Pharmacokinetics and Pharmacodynamics of Cilofexor in Adults With Normal and Impaired Hepatic Function

NCT ID: NCT02808312

Last Updated: 2021-01-07

Study Results

Results available

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

57 participants

Study Classification

INTERVENTIONAL

Study Start Date

2016-07-13

Study Completion Date

2018-10-16

Brief Summary

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The primary objective of this study is to evaluate the single-dose pharmacokinetics of cilofexor in adults with impaired hepatic function relative to matched, healthy controls with normal hepatic function.

Detailed Description

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Conditions

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Nonalcoholic Steatohepatitis (NASH) Primary Sclerosing Cholangitis (PSC)

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Cohort 1: Mild Hepatic Impairment

Participants with mild hepatic impairment will receive a single oral dose of cilofexor 30 mg (3 x 10 mg tablets).

Group Type EXPERIMENTAL

Cilofexor

Intervention Type DRUG

Tablet(s) administered orally in a fed state on Day 1

Cohort 1: Normal Hepatic Function

Matched normal hepatic function participants to mild hepatic impairment participants will receive a single oral dose of cilofexor 30 mg (3 x 10 mg tablets).

Group Type EXPERIMENTAL

Cilofexor

Intervention Type DRUG

Tablet(s) administered orally in a fed state on Day 1

Cohort 2: Moderate Hepatic Impairment

Participants with moderate hepatic impairment will receive a single oral dose of cilofexor 30 mg (3 x 10 mg tablets).

Group Type EXPERIMENTAL

Cilofexor

Intervention Type DRUG

Tablet(s) administered orally in a fed state on Day 1

Cohort 2: Normal Hepatic Function

Matched normal hepatic function participants to moderate hepatic impairment participants will receive a single oral dose of cilofexor 30 mg (3 x 10 mg tablets).

Group Type EXPERIMENTAL

Cilofexor

Intervention Type DRUG

Tablet(s) administered orally in a fed state on Day 1

Cohort 3: Severe Hepatic Impairment

Participants with severe hepatic impairment will receive a single oral dose of cilofexor 10 mg (1 x 10 mg tablet).

Group Type EXPERIMENTAL

Cilofexor

Intervention Type DRUG

Tablet(s) administered orally in a fed state on Day 1

Cohort 3: Normal Hepatic Function

Matched normal hepatic function participants to severe hepatic impairment participants will receive a single oral dose of cilofexor 10 mg (1 x 10 mg tablet).

Group Type EXPERIMENTAL

Cilofexor

Intervention Type DRUG

Tablet(s) administered orally in a fed state on Day 1

Interventions

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Cilofexor

Tablet(s) administered orally in a fed state on Day 1

Intervention Type DRUG

Other Intervention Names

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GS-9674

Eligibility Criteria

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Inclusion Criteria

Cohort 1:

* Individuals with mildly impaired and normal hepatic function.
* Individuals with mild hepatic impairment must have a score of 5-6 on the Child-Pugh-Turcotte (CPT) classification at screening without evidence of worsening clinical and/or laboratory signs of hepatic impairment within 2 months prior or within the screening period.

Cohort 2:

* Individuals with moderately impaired and normal hepatic function.
* Individuals with moderate hepatic impairment must have a score of 7-9 on the CPT classification at screening without evidence of worsening clinical and/or laboratory signs of hepatic impairment within 2 months prior or within the screening period.

Cohort 3:

* Individuals with severely impaired and normal hepatic function.
* Individuals with severe hepatic impairment must have a score of 10-15 on the CPT classification at screening without evidence of worsening clinical and/or laboratory signs of hepatic impairment within 2 months prior or within the screening period.
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

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Gilead Sciences

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Gilead Study Director

Role: STUDY_DIRECTOR

Gilead Sciences

Locations

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Miami, Florida, United States

Site Status

Orlando, Florida, United States

Site Status

Knoxville, Tennessee, United States

Site Status

San Antonio, Texas, United States

Site Status

Auckland, , New Zealand

Site Status

Countries

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United States New Zealand

Provided Documents

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Document Type: Study Protocol

View Document

Document Type: Statistical Analysis Plan

View Document

Other Identifiers

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GS-US-402-3885

Identifier Type: -

Identifier Source: org_study_id

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