Trial Outcomes & Findings for Pharmacokinetics, Safety, and Tolerability Study of the Pen and PFS of SB5 in Healthy Subjects (NCT NCT02326233)

NCT ID: NCT02326233

Last Updated: 2019-03-18

Results Overview

Recruitment status

COMPLETED

Study phase

PHASE1

Target enrollment

190 participants

Primary outcome timeframe

0, 24, 48, 96, 120, 144, 168, 216, 264, 336, 408, 504, 600, 696, 840, 1008, and 1344 h postdose

Results posted on

2019-03-18

Participant Flow

Participant milestones

Participant milestones
Measure
Pen of SB5
Pen of SB5, single-dose of 40 mg via subcutaneous injection (study drug) Pen of SB5
PFS of SB5
PFS of SB5, single-dose of 40 mg via subcutaneous injection (reference drug) PFS of SB5
Overall Study
STARTED
95
95
Overall Study
COMPLETED
95
94
Overall Study
NOT COMPLETED
0
1

Reasons for withdrawal

Withdrawal data not reported

Baseline Characteristics

Pharmacokinetics, Safety, and Tolerability Study of the Pen and PFS of SB5 in Healthy Subjects

Baseline characteristics by cohort

Baseline characteristics by cohort
Measure
Pen of SB5
n=95 Participants
Pen of SB5, single-dose of 40 mg via subcutaneous injection (study drug) Pen of SB5
PFS of SB5
n=95 Participants
PFS of SB5, single-dose of 40 mg via subcutaneous injection (reference drug) PFS of SB5
Total
n=190 Participants
Total of all reporting groups
Age, Continuous
31.2 years
STANDARD_DEVIATION 10.58 • n=5 Participants
30.5 years
STANDARD_DEVIATION 11.41 • n=7 Participants
30.8 years
STANDARD_DEVIATION 10.98 • n=5 Participants
Sex: Female, Male
Female
9 Participants
n=5 Participants
10 Participants
n=7 Participants
19 Participants
n=5 Participants
Sex: Female, Male
Male
86 Participants
n=5 Participants
85 Participants
n=7 Participants
171 Participants
n=5 Participants
Ethnicity (NIH/OMB)
Hispanic or Latino
5 Participants
n=5 Participants
3 Participants
n=7 Participants
8 Participants
n=5 Participants
Ethnicity (NIH/OMB)
Not Hispanic or Latino
90 Participants
n=5 Participants
92 Participants
n=7 Participants
182 Participants
n=5 Participants
Ethnicity (NIH/OMB)
Unknown or Not Reported
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
Race (NIH/OMB)
American Indian or Alaska Native
1 Participants
n=5 Participants
1 Participants
n=7 Participants
2 Participants
n=5 Participants
Race (NIH/OMB)
Asian
6 Participants
n=5 Participants
8 Participants
n=7 Participants
14 Participants
n=5 Participants
Race (NIH/OMB)
Native Hawaiian or Other Pacific Islander
1 Participants
n=5 Participants
4 Participants
n=7 Participants
5 Participants
n=5 Participants
Race (NIH/OMB)
Black or African American
3 Participants
n=5 Participants
1 Participants
n=7 Participants
4 Participants
n=5 Participants
Race (NIH/OMB)
White
78 Participants
n=5 Participants
80 Participants
n=7 Participants
158 Participants
n=5 Participants
Race (NIH/OMB)
More than one race
6 Participants
n=5 Participants
1 Participants
n=7 Participants
7 Participants
n=5 Participants
Race (NIH/OMB)
Unknown or Not Reported
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
Height (cm)
177.63 cm
STANDARD_DEVIATION 7.753 • n=5 Participants
177.89 cm
STANDARD_DEVIATION 7.814 • n=7 Participants
177.76 cm
STANDARD_DEVIATION 7.764 • n=5 Participants

PRIMARY outcome

Timeframe: 0, 24, 48, 96, 120, 144, 168, 216, 264, 336, 408, 504, 600, 696, 840, 1008, and 1344 h postdose

Outcome measures

Outcome measures
Measure
Pen of SB5
n=94 Participants
Pen of SB5, single-dose of 40 mg via subcutaneous injection (study drug) Pen of SB5
PFS of SB5
n=94 Participants
PFS of SB5, single-dose of 40 mg via subcutaneous injection (reference drug) PFS of SB5
Area Under the Concentration-time Curve From Time Zero to Infinity (AUCinf)
2743.2 h·μg/mL
Standard Deviation 1081.76
2503.3 h·μg/mL
Standard Deviation 1043.69

PRIMARY outcome

Timeframe: 0, 24, 48, 96, 120, 144, 168, 216, 264, 336, 408, 504, 600, 696, 840, 1008, and 1344 h postdose

Outcome measures

Outcome measures
Measure
Pen of SB5
n=94 Participants
Pen of SB5, single-dose of 40 mg via subcutaneous injection (study drug) Pen of SB5
PFS of SB5
n=94 Participants
PFS of SB5, single-dose of 40 mg via subcutaneous injection (reference drug) PFS of SB5
Area Under the Concentration-time Curve From Time Zero to the Last Quantifiable Concentration (AUClast)
2329.2 h·μg/mL
Standard Deviation 733.30
2182.2 h·μg/mL
Standard Deviation 724.98

PRIMARY outcome

Timeframe: 0, 24, 48, 96, 120, 144, 168, 216, 264, 336, 408, 504, 600, 696, 840, 1008, and 1344 h postdose

Outcome measures

Outcome measures
Measure
Pen of SB5
n=94 Participants
Pen of SB5, single-dose of 40 mg via subcutaneous injection (study drug) Pen of SB5
PFS of SB5
n=94 Participants
PFS of SB5, single-dose of 40 mg via subcutaneous injection (reference drug) PFS of SB5
Maximum Serum Concentration (Cmax)
3.803 μg/mL
Standard Deviation 1.0697
3.673 μg/mL
Standard Deviation 0.8810

SECONDARY outcome

Timeframe: 0, 24, 48, 96, 120, 144, 168, 216, 264, 336, 408, 504, 600, 696, 840, 1008, and 1344 h postdose

Outcome measures

Outcome measures
Measure
Pen of SB5
n=94 Participants
Pen of SB5, single-dose of 40 mg via subcutaneous injection (study drug) Pen of SB5
PFS of SB5
n=94 Participants
PFS of SB5, single-dose of 40 mg via subcutaneous injection (reference drug) PFS of SB5
Time to Reach Cmax (Tmax)
168.000 h
Interval 24.0 to 504.12
168.000 h
Interval 48.0 to 408.0

Adverse Events

Pen of SB5

Serious events: 1 serious events
Other events: 39 other events
Deaths: 0 deaths

PFS of SB5

Serious events: 2 serious events
Other events: 28 other events
Deaths: 0 deaths

Serious adverse events

Serious adverse events
Measure
Pen of SB5
n=95 participants at risk
Pen of SB5, single-dose of 40 mg via subcutaneous injection (study drug) Pen of SB5
PFS of SB5
n=94 participants at risk
PFS of SB5, single-dose of 40 mg via subcutaneous injection (reference drug) PFS of SB5
Injury, poisoning and procedural complications
Clavicle fracture
0.00%
0/95
1.1%
1/94 • Number of events 1
Injury, poisoning and procedural complications
Hand fracture
0.00%
0/95
1.1%
1/94 • Number of events 1
Psychiatric disorders
Schizophrenia
1.1%
1/95 • Number of events 1
0.00%
0/94

Other adverse events

Other adverse events
Measure
Pen of SB5
n=95 participants at risk
Pen of SB5, single-dose of 40 mg via subcutaneous injection (study drug) Pen of SB5
PFS of SB5
n=94 participants at risk
PFS of SB5, single-dose of 40 mg via subcutaneous injection (reference drug) PFS of SB5
General disorders
Fatigue
7.4%
7/95 • Number of events 7
1.1%
1/94 • Number of events 1
General disorders
Vessel puncture site bruise
5.3%
5/95 • Number of events 5
0.00%
0/94
Infections and infestations
Upper respiratory tract infection
15.8%
15/95 • Number of events 15
19.1%
18/94 • Number of events 19
Musculoskeletal and connective tissue disorders
Back pain
6.3%
6/95 • Number of events 7
1.1%
1/94 • Number of events 1
Nervous system disorders
Headache
6.3%
6/95 • Number of events 6
8.5%
8/94 • Number of events 10

Additional Information

Director of Clinical Trials

Samsung Bioepis Co., Ltd.

Results disclosure agreements

  • Principal investigator is a sponsor employee
  • Publication restrictions are in place