Phase 1 Dose Escalation Study of CGX1321 in Subjects With Advanced Gastrointestinal Tumors

NCT ID: NCT03507998

Last Updated: 2020-07-24

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

Get a concise snapshot of the trial, including recruitment status, study phase, enrollment targets, and key timeline milestones.

Recruitment Status

UNKNOWN

Clinical Phase

PHASE1

Total Enrollment

39 participants

Study Classification

INTERVENTIONAL

Study Start Date

2017-06-17

Study Completion Date

2021-04-01

Brief Summary

Review the sponsor-provided synopsis that highlights what the study is about and why it is being conducted.

This is a multi-center, open label, repeat dose, Phase 1 study consisting of a Dose Escalation Phase and a Dose Expansion Phase to evaluate safety, pharmacokinetics, and clinical activity.

Detailed Description

Dive into the extended narrative that explains the scientific background, objectives, and procedures in greater depth.

The purpose of the Dose Escalation Phase is to examine the safety and determine the maximum tolerated dose of CGX1321 when administered to subjects with advanced GI tumors that have relapsed or are refractory to or not considered medically suitable to receive standard of care treatment.

Once the dose is identified in the Dose Escalation Phase, the Dose Expansion Phase will start. The purpose of the Dose Expansion Phase is to continue to examine the safety and confirm the final Phase 2 dose of CGX1321 when administered to subjects with advanced GI tumors who meet the entry criteria.

Conditions

See the medical conditions and disease areas that this research is targeting or investigating.

Colorectal Adenocarcinoma Gastric Adenocarcinoma Pancreatic Adenocarcinoma Bile Duct Carcinoma Hepatocellular Carcinoma Esophageal Carcinoma Gastrointestinal Cancer

Study Design

Understand how the trial is structured, including allocation methods, masking strategies, primary purpose, and other design elements.

Allocation Method

NA

Intervention Model

SINGLE_GROUP

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

Review each arm or cohort in the study, along with the interventions and objectives associated with them.

CGX1321 Dosing

Dose Escalation Phase: Ascending doses of CGX1321 will be administered by cohort to determine the maximum tolerated dose. Patients will receive CGX1321, once daily, orally, for 3 weeks (21 days) followed by a one week (7 day) washout period in each 28 day cycle, according to the cohort they are assigned.

Dose Expansion Phase: Patients will receive the recommended dose (identified in the Dose Expansion Phase) of CGX1321

Group Type EXPERIMENTAL

CGX1321

Intervention Type DRUG

CGX1321 capsules for oral administration

Interventions

Learn about the drugs, procedures, or behavioral strategies being tested and how they are applied within this trial.

CGX1321

CGX1321 capsules for oral administration

Intervention Type DRUG

Eligibility Criteria

Check the participation requirements, including inclusion and exclusion rules, age limits, and whether healthy volunteers are accepted.

Inclusion Criteria

* Histologically-diagnosed advanced Gl tumors, such as colorectal adenocarcinoma, gastric adenocarcinoma, pancreatic adenocarcinoma, bile duct carcinoma, hepatocellular carcinoma, esophageal carcinoma that have relapsed or are refractory to or are not considered medically suitable to receive standard of care treatment
* Eastern Cooperative Oncology Group (ECOG) score of 0 - 1
* Minimum estimated life expectancy of 3 months
* Adequate organ function
* Recovery from prior treatment-related toxicities
* Ability to swallow capsules
* Willingness for subjects of reproductive potential to use adequate methods of contraception during and for 3 months after study treatment

Exclusion Criteria

* Prior exposure to a WNT inhibitor
* Received previous therapy for malignancy within 21 days
* Major surgery within 4 weeks of first dose of study drug
* Radiotherapy within 2 weeks of first dose of study drug
* Significant GI or variceal bleeding or subdural hematoma within 3 months of treatment start
* Uncontrolled central nervous system metastases or leptomeningeal metastases
* Requirement for immunosuppressive agents (must be off for at least 7 days)
* Currently receiving medications that are known CYP3A4/5 inhibitors. Patients currently receiving medications of known inducers of CYP3A4/5 or substrates of CYP2C8/9 and CYP1A2 may be excluded.
* Bone abnormalities
* Hypercalcemia
* Cardiac abnormalities
* Known human immunodeficiency virus positive, or active hepatitis A, B or C
* History of additional prior malignancy with the exception of surgically cured carcinomas such as skin, prostate, bladder, thyroid, cervix or other carcinomas in situ
* Active systemic infection requiring intravenous antibiotics within 2 weeks of treatment start
* Pregnancy or lactation
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

Meet the organizations funding or collaborating on the study and learn about their roles.

Guangzhou Curegenix Co. Ltd.

UNKNOWN

Sponsor Role collaborator

Curegenix Inc.

INDUSTRY

Sponsor Role lead

Responsible Party

Identify the individual or organization who holds primary responsibility for the study information submitted to regulators.

Responsibility Role SPONSOR

Locations

Explore where the study is taking place and check the recruitment status at each participating site.

Beijing Cancer Hospital

Beijing, , China

Site Status RECRUITING

Cancer Institute and Hospital, Chinese Academy of Medical Sciences

Beijing, , China

Site Status RECRUITING

Countries

Review the countries where the study has at least one active or historical site.

China

Central Contacts

Reach out to these primary contacts for questions about participation or study logistics.

Peter Ding

Role: CONTACT

(86)020-32299929

Facility Contacts

Find local site contact details for specific facilities participating in the trial.

Lin Shen, MD

Role: primary

Jifang Gong

Role: backup

86 13683208528

Aiping Zhou, MD

Role: primary

Wen Zhang, MD

Role: backup

86 18611643302

Other Identifiers

Review additional registry numbers or institutional identifiers associated with this trial.

CGX1321-102

Identifier Type: -

Identifier Source: org_study_id

More Related Trials

Additional clinical trials that may be relevant based on similarity analysis.

Adjuvant Treatment of Digestive Tract Tumors
NCT05742620 NOT_YET_RECRUITING NA