Safety Evaluation of IV Tc 99m Tilmanocept and Comparison of Imaging With Sulfur Colloid in Subjects With and Without NASH

NCT ID: NCT03332940

Last Updated: 2024-12-24

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

TERMINATED

Clinical Phase

PHASE1

Total Enrollment

6 participants

Study Classification

INTERVENTIONAL

Study Start Date

2017-12-06

Study Completion Date

2019-03-10

Brief Summary

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This is a prospective, open-label, multicenter, safety, comparative study of IV administered Tc99m-tilmanocept and unfiltered Tc99m sulfur colloid in the detection of and assessment of three dimensional tessellation localization to the liver in subjects with and without moderate to severe nonalcoholic steatohepatitis (NASH) by planar and SPECT/CT imaging.

This study is designed to evaluate the safety and tolerability of Tc99m-tilmanocept in subjects with NASH.

Detailed Description

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Conditions

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Nonalcoholic Steatohepatitis NASH - Nonalcoholic Steatohepatitis

Keywords

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Tc99m-tilmanocept Tilmanocept NASH Nonalcoholic Steatohepatitis

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

SEQUENTIAL

Primary Study Purpose

DIAGNOSTIC

Blinding Strategy

NONE

Study Groups

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NASH subjects

All subjects will receive a single IV injection of unfiltered sulfur colloid radiolabeled with 8 mCi Tc99m on study day 0. All subjects will receive a single IV injection of 200 mcg tilmanocept radiolabeled with 8 mCi Tc99m on study day 3.

Group Type EXPERIMENTAL

Tc 99M Sulfur Colloid

Intervention Type DRUG

Sulfur colloid is a radiotracer that is indicated for imaging areas of functional reticuloendothelial cells in the liver, spleen, and bone marrow.

Tc99m-tilmanocept

Intervention Type DRUG

Tilmanocept is a radiotracer that accumulates in macrophages by binding to a mannose binding receptor that resides on the surface.

Healthy controls

All subjects will receive a single IV injection of unfiltered sulfur colloid radiolabeled with 8 mCi Tc99m on study day 0. All subjects will receive a single IV injection of 200 mcg tilmanocept radiolabeled with 8 mCi Tc99m on study day 3.

Group Type EXPERIMENTAL

Tc 99M Sulfur Colloid

Intervention Type DRUG

Sulfur colloid is a radiotracer that is indicated for imaging areas of functional reticuloendothelial cells in the liver, spleen, and bone marrow.

Tc99m-tilmanocept

Intervention Type DRUG

Tilmanocept is a radiotracer that accumulates in macrophages by binding to a mannose binding receptor that resides on the surface.

Interventions

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Tc 99M Sulfur Colloid

Sulfur colloid is a radiotracer that is indicated for imaging areas of functional reticuloendothelial cells in the liver, spleen, and bone marrow.

Intervention Type DRUG

Tc99m-tilmanocept

Tilmanocept is a radiotracer that accumulates in macrophages by binding to a mannose binding receptor that resides on the surface.

Intervention Type DRUG

Other Intervention Names

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Sulfur colloid Tilmanocept Lymphoseek

Eligibility Criteria

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Inclusion Criteria

* ALL SUBJECTS:

1. The subject has provided written informed consent with HIPAA (Health Information Portability and Accountability Act) authorization before the initiation of any study-related procedures.
2. The subject is ≥18 years of age at the time of consent.
3. The subject has a body mass index (BMI) between 18 and 45.

CONTROL SUBJECTS:
4. The subject is deemed to be clinically free of any infectious/inflammatory disease(s) for at least 4 weeks prior to the consent date.
5. The subject has not taken any antibiotics for at least 4 weeks prior to the consent date.

NASH SUBJECTS:

4\. The subject has biopsy-confirmed NASH within 12 months prior to enrollment. 5. The subject has a NAFLD Activity Score (NAS) of ≥ 4, with a score of at least 1 for each steatosis, lobular inflammation, and hepatocyte ballooning.

6\. The subject has fibrosis staging of F3-F4.

Exclusion Criteria

* ALL SUBJECTS:

1. The subject is pregnant or lactating.
2. The subject size or weight is not compatible with imaging per the investigator.
3. The subject has received radiation therapy or chemotherapy or has a previous diagnosis of cancer other than basal cell carcinoma.
4. The subject has renal insufficiency as demonstrated by a GFR of \< 60 mL/min.
5. The subject has a chronic or persistent infection or has any condition that would, in the opinion of the examining physician, preclude their participation.
6. The subject has a known allergy to or has had an adverse reaction to dextran exposure.
7. The subject has received an investigational product within 30 days prior to the Tc 99m sulfur colloid administration.
8. The subject has received any radiopharmaceutical within 7 days prior to the administration of Tc 99m sulfur colloid.
9. The subject is HIV positive.
10. The subject has a history of alcohol abuse or currently consumes alcohol in excess of 3 drinks/day for men or 2 drinks/day for women.
11. The subject has hepatitis B or C.

CONTROL SUBJECTS:
12. The subject has hepatic insufficiency as demonstrated by ALT (alanine aminotransferase \[SGPT\]) or AST (aspartate aminotransferase \[SGOT\]) greater than two times the upper limit of normal (ULN).
13. The subject has been diagnosed with NASH, NAFLD, or other chronic liver disease.
14. The subject has been diagnosed with metabolic syndrome or Type I or II diabetes.

NASH SUBJECTS:

12\. The subject has any chronic liver disease aside from NASH/NAFLD.

13\. The subject has uncontrolled diabetes as indicated by an A1c \>9% within the 3 months prior to enrollment.
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

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Navidea Biopharmaceuticals

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Michael Blue, MD

Role: STUDY_DIRECTOR

Navidea Biopharmaceuticals, Inc.

Locations

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Kettering Medical Center

Kettering, Ohio, United States

Site Status

Countries

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United States

References

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Cope FO, Abbruzzese B, Sanders J, Metz W, Sturms K, Ralph D, Blue M, Zhang J, Bracci P, Bshara W, Behr S, Maurer T, Williams K, Walker J, Beverly A, Blay B, Damughatla A, Larsen M, Mountain C, Neylon E, Parcel K, Raghuraman K, Ricks K, Rose L, Sivakumar A, Streck N, Wang B, Wasco C, Williams A, Schlesinger LS, Azad A, Rajaram MVS, Jarjour W, Young N, Rosol T, McGrath M. Corrigendum to the inextricable axis of targeted diagnostic imaging and therapy: An immunological natural history approach [Nucl Med Biol 43 (2016) 215-225]. Nucl Med Biol. 2016 Dec;43(12):837. doi: 10.1016/j.nucmedbio.2016.10.001. No abstract available.

Reference Type BACKGROUND
PMID: 27866590 (View on PubMed)

Cope, F.O., W. Metz, et al. Innovations in receptor-targeted precision imaging at Navidea: diagnosis up close and personal. Nature Outlook (31 October 2013); S125-S129.

Reference Type BACKGROUND

Provided Documents

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Document Type: Study Protocol and Statistical Analysis Plan

View Document

Related Links

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https://www.navidea.com/

Navidea Biopharmaceuticals, Inc.

Other Identifiers

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NAV3-30

Identifier Type: -

Identifier Source: org_study_id