Trial Outcomes & Findings for Tolerability, Safety, and Activity of SRX246 in Irritable Subjects With Huntington's Disease (NCT NCT02507284)

NCT ID: NCT02507284

Last Updated: 2023-07-20

Results Overview

The primary endpoint, tolerability of SRX246, was assessed by the number of completers in each group.

Recruitment status

COMPLETED

Study phase

PHASE2

Target enrollment

106 participants

Primary outcome timeframe

12 weeks

Results posted on

2023-07-20

Participant Flow

Participant milestones

Participant milestones
Measure
SRX246 120mg BID
SRX246 capsules, administered orally, in divided doses twice daily SRX246
SRX246 160mg BID
SRX246 capsules, administered orally, in divided doses twice daily SRX246
Placebo
Placebo capsules, administered orally, in divided doses twice daily Placebo
Overall Study
STARTED
36
34
36
Overall Study
COMPLETED
25
27
30
Overall Study
NOT COMPLETED
11
7
6

Reasons for withdrawal

Withdrawal data not reported

Baseline Characteristics

Tolerability, Safety, and Activity of SRX246 in Irritable Subjects With Huntington's Disease

Baseline characteristics by cohort

Baseline characteristics by cohort
Measure
SRX246 120mg BID
n=36 Participants
SRX246 capsules, administered orally, in divided doses twice daily SRX246
SRX246 160mg BID
n=34 Participants
SRX246 capsules, administered orally, in divided doses twice daily SRX246
Placebo
n=36 Participants
Placebo capsules, administered orally, in divided doses twice daily Placebo
Total
n=106 Participants
Total of all reporting groups
Age, Continuous
51.1 years
STANDARD_DEVIATION 13.2 • n=5 Participants
48.9 years
STANDARD_DEVIATION 12.7 • n=7 Participants
51.7 years
STANDARD_DEVIATION 10.4 • n=5 Participants
50.6 years
STANDARD_DEVIATION 12.1 • n=4 Participants
Sex: Female, Male
Female
18 Participants
n=5 Participants
17 Participants
n=7 Participants
20 Participants
n=5 Participants
55 Participants
n=4 Participants
Sex: Female, Male
Male
18 Participants
n=5 Participants
17 Participants
n=7 Participants
16 Participants
n=5 Participants
51 Participants
n=4 Participants
Race/Ethnicity, Customized
White
36 Participants
n=5 Participants
33 Participants
n=7 Participants
36 Participants
n=5 Participants
105 Participants
n=4 Participants
Race/Ethnicity, Customized
Not White
0 Participants
n=5 Participants
1 Participants
n=7 Participants
0 Participants
n=5 Participants
1 Participants
n=4 Participants
Race/Ethnicity, Customized
Hispanic/Latino
2 Participants
n=5 Participants
4 Participants
n=7 Participants
0 Participants
n=5 Participants
6 Participants
n=4 Participants
Race/Ethnicity, Customized
Not Hispanic/Latino
34 Participants
n=5 Participants
30 Participants
n=7 Participants
35 Participants
n=5 Participants
99 Participants
n=4 Participants
Race/Ethnicity, Customized
Missing
0 Participants
n=5 Participants
0 Participants
n=7 Participants
1 Participants
n=5 Participants
1 Participants
n=4 Participants
Region of Enrollment
United States
36 participants
n=5 Participants
34 participants
n=7 Participants
36 participants
n=5 Participants
106 participants
n=4 Participants

PRIMARY outcome

Timeframe: 12 weeks

The primary endpoint, tolerability of SRX246, was assessed by the number of completers in each group.

Outcome measures

Outcome measures
Measure
SRX246 120mg BID
n=36 Participants
SRX246 capsules, administered orally, in divided doses twice daily SRX246
SRX246 160mg BID
n=34 Participants
SRX246 capsules, administered orally, in divided doses twice daily SRX246
Placebo
n=36 Participants
Placebo capsules, administered orally, in divided doses twice daily Placebo
Tolerability of SRX246
25 Participants
27 Participants
30 Participants

SECONDARY outcome

Timeframe: 12 weeks

The Safety of SRX246 was assessed by the number of participants who experience an adverse event.

Outcome measures

Outcome measures
Measure
SRX246 120mg BID
n=36 Participants
SRX246 capsules, administered orally, in divided doses twice daily SRX246
SRX246 160mg BID
n=34 Participants
SRX246 capsules, administered orally, in divided doses twice daily SRX246
Placebo
n=36 Participants
Placebo capsules, administered orally, in divided doses twice daily Placebo
Safety of SRX246
29 Participants
30 Participants
26 Participants

Adverse Events

SRX246 120mg BID

Serious events: 5 serious events
Other events: 29 other events
Deaths: 0 deaths

SRX246 160mg BID

Serious events: 0 serious events
Other events: 30 other events
Deaths: 0 deaths

Placebo

Serious events: 0 serious events
Other events: 26 other events
Deaths: 0 deaths

Serious adverse events

Serious adverse events
Measure
SRX246 120mg BID
n=36 participants at risk
SRX246 capsules, administered orally, in divided doses twice daily. This group includes those participants that were enrolled and randomized to the group assigned to receive 120mg BID throughout the study. The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of these 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.
SRX246 160mg BID
n=34 participants at risk
SRX246 capsules, administered orally, in divided doses twice daily. This group includes those participants that were enrolled and randomized to the group assigned to receive 160mg BID throughout the study. The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of those 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.
Placebo
n=36 participants at risk
Placebo capsules, administered orally, in divided doses twice daily
Cardiac disorders
Angina pectoris
2.8%
1/36 • Number of events 1 • From first dose of study drug to last date of patient follow-up at end of study (an average of 12-weeks)
The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of those 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.
0.00%
0/34 • From first dose of study drug to last date of patient follow-up at end of study (an average of 12-weeks)
The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of those 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.
0.00%
0/36 • From first dose of study drug to last date of patient follow-up at end of study (an average of 12-weeks)
The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of those 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.
Musculoskeletal and connective tissue disorders
Ankle fracture
2.8%
1/36 • Number of events 1 • From first dose of study drug to last date of patient follow-up at end of study (an average of 12-weeks)
The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of those 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.
0.00%
0/34 • From first dose of study drug to last date of patient follow-up at end of study (an average of 12-weeks)
The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of those 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.
0.00%
0/36 • From first dose of study drug to last date of patient follow-up at end of study (an average of 12-weeks)
The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of those 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.
Neoplasms benign, malignant and unspecified (incl cysts and polyps)
Renal neoplasm
2.8%
1/36 • Number of events 1 • From first dose of study drug to last date of patient follow-up at end of study (an average of 12-weeks)
The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of those 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.
0.00%
0/34 • From first dose of study drug to last date of patient follow-up at end of study (an average of 12-weeks)
The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of those 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.
0.00%
0/36 • From first dose of study drug to last date of patient follow-up at end of study (an average of 12-weeks)
The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of those 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.
Psychiatric disorders
Aggression and Irritability
5.6%
2/36 • Number of events 2 • From first dose of study drug to last date of patient follow-up at end of study (an average of 12-weeks)
The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of those 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.
0.00%
0/34 • From first dose of study drug to last date of patient follow-up at end of study (an average of 12-weeks)
The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of those 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.
0.00%
0/36 • From first dose of study drug to last date of patient follow-up at end of study (an average of 12-weeks)
The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of those 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.

Other adverse events

Other adverse events
Measure
SRX246 120mg BID
n=36 participants at risk
SRX246 capsules, administered orally, in divided doses twice daily. This group includes those participants that were enrolled and randomized to the group assigned to receive 120mg BID throughout the study. The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of these 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.
SRX246 160mg BID
n=34 participants at risk
SRX246 capsules, administered orally, in divided doses twice daily. This group includes those participants that were enrolled and randomized to the group assigned to receive 160mg BID throughout the study. The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of those 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.
Placebo
n=36 participants at risk
Placebo capsules, administered orally, in divided doses twice daily
Gastrointestinal disorders
nausea
19.4%
7/36 • Number of events 13 • From first dose of study drug to last date of patient follow-up at end of study (an average of 12-weeks)
The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of those 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.
26.5%
9/34 • Number of events 13 • From first dose of study drug to last date of patient follow-up at end of study (an average of 12-weeks)
The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of those 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.
11.1%
4/36 • Number of events 4 • From first dose of study drug to last date of patient follow-up at end of study (an average of 12-weeks)
The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of those 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.
General disorders
Fatigue
8.3%
3/36 • Number of events 3 • From first dose of study drug to last date of patient follow-up at end of study (an average of 12-weeks)
The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of those 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.
14.7%
5/34 • Number of events 7 • From first dose of study drug to last date of patient follow-up at end of study (an average of 12-weeks)
The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of those 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.
5.6%
2/36 • Number of events 2 • From first dose of study drug to last date of patient follow-up at end of study (an average of 12-weeks)
The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of those 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.
Infections and infestations
Upper Respiratory Tract Infection
16.7%
6/36 • Number of events 7 • From first dose of study drug to last date of patient follow-up at end of study (an average of 12-weeks)
The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of those 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.
11.8%
4/34 • Number of events 4 • From first dose of study drug to last date of patient follow-up at end of study (an average of 12-weeks)
The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of those 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.
25.0%
9/36 • Number of events 11 • From first dose of study drug to last date of patient follow-up at end of study (an average of 12-weeks)
The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of those 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.
Injury, poisoning and procedural complications
Fall
11.1%
4/36 • Number of events 6 • From first dose of study drug to last date of patient follow-up at end of study (an average of 12-weeks)
The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of those 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.
11.8%
4/34 • Number of events 7 • From first dose of study drug to last date of patient follow-up at end of study (an average of 12-weeks)
The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of those 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.
13.9%
5/36 • Number of events 5 • From first dose of study drug to last date of patient follow-up at end of study (an average of 12-weeks)
The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of those 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.
Musculoskeletal and connective tissue disorders
Arthralgia
13.9%
5/36 • Number of events 5 • From first dose of study drug to last date of patient follow-up at end of study (an average of 12-weeks)
The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of those 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.
14.7%
5/34 • Number of events 6 • From first dose of study drug to last date of patient follow-up at end of study (an average of 12-weeks)
The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of those 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.
2.8%
1/36 • Number of events 1 • From first dose of study drug to last date of patient follow-up at end of study (an average of 12-weeks)
The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of those 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.
Nervous system disorders
headache
16.7%
6/36 • Number of events 7 • From first dose of study drug to last date of patient follow-up at end of study (an average of 12-weeks)
The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of those 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.
11.8%
4/34 • Number of events 6 • From first dose of study drug to last date of patient follow-up at end of study (an average of 12-weeks)
The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of those 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.
22.2%
8/36 • Number of events 9 • From first dose of study drug to last date of patient follow-up at end of study (an average of 12-weeks)
The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of those 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.
Psychiatric disorders
depressed mood
22.2%
8/36 • Number of events 11 • From first dose of study drug to last date of patient follow-up at end of study (an average of 12-weeks)
The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of those 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.
23.5%
8/34 • Number of events 9 • From first dose of study drug to last date of patient follow-up at end of study (an average of 12-weeks)
The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of those 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.
11.1%
4/36 • Number of events 6 • From first dose of study drug to last date of patient follow-up at end of study (an average of 12-weeks)
The data are reported based on 3 arms: SRX246 120mg, SRX246 160mg and Placebo. All subjects were randomized at the beginning of the study to one of those 3 arms. Thus, the data are displayed this way, even though all participants randomized to the SRX246 arms received a starting dose of SRX246 80mg, then escalated to SRX246 120mg, and then the group that was randomized to the SRX246 160mg was dose escalated.

Additional Information

Neal Simon, PhD

Azevan Pharmaceuticals, Inc.

Phone: (610) 419-1057

Results disclosure agreements

  • Principal investigator is a sponsor employee
  • Publication restrictions are in place