Safety and Pharmacokinetic Study of PF-06651600 in Healthy Volunteers

NCT ID: NCT02309827

Last Updated: 2016-09-19

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

80 participants

Study Classification

INTERVENTIONAL

Study Start Date

2014-12-31

Study Completion Date

2016-04-30

Brief Summary

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This study is a first in human study of PF-06651600. PF-06651600 is being developed for treatment of inflammatory bowel disease. This study will test single and multiple doses of PF-06651600. The goal of the study is to assess the safety, tolerability, pharmacokinetics and pharmacodynamics of PF-06651600 in healthy volunteers.

Detailed Description

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Conditions

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Healthy

Study Design

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Allocation Method

RANDOMIZED

Primary Study Purpose

TREATMENT

Blinding Strategy

DOUBLE

Participants Investigators

Study Groups

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Cohort 1: PF-06651600 or Placebo

Single ascending doses of PF-06651600 or placebo to evaluate safety, tolerability and PK.

Group Type EXPERIMENTAL

PF-06651600 or Placebo

Intervention Type DRUG

PF-06651600 or placebo will be administered as an extemporaneously prepared solution in each cohort.

Cohort 2: PF-06651600 or Placebo

Single ascending doses of PF-06651600 or placebo to evaluate safety, tolerability and PK.

Group Type EXPERIMENTAL

PF-06651600 or Placebo

Intervention Type DRUG

PF-06651600 or placebo will be administered as an extemporaneously prepared solution in each cohort.

Cohort 3: PF-06651600 or Placebo

Single ascending doses and multiple ascending doses of PF-06651600 or placebo to evaluate safety, tolerability and PK.

Group Type EXPERIMENTAL

PF-06651600 or Placebo

Intervention Type DRUG

PF-06651600 or placebo will be administered as an extemporaneously prepared solution in each cohort.

Cohort 4: PF-06651600 or Placebo

Single ascending doses and multiple ascending doses of PF-06651600 or placebo to evaluate safety, tolerability and PK.

Group Type EXPERIMENTAL

PF-06651600 or Placebo

Intervention Type DRUG

PF-06651600 or placebo will be administered as an extemporaneously prepared solution in each cohort.

Cohort 5: PF-06651600 or Placebo

Single ascending doses and multiple ascending doses of PF-06651600 or placebo to evaluate safety, tolerability and PK.

Group Type EXPERIMENTAL

PF-06651600 or Placebo

Intervention Type DRUG

PF-06651600 or placebo will be administered as an extemporaneously prepared solution in each cohort.

Cohort 6: PF-06651600 or Placebo

Single ascending doses and multiple ascending doses of PF-06651600 or placebo to evaluate safety, tolerability and PK.

Group Type EXPERIMENTAL

PF-06651600 or Placebo

Intervention Type DRUG

PF-06651600 or placebo will be administered as an extemporaneously prepared solution in each cohort.

Cohort 7: PF-06651600 or Placebo

Single ascending doses and multiple ascending doses of PF-06651600 or placebo to evaluate safety, tolerability and PK.

Group Type EXPERIMENTAL

PF-06651600 or Placebo

Intervention Type DRUG

PF-06651600 or placebo will be administered as an extemporaneously prepared solution in each cohort.

Cohort 8: PF-06651600 or Placebo

Single ascending doses and multiple ascending doses of PF-06651600 or placebo to evaluate safety, tolerability and PK.

Group Type EXPERIMENTAL

PF-06651600 or Placebo

Intervention Type DRUG

PF-06651600 or placebo will be administered as an extemporaneously prepared solution in each cohort.

Cohort 9: PF-06651600 or Placebo

Multiple ascending doses of PF-06651600 or placebo to evaluate safety, tolerability and PK.

Group Type EXPERIMENTAL

PF-06651600 or Placebo

Intervention Type DRUG

PF-06651600 or placebo will be administered as an extemporaneously prepared solution in each cohort.

Interventions

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PF-06651600 or Placebo

PF-06651600 or placebo will be administered as an extemporaneously prepared solution in each cohort.

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Healthy male/female subjects between 18 and 55 years old, inclusive. Females must be of non-child bearing potential.
* BMI of 17.5 to 30.5 kg/m2; and a total body weight \>50 kg (110 lbs).
* Evidence of personally signed and dated informed consent document.
* Willing and able to comply with scheduled visits, treatment plan, lab tests and other study procedures.
* Subjects must avoid high intensity UV light exposure (eg, active sunbathing, tanning beds/booths or sunlamps) from the first dose of study drug and for the duration of the study.

Exclusion Criteria

* Evidence or history of clinically significant hematological, renal, endocrine, pulmonary, GI, cardiovascular, hepatic, psychiatric, neurologic, or allergic disease.
* Use of tobacco/nicotine containing products in excess of 5 cigarettes/day.
* History of regular alcohol consumption exceeding 14 drinks/week for females or 21 drinks/week for males.
* Screening blood pressure \>140/90 mm Hg.
* Screening laboratory abnormalities as defined by the protocol.
* Unwilling or unable to comply with the Lifestyle Guidelines as defined by the protocol.
Minimum Eligible Age

18 Years

Maximum Eligible Age

55 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

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Pfizer

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Pfizer CT.gov Call Center

Role: STUDY_DIRECTOR

Pfizer

Locations

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Pfizer Clinical Research Unit

Brussels, , Belgium

Site Status

Countries

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Belgium

References

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Saadeddin A, Purohit V, Huh Y, Wong M, Maulny A, Dowty ME, Sagawa K. Virtual Bioequivalence Assessment of Ritlecitinib Capsules with Incorporation of Observed Clinical Variability Using a Physiologically Based Pharmacokinetic Model. AAPS J. 2024 Jan 24;26(1):17. doi: 10.1208/s12248-024-00888-9.

Reference Type DERIVED
PMID: 38267790 (View on PubMed)

Wojciechowski J, S Purohit V, Huh Y, Banfield C, Nicholas T. Evolution of Ritlecitinib Population Pharmacokinetic Models During Clinical Drug Development. Clin Pharmacokinet. 2023 Dec;62(12):1765-1779. doi: 10.1007/s40262-023-01318-3. Epub 2023 Nov 2.

Reference Type DERIVED
PMID: 37917289 (View on PubMed)

Purohit V, Huh Y, Wojciechowski J, Plotka A, Salts S, Antinew J, Dimitrova A, Nicholas T. Leveraging Prior Healthy Participant Pharmacokinetic Data to Evaluate the Impact of Renal and Hepatic Impairment on Ritlecitinib Pharmacokinetics. AAPS J. 2023 Mar 28;25(3):32. doi: 10.1208/s12248-023-00792-8.

Reference Type DERIVED
PMID: 36977960 (View on PubMed)

Telliez JB, Dowty ME, Wang L, Jussif J, Lin T, Li L, Moy E, Balbo P, Li W, Zhao Y, Crouse K, Dickinson C, Symanowicz P, Hegen M, Banker ME, Vincent F, Unwalla R, Liang S, Gilbert AM, Brown MF, Hayward M, Montgomery J, Yang X, Bauman J, Trujillo JI, Casimiro-Garcia A, Vajdos FF, Leung L, Geoghegan KF, Quazi A, Xuan D, Jones L, Hett E, Wright K, Clark JD, Thorarensen A. Discovery of a JAK3-Selective Inhibitor: Functional Differentiation of JAK3-Selective Inhibition over pan-JAK or JAK1-Selective Inhibition. ACS Chem Biol. 2016 Dec 16;11(12):3442-3451. doi: 10.1021/acschembio.6b00677. Epub 2016 Nov 10.

Reference Type DERIVED
PMID: 27791347 (View on PubMed)

Related Links

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https://trialinfoemail.pfizer.com/pages/landing.aspx?StudyID=B7981001

To obtain contact information for a study center near you, click here.

Other Identifiers

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2014-004326-17

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

PF-06651600

Identifier Type: OTHER

Identifier Source: secondary_id

JAK3

Identifier Type: OTHER

Identifier Source: secondary_id

B7981001

Identifier Type: -

Identifier Source: org_study_id

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