MSC2364447C Phase 1b in Systemic Lupus Erythematosus

NCT ID: NCT02537028

Last Updated: 2017-10-09

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

24 participants

Study Classification

INTERVENTIONAL

Study Start Date

2015-11-30

Study Completion Date

2016-10-04

Brief Summary

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The primary purpose of this Phase 1b double-blind, randomized, placebo-controlled trial is to evaluate the safety, tolerability, pharmacokinetic (PK), and biological effect of MSC2364447C administered for 4 weeks in systemic lupus erythematosus subjects (SLE).

Detailed Description

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Conditions

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Lupus Erythematosus, Systemic

Keywords

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MSC2364447C Phase 1 BTK inhibitor Systemic Lupus Erythematosus M2951 Lupus

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

TRIPLE

Participants Caregivers Investigators

Study Groups

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MSC2364447C 25 mg

Group Type EXPERIMENTAL

MSC2364447C

Intervention Type DRUG

Subjects will be administered with MSC2364447C 25 milligrams orally once daily for 4 weeks.

MSC2364447C 75 mg

Group Type EXPERIMENTAL

MSC2364447C

Intervention Type DRUG

Subjects will be administered with MSC2364447C 75 milligrams orally once daily for 4 weeks.

Placebo

Group Type PLACEBO_COMPARATOR

Placebo

Intervention Type DRUG

Subjects will be administered with placebo matching to MSC2364447C orally once daily for 4 weeks.

Interventions

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MSC2364447C

Subjects will be administered with MSC2364447C 25 milligrams orally once daily for 4 weeks.

Intervention Type DRUG

MSC2364447C

Subjects will be administered with MSC2364447C 75 milligrams orally once daily for 4 weeks.

Intervention Type DRUG

Placebo

Subjects will be administered with placebo matching to MSC2364447C orally once daily for 4 weeks.

Intervention Type DRUG

Other Intervention Names

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M2951, Evobrutinib M2951, Evobrutinib

Eligibility Criteria

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Inclusion Criteria

* Male or female of 18 to 65 years of age
* Diagnosis of systemic lupus erythematosus (SLE) (at least 4 of the 11 American College of Rheumatology \[ACR\] classification criteria for SLE) of at least 6 months duration at the Screening visit
* Positive test results for anti-nuclear antibody (ANA) (human epithelial cell-2 ANA greater than or equal to \[\>=\] 1:80) and/or anti-dsDNA antibody (\>= 30 international units per milliliter \[IU/mL\]) at the Screening visit
* At least 1 SLE disease manifestation (assessed by Systemic Lupus Erythematosus Disease Activity Index-2000 \[SLEDAI-2K\]) other than positive antidsDNA and no central nervous system (CNS) SLE (psychosis, organic brain syndrome, cranial nerve disorder, lupus headache, or new-onset cerebrovascular accident)
* History of vaccinations as follows or vaccination against these pathogens during Screening:

1. Vaccination against Streptococcus pneumoniae with pneumococcal polysaccharide vaccine 23 or pneumococcal 13-valent conjugate vaccine as per local guidelines, and
2. Vaccination against influenza virus (as per local seasonal recommendations). Subjects receiving 1 or more of these vaccinations during screening must have at least 2 weeks between the vaccination(s) and the date of randomization at Day 1.

Exclusion Criteria

* Active clinically significant CNS SLE
* Initiation or change in dose of anti-malarial treatment after the screening visit
* Within 2 weeks prior to Screening or during Screening: use of oral corticosteroids greater than (\>) 40 mg daily prednisone equivalent, use of any injectable corticosteroids, or change in dose of corticosteroids
* Within 2 weeks prior to Screening, initiation or change in dose of angiotensin-converting enzyme inhibitor or angiotensin receptor blocker, or nonsteroidal anti-inflammatory drugs (NSAIDs).
* Within 2 months prior to Screening or during Screening: initiation of or change in dose of methotrexate, mycophenolate (mofetil or sodium), or azathioprine
* Within 2 months prior to Screening or during Screening, use of cyclosporine, tacrolimus, leflunomide, abatacept, anti-tumor necrosis factor alpha agents, intravenous immunoglobulin, plasmapheresis, or other disease-modifying, immunosuppressive, or immunomodulatory therapies not otherwise specified in protocol
* Within 6 months prior to Screening or during Screening: use of cyclophosphamide or chlorambucil
* Within 12 months prior to screening or during screening: use of rituximab, belimumab, or any other B cell-depleting or modulating therapies
* Within 1 month prior to Screening or during Screening, vaccination with live or live-attenuated virus vaccine.
* Active clinically significant viral, bacterial or fungal infection, or any serious episode of infection requiring hospitalization within the last 6 months - Estimated glomerular filtration rate by the Modification of Diet in Renal Disease equation of less than (\<) 60 milliliter per minute per 1.73 square meter (mL/min/1.73 m\^2), or recent decline in kidney function, or proteinuria \>= 3 gram per day (g/day) (spot urine protein/creatinine ratio \>= 3 mg/mg)
Minimum Eligible Age

18 Years

Maximum Eligible Age

65 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Merck KGaA, Darmstadt, Germany

INDUSTRY

Sponsor Role collaborator

EMD Serono Research & Development Institute, Inc.

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Medical Responsible

Role: STUDY_DIRECTOR

EMD Serono Research & Development Institute, Inc., a business of Merck KGaA, Darmstadt, Germany

Locations

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Research site

Anniston, Alabama, United States

Site Status

Research site

El Cajon, California, United States

Site Status

Research site

Lakewood, California, United States

Site Status

Research site

Los Angeles, California, United States

Site Status

Research site

Clearwater, Florida, United States

Site Status

Research site

DeBary, Florida, United States

Site Status

Research site

Orlando, Florida, United States

Site Status

Research site

Grand Blanc, Michigan, United States

Site Status

Research site

St Louis, Missouri, United States

Site Status

Research site

Austin, Texas, United States

Site Status

Research site

Sofia, , Bulgaria

Site Status

Research site

Sofia, , Bulgaria

Site Status

Research site

Sofia, , Bulgaria

Site Status

Countries

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United States Bulgaria

Other Identifiers

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2015-001891-23

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

EMR200527-002

Identifier Type: -

Identifier Source: org_study_id