Trial Outcomes & Findings for A Study to Assess the Bioavailability and to Compare the Pharmacokinetics of AZD7594 Inhaled Via Monodose Inhaler and Multiple-dose Dry Powder Inhalers (DPI) or Pressurized Metered-dose Inhaler (pMDI) in Healthy Male Subjects (NCT NCT02648438)

NCT ID: NCT02648438

Last Updated: 2017-06-15

Results Overview

For oral and inhalation administrations: pre-dose (0 hour) and post-dose at 15, 30 and 45 minutes and 1.0, 2.0, 4.0, 6.0, 8.0, 12.0, 16.0, 24.0, 36.0, 48.0, 72.0 and 96.0 hours following the administration of the investigational product AZD7594. For IV administration: pre-dose (0 hour) and post-dose at 5, 10, 15 (end of infusion), 30, 45, 60 and 90 minutes and 2.0, 4.0, 6.0, 8.0, 12.0, 16.0, 48.0, 72.0 and 96.0 hours following the start of the IV infusion of the investigational product AZD7594

Recruitment status

COMPLETED

Study phase

PHASE1

Target enrollment

30 participants

Primary outcome timeframe

0-96 hours

Results posted on

2017-06-15

Participant Flow

This study was conducted at PAREXEL International, Early Phase Clinical Unit, Baltimore, United States of America. A total of 30 subjects were enrolled in the study and Twenty-four subjects completed the study.

The IV infusion was fixed as the first treatment (Period 1), the monodose inhaler was fixed as the second treatment (Period 2) and the oral formulation was fixed as the fourth treatment (Period 4). During Period 3, subjects were split into 2 equal cohorts, multiple-dose DPI and pMDI.

Participant milestones

Participant milestones
Measure
IV, DPI 1, DPI 2, Oral
IV formulation, monodose inhaler, multiple-dose DPI, oral formulation
IV, DPI 1, pMDI, Oral
IV formulation, monodose inhaler, pMDI, oral formulation
pMDI (Additional)
Pressurized metered-dose inhaler (pMDI)
Overall Study
STARTED
12
12
6
Overall Study
COMPLETED
9
9
6
Overall Study
NOT COMPLETED
3
3
0

Reasons for withdrawal

Reasons for withdrawal
Measure
IV, DPI 1, DPI 2, Oral
IV formulation, monodose inhaler, multiple-dose DPI, oral formulation
IV, DPI 1, pMDI, Oral
IV formulation, monodose inhaler, pMDI, oral formulation
pMDI (Additional)
Pressurized metered-dose inhaler (pMDI)
Overall Study
Eligibility criteria not fulfilled
0
2
0
Overall Study
Protocol Violation
2
0
0
Overall Study
Withdrawal by Subject
1
1
0

Baseline Characteristics

A Study to Assess the Bioavailability and to Compare the Pharmacokinetics of AZD7594 Inhaled Via Monodose Inhaler and Multiple-dose Dry Powder Inhalers (DPI) or Pressurized Metered-dose Inhaler (pMDI) in Healthy Male Subjects

Baseline characteristics by cohort

Baseline characteristics by cohort
Measure
IV, DPI 1, DPI 2, Oral
n=12 Participants
IV formulation, monodose inhaler, multiple-dose DPI, oral formulation
IV, DPI 1, pMDI, Oral
n=12 Participants
IV formulation, monodose inhaler, pMDI, oral formulation
pMDI (Additional)
n=6 Participants
Pressurized metered-dose inhaler (pMDI)
Total
n=30 Participants
Total of all reporting groups
Age, Continuous
33.3 Years
STANDARD_DEVIATION 7.07 • n=5 Participants
31.3 Years
STANDARD_DEVIATION 4.58 • n=7 Participants
35.5 Years
STANDARD_DEVIATION 2.88 • n=5 Participants
32.9 Years
STANDARD_DEVIATION 5.56 • n=4 Participants
Sex/Gender, Customized
Male
12 Participants
n=5 Participants
12 Participants
n=7 Participants
6 Participants
n=5 Participants
30 Participants
n=4 Participants

PRIMARY outcome

Timeframe: 0-96 hours

Population: The PK analysis set will consist of all subjects in the safety analysis set for whom at least 1 PK parameters can be calculated for at least 1 treatment period and who have no major protocol deviations thought to impact on the analysis of the PK data.

For oral and inhalation administrations: pre-dose (0 hour) and post-dose at 15, 30 and 45 minutes and 1.0, 2.0, 4.0, 6.0, 8.0, 12.0, 16.0, 24.0, 36.0, 48.0, 72.0 and 96.0 hours following the administration of the investigational product AZD7594. For IV administration: pre-dose (0 hour) and post-dose at 5, 10, 15 (end of infusion), 30, 45, 60 and 90 minutes and 2.0, 4.0, 6.0, 8.0, 12.0, 16.0, 48.0, 72.0 and 96.0 hours following the start of the IV infusion of the investigational product AZD7594

Outcome measures

Outcome measures
Measure
400 µg DPI Device 1
n=1 Participants
AZD7594 400 μg delivered dose via Monodose inhaler
400 µg DPI Device 2
n=1 Participants
AZD7594 400 μg delivered dose via Multiple dose inhaler
400 µg pMDI
n=10 Participants
AZD7594 400 μg delivered dose pMDI
400 µg pMDI (Additional)
n=6 Participants
AZD7594 400 μg delivered dose pMDI (Separate treatment)
150 µg IV Formulation
AZD7594 150 µg IV formulation
1200 µg Oral Formulation
AZD7594 1200 μg oral formulation
Pharmacokinetics (PK) of AZD7594 Delivered by Monodose Inhaler and Multiple-dose DPI or pMDI in Terms of Pulmonary Bioavailability After Inhalation (Fpulmonary)
27.49 Percentage
Geometric Coefficient of Variation NA
Insufficient number of participants for CV%.
30.73 Percentage
Geometric Coefficient of Variation NA
Insufficient number of participants for CV%.
NA Percentage
Geometric Coefficient of Variation NA
Plasma levels were too low to be detected hence not calculated.
NA Percentage
Geometric Coefficient of Variation NA
Plasma levels were too low to be detected hence not calculated.

SECONDARY outcome

Timeframe: 0-96 hours

Population: The PK analysis set will consist of all subjects in the safety analysis set for whom at least 1 PK parameters can be calculated for at least 1 treatment period and who have no major protocol deviations thought to impact on the analysis of the PK data.

For oral and inhalation administrations: pre-dose (0 hour) and post-dose at 15, 30 and 45 minutes and 1.0, 2.0, 4.0, 6.0, 8.0, 12.0, 16.0, 24.0, 36.0, 48.0, 72.0 and 96.0 hours following the administration of the investigational product AZD7594. For IV administration: pre-dose (0 hour) and post-dose at 5, 10, 15 (end of infusion), 30, 45, 60 and 90 minutes and 2.0, 4.0, 6.0, 8.0, 12.0, 16.0, 48.0, 72.0 and 96.0 hours following the start of the IV infusion of the investigational product AZD7594

Outcome measures

Outcome measures
Measure
400 µg DPI Device 1
n=24 Participants
AZD7594 400 μg delivered dose via Monodose inhaler
400 µg DPI Device 2
n=1 Participants
AZD7594 400 μg delivered dose via Multiple dose inhaler
400 µg pMDI
AZD7594 400 μg delivered dose pMDI
400 µg pMDI (Additional)
AZD7594 400 μg delivered dose pMDI (Separate treatment)
150 µg IV Formulation
AZD7594 150 µg IV formulation
1200 µg Oral Formulation
AZD7594 1200 μg oral formulation
PK of AZD7594 Following Oral Administration by Assessment of the Absolute Systemic Bioavailability After Oral Administration (Fpo)
NA Percentage
Geometric Coefficient of Variation NA
The Fpo is calculated only after oral administration hence not applicable for IV administration.
0.4543 Percentage
Geometric Coefficient of Variation NA
The Fpo could not be calculated because the plasma levels after oral administration were so low, they could not be quantified.

SECONDARY outcome

Timeframe: 0-96 hours

Population: The PK analysis set will consist of all subjects in the safety analysis set for whom at least 1 PK parameters can be calculated for at least 1 treatment period and who have no major protocol deviations thought to impact on the analysis of the PK data.

For oral and inhalation administrations: pre-dose (0 hour) and post-dose at 15, 30 and 45 minutes and 1.0, 2.0, 4.0, 6.0, 8.0, 12.0, 16.0, 24.0, 36.0, 48.0, 72.0 and 96.0 hours following the administration of the investigational product AZD7594. For IV administration: pre-dose (0 hour) and post-dose at 5, 10, 15 (end of infusion), 30, 45, 60 and 90 minutes and 2.0, 4.0, 6.0, 8.0, 12.0, 16.0, 48.0, 72.0 and 96.0 hours following the start of the IV infusion of the investigational product AZD7594

Outcome measures

Outcome measures
Measure
400 µg DPI Device 1
n=23 Participants
AZD7594 400 μg delivered dose via Monodose inhaler
400 µg DPI Device 2
n=9 Participants
AZD7594 400 μg delivered dose via Multiple dose inhaler
400 µg pMDI
n=3 Participants
AZD7594 400 μg delivered dose pMDI
400 µg pMDI (Additional)
n=3 Participants
AZD7594 400 μg delivered dose pMDI (Separate treatment)
150 µg IV Formulation
n=24 Participants
AZD7594 150 µg IV formulation
1200 µg Oral Formulation
n=2 Participants
AZD7594 1200 μg oral formulation
Observed Maximum Plasma Concentration (Cmax)
112.6 pmol/L
Geometric Coefficient of Variation 28.42
68.88 pmol/L
Geometric Coefficient of Variation 22.16
13.93 pmol/L
Geometric Coefficient of Variation 25.73
15.47 pmol/L
Geometric Coefficient of Variation 11.34
6598 pmol/L
Geometric Coefficient of Variation 27.05
19.31 pmol/L
Geometric Coefficient of Variation 19.90

SECONDARY outcome

Timeframe: 0-96 hours

Population: The PK analysis set will consist of all subjects in the safety analysis set for whom at least 1 PK parameters can be calculated for at least 1 treatment period and who have no major protocol deviations thought to impact on the analysis of the PK data.

For oral and inhalation administrations: pre-dose (0 hour) and post-dose at 15, 30 and 45 minutes and 1.0, 2.0, 4.0, 6.0, 8.0, 12.0, 16.0, 24.0, 36.0, 48.0, 72.0 and 96.0 hours following the administration of the investigational product AZD7594. For IV administration: pre-dose (0 hour) and post-dose at 5, 10, 15 (end of infusion), 30, 45, 60 and 90 minutes and 2.0, 4.0, 6.0, 8.0, 12.0, 16.0, 48.0, 72.0 and 96.0 hours following the start of the IV infusion of the investigational product AZD7594

Outcome measures

Outcome measures
Measure
400 µg DPI Device 1
n=23 Participants
AZD7594 400 μg delivered dose via Monodose inhaler
400 µg DPI Device 2
n=9 Participants
AZD7594 400 μg delivered dose via Multiple dose inhaler
400 µg pMDI
n=1 Participants
AZD7594 400 μg delivered dose pMDI
400 µg pMDI (Additional)
n=3 Participants
AZD7594 400 μg delivered dose pMDI (Separate treatment)
150 µg IV Formulation
n=24 Participants
AZD7594 150 µg IV formulation
1200 µg Oral Formulation
n=1 Participants
AZD7594 1200 μg oral formulation
Area Under the Plasma Concentration-curve From Time Zero to Time of Last Quantifiable Concentration (AUC0-t)
2524 (h*pmol/L)
Geometric Coefficient of Variation 45.16
2648 (h*pmol/L)
Geometric Coefficient of Variation 23.13
42.93 (h*pmol/L)
Geometric Coefficient of Variation NA
Not applicable as n=1
572.7 (h*pmol/L)
Geometric Coefficient of Variation 83.69
3343 (h*pmol/L)
Geometric Coefficient of Variation 19.69
110.1 (h*pmol/L)
Geometric Coefficient of Variation NA
Not applicable as n=1

SECONDARY outcome

Timeframe: 0-96 hours

Population: The PK analysis set will consist of all subjects in the safety analysis set for whom at least 1 PK parameters can be calculated for at least 1 treatment period and who have no major protocol deviations thought to impact on the analysis of the PK data.

For oral and inhalation administrations: pre-dose (0 hour) and post-dose at 15, 30 and 45 minutes and 1.0, 2.0, 4.0, 6.0, 8.0, 12.0, 16.0, 24.0, 36.0, 48.0, 72.0 and 96.0 hours following the administration of the investigational product AZD7594. For IV administration: pre-dose (0 hour) and post-dose at 5, 10, 15 (end of infusion), 30, 45, 60 and 90 minutes and 2.0, 4.0, 6.0, 8.0, 12.0, 16.0, 48.0, 72.0 and 96.0 hours following the start of the IV infusion of the investigational product AZD7594

Outcome measures

Outcome measures
Measure
400 µg DPI Device 1
n=23 Participants
AZD7594 400 μg delivered dose via Monodose inhaler
400 µg DPI Device 2
n=9 Participants
AZD7594 400 μg delivered dose via Multiple dose inhaler
400 µg pMDI
n=1 Participants
AZD7594 400 μg delivered dose pMDI
400 µg pMDI (Additional)
n=6 Participants
AZD7594 400 μg delivered dose pMDI (Separate treatment)
150 µg IV Formulation
AZD7594 150 µg IV formulation
1200 µg Oral Formulation
AZD7594 1200 μg oral formulation
Absolute Systemic Bioavailability After Inhalation (F Inhalation, Total)
28.21 Percentage
Geometric Coefficient of Variation 45.38
30.92 Percentage
Geometric Coefficient of Variation 20.87
0.3560 Percentage
Geometric Coefficient of Variation NA
Plasma levels were too low to be detected hence not calculated.
NA Percentage
Geometric Coefficient of Variation NA
Plasma levels were too low to be detected hence not calculated.

SECONDARY outcome

Timeframe: 0-96 hours

Population: The PK analysis set will consist of all subjects in the safety analysis set for whom at least 1 PK parameters can be calculated for at least 1 treatment period and who have no major protocol deviations thought to impact on the analysis of the PK data.

For oral and inhalation administrations: pre-dose (0 hour) and post-dose at 15, 30 and 45 minutes and 1.0, 2.0, 4.0, 6.0, 8.0, 12.0, 16.0, 24.0, 36.0, 48.0, 72.0 and 96.0 hours following the administration of the investigational product AZD7594. For IV administration: pre-dose (0 hour) and post-dose at 5, 10, 15 (end of infusion), 30, 45, 60 and 90 minutes and 2.0, 4.0, 6.0, 8.0, 12.0, 16.0, 48.0, 72.0 and 96.0 hours following the start of the IV infusion of the investigational product AZD7594

Outcome measures

Outcome measures
Measure
400 µg DPI Device 1
n=1 Participants
AZD7594 400 μg delivered dose via Monodose inhaler
400 µg DPI Device 2
n=1 Participants
AZD7594 400 μg delivered dose via Multiple dose inhaler
400 µg pMDI
n=10 Participants
AZD7594 400 μg delivered dose pMDI
400 µg pMDI (Additional)
n=6 Participants
AZD7594 400 μg delivered dose pMDI (Separate treatment)
150 µg IV Formulation
AZD7594 150 µg IV formulation
1200 µg Oral Formulation
AZD7594 1200 μg oral formulation
Oral Bioavailability After Inhaled Treatment (F Oral)
0.3294 Percentage
Geometric Coefficient of Variation NA
Not applicable as n=1
0.3147 Percentage
Geometric Coefficient of Variation NA
Not applicable as n=1
NA Percentage
Geometric Coefficient of Variation NA
F oral was not calculated for the additional pMDI cohort as this cohort did not receive the oral and IV formulation treatments.
NA Percentage
Geometric Coefficient of Variation NA
F oral was not calculated for the additional pMDI cohort as this cohort did not receive the oral and IV formulation treatments.

SECONDARY outcome

Timeframe: 0-96 hours

Population: The PK analysis set will consist of all subjects in the safety analysis set for whom at least 1 PK parameters can be calculated for at least 1 treatment period and who have no major protocol deviations thought to impact on the analysis of the PK data.

For oral and inhalation administrations: pre-dose (0 hour) and post-dose at 15, 30 and 45 minutes and 1.0, 2.0, 4.0, 6.0, 8.0, 12.0, 16.0, 24.0, 36.0, 48.0, 72.0 and 96.0 hours following the administration of the investigational product AZD7594. For IV administration: pre-dose (0 hour) and post-dose at 5, 10, 15 (end of infusion), 30, 45, 60 and 90 minutes and 2.0, 4.0, 6.0, 8.0, 12.0, 16.0, 48.0, 72.0 and 96.0 hours following the start of the IV infusion of the investigational product AZD7594

Outcome measures

Outcome measures
Measure
400 µg DPI Device 1
n=23 Participants
AZD7594 400 μg delivered dose via Monodose inhaler
400 µg DPI Device 2
n=9 Participants
AZD7594 400 μg delivered dose via Multiple dose inhaler
400 µg pMDI
n=10 Participants
AZD7594 400 μg delivered dose pMDI
400 µg pMDI (Additional)
n=6 Participants
AZD7594 400 μg delivered dose pMDI (Separate treatment)
150 µg IV Formulation
n=24 Participants
AZD7594 150 µg IV formulation
1200 µg Oral Formulation
n=9 Participants
AZD7594 1200 μg oral formulation
Area Under Plasma Concentration-time Curve From Time Zero Extrapolated to Infinity (AUC)
NA (h*pmol/L)
Geometric Coefficient of Variation NA
Not reported since parameter cannot be calculated as per standard criteria.
NA (h*pmol/L)
Geometric Coefficient of Variation NA
Not reported since parameter cannot be calculated as per standard criteria.
NA (h*pmol/L)
Geometric Coefficient of Variation NA
Plasma levels were too low to be detected hence not calculated.
NA (h*pmol/L)
Geometric Coefficient of Variation NA
Plasma levels were too low to be detected hence not calculated.
3465 (h*pmol/L)
Geometric Coefficient of Variation 19.44
NA (h*pmol/L)
Geometric Coefficient of Variation NA
Plasma levels were too low to be detected hence not calculated.

Adverse Events

IV Formulation

Serious events: 0 serious events
Other events: 2 other events
Deaths: 0 deaths

DPI Device 1

Serious events: 0 serious events
Other events: 0 other events
Deaths: 0 deaths

DPI Device 2

Serious events: 0 serious events
Other events: 2 other events
Deaths: 0 deaths

pMDI

Serious events: 0 serious events
Other events: 1 other events
Deaths: 0 deaths

Oral Formulation

Serious events: 0 serious events
Other events: 1 other events
Deaths: 0 deaths

pMDI (Additional)

Serious events: 0 serious events
Other events: 1 other events
Deaths: 0 deaths

Serious adverse events

Adverse event data not reported

Other adverse events

Other adverse events
Measure
IV Formulation
n=24 participants at risk
AZD7594 150 μg IV formulation
DPI Device 1
n=23 participants at risk
AZD7594 400 μg delivered dose monodose inhaler
DPI Device 2
n=9 participants at risk
AZD7594 400 μg delivered dose multiple-dose DPI
pMDI
n=10 participants at risk
AZD7594 400 μg delivered dose pMDI
Oral Formulation
n=18 participants at risk
AZD7594 1200 μg oral formulation
pMDI (Additional)
n=6 participants at risk
AZD7594 400 μg delivered dose pMDI (separate treatment)
Nervous system disorders
Dizziness
0.00%
0/24 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
0.00%
0/23 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
0.00%
0/9 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
10.0%
1/10 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
0.00%
0/18 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
16.7%
1/6 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
Eye disorders
Ocular hyperemia
0.00%
0/24 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
0.00%
0/23 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
0.00%
0/9 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
0.00%
0/10 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
5.6%
1/18 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
0.00%
0/6 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
General disorders
Infusion site pain
4.2%
1/24 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
0.00%
0/23 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
0.00%
0/9 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
0.00%
0/10 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
0.00%
0/18 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
0.00%
0/6 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
Infections and infestations
Viral upper respiratory tract infection
0.00%
0/24 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
0.00%
0/23 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
11.1%
1/9 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
0.00%
0/10 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
0.00%
0/18 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
0.00%
0/6 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
Injury, poisoning and procedural complications
Traumatic hematoma
4.2%
1/24 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
0.00%
0/23 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
0.00%
0/9 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
0.00%
0/10 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
0.00%
0/18 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
0.00%
0/6 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
Musculoskeletal and connective tissue disorders
Myalgia
4.2%
1/24 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
0.00%
0/23 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
0.00%
0/9 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
0.00%
0/10 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
0.00%
0/18 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
0.00%
0/6 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
Respiratory, thoracic and mediastinal disorders
Nasal congestion
0.00%
0/24 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
0.00%
0/23 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
11.1%
1/9 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
0.00%
0/10 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
0.00%
0/18 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.
0.00%
0/6 • Serious adverse events (SAEs) were collected from the signing of informed consent and AEs from check-in for the first treatment period until the final follow-up phone-call i.e., from Visit 1 to Visit 6 (Day -21 to Day 5).
There were no deaths or SAEs reported in this study.

Additional Information

Global Clinical Leader

AstraZeneca AB

Phone: +46 31 7761000

Results disclosure agreements

  • Principal investigator is a sponsor employee If a publication (e.g., in a scientific journal) based on the results of this study is envisaged, approval from AstraZeneca will be obtained and a draft manuscript will be submitted to AstraZeneca for scrutiny and comment. The choice of conduit will be mutually agreed on by the Principal Investigator and AstraZeneca.
  • Publication restrictions are in place

Restriction type: OTHER