Study on Effects of BMS-955176 on the Pharmacokinetics of Probe Substrates

NCT ID: NCT02578277

Last Updated: 2018-07-13

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

59 participants

Study Classification

INTERVENTIONAL

Study Start Date

2015-11-09

Study Completion Date

2015-12-23

Brief Summary

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The purpose of the study is to study the effects of BMS-955176 on the single-dose PK parameters of probe substrates caffeine, metoprolol, montelukast, flurbiprofen, omeprazole, midazolam, digoxin, and pravastatin

Detailed Description

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Conditions

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HIV Infections

Study Design

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Allocation Method

NA

Intervention Model

SINGLE_GROUP

Primary Study Purpose

OTHER

Blinding Strategy

NONE

Study Groups

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Single sequence, 3-period DDI (drug-drug interaction)

Single sequence

Group Type EXPERIMENTAL

CYP and transporter probe substrates

Intervention Type DRUG

Cocktail of CYP (cytochrome P450) and transporter probe substrates

BMS-955176

Intervention Type DRUG

BMS-955176

BMS-955176 plus CYP and transporter probe substrates

Intervention Type DRUG

BMS-955176 plus the cocktail of CYP and transporter probe substrates

Interventions

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CYP and transporter probe substrates

Cocktail of CYP (cytochrome P450) and transporter probe substrates

Intervention Type DRUG

BMS-955176

BMS-955176

Intervention Type DRUG

BMS-955176 plus CYP and transporter probe substrates

BMS-955176 plus the cocktail of CYP and transporter probe substrates

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

1. Written Informed Consent
2. Healthy male and female (not of childbearing potential) subjects as determined by medical history, surgical history, physical examination, vital signs, ECGs, and clinical laboratory determinations
3. Body mass index (BMI) of 18.0 kg/m2 to 32.0 kg/m2, inclusive, at screening and Day 1. BMI = weight (kg)/\[height(m)\]
4. Women must have documented proof that they are not of childbearing potential (eg, surgically sterile, postmenopausal with a documented follicle-stimulating hormone (FSH) \> 40 mIU/mL) and should not be breast feeding
5. Males who are sexually active with WOCBP must agree to follow instructions for method(s) of contraception for the duration of treatment with BMS-955176 in addition to a post-treatment completion period

Exclusion Criteria

1. Any significant acute or chronic medical illness
2. Use of tobacco, excessive alcohol
3. Medical history indicative of an increased risk of a cardiac arrhythmia or cardiac disease and history of asthma, bronchospasm, sleep apnea, rhabdomyolysis, a bleeding disorder, a major depressive disorder within the past 6 months, peptic ulcer or significant GI bleed, Raynaud's disease, or any gastrointestinal surgery that could impact upon the absorption of study drug
4. Evidence of organ dysfunction or any clinically significant deviation from normal in physical examination, vital signs, ECG, or clinical laboratory determinations beyond what is consistent with the target population
5. History of allergy to BMS-955176, digoxin (or any member of the digitalis glycosides class of drugs), caffeine, metoprolol, montelukast, flurbiprofen, omeprazole, midazolam, or pravastatin, or to any related compounds
Minimum Eligible Age

18 Years

Maximum Eligible Age

50 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

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ViiV Healthcare

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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GSK Clinical Trials

Role: STUDY_DIRECTOR

ViiV Healthcare

Locations

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GSK Investigational Site

Austin, Texas, United States

Site Status

Countries

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United States

Other Identifiers

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AI468-063

Identifier Type: OTHER

Identifier Source: secondary_id

206294

Identifier Type: -

Identifier Source: org_study_id

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