PF-06804103 Dose Escalation in HER2 Positive and Negative (Negative Only in Part 2) Solid Tumors

NCT ID: NCT03284723

Last Updated: 2024-09-03

Study Results

Results available

Outcome measurements, participant flow, baseline characteristics, and adverse events have been published for this study.

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Basic Information

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Recruitment Status

TERMINATED

Clinical Phase

PHASE1

Total Enrollment

95 participants

Study Classification

INTERVENTIONAL

Study Start Date

2017-11-01

Study Completion Date

2021-08-31

Brief Summary

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The study will evaluate the safety, pharmacokinetics and pharmacodynamics of increasing doses of PF-06804103 in patients with HER2 positive and negative breast and gastric cancer (HER2 positive only and gastric were studied in Part 1A only). The study will expand to look at selected doses in patients with HER2 positive and negative breast cancer.

Detailed Description

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Conditions

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Breast Neoplasms

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

SEQUENTIAL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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PF-06804103

Study Treatment

Group Type EXPERIMENTAL

PF-06804103

Intervention Type DRUG

Dose Escalation Part - 1A Dose Expansion Part - 2A

PF-06804103+Combination Regimen

Study Treatment

Group Type EXPERIMENTAL

PF-06804103 + Palbociclib +Letrozole

Intervention Type DRUG

Dose Escalation - Part 1B Dose Expansion - Part 2B

Interventions

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PF-06804103

Dose Escalation Part - 1A Dose Expansion Part - 2A

Intervention Type DRUG

PF-06804103 + Palbociclib +Letrozole

Dose Escalation - Part 1B Dose Expansion - Part 2B

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* HER2 positive breast cancer or gastric cancer that is resistant to standard therapy or for which no standard therapy is available (Part 1A only)
* HER2 positive and negative breast cancer (Part 2A)
* HER2 negative breast cancer (Part 1B \& Part 2B)
* Performance status of 0 or 1
* Adequate bone marrow, kidney and liver function

Exclusion Criteria

* Known CNS disease including, but not limited to, metastases
* History of exposure to certain cumulative doses of anthracyclines
* Grade 3 or higher hypersensitivity reaction to prior receipt of any antibody therapy
* Active and clinically significant bacterial, fungal, or viral infection
* Abnormal cardiac function defined by a LVEF \<50% by ECHO or MUGA
* Patients with previous history or active interstitial lung disease or pulmonary fibrosis, or a history of other clinically significant lung diseases
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Pfizer

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Pfizer CT.gov Call Center

Role: STUDY_DIRECTOR

Pfizer

Locations

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Banner-University Medical Center Tucson

Tucson, Arizona, United States

Site Status

The University of Arizona Cancer Center - North Campus

Tucson, Arizona, United States

Site Status

The University of Arizona Cancer Center

Tucson, Arizona, United States

Site Status

Cedars-Sinai Medical Center, Samuel Oschin Comprehensive Cancer Institute

Los Angeles, California, United States

Site Status

UCLA Health (main campus)

Los Angeles, California, United States

Site Status

UCLA Hematology/Oncology

Los Angeles, California, United States

Site Status

Santa Monica - UCLA Medical Center and Orthopaedic Hospital

Santa Monica, California, United States

Site Status

UCLA Dept of Medicine - Hematology/Oncology, Santa Monica

Santa Monica, California, United States

Site Status

UCLA Health, Santa Monica

Santa Monica, California, United States

Site Status

Northside Hospital Inc.- GCS/Athens

Athens, Georgia, United States

Site Status

Atlanta Cancer Care - Atlanta

Atlanta, Georgia, United States

Site Status

Northside Hospital, Inc. - GCS/Northside

Atlanta, Georgia, United States

Site Status

Northside Hospital

Atlanta, Georgia, United States

Site Status

Northside Hospital,Inc.-GCS /Blairsville

Blairsville, Georgia, United States

Site Status

Northside Hospital, Inc. - GCS/Canton

Canton, Georgia, United States

Site Status

Atlanta Cancer Care - Cumming

Cumming, Georgia, United States

Site Status

Northside Hospital, Inc.-GCS/Stemmer

Decatur, Georgia, United States

Site Status

Suburban Hematology-Oncology Associates - Duluth

Duluth, Georgia, United States

Site Status

Atlanta Cancer Care - Lake Spivey

Jonesboro, Georgia, United States

Site Status

Suburban Hematology-Oncology Associates- Lawrenceville

Lawrenceville, Georgia, United States

Site Status

Northside Hospital, Inc. - GCS/Macon

Macon, Georgia, United States

Site Status

Northside Hospital, Inc. GCS/Kennestone

Marietta, Georgia, United States

Site Status

Oncology Hematology West, PC dba Nebraska Cancer Specialists

Omaha, Nebraska, United States

Site Status

The University of Texas MD Anderson Cancer Center

Houston, Texas, United States

Site Status

University of Utah, Huntsman Cancer Hospital

Salt Lake City, Utah, United States

Site Status

University of Utah, Huntsman Cancer Institute

Salt Lake City, Utah, United States

Site Status

Chris O'Brien Lifehouse

Camperdown, New South Wales, Australia

Site Status

Macquarie University

Macquarie Park, New South Wales, Australia

Site Status

Istituto Clinico Humanitas U. O. Oculistica

Milan, Lombardy, Italy

Site Status

Azienda Socio-Sanitaria Territoriale Monza

Monza, MB, Italy

Site Status

Fondazione IRCCS, Istituto Nazionale dei Tumori

Milan, MI, Italy

Site Status

Divisione di Cardiologia - Istituto Europeo di Oncologia Divisione di Medicina Nucleare

Milan, MI, Italy

Site Status

Istituto Europeo di Oncologia

Milan, MI, Italy

Site Status

LLC "Clinica UZI 4D"

Pyatigorsk, Stavropol Kray, Russia

Site Status

Private Healthcare Institution "Clinical hospital "RZD-Medicine" of Saint-Petersburg

Saint Petersburg, , Russia

Site Status

National Cancer Center

Goyang-si, Gyeonggi-do, South Korea

Site Status

Seoul National University Bundang Hospital

Seongnam-si, Gyeonggi-do, South Korea

Site Status

Gachon University Gil Medical Center

Incheon, , South Korea

Site Status

Seoul National University Hospital

Seoul, , South Korea

Site Status

Severance Hospital, Yonsei University Health System

Seoul, , South Korea

Site Status

Samsung Medical Center

Seoul, , South Korea

Site Status

Hospital Universitario Quirón Madrid

Pozuelo de Alarcón, Madrid, Spain

Site Status

Hospital Universitario Vall d'Hebron

Barcelona, , Spain

Site Status

Hospital Clinic de Barcelona

Barcelona, , Spain

Site Status

Hospital Universitario Fundación Jiménez Díaz

Madrid, , Spain

Site Status

Hospital Universitario HM Sanchinarro

Madrid, , Spain

Site Status

Countries

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United States Australia Italy Russia South Korea Spain

References

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Meric-Bernstam F, Calvo E, Lee KS, Moreno V, Park YH, Rha SY, Chalasani P, Zhong W, Zhou L, Pirie-Shepherd S, Leung ACF, Curigliano G. Safety and Tolerability of a Novel Anti-HER2 Antibody-Drug Conjugate (PF-06804103) in Patients with HER2-Expressing Solid Tumors: A Phase 1 Dose-Escalation Study. Mol Cancer Ther. 2023 Oct 2;22(10):1191-1203. doi: 10.1158/1535-7163.MCT-23-0101.

Reference Type DERIVED
PMID: 37420274 (View on PubMed)

Provided Documents

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Document Type: Study Protocol

View Document

Document Type: Statistical Analysis Plan

View Document

Related Links

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https://pmiform.com/clinical-trial-info-request?StudyID=C0541001

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Other Identifiers

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2017-002538-22

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

C0541001

Identifier Type: -

Identifier Source: org_study_id

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