Study to Evaluate Pharmacokinetic Drug Interactions and Safety of Clarithromycin, Amoxicillin and Ilaprazole

NCT ID: NCT02998437

Last Updated: 2017-01-26

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

28 participants

Study Classification

INTERVENTIONAL

Study Start Date

2016-12-31

Study Completion Date

2017-01-31

Brief Summary

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This study evaluate the pharmacokinetic drug interaction in Ilaprazole, Clarithromycin, Amoxicillin.

Detailed Description

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This study evaluate the pharmacokinetic drug interaction and safety in Ilaprazole, Clarithromycin, Amoxicillin.

Conditions

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Drug Interaction Potentiation

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Ilaprazole 10mg

Period 1: Ilaprazole 10mg 1 tab.m one a day

Period 2: Clarithromycin 500mg 1 tab. + Amoxicillin 500mg 2 cap. twice a day, 6 days Ilaprazole 10mg, one a day at the 5 day

Group Type EXPERIMENTAL

Ilaprazole 10mg

Intervention Type DRUG

Period 1: Ilaprazole 10mg, one a day, one day Period 2: Ilaprazole 10mg, twice a day, 6 days

Clarithromycin 500mg

Period 1: Clarithromycin 500mg 1 tab. + Amoxicillin 500mg 2 cap., one a day

Period 2: Ilaprazole 10mg 1 tab., twice a day, 6 days Clarithromycin 500mg 1 tab. + Amoxicillin 500mg 2 cap., one a day at the 5 day

Group Type ACTIVE_COMPARATOR

Clarithromycin 500mg

Intervention Type DRUG

Period 1: Clarithromycin 500mg 1 tab., twice a day, one day Period 2: Clarithromycin 500mg 1 tab., one a day at 5 day

Amoxicillin 500mg

Period 1: Clarithromycin 500mg 1 tab. + Amoxicillin 500mg 2 cap., one a day

Period 2: Ilaprazole 10mg 1 tab., twice a day, 6 days Clarithromycin 500mg 1 tab. + Amoxicillin 500mg 2 cap., one a day at 5 day

Group Type ACTIVE_COMPARATOR

Amoxicillin 500 Mg

Intervention Type DRUG

Period 1: Amoxicillin 500mg 2 cap., one a day, one day Period 2: Amoxicillin 500mg 2 cap., one a day at 5 day

Interventions

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Ilaprazole 10mg

Period 1: Ilaprazole 10mg, one a day, one day Period 2: Ilaprazole 10mg, twice a day, 6 days

Intervention Type DRUG

Clarithromycin 500mg

Period 1: Clarithromycin 500mg 1 tab., twice a day, one day Period 2: Clarithromycin 500mg 1 tab., one a day at 5 day

Intervention Type DRUG

Amoxicillin 500 Mg

Period 1: Amoxicillin 500mg 2 cap., one a day, one day Period 2: Amoxicillin 500mg 2 cap., one a day at 5 day

Intervention Type DRUG

Other Intervention Names

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Noltec(the brand name) Klaricid 500mg(the brand name) Amoxicillin Cap. 500mg Chongkundang(the brand name)

Eligibility Criteria

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Inclusion Criteria

1. Healthy male adults aged ≥19 years and \<50 years at screening
2. Body mass index ≥18.5 and \<25

* Body mass index (kg/m2) = body weight (kg)/\[height (m)\]2
3. Men who have sexual relationship with women of child bearing potential must give consent to using contraceptive measures (condoms, spermicide, and menstrual cycle control) and avoiding sperm donation during the study and up to 28 days following the last dose of IMP (these contraceptive measures are not required if the male subject or female partner is infertile).
4. Those who voluntarily decided to participate in this study and gave written consent to comply with the requirements after receiving sufficient explanation and fully understanding this study.

Exclusion Criteria

1. Hypersensitivity or history of clinically significant hypersensitivity to active ingredients or excipients (in particular, Yellow No. 4 (Tartrazine); Yellow No. 5 (Sunset Yellow FCF); macrolide antibiotics such as Clarithromycin and erythromycin; or Penicillins)
2. History of QT prolongation or ventricular arrhythmia (including Torsadedes de pointes)
3. Clinically significant, current or past disorder of hepatobiliary (severe hepatic impairment, etc.), renal (severe renal impairment, etc.), nervous, immune, respiratory, endocrine, blood•tumor, cardiovascular (heart failure, etc.), or psychiatric system
4. History of gastrointestinal disorder (Crohn's disease, ulcer, etc.) or operation (excluding simple appendectomy or herniotomy) that may affect drug absorption
5. Administration of other IMP from other study (including biological comparability test) within 3 months of the first dose of IMP.
6. Whole blood donation within 60 days, or apheresis donation within 30 days before the first dose of IMP.
7. Constant caffeine intake (\> 5 cups of coffee/day, \> 1250 cc of tea/day, \> 1250 cc of cola/day), constant smoking (more than 10 cigarettes/day) or constant alcohol drinking (more than 210 g/week) or inability to refrain from alcohol consumption from 2 days before the first dose of IMP until the end of PK assessment.
8. Consumption of grapefruit-containing food within 7 days before the first dose of IMP
9. History of drug abuse within 1 year before screening, or positive response in urine drug misuse/abuse screening test
10. Use of medicinal products that are expected to or may affect the metabolism of IMP; St. John's wort; or relevant preparations within 30 days of IMP administration
11. Use of following medicinal products within given time period excluding local preparations, which do not have significant systemic absorption, and hormonal contraceptives

* Prescription drug within 14 days of the first dose of IMP
* OTC including health supplements and vitamins within 7 days of the first dose of IMP
* Medicinal products via depot injection or other implantations within 30 days of the first dose of IMP (excluding contraceptives)
* Drug metabolizing enzyme inducer or inhibitor such as barbiturate within 30 days before the first dose of IMP
12. Stable vital sign measured in sitting position at screening: systolic blood pressure \> 150 mmHg or \< 90 mmHg, diastolic blood pressure \> 100 mmHg or \< 50 mmHg, pulse rate \> 110 bpm or \<40 bpm
13. Following findings at screening

* Blood total bilirubin \> 1.5 x upper limit of normal
* Blood AST (SGOT), ALT (SGPT) \> 1.25 x upper limit of normal
* MDRD-estimated eGFR \< 60 mL/min/1.73m2 eGFR (estimated glomerular filtration rate)(mL/min/1.73m2) = 175 x \[serum creatinine (mg/dL)\]-1.154 x \[age (years)\]-0.203
* Positive serum test (hepatitis B, hepatitis C, HIV, syphilis)
14. Those considered ineligible by the investigator due to other screening results or reasons.
Minimum Eligible Age

19 Years

Maximum Eligible Age

50 Years

Eligible Sex

MALE

Accepts Healthy Volunteers

Yes

Sponsors

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Severance Hospital

OTHER

Sponsor Role collaborator

Il-Yang Pharm. Co., Ltd.

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Min MS Park, PhD

Role: PRINCIPAL_INVESTIGATOR

Severance Hospital

Locations

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Severance Hospital

Seoul, , South Korea

Site Status

Countries

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South Korea

References

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Jin BH, Yoo BW, Park J, Kim JH, Lee JY, Shin JS, Park MS. Pharmacokinetic drug interaction and safety after coadministration of clarithromycin, amoxicillin, and ilaprazole: a randomised, open-label, one-way crossover, two parallel sequences study. Eur J Clin Pharmacol. 2018 Sep;74(9):1149-1157. doi: 10.1007/s00228-018-2489-2. Epub 2018 May 30.

Reference Type DERIVED
PMID: 29846770 (View on PubMed)

Other Identifiers

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IY81149-DI03

Identifier Type: -

Identifier Source: org_study_id

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