Trial Outcomes & Findings for Lubiprostone for Treatment of Chronic Idiopathic Constipation (NCT NCT02695719)

NCT ID: NCT02695719

Last Updated: 2018-12-31

Results Overview

A SBM was defined as any bowel movement (BM) that does not occur within 24 hours after rescue medication use (laxative, suppository, or enema). Participants will be given a diary to complete at home where they will record all details of each SBM including the consistency of the stool and the difficulty they have in passing it.

Recruitment status

COMPLETED

Study phase

PHASE3

Target enrollment

156 participants

Primary outcome timeframe

Week 1

Results posted on

2018-12-31

Participant Flow

Participants took part in the study at 13 investigative sites in Korea from 14 April 2016 to 24 February 2017.

Participants with a diagnosis of chronic idiopathic constipation as determined by the Rome III Diagnostic Criteria for Functional Constipation were enrolled in 1:1 ratio to receive lubiprostone or placebo.

Participant milestones

Participant milestones
Measure
Placebo
Lubiprostone placebo-matching capsules, orally, twice daily, under fed conditions, for up to 4 weeks
Lubiprostone 24 μg
Lubiprostone 24 μg, capsules, orally, twice daily, under fed conditions, for up to 4 weeks
Overall Study
STARTED
74
82
Overall Study
COMPLETED
71
72
Overall Study
NOT COMPLETED
3
10

Reasons for withdrawal

Reasons for withdrawal
Measure
Placebo
Lubiprostone placebo-matching capsules, orally, twice daily, under fed conditions, for up to 4 weeks
Lubiprostone 24 μg
Lubiprostone 24 μg, capsules, orally, twice daily, under fed conditions, for up to 4 weeks
Overall Study
Pretreatment Event/Adverse Event
2
9
Overall Study
Significant Protocol Deviation
0
1
Overall Study
Voluntary Withdrawal
1
0

Baseline Characteristics

Lubiprostone for Treatment of Chronic Idiopathic Constipation

Baseline characteristics by cohort

Baseline characteristics by cohort
Measure
Placebo
n=74 Participants
Lubiprostone placebo-matching capsules, orally, twice daily, under fed conditions, for up to 4 weeks
Lubiprostone 24 μg
n=82 Participants
Lubiprostone 24 μg, capsules, orally, twice daily, under fed conditions, for up to 4 weeks
Total
n=156 Participants
Total of all reporting groups
Age, Continuous
43.9 years
FULL_RANGE 15.95 • n=5 Participants
44.6 years
FULL_RANGE 16.88 • n=7 Participants
44.3 years
n=5 Participants
Sex: Female, Male
Female
59 Participants
n=5 Participants
66 Participants
n=7 Participants
125 Participants
n=5 Participants
Sex: Female, Male
Male
15 Participants
n=5 Participants
16 Participants
n=7 Participants
31 Participants
n=5 Participants
Race/Ethnicity, Customized
Asian
74 participants
n=5 Participants
82 participants
n=7 Participants
156 participants
n=5 Participants
Region of Enrollment
Korea, Republic Of
74 participants
n=5 Participants
82 participants
n=7 Participants
156 participants
n=5 Participants
Height
163.4 cm
STANDARD_DEVIATION 6.65 • n=5 Participants
162.2 cm
STANDARD_DEVIATION 7.83 • n=7 Participants
162.7 cm
STANDARD_DEVIATION 7.30 • n=5 Participants
Weight
60.32 kg
STANDARD_DEVIATION 9.434 • n=5 Participants
59.78 kg
STANDARD_DEVIATION 11.218 • n=7 Participants
60.05 kg
STANDARD_DEVIATION 10.380 • n=5 Participants
Body Mass Index (BMI)
22.531 (kg/m^2)
STANDARD_DEVIATION 2.5836 • n=5 Participants
22.623 (kg/m^2)
STANDARD_DEVIATION 3.1104 • n=7 Participants
22.579 (kg/m^2)
STANDARD_DEVIATION 2.8638 • n=5 Participants
Smokers
Participant has never smoked
64 participants
n=5 Participants
73 participants
n=7 Participants
137 participants
n=5 Participants
Smokers
participant is a current smoker
4 participants
n=5 Participants
3 participants
n=7 Participants
7 participants
n=5 Participants
Smokers
Participant is an ex-smoker
6 participants
n=5 Participants
6 participants
n=7 Participants
12 participants
n=5 Participants

PRIMARY outcome

Timeframe: Week 1

Population: FAS included all participants who were randomized to receive study treatment whether or not they received treatment. Missing values were imputed by last observation carried forward (LOCF) method.

A SBM was defined as any bowel movement (BM) that does not occur within 24 hours after rescue medication use (laxative, suppository, or enema). Participants will be given a diary to complete at home where they will record all details of each SBM including the consistency of the stool and the difficulty they have in passing it.

Outcome measures

Outcome measures
Measure
Placebo
n=74 Participants
Lubiprostone placebo-matching capsules, orally, twice daily, under fed conditions, for up to 4 weeks
Lubiprostone 24 μg
n=82 Participants
Lubiprostone 24 μg, capsules, orally, twice daily, under fed conditions, for up to 4 weeks
Spontaneous Bowel Movement (SBM) Frequency at Week 1
3.1 SBMs/week
Standard Deviation 1.75
4.4 SBMs/week
Standard Deviation 2.65

SECONDARY outcome

Timeframe: Weeks 2, 3 and 4

Population: FAS included all participants who were randomized to receive study treatment whether or not they received treatment. Missing values were imputed by LOCF method.

A SBM was defined as any BM that does not occur within 24 hours after rescue medication use. Participants will be given a diary to complete at home where they will record all details of each SBM including the consistency of the stool and the difficulty they have in passing it.

Outcome measures

Outcome measures
Measure
Placebo
n=74 Participants
Lubiprostone placebo-matching capsules, orally, twice daily, under fed conditions, for up to 4 weeks
Lubiprostone 24 μg
n=82 Participants
Lubiprostone 24 μg, capsules, orally, twice daily, under fed conditions, for up to 4 weeks
SBM Frequency at Weeks 2, 3 and 4
Week 2
3.2 SBMs/week
Standard Deviation 1.80
4.2 SBMs/week
Standard Deviation 2.39
SBM Frequency at Weeks 2, 3 and 4
Week 3
3.4 SBMs/week
Standard Deviation 1.98
4.1 SBMs/week
Standard Deviation 2.42
SBM Frequency at Weeks 2, 3 and 4
Week 4
3.2 SBMs/week
Standard Deviation 1.75
4.0 SBMs/week
Standard Deviation 2.31

SECONDARY outcome

Timeframe: Up to 24 hours after the first dose of study medication

Population: FAS included all participants who were randomized to receive study treatment whether or not they received treatment. Here, number of participants analyzed is the participants who were evaluated for this outcome measure.

A SBM was defined as any BM that does not occur within 24 hours after rescue medication use. Percentage of participants who have an SBM within 24 hours after the first dose will be assessed and derived from the data on SBMs collected in the participant diary.

Outcome measures

Outcome measures
Measure
Placebo
n=74 Participants
Lubiprostone placebo-matching capsules, orally, twice daily, under fed conditions, for up to 4 weeks
Lubiprostone 24 μg
n=81 Participants
Lubiprostone 24 μg, capsules, orally, twice daily, under fed conditions, for up to 4 weeks
Percentage of Participants Who Had a SBM Within 24 Hours After the First Dose of Study Medication
35.1 percentage of participants
56.8 percentage of participants

SECONDARY outcome

Timeframe: Weeks 1, 2, 3 and 4

Population: FAS included all participants who were randomized to receive study treatment whether or not they received treatment. Missing values were imputed by LOCF method.

For each participant, the mean degree of straining was averaged for all SBMs in a given week. The degree of straining for each SBM was collected in the participant diary. The degree of straining is scored on a 5-point scale where: 0=No straining, 1=Mild straining, 2=Moderate straining, 3=Strong straining or 4=Very strong straining with higher scores indicating more severe straining.

Outcome measures

Outcome measures
Measure
Placebo
n=74 Participants
Lubiprostone placebo-matching capsules, orally, twice daily, under fed conditions, for up to 4 weeks
Lubiprostone 24 μg
n=82 Participants
Lubiprostone 24 μg, capsules, orally, twice daily, under fed conditions, for up to 4 weeks
Mean Degree of Straining Score
Week 4
2.1 scores on a scale
Standard Deviation 0.88
1.9 scores on a scale
Standard Deviation 1.03
Mean Degree of Straining Score
Week 1
2.3 scores on a scale
Standard Deviation 0.93
2.0 scores on a scale
Standard Deviation 1.01
Mean Degree of Straining Score
Week 2
2.2 scores on a scale
Standard Deviation 0.92
2.0 scores on a scale
Standard Deviation 1.02
Mean Degree of Straining Score
Week 3
2.1 scores on a scale
Standard Deviation 0.87
2.0 scores on a scale
Standard Deviation 1.04

SECONDARY outcome

Timeframe: Weeks 1, 2, 3 and 4

Population: FAS included all participants who were randomized to receive study treatment whether or not they received treatment. Missing values were imputed by LOCF method.

For each participant, the mean stool consistency score was averaged for all SBMs in a given week. The mean degree of stool consistency for each SBM was collected in the participant diary based on the Bristol Stool Chart. The Bristol Stool Chart is a visual medical aid designed to classify the form of human feces into seven categories where: 1=Hard and round (difficult-to-pass), 2=Sausage-shaped but hard stool, 3=Sausage-shaped stool with cracks on the surface, 4=Sausage-shaped, soft stool with smooth surface, or coiled stool, 5=Soft, half-solid (and easy-to-pass) stool with clear crease, 6=Unshaped, loose stool with small, irregular-shaped pieces, or mushy stool or 7=Watery stool without solid pieces (entirely liquid).

Outcome measures

Outcome measures
Measure
Placebo
n=74 Participants
Lubiprostone placebo-matching capsules, orally, twice daily, under fed conditions, for up to 4 weeks
Lubiprostone 24 μg
n=82 Participants
Lubiprostone 24 μg, capsules, orally, twice daily, under fed conditions, for up to 4 weeks
Mean Degree Stool Consistency Score
Week 1
3.2 scores on a scale
Standard Deviation 1.04
4.2 scores on a scale
Standard Deviation 1.38
Mean Degree Stool Consistency Score
Week 2
3.3 scores on a scale
Standard Deviation 1.19
4.3 scores on a scale
Standard Deviation 1.27
Mean Degree Stool Consistency Score
Week 3
3.3 scores on a scale
Standard Deviation 1.04
4.1 scores on a scale
Standard Deviation 1.21
Mean Degree Stool Consistency Score
Week 4
3.3 scores on a scale
Standard Deviation 1.08
4.1 scores on a scale
Standard Deviation 1.22

SECONDARY outcome

Timeframe: Weeks 1, 2, 3 and 4

Population: FAS included all participants who were randomized to receive study treatment whether or not they received treatment. Missing values were imputed by LOCF method.

The abdominal symptoms (bloating and discomfort upon waking in the morning) were scored weekly on a 5-point scale, where: 0=None, 1=Mild, 2=Moderate, 3=Severe or 4=Very severe, with a higher score indicating more severe symptoms. Assessment of weekly abdominal symptoms were recorded by the participant in the diary.

Outcome measures

Outcome measures
Measure
Placebo
n=74 Participants
Lubiprostone placebo-matching capsules, orally, twice daily, under fed conditions, for up to 4 weeks
Lubiprostone 24 μg
n=82 Participants
Lubiprostone 24 μg, capsules, orally, twice daily, under fed conditions, for up to 4 weeks
Weekly Abdominal Symptoms Score
Abdominal Bloating, Week 1
1.9 scores on a sclae
Standard Deviation 1.03
1.7 scores on a sclae
Standard Deviation 0.93
Weekly Abdominal Symptoms Score
Abdominal Bloating, Week 2
1.8 scores on a sclae
Standard Deviation 0.96
1.5 scores on a sclae
Standard Deviation 1.00
Weekly Abdominal Symptoms Score
Abdominal Bloating, Week 3
1.7 scores on a sclae
Standard Deviation 0.90
1.5 scores on a sclae
Standard Deviation 1.05
Weekly Abdominal Symptoms Score
Abdominal Bloating, Week 4
1.6 scores on a sclae
Standard Deviation 1.05
1.4 scores on a sclae
Standard Deviation 0.98
Weekly Abdominal Symptoms Score
Abdominal Discomfort, Week 1
1.9 scores on a sclae
Standard Deviation 1.13
1.5 scores on a sclae
Standard Deviation 1.01
Weekly Abdominal Symptoms Score
Abdominal Discomfort, Week 2
1.7 scores on a sclae
Standard Deviation 1.04
1.5 scores on a sclae
Standard Deviation 1.02
Weekly Abdominal Symptoms Score
Abdominal Discomfort, Week 3
1.6 scores on a sclae
Standard Deviation 1.03
1.4 scores on a sclae
Standard Deviation 1.07
Weekly Abdominal Symptoms Score
Abdominal Discomfort, Week 4
1.5 scores on a sclae
Standard Deviation 1.09
1.4 scores on a sclae
Standard Deviation 1.09

SECONDARY outcome

Timeframe: Weeks 1, 2, 3 and 4

Population: FAS included all participants who were randomized to receive study treatment whether or not they received treatment. Missing values were imputed by LOCF method.

The responder rate was assessed each week and was derived from the data on SBMs collected in the diary. A non-responder was defined as any participant with a spontaneous BM frequency rate of less than 3 for a given week, any participant who dropped out during or before the given week due to lack of efficacy, or any participant who used rescue medication during or within 24 hours before the given week. Otherwise, the participant subject was considered a responder. A responder with a spontaneous BM frequency rate ≥3 but \<4 was considered a moderate responder. Otherwise, the participant was a full responder (≥4 SBM).

Outcome measures

Outcome measures
Measure
Placebo
n=74 Participants
Lubiprostone placebo-matching capsules, orally, twice daily, under fed conditions, for up to 4 weeks
Lubiprostone 24 μg
n=82 Participants
Lubiprostone 24 μg, capsules, orally, twice daily, under fed conditions, for up to 4 weeks
Weekly Responder Rate
Moderate Responders, Week 1
27.0 percentage of participants
18.3 percentage of participants
Weekly Responder Rate
Moderate Responders, Week 2
24.3 percentage of participants
23.2 percentage of participants
Weekly Responder Rate
Moderate Responders, Week 3
24.3 percentage of participants
24.4 percentage of participants
Weekly Responder Rate
Moderate Responders, Week 4
20.3 percentage of participants
24.4 percentage of participants
Weekly Responder Rate
Full Responders, Week 1
31.1 percentage of participants
56.1 percentage of participants
Weekly Responder Rate
Full Responders, Week 2
32.4 percentage of participants
58.5 percentage of participants
Weekly Responder Rate
Full Responders, Week 3
37.8 percentage of participants
52.4 percentage of participants
Weekly Responder Rate
Full Responders, Week 4
35.1 percentage of participants
50.0 percentage of participants

Adverse Events

Placebo

Serious events: 0 serious events
Other events: 8 other events
Deaths: 0 deaths

Lubiprostone 24 μg

Serious events: 0 serious events
Other events: 28 other events
Deaths: 0 deaths

Serious adverse events

Adverse event data not reported

Other adverse events

Other adverse events
Measure
Placebo
n=74 participants at risk
Lubiprostone placebo-matching capsules, orally, twice daily, under fed conditions, for up to 4 weeks
Lubiprostone 24 μg
n=81 participants at risk
Lubiprostone 24 μg, capsules, orally, twice daily, under fed conditions, for up to 4 weeks
Gastrointestinal disorders
Nausea
4.1%
3/74 • Baseline and up to Week 6
At each visit the investigator had to document any occurrence of adverse events and abnormal laboratory findings. Any event spontaneously reported by the participant or observed by the investigator was recorded, irrespective of the relation to study treatment.
23.5%
19/81 • Baseline and up to Week 6
At each visit the investigator had to document any occurrence of adverse events and abnormal laboratory findings. Any event spontaneously reported by the participant or observed by the investigator was recorded, irrespective of the relation to study treatment.
Gastrointestinal disorders
Dyspepsia
6.8%
5/74 • Baseline and up to Week 6
At each visit the investigator had to document any occurrence of adverse events and abnormal laboratory findings. Any event spontaneously reported by the participant or observed by the investigator was recorded, irrespective of the relation to study treatment.
7.4%
6/81 • Baseline and up to Week 6
At each visit the investigator had to document any occurrence of adverse events and abnormal laboratory findings. Any event spontaneously reported by the participant or observed by the investigator was recorded, irrespective of the relation to study treatment.
Gastrointestinal disorders
Diarrhoea
2.7%
2/74 • Baseline and up to Week 6
At each visit the investigator had to document any occurrence of adverse events and abnormal laboratory findings. Any event spontaneously reported by the participant or observed by the investigator was recorded, irrespective of the relation to study treatment.
6.2%
5/81 • Baseline and up to Week 6
At each visit the investigator had to document any occurrence of adverse events and abnormal laboratory findings. Any event spontaneously reported by the participant or observed by the investigator was recorded, irrespective of the relation to study treatment.
Nervous system disorders
Headache
0.00%
0/74 • Baseline and up to Week 6
At each visit the investigator had to document any occurrence of adverse events and abnormal laboratory findings. Any event spontaneously reported by the participant or observed by the investigator was recorded, irrespective of the relation to study treatment.
6.2%
5/81 • Baseline and up to Week 6
At each visit the investigator had to document any occurrence of adverse events and abnormal laboratory findings. Any event spontaneously reported by the participant or observed by the investigator was recorded, irrespective of the relation to study treatment.

Additional Information

Medical Director

Takeda

Phone: +1-877-825-3327

Results disclosure agreements

  • Principal investigator is a sponsor employee The first study related publication will be a multi-center publication submitted within 24 months after conclusion or termination of a study at all sites. After such multi site publication, all proposed site publications and presentations will be submitted to sponsor for review 60 days in advance of publication. Site will remove Sponsor confidential information unrelated to study results. Sponsor can delay a proposed publication for another 60 days to preserve intellectual property.
  • Publication restrictions are in place

Restriction type: OTHER