Safety and Tolerability of MSI-1436C in Metastatic Breast Cancer

NCT ID: NCT02524951

Last Updated: 2018-05-18

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

TERMINATED

Clinical Phase

PHASE1

Total Enrollment

5 participants

Study Classification

INTERVENTIONAL

Study Start Date

2016-04-30

Study Completion Date

2018-05-14

Brief Summary

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This is a Phase I, open-label, dose escalation study. MSI-1436 will be administered as a single intravenous infusion twice a week for 3 weeks on a 4-week cycle.

Detailed Description

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This is a Phase I, open-label, dose escalation study. MSI-1436 will be administered as a single intravenous infusion twice a week for 3 weeks on a 4-week cycle. Subjects will be enrolled according to a standard Phase I Fibonacci design to receive MSI-1436. Drug infusions will last approximately 2 hours. If a subject has a dose-limiting toxicity (DLT) at any time during the study, MSI-1436 will be held and either re-started or discontinued in that subject as per the Dose Adjustments and Toxicities Guidelines.

Conditions

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Metastatic Breast Cancer

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

SINGLE_GROUP

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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MSI-1436C (Trodusquemine) 20 mg/m2 IV

Open label, interventional, dose escalation of MSI-1436 (Trodusquemine), single intravenous infusion twice a week for 3 weeks on a 4-week cycle. Subjects will receive MSI-1436 at a dose of 20 mg/m2. Drug infusions will last approximately 2 hours.

Group Type EXPERIMENTAL

MSI-1436C

Intervention Type DRUG

Dose escalation, single intravenous infusion twice a week for 3 weeks on a 4-week cycle.

MSI-1436C (Trodusquemine) 26 mg/m2 IV

Open label, interventional, dose escalation of MSI-1436 (Trodusquemine), single intravenous infusion twice a week for 3 weeks on a 4-week cycle. Subjects will receive MSI-1436 at a dose of 26 mg/m2. Drug infusions will last approximately 2 hours.

Group Type EXPERIMENTAL

MSI-1436C

Intervention Type DRUG

Dose escalation, single intravenous infusion twice a week for 3 weeks on a 4-week cycle.

MSI-1436C (Trodusquemine) 34 mg/m2 IV

Open label, interventional, dose escalation of MSI-1436 (Trodusquemine), single intravenous infusion twice a week for 3 weeks on a 4-week cycle. Subjects will receive MSI-1436 at a dose of 34 mg/m2 . Drug infusions will last approximately 2 hours.

Group Type EXPERIMENTAL

MSI-1436C

Intervention Type DRUG

Dose escalation, single intravenous infusion twice a week for 3 weeks on a 4-week cycle.

MSI-1436C (Trodusquemine) 44 mg/m2 IV

Open label, interventional, dose escalation of MSI-1436 (Trodusquemine), single intravenous infusion twice a week for 3 weeks on a 4-week cycle. Subjects will receive MSI-1436 at a dose of 44 mg/m2 . Drug infusions will last approximately 2 hours.

Group Type EXPERIMENTAL

MSI-1436C

Intervention Type DRUG

Dose escalation, single intravenous infusion twice a week for 3 weeks on a 4-week cycle.

MSI-1436C (Trodusquemine) 57 mg/m2 IV

Open label, interventional, dose escalation of MSI-1436 (Trodusquemine), single intravenous infusion twice a week for 3 weeks on a 4-week cycle. Subjects will receive MSI-1436 at a dose of 57 mg/m2. Drug infusions will last approximately 2 hours.

Group Type EXPERIMENTAL

MSI-1436C

Intervention Type DRUG

Dose escalation, single intravenous infusion twice a week for 3 weeks on a 4-week cycle.

MSI-1436C (Trodusquemine) 74 mg/m2 IV

Open label, interventional, dose escalation of MSI-1436 (Trodusquemine), single intravenous infusion twice a week for 3 weeks on a 4-week cycle. Subjects will receive MSI-1436 at a dose of 74 mg/m2 . Drug infusions will last approximately 2 hours.

Group Type EXPERIMENTAL

MSI-1436C

Intervention Type DRUG

Dose escalation, single intravenous infusion twice a week for 3 weeks on a 4-week cycle.

MSI-1436C (Trodusquemine) 96 mg/m2 IV

Open label, interventional, dose escalation of MSI-1436 (Trodusquemine), single intravenous infusion twice a week for 3 weeks on a 4-week cycle. Subjects will receive MSI-1436 at a dose of 96 mg/m2 . Drug infusions will last approximately 2 hours.

Group Type EXPERIMENTAL

MSI-1436C

Intervention Type DRUG

Dose escalation, single intravenous infusion twice a week for 3 weeks on a 4-week cycle.

Interventions

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MSI-1436C

Dose escalation, single intravenous infusion twice a week for 3 weeks on a 4-week cycle.

Intervention Type DRUG

Other Intervention Names

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Trodusquemine

Eligibility Criteria

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Inclusion Criteria

* Signed, witnessed, and dated Institutional Review Board (IRB) approved Informed Consent Form (ICF).
* Pathologically confirmed metastatic breast cancer with measurable disease. Metastatic sites must be measurable on CT, MRI, or FDG-PET/CT as per the revised RECIST v1.1 criteria or measurable disease on physical examination.

A metastatic site must be biopsy proven

* Life expectancy ≥3 months.
* Patients enrolled must have received 2 or more lines of therapy and all patients with HER2 expressing tumors must have received HER2 targeted therapy.
* Female Age ≥18 years.
* Stable brain metastasis is permitted. This is not considered measurable disease.

Stable brain metastasis is defined as no change on CT scan or MRI for minimum of 2 months AND no change in steroid dose for a minimum of 4 weeks

* A negative serum pregnancy test, if female of reproductive potential. Reproductive potential defined as age \< 55 or with no menses for \< 1 year
* Screening laboratory values as follows:

Total bilirubin ≤1.5 times upper limit of normal (ULN). Aspartate aminotransferase (serum glutamic oxaloacetic transaminase) and alanine aminotransferase (serum glutamic pyruvate transaminase)≤ 2.5 times ULN.

Serum creatinine ≤2.0 mg/dL or calculated creatinine clearance ≥60 mL/min. Absolute neutrophil count \>1,500 cells/mm3. Platelet count ≥100,000 plt/mm3. Hemoglobin ≥ 8 g/dL. Non-diabetic

Exclusion Criteria

* Pregnant or breast-feeding
* ECOG Performance Status greater than 2
Minimum Eligible Age

18 Years

Eligible Sex

FEMALE

Accepts Healthy Volunteers

No

Sponsors

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DepYmed Inc.

INDUSTRY

Sponsor Role collaborator

Northwell Health

OTHER

Sponsor Role lead

Responsible Party

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Daniel Budman

Director Translational Research, Cancer Institute

Responsibility Role PRINCIPAL_INVESTIGATOR

Principal Investigators

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Daniel Budman, MD

Role: PRINCIPAL_INVESTIGATOR

North Shore LIJ Cancer Institute

Locations

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CFAM / Monter Cancer Center

Lake Success, New York, United States

Site Status

Countries

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United States

Other Identifiers

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IIS-0039

Identifier Type: -

Identifier Source: org_study_id

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