Study of Acute Uncomplicated Seasonal Influenza A in Adult Subjects

NCT ID: NCT02342249

Last Updated: 2025-02-04

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE2

Total Enrollment

292 participants

Study Classification

INTERVENTIONAL

Study Start Date

2014-12-11

Study Completion Date

2016-05-25

Brief Summary

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The purpose of this study is to evaluate the antiviral effect, as measured by viral titer in nasal secretions in adults with acute uncomplicated seasonal influenza A following administration of VX-787.

Detailed Description

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Conditions

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Influenza A

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

QUADRUPLE

Participants Caregivers Investigators Outcome Assessors

Study Groups

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VX-787 Placebo BID + Oseltamivir Placebo BID

Subjects will receive 10 doses of matching placebo of VX-787 and Oseltamivir twice daily (BID) with approximately 12 hour (+/- 2) intervals, over 5-6 days.

Group Type PLACEBO_COMPARATOR

Placebo

Intervention Type DRUG

Subjects will receive matching placebo of Oseltamivir

VX-787 300 mg BID + Oseltamivir Placebo BID

Subjects will receive 10 doses of VX-787 300 milligram (mg) tablet along with matching placebo of Oseltamivir twice daily (BID) with approximately 12 hour (+/- 2) intervals, over 5-6 days.

Group Type ACTIVE_COMPARATOR

VX-787 300 mg

Intervention Type DRUG

A oral dose of 300 mg VX-787 tablet will be administered over 5-6 days.

Placebo

Intervention Type DRUG

Subjects will receive matching placebo of Oseltamivir

VX-787 600 mg BID + Oseltamivir Placebo BID

Subjects will receive 10 doses of VX-787 600 mg (2\*300 mg tablets) along with matching placebo of Oseltamivir twice daily (BID) with approximately 12 hour (+/- 2) intervals, over 5-6 days.

Group Type ACTIVE_COMPARATOR

VX-787 600 mg

Intervention Type DRUG

A oral dose of VX-787 600 mg (formulated as 2\*300 mg tablets) will be administered over 5-6 days.

Placebo

Intervention Type DRUG

Subjects will receive matching placebo of Oseltamivir

VX-787 600 mg BID + Oseltamivir 75 mg BID

Subjects will receive 10 doses of VX-787 600 mg tablets (2\*300 mg tablets) along with 75 mg Oseltamivir capsule twice daily (BID) with approximately 12 hour (+/- 2) intervals, over 5-6 days.

Group Type ACTIVE_COMPARATOR

VX-787 600 mg

Intervention Type DRUG

A oral dose of VX-787 600 mg (formulated as 2\*300 mg tablets) will be administered over 5-6 days.

Oseltamivir 75 mg

Intervention Type DRUG

A oral dose of 75 mg Oseltamivir capsule will be administered over 5-6 days.

Interventions

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VX-787 300 mg

A oral dose of 300 mg VX-787 tablet will be administered over 5-6 days.

Intervention Type DRUG

VX-787 600 mg

A oral dose of VX-787 600 mg (formulated as 2\*300 mg tablets) will be administered over 5-6 days.

Intervention Type DRUG

Oseltamivir 75 mg

A oral dose of 75 mg Oseltamivir capsule will be administered over 5-6 days.

Intervention Type DRUG

Placebo

Subjects will receive matching placebo of Oseltamivir

Intervention Type DRUG

Other Intervention Names

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JNJ-63623872 JNJ-63623872

Eligibility Criteria

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Inclusion Criteria

1. Willing and able to comply with the NP swab procedure
2. Subject will sign and date an informed consent form (ICF)
3. Presenting to the clinic with symptoms suggestive of a diagnosis of acute influenza. Symptoms include oral temperature ≥38°C (100.4°F) within the prior 24 hours, at least 1 respiratory symptom AND at least 1 systemic symptom.
4. Understand that no study treatment will be provided to subjects in Part A but that they are free to receive any treatment considered appropriate by their physician

Part B

1. Willing and able to comply with study requirements including treatment plan, study restrictions, laboratory tests, contraceptive guidelines, and other study procedures
2. Subject will sign and date an ICF
3. Present to the clinic with symptoms suggestive of a diagnosis of acute influenza. Symptoms include documented oral temperature ≥38°C (100.4°F) any time during the screening process, at least 1 respiratory symptom AND at least 1 systemic symptom, both scored as at least "moderate".
4. The time of onset of flu-like symptoms to the time anticipated for the start of treatment must be ≤48 hours. Onset of symptoms is defined as the first time (within 1 hour) the subject becomes aware of respiratory or systemic symptoms compatible with the flu or experiences an oral temperature ≥38°C (100.4°F)
5. Positive Rapid Influenza Diagnostic Test for influenza type A
6. Body mass index (BMI) of 18.0 to 33.0 kg/m2, inclusive, and a total body weight \>50 kg

Exclusion Criteria

1. History of any illness or any clinical condition that, in the opinion of the investigator or the subject's general practitioner, might confound the results of the study or pose an additional risk in administering study drug(s) to the subject.
2. Any condition possibly affecting drug absorption (e.g., gastrectomy, cholecystectomy, or other gastrointestinal tract surgery, except appendectomy).
3. Immunized (intranasal or injected vaccine) against influenza in the 6 months before study entry.
4. At Screening, an ECG that is abnormal and deemed by the investigator(s) to be clinically significant.
5. For female subjects: Pregnant or nursing subjects and female subjects of childbearing potential who are unwilling or unable to use an acceptable method of contraception as outlined in this protocol.
6. For male subjects, unwilling to comply with contraception requirements as outlined in the study protocol.
7. Blood donation (of approximately 1 pint \[500 mL\] or more) within 56 days before the first study drug dose.
8. Use of the following medications:

* Influenza antiviral medication (oseltamivir, zanamivir, rimantidine, or amantadine) within 14 days or ribavirin within 6 months of screening.
* Substrates of OATP1B1 and/or OATP1B3, including atrasentan, bosentan, ezetimibe, glyburide, irinotecan, repaglinide, rifampin, telmisartan, valsartan, and olmesartan, from Day 1 through the last dose of study drug. "Statins" (i.e., HMG CoA reductase inhibitors) may be continued, but subjects should be cautioned and observed for potential "statin"-related toxicity. Alternatively, subjects can abstain from statins for the duration of study drug dosing.
* Strong inhibitors or inducers of CYP3A metabolism, including carbamazepine, clarithromycin, HIV and HCV protease inhibitors, itraconazole, ketoconazole, nefazodone, phenytoin, posaconazole, rifampin, St. John's wort, telithromycin, and voriconazole from 2 weeks prior to the first dose of study drug until the last PK sample is collected on Day 8.
* An investigational drug or device 30 days before the first dose of study drug, 5 half lives before the first dose of study drug, or time determined by local requirements, whichever is longest.
9. History of excessive alcohol consumption.
10. History of known or current usage of drugs of abuse.
11. Hospitalized subjects and subjects with bacterial infections requiring systemic antibacterial agents at the time of screening.
Minimum Eligible Age

18 Years

Maximum Eligible Age

64 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Janssen Pharmaceuticals

INDUSTRY

Sponsor Role collaborator

Janssen Research & Development, LLC

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Janssen Research & Development, LLC Clinical Trial

Role: STUDY_DIRECTOR

Janssen Research & Development, LLC

Locations

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Athens, Alabama, United States

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Birmingham, Alabama, United States

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Gulf Shores, Alabama, United States

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Huntsville, Alabama, United States

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Scottsboro, Alabama, United States

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Harrisburg, Arkansas, United States

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Phoenix, Arkansas, United States

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Anaheim, California, United States

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Burbank, California, United States

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Canoga Park, California, United States

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Chula Vista, California, United States

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El Cajon, California, United States

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Encino, California, United States

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Fresno, California, United States

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Garden Grove, California, United States

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Harbor City, California, United States

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Huntington Beach, California, United States

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La Mesa, California, United States

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Lomita, California, United States

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Long Beach, California, United States

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Norwalk, California, United States

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Oakland, California, United States

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Oceanside, California, United States

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Paramount, California, United States

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San Diego, California, United States

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Santa Monica, California, United States

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Tustin, California, United States

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Upland, California, United States

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Colorado Springs, Colorado, United States

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Northglenn, Colorado, United States

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Washington D.C., District of Columbia, United States

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Boca Raton, Florida, United States

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Boynton Beach, Florida, United States

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Bradenton, Florida, United States

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Brooksville, Florida, United States

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Chiefland, Florida, United States

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Clearwater, Florida, United States

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Coral Gables, Florida, United States

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Doral, Florida, United States

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Edgewater, Florida, United States

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Fort Myers, Florida, United States

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Hialeah, Florida, United States

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Homestead, Florida, United States

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Jacksonville, Florida, United States

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Kissimmee, Florida, United States

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Lake Worth, Florida, United States

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Lakeland, Florida, United States

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Long Beach Resort, Florida, United States

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Miami, Florida, United States

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New Port Richey, Florida, United States

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North Miami Beach, Florida, United States

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Orlando, Florida, United States

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Ormond Beach, Florida, United States

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Pembroke Pines, Florida, United States

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Sarasota, Florida, United States

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St. Petersburg, Florida, United States

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Tampa, Florida, United States

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West Palm Beach, Florida, United States

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Atlanta, Georgia, United States

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Columbus, Georgia, United States

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Anderson, Idaho, United States

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Idaho Falls, Idaho, United States

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Meridian, Idaho, United States

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Anderson, Indiana, United States

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Muncie, Indiana, United States

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Newburgh, Indiana, United States

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Council Bluffs, Iowa, United States

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Overland Park, Kansas, United States

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Bardstown, Kentucky, United States

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Hazard, Kentucky, United States

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Eunice, Louisiana, United States

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Mandeville, Louisiana, United States

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Shreveport, Louisiana, United States

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Oxon Hill, Maryland, United States

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Worcester, Massachusetts, United States

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Belton, Michigan, United States

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Niles, Michigan, United States

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Troy, Michigan, United States

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St Louis, Missouri, United States

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Fremont, Nebraska, United States

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Las Vegas, Nevada, United States

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Berlin, New Jersey, United States

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Brooklyn, New York, United States

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New York, New York, United States

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Rochester, New York, United States

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Rosedale, New York, United States

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Advance, North Carolina, United States

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Hickory, North Carolina, United States

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Morehead City, North Carolina, United States

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Morganton, North Carolina, United States

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Salisbury, North Carolina, United States

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Akron, Ohio, United States

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Dayton, Ohio, United States

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Hilliard, Ohio, United States

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Huber Heights, Ohio, United States

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Tulsa, Oklahoma, United States

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Harleysville, Pennsylvania, United States

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Jenkintown, Pennsylvania, United States

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Philadelphia, Pennsylvania, United States

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Warminster, Pennsylvania, United States

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East Providence, Rhode Island, United States

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Johnston, Rhode Island, United States

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Greer, South Carolina, United States

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Laurens, South Carolina, United States

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Mt. Pleasant, South Carolina, United States

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Rock Hill, South Carolina, United States

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Simpsonville, South Carolina, United States

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Rapid City, South Dakota, United States

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Bristol, Tennessee, United States

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Amarillo, Texas, United States

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Arlington, Texas, United States

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Austin, Texas, United States

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Baytown, Texas, United States

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Carrollton, Texas, United States

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Corpus Christi, Texas, United States

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Dallas, Texas, United States

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Fort Worth, Texas, United States

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Houston, Texas, United States

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Humble, Texas, United States

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Katy, Texas, United States

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Plano, Texas, United States

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San Antonio, Texas, United States

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Tomball, Texas, United States

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Clinton, Utah, United States

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Salt Lake City, Utah, United States

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South Jordan, Utah, United States

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Alexandria, Virginia, United States

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La Crosse, Wisconsin, United States

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Milwaukee, Wisconsin, United States

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Borgerhout, , Belgium

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Linkebeek, , Belgium

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Massemen, , Belgium

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Wichelen, , Belgium

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Sofia, , Bulgaria

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Veliko Tarnovo, , Bulgaria

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Calgary, Alberta, Canada

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West Vancouver, British Columbia, Canada

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Mount Pearl, Newfoundland and Labrador, Canada

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Brampton, Ontario, Canada

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Newmarket, Ontario, Canada

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Toronto, Ontario, Canada

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Mirabel, Quebec, Canada

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Montreal, Quebec, Canada

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Saint-Jérôme, Quebec, Canada

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Trois-Rivières, Quebec, Canada

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Paide, , Estonia

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Saku, , Estonia

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Tallinn, , Estonia

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Tartu, , Estonia

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Võru, , Estonia

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Berlin, , Germany

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Essen, , Germany

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Goch, , Germany

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Hamburg, , Germany

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Stuhr, , Germany

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Balvi, , Latvia

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Daugavpils, , Latvia

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Jelgava, , Latvia

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Jēkabpils, , Latvia

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Kuldīga, , Latvia

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Lielvārde, , Latvia

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Riga, , Latvia

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Toa Baja, , Puerto Rico

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Boksburg, , South Africa

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Breyten, , South Africa

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Cape Town, , South Africa

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Durban, , South Africa

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Johannesburg, , South Africa

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Kempton Park, , South Africa

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Krugersdorp, , South Africa

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Middelburg, , South Africa

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Moloto South, , South Africa

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Pretoria, , South Africa

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Thabazimbi, , South Africa

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Vanderbijlpark, , South Africa

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Worcester, , South Africa

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Countries

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United States Belgium Bulgaria Canada Estonia Germany Latvia Puerto Rico South Africa

References

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Finberg RW, Lanno R, Anderson D, Fleischhackl R, van Duijnhoven W, Kauffman RS, Kosoglou T, Vingerhoets J, Leopold L. Phase 2b Study of Pimodivir (JNJ-63623872) as Monotherapy or in Combination With Oseltamivir for Treatment of Acute Uncomplicated Seasonal Influenza A: TOPAZ Trial. J Infect Dis. 2019 Mar 15;219(7):1026-1034. doi: 10.1093/infdis/jiy547.

Reference Type DERIVED
PMID: 30428049 (View on PubMed)

Other Identifiers

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CR107745

Identifier Type: -

Identifier Source: org_study_id

VX-787FLZ2001

Identifier Type: OTHER

Identifier Source: secondary_id

VX14-787-103

Identifier Type: OTHER

Identifier Source: secondary_id

2014-004068-39

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

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