Efficacy and Tolerability of the Nutraceutical Formulation Coleosoma in Dyslipidemic Subjects

NCT ID: NCT03027336

Last Updated: 2017-01-23

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE2

Total Enrollment

39 participants

Study Classification

INTERVENTIONAL

Study Start Date

2016-01-31

Study Completion Date

2016-10-31

Brief Summary

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The overall objective of the study is to assess the efficacy of Coleosoma formulation (fermented red rice, berberine and chitosan) in reducing non-HDL cholesterol in dyslipidemic patients.

Detailed Description

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The incidence of cardiovascular diseases related to atherosclerosis is the leading cause of death in industrialized countries and in many developing countries. It becomes, therefore, essential to implement preventive strategies with lifestyle changes in order to prevent / control the risk factors related to cardiovascular disease.

Dyslipidemia is characterized by qualitative and quantitative alterations of plasma lipids and lipoproteins. In subjects where it is not yet indicated a statin therapy, the guidelines recommend a lifestyle (diet and exercise) act to control cardiovascular risk factors.

The formulation Coleosoma is a supplement composed of fermented red rice, berberine and chitosan. Aim of the study is to evaluate the effectiveness of coleosoma formulation in reducing non-HDL cholesterol (Non-HDL-C), which provides a measure of the cholesterol content in all atherogenic particles.

This is a single-center, randomized (3:1) and controlled double-blind phase II study that involve dyslipidemic patients with non-HDL cholesterol levels ≥ 160 mg / dl.

The study included a maximum of 4 visits for all subjects enrolled. All eligible patients at V0 (screening) undergo baseline assessments (V1) and have been allocated according to the procedure of randomization to one of the study arms. Follow-up (FU) visits for all subjects was at 4 (V2) and at 12 weeks (V3) after randomization.

Laboratory and diagnostic:

At each visits patients undergo: anthropometric and hemodynamic assessment: weight and height for Body Mass Index (BMI) calculation, waist circumference, blood pressure, heart rate; blood collection for metabolic/hormonal profile: fasting plasma glucose, HbA1c, insulin, glucagon, active glucagon-like peptide-1 (GLP-1), total gastric inhibitory polypeptide (GIP), total cholesterol, HDL-cholesterol, triglycerides, aspartate aminotransferase (AST), alanine aminotransferase (ALT), creatinine, creatine phosphokinase (CPK), apolipoprotein (Apo) B, Apo A1, and inflammatory cytokines (IL-1, IL-6, IL-10, high-sensitivity C Reactive Protein (hsPCR), TNFalpha).

At V1 and V2 the Endothelial Progenitor Cells (EPC) number was evaluated with a cytofluorimetric assay.

Safety analysis has been conducted after 12 weeks treatment by determining ALT, CPK and estimated Glomerular filtration rate (eGFR) values.

This study has been sponsored by DOC generici s.r.l.

Conditions

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Dyslipidemias

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

The study included two arms: a treatment arm with dietary supplement (Coleosoma) and a placebo arm.

Coleosoma is the name of a new patented dietary supplement composed by Berberin 200 mg, Fermented Red Rice from Monascus purpureus 100 mg (correspondiing at 3 mg of monacolin K), Chitosan 100 mg e Q10 Coenzyme10 mg
Primary Study Purpose

TREATMENT

Blinding Strategy

QUADRUPLE

Participants Caregivers Investigators Outcome Assessors

Study Groups

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coleosoma

coleosoma 500mg tablet daily

Group Type EXPERIMENTAL

Coleosoma

Intervention Type DIETARY_SUPPLEMENT

patients will take one tablet of 500mg daily for 12 weeks. No dose titration is foreseen.

placebo

placebo tablets

Group Type PLACEBO_COMPARATOR

Placebo

Intervention Type DIETARY_SUPPLEMENT

patients will take one tablet daily for 12 weeks.

Interventions

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Coleosoma

patients will take one tablet of 500mg daily for 12 weeks. No dose titration is foreseen.

Intervention Type DIETARY_SUPPLEMENT

Placebo

patients will take one tablet daily for 12 weeks.

Intervention Type DIETARY_SUPPLEMENT

Other Intervention Names

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TegraDOC

Eligibility Criteria

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Inclusion Criteria

* non-HDL cholesterol ≥ 160 mg/dl;
* providing their written Informed Consent;
* capable of understanding the nature, purpose and study procedures

Exclusion Criteria

* diabetes (ADA criteria)
* reduced renal (GFR\<60 mL/min/1.73m2) or hepatic (transaminase levels \>2.5 folds the upper reference limit) function;
* present or past history of alcohol or drug abuse
* cerebro-vascular and neoplastic diseases in the 5 years prior to study visit
* use of drugs or food supplements interfering with cholesterol levels
* pregnancy or breastfeeding;
* monogenic dyslipidemia;
* participation in other clinical trials in the previous 30 days;
* uncompensated hypothyroidism
Minimum Eligible Age

18 Years

Maximum Eligible Age

75 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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DOC generici srl

UNKNOWN

Sponsor Role collaborator

Azienda Ospedaliero-Universitaria di Parma

OTHER

Sponsor Role lead

Responsible Party

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Alessandra Dei Cas

Research Assistant, MD, PhD

Responsibility Role PRINCIPAL_INVESTIGATOR

Principal Investigators

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Alessandra Dei Cas, MD

Role: PRINCIPAL_INVESTIGATOR

University of Parma

Locations

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Endocrinology Unit

Parma, Italy, Italy

Site Status

Countries

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Italy

References

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Reference Type BACKGROUND
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Reference Type BACKGROUND
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Dei Cas A, Spigoni V, Ardigo D, Pedrazzi G, Franzini L, Derlindati E, Urbani S, Monti L, Gnudi L, Zavaroni I. Reduced circulating endothelial progenitor cell number in healthy young adult hyperinsulinemic men. Nutr Metab Cardiovasc Dis. 2011 Jul;21(7):512-7. doi: 10.1016/j.numecd.2009.11.011. Epub 2010 Mar 15.

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Reference Type BACKGROUND
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Other Identifiers

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COLEOSOMA 29-06

Identifier Type: -

Identifier Source: org_study_id

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