Pharmacokinetic Study of Alpelisib in Subjects With Hepatic Impairment.

NCT ID: NCT02624557

Last Updated: 2020-12-09

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

23 participants

Study Classification

INTERVENTIONAL

Study Start Date

2015-12-21

Study Completion Date

2017-10-01

Brief Summary

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To characterize the pharmacokinetics and safety of alpelisib in subjects with hepatic impairment compared to matched healthy control subjects.

Detailed Description

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Conditions

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Hepatic Impairment

Keywords

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Hepatic impairment Healthy volunteers Clinical pharmacology study BYL719 alpelisib

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

BASIC_SCIENCE

Blinding Strategy

NONE

Study Groups

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Moderate hepatic impairment group

Subjects with moderate hepatic impairment with Child-Pugh score 7 - 9

Group Type EXPERIMENTAL

Alpelisib

Intervention Type DRUG

Subjects will receive a single dose of 300 mg alpelisib.

Severe hepatic impairment group

Subjects with severe hepatic impairment with Child-Pugh score 10 - 15

Group Type EXPERIMENTAL

Alpelisib

Intervention Type DRUG

Subjects will receive a single dose of 300 mg alpelisib.

Matching healthy control group

Subjects with apparent normal liver function matched to the hepatic impairment subjects by sex, race, age, and weight.

Group Type EXPERIMENTAL

Alpelisib

Intervention Type DRUG

Subjects will receive a single dose of 300 mg alpelisib.

Interventions

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Alpelisib

Subjects will receive a single dose of 300 mg alpelisib.

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

Additional criteria for hepatic impaired subjects: -Subjects must have a score clinically determined and calculated as per the Child-Pugh classification and consistent with the degree of hepatic impairment in which study is currently enrolling. -Stable Child-Pugh status within 28 days prior to dosing.

Exclusion Criteria

* Subject has received a liver transplant at any time in the past and is on immunosuppressant therapy.
* Smokers not willing to limit the use of tobacco to 10 cigarettes per day. -Surgical or medical condition which might significantly alter the absorption, distribution, metabolism, or excretion of drugs, or which may jeopardize the subject's safety in case of participation in the study. -Use of any herbal medications/supplements.

History of acute pancreatitis within 1 year of study entry.

Additional criteria for subjects with normal liver function:

-Use of any prescription or non-prescription medication. -Positive Hepatitis B surface antigen (HBsAg) or Hepatitis C test result.

Additional criteria for hepatic impaired subjects: -Use of any prescription or non-prescription medication, that has the potential to interact with alpelisb. Concomitant medications without potential to interact with alpelisib must be stable in dose. -Encephalopathy grade 3 or worse. -Total bilirubin \> 6 mg/dl. Screening or baseline ECG: QTcF\>480msec for both genders
Minimum Eligible Age

18 Years

Maximum Eligible Age

75 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

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Novartis Pharmaceuticals

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Novartis Pharmaceuticals

Role: STUDY_DIRECTOR

Novartis Pharmaceuticals

Locations

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DaVita Clinical Research-Denver

Lakewood, Colorado, United States

Site Status

University of Miami / Clinical Research Services, Inc.

Miami, Florida, United States

Site Status

Orlando Clinical Research Center

Orlando, Florida, United States

Site Status

DaVita Clinical Research

Minneapolis, Minnesota, United States

Site Status

Countries

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United States

Related Links

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https://www.novctrd.com/ctrdweb/trialresult/trialresults/pdf?trialResultId=17198

Results for CBYL719A2105 can be found on the Novartis Clinical Trial Results Website

Other Identifiers

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CBYL719A2105

Identifier Type: -

Identifier Source: org_study_id