Trial Outcomes & Findings for Use of F-652 in Patients With Alcoholic Hepatitis (NCT NCT02655510)

NCT ID: NCT02655510

Last Updated: 2019-09-09

Results Overview

The count of subjects who experience serious adverse events

Recruitment status

COMPLETED

Study phase

PHASE1/PHASE2

Target enrollment

18 participants

Primary outcome timeframe

From day 1 up to 42 days following administration of last dose of study drug

Results posted on

2019-09-09

Participant Flow

Participant milestones

Participant milestones
Measure
Period 1: F-652 10 μg/kg
Participants will receive 10 μg/kg of F-652 on Day 1 and Day 7 via slow intravenous infusion.
Period 2: F-652 30 μg/kg
Participants will receive 30 μg/kg of F-652 on Day 1 and Day 7 via slow intravenous infusion.
Period 3: F-652 45 μg/kg
Participants will receive 45 μg/kg of F-652 on Day 1 and Day 7 via slow intravenous infusion.
Overall Study
STARTED
6
6
6
Overall Study
COMPLETED
6
6
6
Overall Study
NOT COMPLETED
0
0
0

Reasons for withdrawal

Withdrawal data not reported

Baseline Characteristics

The six participants in each period were further defined by MELD grouping, where three participants had a MELD score of 11-20 and three participants had a MELD score of 21-28; resulting in a total of six participants in each period, a total of 18 subjects overall.

Baseline characteristics by cohort

Baseline characteristics by cohort
Measure
Period 1: F-652 10 μg/kg
n=6 Participants
Participants will receive 10 μg/kg of F-652 on Day 1 and Day 7 via slow intravenous infusion.
Period 2: F-652 30 μg/kg
n=6 Participants
Participants will receive 30 μg/kg of F-652 on Day 1 and Day 7 via slow intravenous infusion
Period 3: F-652 45 μg/kg
n=6 Participants
Participants will receive 45 μg/kg of F-652 on Day 1 and Day 7 via slow intravenous infusion.
Total
n=18 Participants
Total of all reporting groups
Age, Continuous
46.8 years
STANDARD_DEVIATION 6.9 • n=6 Participants
50.5 years
STANDARD_DEVIATION 12.0 • n=6 Participants
50.3 years
STANDARD_DEVIATION 11.3 • n=6 Participants
49.1 years
STANDARD_DEVIATION 9.8 • n=18 Participants
Sex: Female, Male
Female
2 Participants
n=6 Participants
2 Participants
n=6 Participants
2 Participants
n=6 Participants
6 Participants
n=18 Participants
Sex: Female, Male
Male
4 Participants
n=6 Participants
4 Participants
n=6 Participants
4 Participants
n=6 Participants
12 Participants
n=18 Participants
Race (NIH/OMB)
American Indian or Alaska Native
1 Participants
n=6 Participants
0 Participants
n=6 Participants
0 Participants
n=6 Participants
1 Participants
n=18 Participants
Race (NIH/OMB)
Asian
0 Participants
n=6 Participants
0 Participants
n=6 Participants
0 Participants
n=6 Participants
0 Participants
n=18 Participants
Race (NIH/OMB)
Native Hawaiian or Other Pacific Islander
0 Participants
n=6 Participants
0 Participants
n=6 Participants
0 Participants
n=6 Participants
0 Participants
n=18 Participants
Race (NIH/OMB)
Black or African American
0 Participants
n=6 Participants
0 Participants
n=6 Participants
0 Participants
n=6 Participants
0 Participants
n=18 Participants
Race (NIH/OMB)
White
5 Participants
n=6 Participants
6 Participants
n=6 Participants
6 Participants
n=6 Participants
17 Participants
n=18 Participants
Race (NIH/OMB)
More than one race
0 Participants
n=6 Participants
0 Participants
n=6 Participants
0 Participants
n=6 Participants
0 Participants
n=18 Participants
Race (NIH/OMB)
Unknown or Not Reported
0 Participants
n=6 Participants
0 Participants
n=6 Participants
0 Participants
n=6 Participants
0 Participants
n=18 Participants
Region of Enrollment
United States
6 participants
n=6 Participants
6 participants
n=6 Participants
6 participants
n=6 Participants
18 participants
n=18 Participants
Alcohol Consumption by MELD grouping
MELD 11-20
143.3 grams per day
STANDARD_DEVIATION 75.0 • n=3 Participants • The six participants in each period were further defined by MELD grouping, where three participants had a MELD score of 11-20 and three participants had a MELD score of 21-28; resulting in a total of six participants in each period, a total of 18 subjects overall.
151.3 grams per day
STANDARD_DEVIATION 28.8 • n=3 Participants • The six participants in each period were further defined by MELD grouping, where three participants had a MELD score of 11-20 and three participants had a MELD score of 21-28; resulting in a total of six participants in each period, a total of 18 subjects overall.
186.6 grams per day
STANDARD_DEVIATION 88.9 • n=3 Participants • The six participants in each period were further defined by MELD grouping, where three participants had a MELD score of 11-20 and three participants had a MELD score of 21-28; resulting in a total of six participants in each period, a total of 18 subjects overall.
160.4 grams per day
STANDARD_DEVIATION 63.1 • n=9 Participants • The six participants in each period were further defined by MELD grouping, where three participants had a MELD score of 11-20 and three participants had a MELD score of 21-28; resulting in a total of six participants in each period, a total of 18 subjects overall.
Alcohol Consumption by MELD grouping
MELD 21-28
181.3 grams per day
STANDARD_DEVIATION 140.0 • n=3 Participants • The six participants in each period were further defined by MELD grouping, where three participants had a MELD score of 11-20 and three participants had a MELD score of 21-28; resulting in a total of six participants in each period, a total of 18 subjects overall.
212.6 grams per day
STANDARD_DEVIATION 141.7 • n=3 Participants • The six participants in each period were further defined by MELD grouping, where three participants had a MELD score of 11-20 and three participants had a MELD score of 21-28; resulting in a total of six participants in each period, a total of 18 subjects overall.
57.3 grams per day
STANDARD_DEVIATION 28.0 • n=3 Participants • The six participants in each period were further defined by MELD grouping, where three participants had a MELD score of 11-20 and three participants had a MELD score of 21-28; resulting in a total of six participants in each period, a total of 18 subjects overall.
150.4 grams per day
STANDARD_DEVIATION 123.2 • n=9 Participants • The six participants in each period were further defined by MELD grouping, where three participants had a MELD score of 11-20 and three participants had a MELD score of 21-28; resulting in a total of six participants in each period, a total of 18 subjects overall.
Hospitalized at screening by MELD grouping
MELD 11-20
3 Participants
n=3 Participants • The six participants in each period were further defined by MELD grouping, where three participants had a MELD score of 11-20 and three participants had a MELD score of 21-28; resulting in a total of six participants in each period, a total of 18 subjects overall.
3 Participants
n=3 Participants • The six participants in each period were further defined by MELD grouping, where three participants had a MELD score of 11-20 and three participants had a MELD score of 21-28; resulting in a total of six participants in each period, a total of 18 subjects overall.
2 Participants
n=3 Participants • The six participants in each period were further defined by MELD grouping, where three participants had a MELD score of 11-20 and three participants had a MELD score of 21-28; resulting in a total of six participants in each period, a total of 18 subjects overall.
8 Participants
n=9 Participants • The six participants in each period were further defined by MELD grouping, where three participants had a MELD score of 11-20 and three participants had a MELD score of 21-28; resulting in a total of six participants in each period, a total of 18 subjects overall.
Hospitalized at screening by MELD grouping
MELD 21-28
1 Participants
n=3 Participants • The six participants in each period were further defined by MELD grouping, where three participants had a MELD score of 11-20 and three participants had a MELD score of 21-28; resulting in a total of six participants in each period, a total of 18 subjects overall.
1 Participants
n=3 Participants • The six participants in each period were further defined by MELD grouping, where three participants had a MELD score of 11-20 and three participants had a MELD score of 21-28; resulting in a total of six participants in each period, a total of 18 subjects overall.
3 Participants
n=3 Participants • The six participants in each period were further defined by MELD grouping, where three participants had a MELD score of 11-20 and three participants had a MELD score of 21-28; resulting in a total of six participants in each period, a total of 18 subjects overall.
5 Participants
n=9 Participants • The six participants in each period were further defined by MELD grouping, where three participants had a MELD score of 11-20 and three participants had a MELD score of 21-28; resulting in a total of six participants in each period, a total of 18 subjects overall.

PRIMARY outcome

Timeframe: From day 1 up to 42 days following administration of last dose of study drug

The count of subjects who experience serious adverse events

Outcome measures

Outcome measures
Measure
Period 1: F-652 10 μg/kg
n=6 Participants
Participants will receive 10 μg/kg of F-652 on Day 1 and Day 7 via slow intravenous infusion.
Period 2: F-652 30 μg/kg
n=6 Participants
Participants will receive 30 μg/kg of F-652 on Day 1 and Day 7 via slow intravenous infusion.
Period 3: F-652 45 μg/kg
n=6 Participants
Participants will receive 45 μg/kg of F-652 on Day 1 and Day 7 via slow intravenous infusion.
The Number of Subjects With Unexpected Serious Adverse Events.
0 Participants
0 Participants
0 Participants

Adverse Events

Period 1: F-652 10 μg/kg

Serious events: 0 serious events
Other events: 2 other events
Deaths: 0 deaths

Period 2: F-652 30 μg/kg

Serious events: 0 serious events
Other events: 5 other events
Deaths: 1 deaths

Period 3: F-652 45 μg/kg

Serious events: 0 serious events
Other events: 4 other events
Deaths: 0 deaths

Serious adverse events

Adverse event data not reported

Other adverse events

Other adverse events
Measure
Period 1: F-652 10 μg/kg
n=6 participants at risk
Participants will receive 10 μg/kg of F-652 on Day 1 and Day 7 via slow intravenous infusion.
Period 2: F-652 30 μg/kg
n=6 participants at risk
Participants will receive 30 μg/kg of F-652 on Day 1 and Day 7 via slow intravenous infusion.
Period 3: F-652 45 μg/kg
n=6 participants at risk
Participants will receive 45 μg/kg of F-652 on Day 1 and Day 7 via slow intravenous infusion.
Skin and subcutaneous tissue disorders
Pruritus
0.00%
0/6 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
33.3%
2/6 • Number of events 3 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
16.7%
1/6 • Number of events 1 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
Investigations
Leukocytosis
0.00%
0/6 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
16.7%
1/6 • Number of events 1 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
0.00%
0/6 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
Cardiac disorders
Arrhythmia
0.00%
0/6 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
0.00%
0/6 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
16.7%
1/6 • Number of events 1 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
General disorders
Fever
0.00%
0/6 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
16.7%
1/6 • Number of events 1 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
0.00%
0/6 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
General disorders
Nausea
0.00%
0/6 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
16.7%
1/6 • Number of events 1 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
0.00%
0/6 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
Gastrointestinal disorders
Diarrhea
0.00%
0/6 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
0.00%
0/6 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
16.7%
1/6 • Number of events 1 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
Cardiac disorders
Hypertension
0.00%
0/6 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
16.7%
1/6 • Number of events 1 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
0.00%
0/6 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
Skin and subcutaneous tissue disorders
Rash
16.7%
1/6 • Number of events 1 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
0.00%
0/6 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
16.7%
1/6 • Number of events 1 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
General disorders
Tremors
16.7%
1/6 • Number of events 1 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
0.00%
0/6 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
0.00%
0/6 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
General disorders
Muscle Weakness
0.00%
0/6 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
16.7%
1/6 • Number of events 1 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
0.00%
0/6 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
General disorders
Increased body temperature
0.00%
0/6 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
16.7%
1/6 • Number of events 1 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
0.00%
0/6 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
Gastrointestinal disorders
Constipation
0.00%
0/6 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
16.7%
1/6 • Number of events 1 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
0.00%
0/6 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
Hepatobiliary disorders
Hyperbilirubinaemia
0.00%
0/6 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
16.7%
1/6 • Number of events 1 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
0.00%
0/6 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
General disorders
Thrombocytosis
0.00%
0/6 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
16.7%
1/6 • Number of events 1 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
0.00%
0/6 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
Cardiac disorders
Atrioventricular block
0.00%
0/6 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
0.00%
0/6 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days
16.7%
1/6 • Number of events 1 • Adverse Events were collected up to 42 days following the last administration of study treatment for each subject, an average of 56 days

Additional Information

Vijay Shah, M.D.

Mayo Clinic

Phone: 507-284-3917

Results disclosure agreements

  • Principal investigator is a sponsor employee
  • Publication restrictions are in place