Trial Outcomes & Findings for Efficacy/Safety of CPI-613 in Combination With HD Cyt. and Mito. vs HD Cyt. and Mito. in Older Patients With R/R AML (NCT NCT03504410)

NCT ID: NCT03504410

Last Updated: 2023-02-08

Results Overview

Complete disappearance of all clinical evidence of disease

Recruitment status

TERMINATED

Study phase

PHASE3

Target enrollment

200 participants

Primary outcome timeframe

12 months

Results posted on

2023-02-08

Participant Flow

Participant milestones

Participant milestones
Measure
CPI-613 + HD Cytarabine and Mitoxantrone
CPI-613 at 2,000 mg/m2/day from day 1 to 5. Cytarabine at 1gm/m2 (5 doses), every 12 hours starting day 3. Mitoxantrone at 6gm/m2 (3 doses), everyday following the 1st, 2nd and 5th doses of Cytarabine.
Control (HAM) and Control Sub-groups (MEC and FLAG)
Cytarabine at 1gm/m2 (5 doses), every 12 hours starting day 3. Mitoxantrone at 6gm/m2 (3 doses), everyday following the 1st, 3rd and 5th doses of Cytarabine. Mitoxantrone, Etoposide and Cytarabine Etoposide 80mg/m over 60 minutes as a central line IV infusion; 6 doses Day 1 though 6 Cytarabine 1000mg/m2 over 3 hours as a central line IV infusion: 6 doses, Day 1 through 6 Mitoxantrone 6 mg/m2 over 30 minutes as a central line IV infusion: 6 dose, Day 1 through 6 Fludarabine, Cytarabine and Filgrastim Fludarabine 30mg/m2/day over 30 minutes as a central line IV infusion; 5 doses Day 1 though 5 Cytarabine 2g/m2 over 4 hours as a central line IV infusion: 4 hours after Fludarabine: 5 doses, Day 1 through 5 Filgrastim 5µg/kg/day by SQ or as per institutional guidelines starting from Day 1 through Day 5
Overall Study
STARTED
98
102
Overall Study
COMPLETED
11
11
Overall Study
NOT COMPLETED
87
91

Reasons for withdrawal

Withdrawal data not reported

Baseline Characteristics

Efficacy/Safety of CPI-613 in Combination With HD Cyt. and Mito. vs HD Cyt. and Mito. in Older Patients With R/R AML

Baseline characteristics by cohort

Baseline characteristics by cohort
Measure
CPI-613 + HD Cytarabine and Mitoxantrone
n=98 Participants
CPI-613 + High Dose Cytarabine and Mitoxantrone CPI-613 at 2,000 mg/m2/day from day 1 to 5. Cytarabine at 1gm/m2 (5 doses), every 12 hours starting day 3. Mitoxantrone at 6gm/m2 (3 doses), everyday following the 1st, 2nd and 5th doses of Cytarabine. CPI-613 + High Dose Cytarabine and Mitoxantrone: CPI-613 + High Dose Cytarabine and Mitoxantrone CPI-613: 2000mg/m2, 5 doses once a day, days 1-5 Cytarabine 1gm/m2, 5 doses every 12hrs starting day 3 through day 5 Mitoxantrone 6mg/m2, 3 doses, once a day following the first, third and fifth doses of Cytarabine
Control (HAM) and Control Sub-groups (MEC and FLAG)
n=102 Participants
High Dose Cytarabine and Mitoxantrone Cytarabine at 1gm/m2 (5 doses), every 12 hours starting day 3. Mitoxantrone at 6gm/m2 (3 doses), everyday following the 1st, 3rd and 5th doses of Cytarabine. Mitoxantrone, Etoposide and Cytarabine Etoposide 80mg/m over 60 minutes as a central line IV infusion; 6 doses Day 1 though 6 Cytarabine 1000mg/m2 over 3 hours as a central line IV infusion: 6 doses, Day 1 through 6 Mitoxantrone 6 mg/m2 over 30 minutes as a central line IV infusion: 6 dose, Day 1 through 6 Fludarabine, Cytarabine and Filgrastim Fludarabine 30mg/m2/day over 30 minutes as a central line IV infusion; 5 doses Day 1 though 5 Cytarabine 2g/m2 over 4 hours as a central line IV infusion: 4 hours after Fludarabine: 5 doses, Day 1 through 5 Filgrastim 5µg/kg/day by SQ or as per institutional guidelines starting from Day 1 through Day 5
Total
n=200 Participants
Total of all reporting groups
Age, Categorical
<=18 years
0 Participants
n=93 Participants
0 Participants
n=4 Participants
0 Participants
n=27 Participants
Age, Categorical
Between 18 and 65 years
42 Participants
n=93 Participants
46 Participants
n=4 Participants
88 Participants
n=27 Participants
Age, Categorical
>=65 years
56 Participants
n=93 Participants
56 Participants
n=4 Participants
112 Participants
n=27 Participants
Sex: Female, Male
Female
37 Participants
n=93 Participants
42 Participants
n=4 Participants
79 Participants
n=27 Participants
Sex: Female, Male
Male
61 Participants
n=93 Participants
60 Participants
n=4 Participants
121 Participants
n=27 Participants
Ethnicity (NIH/OMB)
Hispanic or Latino
8 Participants
n=93 Participants
3 Participants
n=4 Participants
11 Participants
n=27 Participants
Ethnicity (NIH/OMB)
Not Hispanic or Latino
72 Participants
n=93 Participants
81 Participants
n=4 Participants
153 Participants
n=27 Participants
Ethnicity (NIH/OMB)
Unknown or Not Reported
18 Participants
n=93 Participants
18 Participants
n=4 Participants
36 Participants
n=27 Participants

PRIMARY outcome

Timeframe: 12 months

Population: Number of Participants with Complete Remission (CR)

Complete disappearance of all clinical evidence of disease

Outcome measures

Outcome measures
Measure
CPI-613 + HD Cytarabine and Mitoxantrone
n=98 Participants
CPI-613 + High Dose Cytarabine and Mitoxantrone CPI-613 at 2,000 mg/m2/day from day 1 to 5. Cytarabine at 1gm/m2 (5 doses), every 12 hours starting day 3. Mitoxantrone at 6gm/m2 (3 doses), everyday following the 1st, 2nd and 5th doses of Cytarabine. CPI-613 + High Dose Cytarabine and Mitoxantrone: CPI-613 + High Dose Cytarabine and Mitoxantrone CPI-613: 2000mg/m2, 5 doses once a day, days 1-5 Cytarabine 1gm/m2, 5 doses every 12hrs starting day 3 through day 5 Mitoxantrone 6mg/m2, 3 doses, once a day following the first, third and fifth doses of Cytarabine
Control (HAM) and Control Sub-groups (MEC and FLAG)
n=102 Participants
High Dose Cytarabine and Mitoxantrone Cytarabine at 1gm/m2 (5 doses), every 12 hours starting day 3. Mitoxantrone at 6gm/m2 (3 doses), everyday following the 1st, 3rd and 5th doses of Cytarabine. Mitoxantrone, Etoposide and Cytarabine Etoposide 80mg/m over 60 minutes as a central line IV infusion; 6 doses Day 1 though 6 Cytarabine 1000mg/m2 over 3 hours as a central line IV infusion: 6 doses, Day 1 through 6 Mitoxantrone 6 mg/m2 over 30 minutes as a central line IV infusion: 6 dose, Day 1 through 6 Fludarabine, Cytarabine and Filgrastim Fludarabine 30mg/m2/day over 30 minutes as a central line IV infusion; 5 doses Day 1 though 5 Cytarabine 2g/m2 over 4 hours as a central line IV infusion: 4 hours after Fludarabine: 5 doses, Day 1 through 5 Filgrastim 5µg/kg/day by SQ or as per institutional guidelines starting from Day 1 through Day 5
Complete Remission (CR)
20 Participants
22 Participants

Adverse Events

CPI-613 + HD Cytarabine and Mitoxantrone

Serious events: 36 serious events
Other events: 93 other events
Deaths: 52 deaths

Control (HAM) and Control Sub-groups (MEC and FLAG)

Serious events: 34 serious events
Other events: 94 other events
Deaths: 55 deaths

Serious adverse events

Serious adverse events
Measure
CPI-613 + HD Cytarabine and Mitoxantrone
n=96 participants at risk
CPI-613 + High Dose Cytarabine and Mitoxantrone CPI-613 at 2,000 mg/m2/day from day 1 to 5. Cytarabine at 1gm/m2 (5 doses), every 12 hours starting day 3. Mitoxantrone at 6gm/m2 (3 doses), everyday following the 1st, 2nd and 5th doses of Cytarabine.
Control (HAM) and Control Sub-groups (MEC and FLAG)
n=97 participants at risk
High Dose Cytarabine and Mitoxantrone Cytarabine at 1gm/m2 (5 doses), every 12 hours starting day 3. Mitoxantrone at 6gm/m2 (3 doses), everyday following the 1st, 3rd and 5th doses of Cytarabine. Mitoxantrone, Etoposide and Cytarabine Etoposide 80mg/m over 60 minutes as a central line IV infusion; 6 doses Day 1 though 6 Cytarabine 1000mg/m2 over 3 hours as a central line IV infusion: 6 doses, Day 1 through 6 Mitoxantrone 6 mg/m2 over 30 minutes as a central line IV infusion: 6 dose, Day 1 through 6 Fludarabine, Cytarabine and Filgrastim Fludarabine 30mg/m2/day over 30 minutes as a central line IV infusion; 5 doses Day 1 though 5 Cytarabine 2g/m2 over 4 hours as a central line IV infusion: 4 hours after Fludarabine: 5 doses, Day 1 through 5 Filgrastim 5µg/kg/day by SQ or as per institutional guidelines starting from Day 1 through Day 5
Blood and lymphatic system disorders
disseminated intravascular coagulation
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Blood and lymphatic system disorders
Febrile Neutropenia
2.1%
2/96 • 38 months
6.2%
6/97 • 38 months
Blood and lymphatic system disorders
Hemolysis
2.1%
2/96 • 38 months
0.00%
0/97 • 38 months
Blood and lymphatic system disorders
Leukostasis syndrome
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Cardiac disorders
Atrial Fibrillation
3.1%
3/96 • 38 months
1.0%
1/97 • 38 months
Cardiac disorders
Atrial Flutter
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Cardiac disorders
Cardiac arrest
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Cardiac disorders
Cardiac failure
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Cardiac disorders
cardiac failure acute
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Eye disorders
Photophobia
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Gastrointestinal disorders
Anal fistula
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Gastrointestinal disorders
Colitis
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Gastrointestinal disorders
Enterocolitis
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Gastrointestinal disorders
Ileus
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Gastrointestinal disorders
small intestinal obstruction
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Gastrointestinal disorders
Stomatitis
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Infections and infestations
Achromobacter infection
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Infections and infestations
Anal Abscess
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Infections and infestations
Bacillus bacteraemia
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Infections and infestations
Bacteraemia
0.00%
0/96 • 38 months
2.1%
2/97 • 38 months
Infections and infestations
Covid-19
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Infections and infestations
COVID-19 pneumonia
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Infections and infestations
Candida infection
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Infections and infestations
Cellulitis
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Infections and infestations
Device related infection
0.00%
0/96 • 38 months
2.1%
2/97 • 38 months
Infections and infestations
Encephalitis
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Infections and infestations
Enterococcal infection
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Infections and infestations
Fungal oesophagitis
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Infections and infestations
Klebsiella sepsis
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Infections and infestations
Neutropenic sepsis
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Infections and infestations
Pneumococcal infection
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Infections and infestations
Pneumonia
4.2%
4/96 • 38 months
5.2%
5/97 • 38 months
Infections and infestations
Pseudomonal sepsis
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Infections and infestations
Scrotal infection
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Infections and infestations
Sepsis
6.2%
6/96 • 38 months
5.2%
5/97 • 38 months
Infections and infestations
Septic Shock
3.1%
3/96 • 38 months
1.0%
1/97 • 38 months
Infections and infestations
Staphylococcal infection
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Infections and infestations
Stenotrophomonas infection
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Injury, poisoning and procedural complications
Fall
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Metabolism and nutrition disorders
Fluid Overload
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Neoplasms benign, malignant and unspecified (incl cysts and polyps)
Basal Cell Carcinoma
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Nervous system disorders
Aphasia
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Nervous system disorders
Cerebrovascular accident
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Product Issues
device occlusion
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Renal and urinary disorders
Acute Kidney Injury
2.1%
2/96 • 38 months
0.00%
0/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Acute respiratory failure
2.1%
2/96 • 38 months
2.1%
2/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Pulmonary Oedema
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Respiratory Failure
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Vascular disorders
Hypotension
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months

Other adverse events

Other adverse events
Measure
CPI-613 + HD Cytarabine and Mitoxantrone
n=96 participants at risk
CPI-613 + High Dose Cytarabine and Mitoxantrone CPI-613 at 2,000 mg/m2/day from day 1 to 5. Cytarabine at 1gm/m2 (5 doses), every 12 hours starting day 3. Mitoxantrone at 6gm/m2 (3 doses), everyday following the 1st, 2nd and 5th doses of Cytarabine.
Control (HAM) and Control Sub-groups (MEC and FLAG)
n=97 participants at risk
High Dose Cytarabine and Mitoxantrone Cytarabine at 1gm/m2 (5 doses), every 12 hours starting day 3. Mitoxantrone at 6gm/m2 (3 doses), everyday following the 1st, 3rd and 5th doses of Cytarabine. Mitoxantrone, Etoposide and Cytarabine Etoposide 80mg/m over 60 minutes as a central line IV infusion; 6 doses Day 1 though 6 Cytarabine 1000mg/m2 over 3 hours as a central line IV infusion: 6 doses, Day 1 through 6 Mitoxantrone 6 mg/m2 over 30 minutes as a central line IV infusion: 6 dose, Day 1 through 6 Fludarabine, Cytarabine and Filgrastim Fludarabine 30mg/m2/day over 30 minutes as a central line IV infusion; 5 doses Day 1 though 5 Cytarabine 2g/m2 over 4 hours as a central line IV infusion: 4 hours after Fludarabine: 5 doses, Day 1 through 5 Filgrastim 5µg/kg/day by SQ or as per institutional guidelines starting from Day 1 through Day 5
Skin and subcutaneous tissue disorders
Rash morbilliform
1.0%
1/96 • 38 months
9.3%
9/97 • 38 months
Skin and subcutaneous tissue disorders
Rash pruritic
1.0%
1/96 • 38 months
2.1%
2/97 • 38 months
Infections and infestations
Rash pustular
2.1%
2/96 • 38 months
0.00%
0/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Respiratory depression
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Respiratory failure
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Nervous system disorders
Restless legs syndrome
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Rhinitis allergic
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Rhinorrhoea
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Infections and infestations
Rhinovirus infection
0.00%
0/96 • 38 months
2.1%
2/97 • 38 months
Infections and infestations
Root canal infection
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Infections and infestations
Scrotal infection
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Reproductive system and breast disorders
Scrotal pain
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Infections and infestations
Sepsis
10.4%
10/96 • 38 months
1.0%
1/97 • 38 months
Infections and infestations
Septic shock
5.2%
5/96 • 38 months
0.00%
0/97 • 38 months
Cardiac disorders
Sinus bradycardia
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Infections and infestations
Abdominal abscess
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Gastrointestinal disorders
Abdominal distension
3.1%
3/96 • 38 months
3.1%
3/97 • 38 months
Gastrointestinal disorders
Abdominal pain
5.2%
5/96 • 38 months
7.2%
7/97 • 38 months
Gastrointestinal disorders
Abdominal pain upper
3.1%
3/96 • 38 months
1.0%
1/97 • 38 months
Metabolism and nutrition disorders
Abnormal loss of weight
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Infections and infestations
Abscess limb
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Infections and infestations
Achromobacter infection
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Metabolism and nutrition disorders
Acidosis
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Investigations
Activated partial thromboplastin time prolonged
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Renal and urinary disorders
Acute kidney injury
8.3%
8/96 • 38 months
0.00%
0/97 • 38 months
Cardiac disorders
Acute myocardial infarction
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Acute pulmonary oedema
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Acute respiratory failure
3.1%
3/96 • 38 months
2.1%
2/97 • 38 months
Nervous system disorders
Ageusia
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Psychiatric disorders
Agitation
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Investigations
Alanine aminotransferase increased
9.4%
9/96 • 38 months
14.4%
14/97 • 38 months
Skin and subcutaneous tissue disorders
Alopecia
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Infections and infestations
Anal abscess
1.0%
1/96 • 38 months
36.1%
35/97 • 38 months
Gastrointestinal disorders
Anal fistula
2.1%
2/96 • 38 months
0.00%
0/97 • 38 months
Gastrointestinal disorders
Anal incontinence
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Gastrointestinal disorders
Anal inflammation
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Cardiac disorders
Angina pectoris
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Gastrointestinal disorders
Anorectal discomfort
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Psychiatric disorders
Anxiety
2.1%
2/96 • 38 months
0.00%
0/97 • 38 months
Nervous system disorders
Aphasia
1.0%
1/96 • 38 months
2.1%
2/97 • 38 months
Cardiac disorders
Arrhythmia
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Musculoskeletal and connective tissue disorders
Arthralgia
5.2%
5/96 • 38 months
0.00%
0/97 • 38 months
Investigations
Aspartate aminotransferase increased
8.3%
8/96 • 38 months
6.2%
6/97 • 38 months
Infections and infestations
Aspergilloma
1.0%
1/96 • 38 months
9.3%
9/97 • 38 months
Infections and infestations
Aspergillus infection
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
General disorders
Asthenia
3.1%
3/96 • 38 months
0.00%
0/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Atelectasis
0.00%
0/96 • 38 months
6.2%
6/97 • 38 months
Cardiac disorders
Atrial fibrillation
7.3%
7/96 • 38 months
1.0%
1/97 • 38 months
Cardiac disorders
Atrial flutter
1.0%
1/96 • 38 months
4.1%
4/97 • 38 months
Cardiac disorders
Atrioventricular block first degree
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Infections and infestations
Bacillus bacteraemia
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Infections and infestations
Bacillus infection
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Musculoskeletal and connective tissue disorders
Back pain
6.2%
6/96 • 38 months
0.00%
0/97 • 38 months
Infections and infestations
Bacteraemia
3.1%
3/96 • 38 months
8.2%
8/97 • 38 months
Reproductive system and breast disorders
Benign prostatic hyperplasia
1.0%
1/96 • 38 months
7.2%
7/97 • 38 months
Investigations
Blood alkaline phosphatase increased
4.2%
4/96 • 38 months
0.00%
0/97 • 38 months
Investigations
Blood bilirubin increased
10.4%
10/96 • 38 months
1.0%
1/97 • 38 months
Investigations
Blood creatinine increased
2.1%
2/96 • 38 months
5.2%
5/97 • 38 months
Investigations
Blood fibrinogen decreased
0.00%
0/96 • 38 months
7.2%
7/97 • 38 months
Investigations
Blood fibrinogen increased
1.0%
1/96 • 38 months
6.2%
6/97 • 38 months
Investigations
Blood folate decreased
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Investigations
Blood lactate dehydrogenase increased
2.1%
2/96 • 38 months
0.00%
0/97 • 38 months
Investigations
Blood phosphorus increased
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Investigations
Blood uric acid increased
0.00%
0/96 • 38 months
2.1%
2/97 • 38 months
Investigations
Body temperature increased
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Infections and infestations
Bone abscess
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Musculoskeletal and connective tissue disorders
Bone pain
3.1%
3/96 • 38 months
1.0%
1/97 • 38 months
Cardiac disorders
Bradycardia
4.2%
4/96 • 38 months
0.00%
0/97 • 38 months
Investigations
Breath sounds abnormal
0.00%
0/96 • 38 months
2.1%
2/97 • 38 months
Infections and infestations
Bronchopulmonary aspergillosis
2.1%
2/96 • 38 months
2.1%
2/97 • 38 months
Injury, poisoning and procedural complications
Burns second degree
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Investigations
C-reactive protein increased
5.2%
5/96 • 38 months
1.0%
1/97 • 38 months
Infections and infestations
Candida infection
3.1%
3/96 • 38 months
1.0%
1/97 • 38 months
Cardiac disorders
Cardiac arrest
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Cardiac disorders
Cardiac failure
2.1%
2/96 • 38 months
1.0%
1/97 • 38 months
Cardiac disorders
Cardiac failure acute
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Surgical and medical procedures
Catheter management
0.00%
0/96 • 38 months
3.1%
3/97 • 38 months
General disorders
Catheter site erythema
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
General disorders
Catheter site haemorrhage
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
General disorders
Catheter site induration
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
General disorders
Catheter site pain
1.0%
1/96 • 38 months
2.1%
2/97 • 38 months
Infections and infestations
Cellulitis
5.2%
5/96 • 38 months
0.00%
0/97 • 38 months
Nervous system disorders
Cerebral atrophy
0.00%
0/96 • 38 months
2.1%
2/97 • 38 months
Nervous system disorders
Cerebral haemorrhage
1.0%
1/96 • 38 months
4.1%
4/97 • 38 months
Nervous system disorders
Cerebrovascular accident
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Gastrointestinal disorders
Cheilitis
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
General disorders
Chills
5.2%
5/96 • 38 months
0.00%
0/97 • 38 months
Hepatobiliary disorders
Cholestasis
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Renal and urinary disorders
Chromaturia
1.0%
1/96 • 38 months
10.3%
10/97 • 38 months
Vascular disorders
Circulatory collapse
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Infections and infestations
Citrobacter infection
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Infections and infestations
Clostridium difficile colitis
4.2%
4/96 • 38 months
0.00%
0/97 • 38 months
Infections and infestations
Clostridium difficile infection
4.2%
4/96 • 38 months
1.0%
1/97 • 38 months
Musculoskeletal and connective tissue disorders
Coccydynia
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Gastrointestinal disorders
Colitis
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Psychiatric disorders
Confusional state
6.2%
6/96 • 38 months
0.00%
0/97 • 38 months
Infections and infestations
Conjunctivitis
0.00%
0/96 • 38 months
2.1%
2/97 • 38 months
Gastrointestinal disorders
Constipation
21.9%
21/96 • 38 months
0.00%
0/97 • 38 months
Injury, poisoning and procedural complications
Contusion
2.1%
2/96 • 38 months
1.0%
1/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Cough
9.4%
9/96 • 38 months
20.6%
20/97 • 38 months
Infections and infestations
COVID-19
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Infections and infestations
COVID-19 pneumonia
0.00%
0/96 • 38 months
9.3%
9/97 • 38 months
Investigations
Creatinine renal clearance decreased
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Metabolism and nutrition disorders
Decreased appetite
12.5%
12/96 • 38 months
1.0%
1/97 • 38 months
Skin and subcutaneous tissue disorders
Decubitus ulcer
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Vascular disorders
Deep vein thrombosis
1.0%
1/96 • 38 months
12.4%
12/97 • 38 months
Metabolism and nutrition disorders
Dehydration
1.0%
1/96 • 38 months
2.1%
2/97 • 38 months
Psychiatric disorders
Delirium
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Nervous system disorders
Depressed level of consciousness
1.0%
1/96 • 38 months
2.1%
2/97 • 38 months
Psychiatric disorders
Depression
2.1%
2/96 • 38 months
3.1%
3/97 • 38 months
Skin and subcutaneous tissue disorders
Dermal cyst
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Skin and subcutaneous tissue disorders
Dermatitis contact
1.0%
1/96 • 38 months
2.1%
2/97 • 38 months
Skin and subcutaneous tissue disorders
Dermatitis psoriasiform
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Infections and infestations
Device related infection
3.1%
3/96 • 38 months
0.00%
0/97 • 38 months
General disorders
Device related thrombosis
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Metabolism and nutrition disorders
Diabetes mellitus
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Gastrointestinal disorders
Diarrhoea
44.8%
43/96 • 38 months
4.1%
4/97 • 38 months
Psychiatric disorders
Disorientation
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Blood and lymphatic system disorders
Disseminated intravascular coagulation
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Nervous system disorders
Dizziness
6.2%
6/96 • 38 months
22.7%
22/97 • 38 months
Skin and subcutaneous tissue disorders
Drug eruption
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Immune system disorders
Drug hypersensitivity
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Eye disorders
Dry eye
1.0%
1/96 • 38 months
8.2%
8/97 • 38 months
Gastrointestinal disorders
Dry mouth
3.1%
3/96 • 38 months
0.00%
0/97 • 38 months
Skin and subcutaneous tissue disorders
Dry skin
4.2%
4/96 • 38 months
0.00%
0/97 • 38 months
Nervous system disorders
Dysgeusia
3.1%
3/96 • 38 months
2.1%
2/97 • 38 months
Nervous system disorders
Dyskinesia
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Nervous system disorders
Dysmetria
0.00%
0/96 • 38 months
2.1%
2/97 • 38 months
Gastrointestinal disorders
Dyspepsia
4.2%
4/96 • 38 months
3.1%
3/97 • 38 months
Gastrointestinal disorders
Dysphagia
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Dyspnoea
8.3%
8/96 • 38 months
1.0%
1/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Dyspnoea exertional
0.00%
0/96 • 38 months
4.1%
4/97 • 38 months
Renal and urinary disorders
Dysuria
3.1%
3/96 • 38 months
1.0%
1/97 • 38 months
Skin and subcutaneous tissue disorders
Ecchymosis
1.0%
1/96 • 38 months
12.4%
12/97 • 38 months
Infections and infestations
Ecthyma
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Investigations
Ejection fraction decreased
3.1%
3/96 • 38 months
3.1%
3/97 • 38 months
Investigations
Electrocardiogram abnormal
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Investigations
Electrocardiogram QT prolonged
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Infections and infestations
Encephalitis
1.0%
1/96 • 38 months
2.1%
2/97 • 38 months
Infections and infestations
Endocarditis
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Infections and infestations
Enterococcal infection
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Gastrointestinal disorders
Enterocolitis
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Infections and infestations
Enterocolitis infectious
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Gastrointestinal disorders
Epigastric discomfort
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Epistaxis
8.3%
8/96 • 38 months
0.00%
0/97 • 38 months
Skin and subcutaneous tissue disorders
Erythema
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Infections and infestations
Escherichia bacteraemia
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Eye disorders
Extraocular muscle paresis
0.00%
0/96 • 38 months
12.4%
12/97 • 38 months
Eye disorders
Eye haemorrhage
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Eye disorders
Eye inflammation
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Eye disorders
Eye pain
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Eye disorders
Eye pruritus
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Eye disorders
Eye swelling
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
General disorders
Face oedema
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Injury, poisoning and procedural complications
Fall
4.2%
4/96 • 38 months
0.00%
0/97 • 38 months
General disorders
Fatigue
15.6%
15/96 • 38 months
0.00%
0/97 • 38 months
Blood and lymphatic system disorders
Febrile neutropenia
36.5%
35/96 • 38 months
2.1%
2/97 • 38 months
Investigations
Fibrin D dimer increased
2.1%
2/96 • 38 months
5.2%
5/97 • 38 months
Musculoskeletal and connective tissue disorders
Flank pain
4.2%
4/96 • 38 months
13.4%
13/97 • 38 months
Gastrointestinal disorders
Flatulence
3.1%
3/96 • 38 months
33.0%
32/97 • 38 months
Metabolism and nutrition disorders
Fluid overload
4.2%
4/96 • 38 months
3.1%
3/97 • 38 months
Metabolism and nutrition disorders
Fluid retention
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Vascular disorders
Flushing
0.00%
0/96 • 38 months
5.2%
5/97 • 38 months
Infections and infestations
Folliculitis
1.0%
1/96 • 38 months
6.2%
6/97 • 38 months
Infections and infestations
Fungal oesophagitis
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
General disorders
Gait disturbance
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Investigations
Gamma-glutamyltransferase increased
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Gastrointestinal disorders
Gastrointestinal pain
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Gastrointestinal disorders
Gastrooesophageal reflux disease
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
General disorders
Generalised oedema
2.1%
2/96 • 38 months
2.1%
2/97 • 38 months
Gastrointestinal disorders
Gingival bleeding
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Gastrointestinal disorders
Gingival erythema
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Gastrointestinal disorders
Gingival pain
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Infections and infestations
Gingivitis
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Investigations
Glomerular filtration rate decreased
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Metabolism and nutrition disorders
Gout
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Immune system disorders
Graft versus host disease in skin
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Reproductive system and breast disorders
Gynaecomastia
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Musculoskeletal and connective tissue disorders
Haemarthrosis
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Gastrointestinal disorders
Haematochezia
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Vascular disorders
Haematoma
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Renal and urinary disorders
Haematuria
6.2%
6/96 • 38 months
0.00%
0/97 • 38 months
Blood and lymphatic system disorders
Haemolysis
2.1%
2/96 • 38 months
1.0%
1/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Haemoptysis
1.0%
1/96 • 38 months
2.1%
2/97 • 38 months
Gastrointestinal disorders
Haemorrhoidal haemorrhage
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Gastrointestinal disorders
Haemorrhoids
5.2%
5/96 • 38 months
0.00%
0/97 • 38 months
Psychiatric disorders
Hallucination
2.1%
2/96 • 38 months
2.1%
2/97 • 38 months
Psychiatric disorders
Hallucination, visual
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Injury, poisoning and procedural complications
Head injury
1.0%
1/96 • 38 months
3.1%
3/97 • 38 months
Nervous system disorders
Headache
19.8%
19/96 • 38 months
0.00%
0/97 • 38 months
Investigations
Heart rate increased
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Investigations
Heart rate irregular
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Nervous system disorders
Hemiparesis
1.0%
1/96 • 38 months
23.7%
23/97 • 38 months
Hepatobiliary disorders
Hepatic cyst
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Infections and infestations
Hepatosplenic candidiasis
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Infections and infestations
Herpes simplex
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Infections and infestations
Herpes simplex reactivation
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Infections and infestations
Herpes zoster
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Hiccups
4.2%
4/96 • 38 months
1.0%
1/97 • 38 months
Hepatobiliary disorders
Hyperbilirubinaemia
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Metabolism and nutrition disorders
Hyperglycaemia
12.5%
12/96 • 38 months
0.00%
0/97 • 38 months
Skin and subcutaneous tissue disorders
Hyperhidrosis
2.1%
2/96 • 38 months
4.1%
4/97 • 38 months
Metabolism and nutrition disorders
Hyperkalaemia
3.1%
3/96 • 38 months
1.0%
1/97 • 38 months
Nervous system disorders
Hyperkinesia
0.00%
0/96 • 38 months
10.3%
10/97 • 38 months
Metabolism and nutrition disorders
Hypermagnesaemia
2.1%
2/96 • 38 months
3.1%
3/97 • 38 months
Metabolism and nutrition disorders
Hypernatraemia
1.0%
1/96 • 38 months
4.1%
4/97 • 38 months
Metabolism and nutrition disorders
Hyperphosphataemia
4.2%
4/96 • 38 months
1.0%
1/97 • 38 months
Immune system disorders
Hypersensitivity
1.0%
1/96 • 38 months
2.1%
2/97 • 38 months
Vascular disorders
Hypertension
5.2%
5/96 • 38 months
0.00%
0/97 • 38 months
Vascular disorders
Hypertensive crisis
1.0%
1/96 • 38 months
8.2%
8/97 • 38 months
General disorders
Hyperthermia
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Metabolism and nutrition disorders
Hyperuricaemia
0.00%
0/96 • 38 months
10.3%
10/97 • 38 months
Metabolism and nutrition disorders
Hypervolaemia
2.1%
2/96 • 38 months
0.00%
0/97 • 38 months
Nervous system disorders
Hypoaesthesia
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Metabolism and nutrition disorders
Hypoalbuminaemia
11.5%
11/96 • 38 months
2.1%
2/97 • 38 months
Metabolism and nutrition disorders
Hypocalcaemia
16.7%
16/96 • 38 months
0.00%
0/97 • 38 months
Metabolism and nutrition disorders
Hypoglycaemia
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Metabolism and nutrition disorders
Hypokalaemia
29.2%
28/96 • 38 months
14.4%
14/97 • 38 months
Metabolism and nutrition disorders
Hypomagnesaemia
14.6%
14/96 • 38 months
16.5%
16/97 • 38 months
Metabolism and nutrition disorders
Hyponatraemia
9.4%
9/96 • 38 months
1.0%
1/97 • 38 months
Metabolism and nutrition disorders
Hypophagia
0.00%
0/96 • 38 months
37.1%
36/97 • 38 months
Metabolism and nutrition disorders
Hypophosphataemia
15.6%
15/96 • 38 months
15.5%
15/97 • 38 months
Vascular disorders
Hypotension
10.4%
10/96 • 38 months
4.1%
4/97 • 38 months
General disorders
Hypothermia
1.0%
1/96 • 38 months
2.1%
2/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Hypoxia
6.2%
6/96 • 38 months
14.4%
14/97 • 38 months
Gastrointestinal disorders
Ileus
1.0%
1/96 • 38 months
14.4%
14/97 • 38 months
Infections and infestations
Infection
3.1%
3/96 • 38 months
0.00%
0/97 • 38 months
General disorders
Inflammation
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
General disorders
Influenza like illness
0.00%
0/96 • 38 months
4.1%
4/97 • 38 months
Injury, poisoning and procedural complications
Infusion related reaction
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
General disorders
Injection site reaction
1.0%
1/96 • 38 months
2.1%
2/97 • 38 months
Psychiatric disorders
Insomnia
10.4%
10/96 • 38 months
1.0%
1/97 • 38 months
Reproductive system and breast disorders
Intermenstrual bleeding
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Investigations
International normalised ratio increased
1.0%
1/96 • 38 months
2.1%
2/97 • 38 months
Injury, poisoning and procedural complications
Joint injury
1.0%
1/96 • 38 months
2.1%
2/97 • 38 months
Vascular disorders
Jugular vein thrombosis
1.0%
1/96 • 38 months
8.2%
8/97 • 38 months
Infections and infestations
Klebsiella bacteraemia
2.1%
2/96 • 38 months
1.0%
1/97 • 38 months
Infections and infestations
Klebsiella sepsis
1.0%
1/96 • 38 months
2.1%
2/97 • 38 months
Infections and infestations
Leptotrichia infection
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Nervous system disorders
Lethargy
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Infections and infestations
Leuconostoc infection
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Blood and lymphatic system disorders
Leukopenia
4.2%
4/96 • 38 months
0.00%
0/97 • 38 months
Blood and lymphatic system disorders
Leukostasis syndrome
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Gastrointestinal disorders
Lip pain
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Gastrointestinal disorders
Lip swelling
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Gastrointestinal disorders
Lip ulceration
1.0%
1/96 • 38 months
4.1%
4/97 • 38 months
General disorders
Localised oedema
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Lung opacity
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Blood and lymphatic system disorders
Lymph node pain
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Blood and lymphatic system disorders
Lymphadenopathy
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Investigations
Lymphocyte count decreased
12.5%
12/96 • 38 months
3.1%
3/97 • 38 months
Blood and lymphatic system disorders
Lymphopenia
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Skin and subcutaneous tissue disorders
Macule
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
General disorders
Malaise
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Metabolism and nutrition disorders
Malnutrition
2.1%
2/96 • 38 months
11.3%
11/97 • 38 months
General disorders
Medical device site pain
2.1%
2/96 • 38 months
0.00%
0/97 • 38 months
General disorders
Medical device site pruritus
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Gastrointestinal disorders
Mesenteric panniculitis
1.0%
1/96 • 38 months
2.1%
2/97 • 38 months
Renal and urinary disorders
Micturition urgency
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Cardiac disorders
Mitral valve incompetence
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Infections and infestations
Moraxella infection
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Infections and infestations
Morganella infection
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Gastrointestinal disorders
Mouth haemorrhage
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Gastrointestinal disorders
Mouth ulceration
3.1%
3/96 • 38 months
1.0%
1/97 • 38 months
Musculoskeletal and connective tissue disorders
Muscle spasms
2.1%
2/96 • 38 months
1.0%
1/97 • 38 months
Musculoskeletal and connective tissue disorders
Muscular weakness
3.1%
3/96 • 38 months
1.0%
1/97 • 38 months
Musculoskeletal and connective tissue disorders
Musculoskeletal chest pain
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Musculoskeletal and connective tissue disorders
Musculoskeletal pain
0.00%
0/96 • 38 months
3.1%
3/97 • 38 months
Musculoskeletal and connective tissue disorders
Myalgia
3.1%
3/96 • 38 months
1.0%
1/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Nasal cavity mass
0.00%
0/96 • 38 months
3.1%
3/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Nasal congestion
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Nasal discomfort
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Nasal disorder
1.0%
1/96 • 38 months
2.1%
2/97 • 38 months
Infections and infestations
Nasal herpes
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Gastrointestinal disorders
Nausea
32.3%
31/96 • 38 months
4.1%
4/97 • 38 months
Musculoskeletal and connective tissue disorders
Neck pain
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Nervous system disorders
Neuralgia
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Nervous system disorders
Neuropathy peripheral
2.1%
2/96 • 38 months
1.0%
1/97 • 38 months
Blood and lymphatic system disorders
Neutropenia
7.3%
7/96 • 38 months
25.8%
25/97 • 38 months
Gastrointestinal disorders
Neutropenic colitis
1.0%
1/96 • 38 months
2.1%
2/97 • 38 months
Infections and infestations
Neutropenic sepsis
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Investigations
Neutrophil count decreased
12.5%
12/96 • 38 months
2.1%
2/97 • 38 months
Skin and subcutaneous tissue disorders
Night sweats
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Renal and urinary disorders
Nocturia
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
General disorders
Non-cardiac chest pain
1.0%
1/96 • 38 months
2.1%
2/97 • 38 months
Eye disorders
Ocular discomfort
1.0%
1/96 • 38 months
15.5%
15/97 • 38 months
Eye disorders
Ocular hyperaemia
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
General disorders
Oedema peripheral
19.8%
19/96 • 38 months
1.0%
1/97 • 38 months
Infections and infestations
Oral candidiasis
1.0%
1/96 • 38 months
3.1%
3/97 • 38 months
Gastrointestinal disorders
Oral dysaesthesia
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Infections and infestations
Oral herpes
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Infections and infestations
Oral infection
2.1%
2/96 • 38 months
20.6%
20/97 • 38 months
Gastrointestinal disorders
Oral pain
3.1%
3/96 • 38 months
0.00%
0/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Oropharyngeal pain
2.1%
2/96 • 38 months
1.0%
1/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Oropharyngeal plaque
1.0%
1/96 • 38 months
5.2%
5/97 • 38 months
Vascular disorders
Orthostatic hypotension
2.1%
2/96 • 38 months
0.00%
0/97 • 38 months
General disorders
Pain
2.1%
2/96 • 38 months
4.1%
4/97 • 38 months
Musculoskeletal and connective tissue disorders
Pain in extremity
3.1%
3/96 • 38 months
3.1%
3/97 • 38 months
Musculoskeletal and connective tissue disorders
Pain in jaw
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Blood and lymphatic system disorders
Pancytopenia
3.1%
3/96 • 38 months
1.0%
1/97 • 38 months
Nervous system disorders
Paraesthesia
1.0%
1/96 • 38 months
4.1%
4/97 • 38 months
Infections and infestations
Pathogen resistance
0.00%
0/96 • 38 months
5.2%
5/97 • 38 months
Cardiac disorders
Pericardial effusion
2.1%
2/96 • 38 months
2.1%
2/97 • 38 months
General disorders
Peripheral swelling
0.00%
0/96 • 38 months
2.1%
2/97 • 38 months
Skin and subcutaneous tissue disorders
Petechiae
2.1%
2/96 • 38 months
1.0%
1/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Pharyngeal oedema
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Vascular disorders
Phlebitis
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Eye disorders
Photophobia
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Investigations
Platelet count decreased
19.8%
19/96 • 38 months
7.2%
7/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Pleural effusion
6.2%
6/96 • 38 months
1.0%
1/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Pleuritic pain
2.1%
2/96 • 38 months
1.0%
1/97 • 38 months
Infections and infestations
Pneumococcal infection
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Infections and infestations
Pneumonia
8.3%
8/96 • 38 months
20.6%
20/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Pneumonia aspiration
1.0%
1/96 • 38 months
3.1%
3/97 • 38 months
Infections and infestations
Pneumonia fungal
2.1%
2/96 • 38 months
1.0%
1/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Pneumonitis
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Renal and urinary disorders
Pollakiuria
2.1%
2/96 • 38 months
10.3%
10/97 • 38 months
Nervous system disorders
Polyneuropathy
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Injury, poisoning and procedural complications
Post procedural haematoma
1.0%
1/96 • 38 months
5.2%
5/97 • 38 months
Injury, poisoning and procedural complications
Post procedural swelling
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Nervous system disorders
Presyncope
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Injury, poisoning and procedural complications
Procedural pain
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Gastrointestinal disorders
Proctalgia
2.1%
2/96 • 38 months
0.00%
0/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Productive cough
2.1%
2/96 • 38 months
1.0%
1/97 • 38 months
Surgical and medical procedures
Prophylaxis of nausea and vomiting
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Investigations
Prothrombin time prolonged
0.00%
0/96 • 38 months
2.1%
2/97 • 38 months
Skin and subcutaneous tissue disorders
Pruritus
7.3%
7/96 • 38 months
1.0%
1/97 • 38 months
Infections and infestations
Pseudomonal bacteraemia
2.1%
2/96 • 38 months
4.1%
4/97 • 38 months
Infections and infestations
Pseudomonal sepsis
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Infections and infestations
Pseudomonal skin infection
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Nervous system disorders
Psychogenic seizure
0.00%
0/96 • 38 months
4.1%
4/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Pulmonary cavitation
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Pulmonary mass
3.1%
3/96 • 38 months
0.00%
0/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Pulmonary oedema
4.2%
4/96 • 38 months
1.0%
1/97 • 38 months
Investigations
Pulse abnormal
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
General disorders
Pyrexia
22.9%
22/96 • 38 months
0.00%
0/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Rales
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Skin and subcutaneous tissue disorders
Rash
6.2%
6/96 • 38 months
4.1%
4/97 • 38 months
Skin and subcutaneous tissue disorders
Rash erythematous
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Skin and subcutaneous tissue disorders
Rash macular
1.0%
1/96 • 38 months
22.7%
22/97 • 38 months
Skin and subcutaneous tissue disorders
Rash maculo-papular
3.1%
3/96 • 38 months
4.1%
4/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Sinus pain
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Cardiac disorders
Sinus tachycardia
3.1%
3/96 • 38 months
10.3%
10/97 • 38 months
Infections and infestations
Sinusitis
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Injury, poisoning and procedural complications
Skin abrasion
1.0%
1/96 • 38 months
2.1%
2/97 • 38 months
Skin and subcutaneous tissue disorders
Skin exfoliation
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Infections and infestations
Skin infection
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Injury, poisoning and procedural complications
Skin laceration
1.0%
1/96 • 38 months
2.1%
2/97 • 38 months
Skin and subcutaneous tissue disorders
Skin lesion
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Skin and subcutaneous tissue disorders
Skin mass
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Skin and subcutaneous tissue disorders
Skin ulcer
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Injury, poisoning and procedural complications
Skin wound
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Sleep apnoea syndrome
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Psychiatric disorders
Sleep disorder
2.1%
2/96 • 38 months
1.0%
1/97 • 38 months
Gastrointestinal disorders
Small intestinal obstruction
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Sneezing
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Nervous system disorders
Somnolence
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Blood and lymphatic system disorders
Splenomegaly
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Sputum retention
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Infections and infestations
Staphylococcal bacteraemia
3.1%
3/96 • 38 months
0.00%
0/97 • 38 months
Infections and infestations
Staphylococcal infection
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Infections and infestations
Stenotrophomonas infection
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Infections and infestations
Stenotrophomonas sepsis
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Gastrointestinal disorders
Stomatitis
10.4%
10/96 • 38 months
2.1%
2/97 • 38 months
Infections and infestations
Stomatococcal infection
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Infections and infestations
Streptococcal bacteraemia
2.1%
2/96 • 38 months
0.00%
0/97 • 38 months
Infections and infestations
Streptococcal infection
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Infections and infestations
Subcutaneous abscess
1.0%
1/96 • 38 months
15.5%
15/97 • 38 months
Injury, poisoning and procedural complications
Subdural haematoma
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Cardiac disorders
Supraventricular tachycardia
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
General disorders
Swelling face
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Eye disorders
Swelling of eyelid
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Nervous system disorders
Syncope
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Cardiac disorders
Tachycardia
2.1%
2/96 • 38 months
1.0%
1/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Tachypnoea
2.1%
2/96 • 38 months
1.0%
1/97 • 38 months
Nervous system disorders
Taste disorder
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Gastrointestinal disorders
Terminal ileitis
1.0%
1/96 • 38 months
2.1%
2/97 • 38 months
General disorders
Thirst
0.00%
0/96 • 38 months
4.1%
4/97 • 38 months
Injury, poisoning and procedural complications
Thoracic vertebral fracture
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Throat irritation
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Blood and lymphatic system disorders
Thrombocytopenia
18.8%
18/96 • 38 months
0.00%
0/97 • 38 months
Vascular disorders
Thrombophlebitis
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Vascular disorders
Thrombophlebitis superficial
2.1%
2/96 • 38 months
0.00%
0/97 • 38 months
Infections and infestations
Tooth abscess
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Gastrointestinal disorders
Tooth disorder
0.00%
0/96 • 38 months
14.4%
14/97 • 38 months
Infections and infestations
Tooth infection
2.1%
2/96 • 38 months
0.00%
0/97 • 38 months
Gastrointestinal disorders
Toothache
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Investigations
Transaminases increased
2.1%
2/96 • 38 months
1.0%
1/97 • 38 months
Injury, poisoning and procedural complications
Transfusion reaction
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Investigations
Troponin I increased
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Metabolism and nutrition disorders
Tumour lysis syndrome
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Upper-airway cough syndrome
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Renal and urinary disorders
Urethral pain
1.0%
1/96 • 38 months
2.1%
2/97 • 38 months
Renal and urinary disorders
Urinary hesitation
1.0%
1/96 • 38 months
2.1%
2/97 • 38 months
Renal and urinary disorders
Urinary incontinence
0.00%
0/96 • 38 months
6.2%
6/97 • 38 months
Renal and urinary disorders
Urinary retention
3.1%
3/96 • 38 months
2.1%
2/97 • 38 months
Infections and infestations
Urinary tract infection
2.1%
2/96 • 38 months
0.00%
0/97 • 38 months
Skin and subcutaneous tissue disorders
Urticaria
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Reproductive system and breast disorders
Vaginal haemorrhage
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Infections and infestations
Vaginal infection
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Cardiac disorders
Ventricular arrhythmia
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Eye disorders
Vision blurred
2.1%
2/96 • 38 months
3.1%
3/97 • 38 months
Eye disorders
Visual acuity reduced
1.0%
1/96 • 38 months
0.00%
0/97 • 38 months
Eye disorders
Visual field defect
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Eye disorders
Visual impairment
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Metabolism and nutrition disorders
Vitamin D deficiency
0.00%
0/96 • 38 months
1.0%
1/97 • 38 months
Gastrointestinal disorders
Vomiting
10.4%
10/96 • 38 months
1.0%
1/97 • 38 months
Gastrointestinal disorders
Vomiting projectile
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months
Investigations
Weight decreased
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Investigations
Weight increased
2.1%
2/96 • 38 months
1.0%
1/97 • 38 months
Respiratory, thoracic and mediastinal disorders
Wheezing
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Investigations
White blood cell count decreased
15.6%
15/96 • 38 months
14.4%
14/97 • 38 months
Injury, poisoning and procedural complications
Wound
1.0%
1/96 • 38 months
1.0%
1/97 • 38 months
Endocrine disorders
Hypothyroidism
0.00%
0/96 • 38 months
2.1%
2/97 • 38 months
Blood and lymphatic system disorders
Anaemia
34.4%
33/96 • 38 months
2.1%
2/97 • 38 months
Neoplasms benign, malignant and unspecified (incl cysts and polyps)
Basal cell carcinoma
1.0%
1/96 • 38 months
4.1%
4/97 • 38 months
Product Issues
Device occlusion
0.00%
0/96 • 38 months
13.4%
13/97 • 38 months
Ear and labyrinth disorders
Vertigo positional
0.00%
0/96 • 38 months
0.00%
0/97 • 38 months

Additional Information

Sanejev Luther

Cornerstone Pharmaceuticals Inc

Phone: 585-978-1351

Results disclosure agreements

  • Principal investigator is a sponsor employee
  • Publication restrictions are in place