Type PLACEBO_COMPARATOR

MAD: Placebo

Intervention Type DRUG

Matching study drug will be repeatedly administered.

Food effect - Fasting condition

Experimental: APX-115 under fasting condition

Group Type ACTIVE_COMPARATOR

Food effect: fasted and fed

Intervention Type OTHER

A single dose of APX-115, selected from the SAD study, will be administered under fasted and fed condition.

Food effect - fed condition

Experimental: APX-115 under fed condition

Group Type ACTIVE_COMPARATOR

Food effect: fasted and fed

Intervention Type OTHER

A single dose of APX-115, selected from the SAD study, will be administered under fasted and fed condition.

Drug Interaction - metabolic probe

Experimental: metabolic probe

Group Type PLACEBO_COMPARATOR

Metabolic probe with or without APX-115

Intervention Type OTHER

A metabolic probe will be administered with and without APX-115.

Interventions

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SAD: APX-115

Drug: APX-115 SAD APX-115 SAD for 1day

Intervention Type DRUG

SAD: Placebo

Drug: Placebo Placebo for 1day

Intervention Type DRUG

MAD: APX-115

Drug: APX-115 MAD APX-115 MAD repeatedly administered.

Intervention Type DRUG

MAD: Placebo

Matching study drug will be repeatedly administered.

Intervention Type DRUG

Food effect: fasted and fed

A single dose of APX-115, selected from the SAD study, will be administered under fasted and fed condition.

Intervention Type OTHER

Metabolic probe with or without APX-115

A metabolic probe will be administered with and without APX-115.

Intervention Type OTHER

Eligibility Criteria

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Inclusion Criteria

* Healthy male subject, aged between 18 and 45 years inclusive
* Certified as healthy by a comprehensive clinical assessment
* Normal dietary habits
* Normal ECG recording on a 12-lead ECG
* Signing a written informed consent prior to selection

Exclusion:

* Any history or presence of cardiovascular, pulmonary, gastro-intestinal, hepatic, renal, metabolic, haematological, neurologic, psychiatric, systemic, infectious or ocular disease
* Frequent headaches and / or migraine, recurrent nausea and / or vomiting
* Symptomatic hypotension whatever the decrease of blood pressure or asymptomatic postural hypotension defined by a decrease in SBP or DBP equal to or greater than 20 mmHg within two minutes when changing from the supine to the standing position
* Blood donation (including in the frame of a clinical trial) within 2 months before administration
* General anaesthesia within 3 months before administration
* Presence or history of drug hypersensitivity, or allergic disease diagnosed and treated by a physician
* Inability to abstain from intensive muscular effort
* No possibility of contact in case of emergency
* Any drug intake (except paracetamol or contraception) during the last month prior to the first administration
* History or presence of drug or alcohol abuse (alcohol consumption \> 30 grams / day)
* Excessive consumption of beverages with xanthine bases (\> 4 cups or glasses / day)
* Positive Hepatitis B surface (HBs) antigen or anti Hepatitis C Virus (HCV) antibody, or positive results for Human Immunodeficiency Virus (HIV) 1 or 2 tests
* Positive results of screening for drugs of abuse
* Subject who, in the judgment of the Investigator, is likely to be non-compliant or uncooperative during the study, or unable to cooperate because of a language problem, poor mental development
* Administrative or legal supervision
Minimum Eligible Age

18 Years

Maximum Eligible Age

45 Years

Eligible Sex

MALE

Accepts Healthy Volunteers

Yes

Sponsors

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Aptabio Therapeutics, Inc.

INDIV

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Yves Donazzolo, MD

Role: PRINCIPAL_INVESTIGATOR

Eurofins Optimed

Locations

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Eurofins Optimed

Gières, , France

Site Status

Countries

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France

Other Identifiers

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2017-004252-30

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

OP101817.APT

Identifier Type: -

Identifier Source: org_study_id

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