Trial Outcomes & Findings for Efficacy & Safety of OPN-375 Adults With Bilateral Nasal Polyps Using Nasoendoscopic Video (NCT NCT03591068)

NCT ID: NCT03591068

Last Updated: 2020-08-03

Results Overview

: Polyp grading of each nasal cavity was determined by a nasal polyp grading scale score measured by nasoendoscopy. 0: No polyps 1. Mild polyposis: polyps not reaching below the inferior border of the middle turbinate 2. Moderate polyposis: polyps reaching below the inferior border of the middle concha, but not the inferior border of the inferior turbinate 3. Severe polyposis large polyps reaching below the lower inferior border of the inferior turbinate

Recruitment status

COMPLETED

Study phase

PHASE3

Target enrollment

11 participants

Primary outcome timeframe

Week 24

Results posted on

2020-08-03

Participant Flow

Participant milestones

Participant milestones
Measure
OPN-375 186 mcg BID
Fluticasone Propionate: OPN-375 186 μg BID, Delivered via exhalation delivery system
Overall Study
STARTED
11
Overall Study
COMPLETED
9
Overall Study
NOT COMPLETED
2

Reasons for withdrawal

Withdrawal data not reported

Baseline Characteristics

Efficacy & Safety of OPN-375 Adults With Bilateral Nasal Polyps Using Nasoendoscopic Video

Baseline characteristics by cohort

Baseline characteristics by cohort
Measure
OPN-375 186 mcg BID
n=11 Participants
Fluticasone Propionate: OPN-375 186 μg BID, Delivered via exhalation delivery system
Age, Continuous
54.6 years
STANDARD_DEVIATION 14.5 • n=5 Participants
Sex: Female, Male
Female
3 Participants
n=5 Participants
Sex: Female, Male
Male
8 Participants
n=5 Participants
Race (NIH/OMB)
American Indian or Alaska Native
0 Participants
n=5 Participants
Race (NIH/OMB)
Asian
0 Participants
n=5 Participants
Race (NIH/OMB)
Native Hawaiian or Other Pacific Islander
0 Participants
n=5 Participants
Race (NIH/OMB)
Black or African American
1 Participants
n=5 Participants
Race (NIH/OMB)
White
10 Participants
n=5 Participants
Race (NIH/OMB)
More than one race
0 Participants
n=5 Participants
Race (NIH/OMB)
Unknown or Not Reported
0 Participants
n=5 Participants
Region of Enrollment
United States
11 participants
n=5 Participants
Total Polyp Grading Score (sum of scores from both nasal cavities)
3.1 units on a scale
n=5 Participants
Sinonasal Outcome Test 22 (SNOT-22) Total Score
48.8 units on a scale
n=5 Participants
Sniffin' Sticks n-butanol tests
11.8 units on a scale
STANDARD_DEVIATION 6.5 • n=5 Participants

PRIMARY outcome

Timeframe: Week 24

: Polyp grading of each nasal cavity was determined by a nasal polyp grading scale score measured by nasoendoscopy. 0: No polyps 1. Mild polyposis: polyps not reaching below the inferior border of the middle turbinate 2. Moderate polyposis: polyps reaching below the inferior border of the middle concha, but not the inferior border of the inferior turbinate 3. Severe polyposis large polyps reaching below the lower inferior border of the inferior turbinate

Outcome measures

Outcome measures
Measure
OPN-375 186 mcg BID
n=11 Participants
Fluticasone Propionate: OPN-375 186 μg BID, Delivered via exhalation delivery system
OPN-375 186 mcg BID - Diastolic BP
Fluticasone Propionate: OPN-375 186 μg BID, Delivered via exhalation delivery system
Change From Visit 1 at End of Study in Bilateral Nasal Polyp Grade Using Endoscopic Video
-0.7 units on a scale
Standard Deviation 0.9

SECONDARY outcome

Timeframe: 24 Weeks, up to 30 days after last dose

Population: No TEAE was experienced by more than a single subject

Outcome measures

Outcome measures
Measure
OPN-375 186 mcg BID
n=11 Participants
Fluticasone Propionate: OPN-375 186 μg BID, Delivered via exhalation delivery system
OPN-375 186 mcg BID - Diastolic BP
Fluticasone Propionate: OPN-375 186 μg BID, Delivered via exhalation delivery system
Assessment for Safety by Recording Adverse Events and Adverse Events of Special Interests
Asthma
1 Participants
Assessment for Safety by Recording Adverse Events and Adverse Events of Special Interests
Back pain
1 Participants
Assessment for Safety by Recording Adverse Events and Adverse Events of Special Interests
Dizziness
1 Participants
Assessment for Safety by Recording Adverse Events and Adverse Events of Special Interests
Dyspnoea
1 Participants
Assessment for Safety by Recording Adverse Events and Adverse Events of Special Interests
Fungal skin infection
1 Participants
Assessment for Safety by Recording Adverse Events and Adverse Events of Special Interests
Hypotension
1 Participants
Assessment for Safety by Recording Adverse Events and Adverse Events of Special Interests
Influenza
1 Participants
Assessment for Safety by Recording Adverse Events and Adverse Events of Special Interests
Lacrimation increased
1 Participants
Assessment for Safety by Recording Adverse Events and Adverse Events of Special Interests
Nasal discharge discolouration
1 Participants
Assessment for Safety by Recording Adverse Events and Adverse Events of Special Interests
Sinusitis
1 Participants
Assessment for Safety by Recording Adverse Events and Adverse Events of Special Interests
Tension headache
1 Participants
Assessment for Safety by Recording Adverse Events and Adverse Events of Special Interests
Upper respiratory tract infection
1 Participants
Assessment for Safety by Recording Adverse Events and Adverse Events of Special Interests
Vasomotor rhinitis
1 Participants

SECONDARY outcome

Timeframe: 24 Weeks, up to 30 days after last dose

Assessed in nasal examination worksheet which includes recording the presence of any epistaxis, septal erosion/perforation, ulceration/erosion of area other than septum. If present, the nostril location is also recorded, along with severity, and if there is any relation to an injury or trauma

Outcome measures

Outcome measures
Measure
OPN-375 186 mcg BID
n=11 Participants
Fluticasone Propionate: OPN-375 186 μg BID, Delivered via exhalation delivery system
OPN-375 186 mcg BID - Diastolic BP
Fluticasone Propionate: OPN-375 186 μg BID, Delivered via exhalation delivery system
Assessment for Safety Through Nasal Examination
Epistaxis
1 Participants
Assessment for Safety Through Nasal Examination
Septal erosion/perforation
0 Participants
Assessment for Safety Through Nasal Examination
Ulceration/erosion
0 Participants

SECONDARY outcome

Timeframe: Baseline, Week 12, Week 24

Includes systolic and diastolic blood pressure measurements in millimeter of mercury (mmHg)

Outcome measures

Outcome measures
Measure
OPN-375 186 mcg BID
n=11 Participants
Fluticasone Propionate: OPN-375 186 μg BID, Delivered via exhalation delivery system
OPN-375 186 mcg BID - Diastolic BP
n=11 Participants
Fluticasone Propionate: OPN-375 186 μg BID, Delivered via exhalation delivery system
Assessment for Safety From Recording Vital Sign - Blood Pressure
Baseline
130.1 mmHg
Standard Deviation 14.3
83.3 mmHg
Standard Deviation 9.3
Assessment for Safety From Recording Vital Sign - Blood Pressure
Week 12
127.4 mmHg
Standard Deviation 19.6
82.0 mmHg
Standard Deviation 12.9
Assessment for Safety From Recording Vital Sign - Blood Pressure
Week 24
131.9 mmHg
Standard Deviation 18.8
81.4 mmHg
Standard Deviation 8.7

SECONDARY outcome

Timeframe: Baseline, Week 12, Week 24

measure pulse in beats per minute (bpm)

Outcome measures

Outcome measures
Measure
OPN-375 186 mcg BID
n=11 Participants
Fluticasone Propionate: OPN-375 186 μg BID, Delivered via exhalation delivery system
OPN-375 186 mcg BID - Diastolic BP
Fluticasone Propionate: OPN-375 186 μg BID, Delivered via exhalation delivery system
Assessment for Safety From Recording Vital Sign - Pulse
Baseline
71.5 bpm
Standard Deviation 7.1
Assessment for Safety From Recording Vital Sign - Pulse
Week 12
73.5 bpm
Standard Deviation 9.1
Assessment for Safety From Recording Vital Sign - Pulse
Week 24
76.4 bpm
Standard Deviation 7.4

SECONDARY outcome

Timeframe: 24 Weeks, up to 30 days after last dose

Outcome measures

Outcome measures
Measure
OPN-375 186 mcg BID
n=11 Participants
Fluticasone Propionate: OPN-375 186 μg BID, Delivered via exhalation delivery system
OPN-375 186 mcg BID - Diastolic BP
Fluticasone Propionate: OPN-375 186 μg BID, Delivered via exhalation delivery system
Assessment for Safety From the Collection of Information for Concomitant Medications Usage
Selective serotonin reuptake inhibitor
1 Participants
Assessment for Safety From the Collection of Information for Concomitant Medications Usage
ACE Inhibitor
1 Participants
Assessment for Safety From the Collection of Information for Concomitant Medications Usage
Angiotensin II Receptor Antagonist
1 Participants
Assessment for Safety From the Collection of Information for Concomitant Medications Usage
Antianginal
1 Participants
Assessment for Safety From the Collection of Information for Concomitant Medications Usage
Anticoagulant
1 Participants
Assessment for Safety From the Collection of Information for Concomitant Medications Usage
Antihistamine
4 Participants
Assessment for Safety From the Collection of Information for Concomitant Medications Usage
Antifungal Cream
1 Participants
Assessment for Safety From the Collection of Information for Concomitant Medications Usage
Ascorbic Acid
1 Participants
Assessment for Safety From the Collection of Information for Concomitant Medications Usage
Beta Blocking Agent, selective
2 Participants
Assessment for Safety From the Collection of Information for Concomitant Medications Usage
Beta2 Adrenergic Agonist
6 Participants
Assessment for Safety From the Collection of Information for Concomitant Medications Usage
Biguanide
1 Participants
Assessment for Safety From the Collection of Information for Concomitant Medications Usage
Calcium Channel Blocker
1 Participants
Assessment for Safety From the Collection of Information for Concomitant Medications Usage
CNS Muscle Relaxant
1 Participants
Assessment for Safety From the Collection of Information for Concomitant Medications Usage
Diuretic
2 Participants
Assessment for Safety From the Collection of Information for Concomitant Medications Usage
Electolytes
1 Participants
Assessment for Safety From the Collection of Information for Concomitant Medications Usage
HMG CoA Reductase Inhibitors
1 Participants
Assessment for Safety From the Collection of Information for Concomitant Medications Usage
Inhaled Corticosteroid
2 Participants
Assessment for Safety From the Collection of Information for Concomitant Medications Usage
Inhaled Corticosteroid/Long-acting beta-agonist
6 Participants
Assessment for Safety From the Collection of Information for Concomitant Medications Usage
Leukotriene Receptor Antagonists
3 Participants
Assessment for Safety From the Collection of Information for Concomitant Medications Usage
Multivitamin
2 Participants
Assessment for Safety From the Collection of Information for Concomitant Medications Usage
Nitrate
1 Participants
Assessment for Safety From the Collection of Information for Concomitant Medications Usage
Non-steroidal anti-inflammatory drug
3 Participants
Assessment for Safety From the Collection of Information for Concomitant Medications Usage
Nuclear factor erythroid-2-related factor
1 Participants
Assessment for Safety From the Collection of Information for Concomitant Medications Usage
Synthetic nucleoside analogue
1 Participants
Assessment for Safety From the Collection of Information for Concomitant Medications Usage
Other analgesics
1 Participants
Assessment for Safety From the Collection of Information for Concomitant Medications Usage
Other antiinflammatorys
1 Participants
Assessment for Safety From the Collection of Information for Concomitant Medications Usage
Topical antibiotics
2 Participants
Assessment for Safety From the Collection of Information for Concomitant Medications Usage
Proton pump inhibitors
1 Participants
Assessment for Safety From the Collection of Information for Concomitant Medications Usage
Testosterone
1 Participants
Assessment for Safety From the Collection of Information for Concomitant Medications Usage
Thyroid Hormone
2 Participants

SECONDARY outcome

Timeframe: Week 24

Polyp grading of each nasal cavity was determined by a nasal polyp grading scale score measured by nasoendoscopy. 0: No polyps 1. Mild polyposis: polyps not reaching below the inferior border of the middle turbinate 2. Moderate polyposis: polyps reaching below the inferior border of the middle concha, but not the inferior border of the inferior turbinate 3. Severe polyposis large polyps reaching below the lower inferior border of the inferior turbinate

Outcome measures

Outcome measures
Measure
OPN-375 186 mcg BID
n=11 Participants
Fluticasone Propionate: OPN-375 186 μg BID, Delivered via exhalation delivery system
OPN-375 186 mcg BID - Diastolic BP
Fluticasone Propionate: OPN-375 186 μg BID, Delivered via exhalation delivery system
Total Polyp Grading Score (Sum of Scores From Both Nasal Cavities)
2.4 units on a scale
Interval 2.0 to 4.0

SECONDARY outcome

Timeframe: Week 24

Polyp grading of each nasal cavity was determined by a nasal polyp grading scale score measured by nasoendoscopy. 0: No polyps 1. Mild polyposis: polyps not reaching below the inferior border of the middle turbinate 2. Moderate polyposis: polyps reaching below the inferior border of the middle concha, but not the inferior border of the inferior turbinate 3. Severe polyposis large polyps reaching below the lower inferior border of the inferior turbinate

Outcome measures

Outcome measures
Measure
OPN-375 186 mcg BID
n=11 Participants
Fluticasone Propionate: OPN-375 186 μg BID, Delivered via exhalation delivery system
OPN-375 186 mcg BID - Diastolic BP
Fluticasone Propionate: OPN-375 186 μg BID, Delivered via exhalation delivery system
Number of Subjects With a Change of Greater Than or Equal to 1 Point in Bilateral Polyp Grade
5 Participants

SECONDARY outcome

Timeframe: Week 24

Polyp grading of each nasal cavity was determined by a nasal polyp grading scale score measured by nasoendoscopy. 0: No polyps 1. Mild polyposis: polyps not reaching below the inferior border of the middle turbinate 2. Moderate polyposis: polyps reaching below the inferior border of the middle concha, but not the inferior border of the inferior turbinate 3. Severe polyposis large polyps reaching below the lower inferior border of the inferior turbinate

Outcome measures

Outcome measures
Measure
OPN-375 186 mcg BID
n=11 Participants
Fluticasone Propionate: OPN-375 186 μg BID, Delivered via exhalation delivery system
OPN-375 186 mcg BID - Diastolic BP
Fluticasone Propionate: OPN-375 186 μg BID, Delivered via exhalation delivery system
Number of Subjects With a Polyp Grade of 0 on at Least One Side of the Nose at Each Visit
1 Participants

SECONDARY outcome

Timeframe: Week 24

SNOT-22 is a subject-completed questionnaire that consists of 22 questions. The questions on the SNOT-22 efficacy evaluation were used to calculate a total score. 22 questions are divided among 4 subscales: Rhinologic (7 questions), Ear/Facial Symptoms (4 questions), Sleep Function (3 questions), and Psychological Issues (6 questions). Each item was rated on the 5-point scale. The total score can range from 0-110, 0 being the best and 110 being the worst. 0: No problem 1. Very mild problem 2. Mild or slight problem 3. Moderate problem 4. Severe problem 5. Problem as bad as can be

Outcome measures

Outcome measures
Measure
OPN-375 186 mcg BID
n=11 Participants
Fluticasone Propionate: OPN-375 186 μg BID, Delivered via exhalation delivery system
OPN-375 186 mcg BID - Diastolic BP
Fluticasone Propionate: OPN-375 186 μg BID, Delivered via exhalation delivery system
Sinonasal Outcome Test 22 (SNOT-22) Total Score
27.8 units on a scale
Standard Deviation 16.1

SECONDARY outcome

Timeframe: Week 24

The Sniffin' Sticks n-butanol (Extended test) are used to investigate human olfactory performance by use of odor pens. the Extended Test consists of 3 different subtests: Threshold, Discrimination and Identification. the Threshold test is used to ascertain the patient's olfactory threshold. the Discrimination test requires the patient to differentiate smells. The Identification test requires the patient to identify everyday smells by means of a card with different choices. The result of this test is expressed as the sum of the results of the 3 subtests, the so called TDI score (threshold, discrimination, identification). A score of more than 30 rates as normal, a score of 30 or less indicates hyposmia and a score of 15 and below point to functional anosmia in form of complete loss of the sense of smell or an extremely weakened smell ability.

Outcome measures

Outcome measures
Measure
OPN-375 186 mcg BID
n=11 Participants
Fluticasone Propionate: OPN-375 186 μg BID, Delivered via exhalation delivery system
OPN-375 186 mcg BID - Diastolic BP
Fluticasone Propionate: OPN-375 186 μg BID, Delivered via exhalation delivery system
Sniffin' Sticks N-butanol Test
16.5 units on a scale
Standard Deviation 6.9

SECONDARY outcome

Timeframe: Week 24

Population: Number of participants who responded that they had some degree of improvement in their symptoms (minimally/much/very much improved)

The Patient Global Impression of Change (PGIC), is a questionnaire where the patient rates the change in their symptoms. Score range is from 1 (very much improved) to 7 (very much worse)

Outcome measures

Outcome measures
Measure
OPN-375 186 mcg BID
n=11 Participants
Fluticasone Propionate: OPN-375 186 μg BID, Delivered via exhalation delivery system
OPN-375 186 mcg BID - Diastolic BP
Fluticasone Propionate: OPN-375 186 μg BID, Delivered via exhalation delivery system
Number of Participants With a PGIC Score of Minimally/Much/Very Much Improved
9 Participants

Adverse Events

OPN-375 186 mcg BID

Serious events: 0 serious events
Other events: 1 other events
Deaths: 0 deaths

Serious adverse events

Adverse event data not reported

Other adverse events

Other adverse events
Measure
OPN-375 186 mcg BID
n=11 participants at risk
Fluticasone Propionate: OPN-375 186 μg BID, Delivered via exhalation delivery system
Cardiac disorders
Dyspnea
9.1%
1/11 • 24 weeks, and up to 30 days after the last dose
Respiratory, thoracic and mediastinal disorders
Asthma
9.1%
1/11 • 24 weeks, and up to 30 days after the last dose
Musculoskeletal and connective tissue disorders
Back Pain
9.1%
1/11 • 24 weeks, and up to 30 days after the last dose
Nervous system disorders
Dizziness
9.1%
1/11 • 24 weeks, and up to 30 days after the last dose
Infections and infestations
Fungal Skin Infection
9.1%
1/11 • 24 weeks, and up to 30 days after the last dose
Cardiac disorders
Hypotension
9.1%
1/11 • 24 weeks, and up to 30 days after the last dose
Infections and infestations
Influenza
9.1%
1/11 • 24 weeks, and up to 30 days after the last dose
Eye disorders
Lacrimation Increased
9.1%
1/11 • 24 weeks, and up to 30 days after the last dose
Respiratory, thoracic and mediastinal disorders
Nasal Discharge Discolouration
9.1%
1/11 • 24 weeks, and up to 30 days after the last dose
Infections and infestations
Sinusitis
9.1%
1/11 • 24 weeks, and up to 30 days after the last dose
Nervous system disorders
Tension Headache
9.1%
1/11 • 24 weeks, and up to 30 days after the last dose
Infections and infestations
Upper Respiratory Tract Infection
9.1%
1/11 • 24 weeks, and up to 30 days after the last dose
Respiratory, thoracic and mediastinal disorders
Vasomotor Rhinitis
9.1%
1/11 • 24 weeks, and up to 30 days after the last dose
Respiratory, thoracic and mediastinal disorders
Epistaxis
9.1%
1/11 • 24 weeks, and up to 30 days after the last dose

Additional Information

Jennifer Carothers

Optinose

Phone: 908-432-3061

Results disclosure agreements

  • Principal investigator is a sponsor employee Disclosure agreement is described in CTA between sponsor and PI
  • Publication restrictions are in place

Restriction type: OTHER