A Study of FT-2102 in Patients With Advanced Solid Tumors and Gliomas With an IDH1 Mutation

NCT ID: NCT03684811

Last Updated: 2023-11-18

Study Results

Results available

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1/PHASE2

Total Enrollment

93 participants

Study Classification

INTERVENTIONAL

Study Start Date

2018-11-01

Study Completion Date

2022-06-13

Brief Summary

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This Phase 1/2 study will evaluate the safety, efficacy, PK, and PD of FT-2102 as a single agent and in combination with other anti-cancer drugs in patients with advanced solid tumors and gliomas.

The study is divided into two parts: single agent FT-2102 followed by combination therapy.

Part 1: A single agent, open-label study in up to five cohorts (glioma, hepatobiliary tumors, chondrosarcoma, intrahepatic cholangiocarcinoma, and other IDH1 mutant solid tumors) that will include a Phase 1 dose confirmation followed by a Phase 2 investigation of clinical activity in up to 4 cohorts. During the dose confirmation, additional doses or altered dose schedules may be explored.

Part 2: An open-label study of FT-2102 in combination with other anti-cancer agents. Patients will be enrolled across 4 different disease cohorts, examining the effect of FT-2102 + azacitidine (glioma and chondrosarcoma), FT-2102 + nivolumab (hepatobiliary tumors), and FT-2102 + gemcitabine/cisplatin (intrahepatic cholangiocarcinoma). There will be a safety lead-in followed by a Phase 2 evaluation in up to four cohorts of patients.

Detailed Description

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Conditions

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Cohort 1a and 1b: Glioma (Advanced Gliomas and Glioblastoma Multiforme) Cohort 2a and 2b: Hepatobiliary Tumors (Hepatocellular Carcinoma, Bile Duct Carcinoma, Intrahepatic Cholangiocarcinoma, Other Hepatobiliary Carcinomas) Cohort 3a and 3b: Chondrosarcoma Cohort 4a and 4b: Intrahepatic Cholangiocarcinoma Cohort 5a: Other Non-Central Nervous System Solid Tumors With IDH1 Mutations

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Phase 1b Dose Confirmation Single Agent (Cohorts 1a-5a)

Group Type EXPERIMENTAL

FT-2102

Intervention Type DRUG

FT-2102 will be supplied as a 150 mg capsule and will be administered per the protocol defined frequency and dose level.

Phase 2 Cohorts FT-2102 Single Agent (Cohorts 1a-5a)

Group Type EXPERIMENTAL

FT-2102

Intervention Type DRUG

FT-2102 will be supplied as a 150 mg capsule and will be administered per the protocol defined frequency and dose level.

Phase 1b and 2 Cohorts Combination (Cohorts 1b and 3b)

Group Type EXPERIMENTAL

FT-2102

Intervention Type DRUG

FT-2102 will be supplied as a 150 mg capsule and will be administered per the protocol defined frequency and dose level.

Azacitidine

Intervention Type DRUG

Azacitidine will be administered per the site's standard of care.

Phase 1b and 2 Cohort Combination (Cohort 2b)

Group Type EXPERIMENTAL

FT-2102

Intervention Type DRUG

FT-2102 will be supplied as a 150 mg capsule and will be administered per the protocol defined frequency and dose level.

Nivolumab

Intervention Type BIOLOGICAL

Nivolumab will be administered per the site's standard of care.

Phase 1b and 2 Cohort Combination (Cohort 4b)

Group Type EXPERIMENTAL

FT-2102

Intervention Type DRUG

FT-2102 will be supplied as a 150 mg capsule and will be administered per the protocol defined frequency and dose level.

Gemcitabine and Cisplatin

Intervention Type DRUG

Gemcitabine and cisplatin will be administered per the site's standard of care.

Interventions

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FT-2102

FT-2102 will be supplied as a 150 mg capsule and will be administered per the protocol defined frequency and dose level.

Intervention Type DRUG

Azacitidine

Azacitidine will be administered per the site's standard of care.

Intervention Type DRUG

Nivolumab

Nivolumab will be administered per the site's standard of care.

Intervention Type BIOLOGICAL

Gemcitabine and Cisplatin

Gemcitabine and cisplatin will be administered per the site's standard of care.

Intervention Type DRUG

Other Intervention Names

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Vidaza Opdivo Gemzar and Platinol

Eligibility Criteria

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Inclusion Criteria

* Patients must have documented IDH1-R132 gene-mutated disease as evaluated by site
* Glioma: Advanced glioma that has recurred or progressed following standard therapy, or that has not responded to standard therapy.
* Hepatobiliary cancer that is relapsed/refractory or intolerant to approved standard-of-care therapy (including: hepatocellular carcinoma, bile duct carcinoma, intrahepatic cholangiocarcinoma or other hepatobiliary carcinomas)
* Chondrosarcoma that is relapsed or refractory and either locally advanced or metastatic and not amenable to complete surgical excision
* Intrahepatic cholangiocarcinoma that is advanced nonresectable or metastatic cholangiocarcinoma not eligible for curative resection or transplantation. Phase 1b/Safety Lead-in of Phase 2: relapsed or refractory disease. Combination Phase 2 (beyond Safety Lead-in): have received no more than 1 cycle of gemcitabine/cisplatin therapy
* Other solid tumors that have relapsed or refractory to standard-of-care therapy with no other available therapeutic options
* Good performance status
* Good kidney and liver function

Exclusion Criteria

* Prior solid organ or hematopoietic cell transplant
* Prior treatment with IDH1 inhibitor (single agent cohorts only)
* Congestive heart failure (New York Heart Association Class III or IV) or unstable angina pectoris. Previous history of myocardial infarction within 1 year prior to study entry, uncontrolled hypertension or uncontrolled arrhythmias
* Unstable or severe, uncontrolled medical condition (e.g., unstable cardiac function, unstable pulmonary condition, including pneumonitis and/or interstitial lung disease, and uncontrolled diabetes)
* Active, uncontrolled bacterial, viral, or fungal infections, requiring systemic therapy
* PD-1 only: active autoimmune disease
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Forma Therapeutics, Inc.

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Emma Barrett

Role: STUDY_DIRECTOR

Forma Therapeutics

Locations

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Banner MD Anderson

Gilbert, Arizona, United States

Site Status

University of Colorado Anschutz Medical Campus

Aurora, Colorado, United States

Site Status

University of Miami, Sylvester Comprehensive Cancer Center

Miami, Florida, United States

Site Status

Northwestern University, Lurie Comprehensive Cancer Center

Chicago, Illinois, United States

Site Status

University of Iowa, Holden Comprehensive Cancer Institute

Iowa City, Iowa, United States

Site Status

Massachusetts General Hospital

Boston, Massachusetts, United States

Site Status

Dana Farber Cancer Institute

Boston, Massachusetts, United States

Site Status

Henry Ford Hospital

Detroit, Michigan, United States

Site Status

Washington University School of Medicine

St Louis, Missouri, United States

Site Status

Rutgers Cancer Institute of New Jersey

New Brunswick, New Jersey, United States

Site Status

Columbia University Medical Center

New York, New York, United States

Site Status

Baylor Scott and White Medical Center

Temple, Texas, United States

Site Status

University of Utah, Huntsman Cancer Hospital

Salt Lake City, Utah, United States

Site Status

Medical College of Wisconsin, Froedtert Hospital

Milwaukee, Wisconsin, United States

Site Status

Austin Hospital

Heidelberg, Victoria, Australia

Site Status

Peter MacCallum Cancer Centre

Melbourne, , Australia

Site Status

Centre de Lutte Contre Cancer (CLCC) - Institute Bergonie

Bordeaux, , France

Site Status

Centre de Lutte Cancre (CLCC) - Lyon

Lyon, , France

Site Status

Hospital de la Timone

Marseille, , France

Site Status

Institut Gustave Roussy Cancer Campus

Villejuif, , France

Site Status

Seoul National University Hospital

Seoul, , South Korea

Site Status

Asan Medical Center

Seoul, , South Korea

Site Status

Samsung Medical Center

Seoul, , South Korea

Site Status

Vall D'Hebron University Hospital

Barcelona, , Spain

Site Status

Cancer Research Beatson Institute

Glasgow, , United Kingdom

Site Status

The Royal Marsden Hospital

London, , United Kingdom

Site Status

Countries

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United States Australia France South Korea Spain United Kingdom

Provided Documents

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Document Type: Study Protocol

View Document

Document Type: Statistical Analysis Plan

View Document

Other Identifiers

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2102-ONC-102

Identifier Type: -

Identifier Source: org_study_id

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