A Study of Efficacy and Safety of Intravenous Cefiderocol (S-649266) Versus Imipenem/Cilastatin in Complicated Urinary Tract Infections

NCT ID: NCT02321800

Last Updated: 2019-12-12

Study Results

Results available

Outcome measurements, participant flow, baseline characteristics, and adverse events have been published for this study.

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE2

Total Enrollment

452 participants

Study Classification

INTERVENTIONAL

Study Start Date

2015-02-05

Study Completion Date

2016-08-16

Brief Summary

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The purpose of this study was to determine the efficacy and safety of intravenous cefiderocol (S-649266) in hospitalized adults with complicated urinary tract infections caused by Gram-negative pathogens.

Detailed Description

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Conditions

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Urinary Tract Infections

Keywords

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S-649266 complicated urinary tract infection cefiderocol acute uncomplicated pyelonephritis Gram-negative pathogens imipenem/cilastatin

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

QUADRUPLE

Participants Caregivers Investigators Outcome Assessors

Study Groups

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Cefiderocol

Participants received 2 g cefiderocol by intravenous injection once every 8 hours for 7 to 14 days.

Group Type EXPERIMENTAL

Cefiderocol

Intervention Type DRUG

2000 mg intravenously every 8 hours for 7 to 14 days; dose adjustments for participants with reduced renal function (estimated CrCl ≤ 70 mL/minute) and/or body weight (\< 70 kg) included every 6-hour dosing intervals and/or reduced doses.

Imipenem/cilastatin

Participants received 1 g each of imipenem/cilastatin by intravenous injection once every 8 hours for 7 to 14 days.

Group Type ACTIVE_COMPARATOR

Imipenem/cilastatin

Intervention Type DRUG

1000 mg of each intravenously every 8 hours for 7 to 14 days; dose adjustments for participants with reduced renal function (estimated CrCl ≤ 70 mL/minute) and/or body weight (\< 70 kg) included every 6-hour dosing intervals and/or reduced doses.

Interventions

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Cefiderocol

2000 mg intravenously every 8 hours for 7 to 14 days; dose adjustments for participants with reduced renal function (estimated CrCl ≤ 70 mL/minute) and/or body weight (\< 70 kg) included every 6-hour dosing intervals and/or reduced doses.

Intervention Type DRUG

Imipenem/cilastatin

1000 mg of each intravenously every 8 hours for 7 to 14 days; dose adjustments for participants with reduced renal function (estimated CrCl ≤ 70 mL/minute) and/or body weight (\< 70 kg) included every 6-hour dosing intervals and/or reduced doses.

Intervention Type DRUG

Other Intervention Names

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FETROJA® S-649266 PRIMAXIN®

Eligibility Criteria

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Inclusion Criteria

* Hospitalized male and female patients ≥ 18 years
* Clinical diagnosis of either complicated urinary tract infections (cUTI) with or without pyelonephritis or acute uncomplicated pyelonephritis
* cUTI diagnosed with a history of ≥ 1 of the following:

* Indwelling urinary catheter or recent instrumentation of the urinary tract
* Urinary retention (caused by benign prostatic hypertrophy)
* Urinary retention of at least 100 mL or more of residual urine after voiding (neurogenic bladder)
* Obstructive uropathy
* Azotemia caused by intrinsic renal disease (blood urea nitrogen and creatinine values greater than normal laboratory values) OR Pyelonephritis and normal urinary tract anatomy, ie, acute uncomplicated pyelonephritis AND

At least 2 of the following signs or symptoms:

* Chills or rigors or warmth associated with fever (temperature greater than or equal to 38 degrees Celsius)
* Flank pain (pyelonephritis) or suprapubic/pelvic pain (cUTI)
* Nausea or vomiting
* Dysuria, urinary frequency, or urinary urgency
* Costo-vertebral angle tenderness on physical examination AND

All subjects had to have urinalysis evidence of pyuria demonstrated by 1 of the following:

* Dipstick analysis positive for leukocyte esterase
* ≥ 10 white blood cells (WBCs) per μL in unspun urine, or ≥ 10 WBCs per high power field in spun urine

* Positive urine culture within 48 hours prior to randomization containing ≥10\^5 colony forming unit (CFU)/mL of a Gram-negative uropathogen likely to be susceptible to imipenem (IPM)
* Patients who were treated previously with an empiric antibiotic other than the study drugs but failed treatment, both clinically and microbiologically, were eligible for the study if they had an identified Gram-negative uropathogen that was not susceptible to the previously used empiric treatment and likely to be susceptible to IPM
* Subjects receiving antibiotic prophylaxis for UTI who present with signs and symptoms consistent with an active new UTI

Exclusion Criteria

* Urine culture identifies only a Gram-positive pathogen and/or a Gram-negative uropathogen resistant to IPM
* Urine culture at study entry isolates more than 2 uropathogens or patient has a confirmed fungal UTI
* Asymptomatic bacteriuria, the presence of \>10\^5 CFU/mL of a uropathogen and pyuria but without local or systemic symptoms
* Patient is receiving hemodialysis or peritoneal dialysis
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Shionogi

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Shionogi Clinical Trials Administrator Clinical Support Help Line

Role: STUDY_DIRECTOR

Shionogi

Countries

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Bulgaria Croatia Czechia Georgia Germany Hungary Italy Japan Latvia Poland Romania Russia Spain United States

References

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Portsmouth S, van Veenhuyzen D, Echols R, Machida M, Ferreira JCA, Ariyasu M, Tenke P, Nagata TD. Cefiderocol versus imipenem-cilastatin for the treatment of complicated urinary tract infections caused by Gram-negative uropathogens: a phase 2, randomised, double-blind, non-inferiority trial. Lancet Infect Dis. 2018 Dec;18(12):1319-1328. doi: 10.1016/S1473-3099(18)30554-1. Epub 2018 Oct 25.

Reference Type RESULT
PMID: 30509675 (View on PubMed)

Portsmouth S, Echols R, Toyoizumi K, Tillotson G, Nagata TD. Structured patient interview to assess clinical outcomes in complicated urinary tract infections in the APEKS-cUTI study: pilot investigation. Ther Adv Infect Dis. 2021 Nov 24;8:20499361211058257. doi: 10.1177/20499361211058257. eCollection 2021 Jan-Dec.

Reference Type DERIVED
PMID: 34868583 (View on PubMed)

Wenzler E, Butler D, Tan X, Katsube T, Wajima T. Pharmacokinetics, Pharmacodynamics, and Dose Optimization of Cefiderocol during Continuous Renal Replacement Therapy. Clin Pharmacokinet. 2022 Apr;61(4):539-552. doi: 10.1007/s40262-021-01086-y. Epub 2021 Nov 18.

Reference Type DERIVED
PMID: 34792787 (View on PubMed)

Naseer S, Weinstein EA, Rubin DB, Suvarna K, Wei X, Higgins K, Goodwin A, Jang SH, Iarikov D, Farley J, Nambiar S. US Food and Drug Administration (FDA): Benefit-Risk Considerations for Cefiderocol (Fetroja(R)). Clin Infect Dis. 2021 Jun 15;72(12):e1103-e1111. doi: 10.1093/cid/ciaa1799.

Reference Type DERIVED
PMID: 33393598 (View on PubMed)

Other Identifiers

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1409R2121

Identifier Type: -

Identifier Source: org_study_id