Trial Outcomes & Findings for Open-label Study of ASP2151 in Herpes Simplex Patients (NCT NCT02209324)

NCT ID: NCT02209324

Last Updated: 2024-09-27

Results Overview

The percentage of participants achieving lesion healing by Day 8 of study treatment

Recruitment status

COMPLETED

Study phase

PHASE3

Target enrollment

275 participants

Primary outcome timeframe

8 days

Results posted on

2024-09-27

Participant Flow

Participant milestones

Participant milestones
Measure
ASP2151
200mg once daily
Overall Study
STARTED
275
Overall Study
COMPLETED
230
Overall Study
NOT COMPLETED
45

Reasons for withdrawal

Reasons for withdrawal
Measure
ASP2151
200mg once daily
Overall Study
Adverse Event
2
Overall Study
Lack of Efficacy
1
Overall Study
Lost to Follow-up
1
Overall Study
Physician Decision
3
Overall Study
Protocol Violation
14
Overall Study
Withdrawal by Subject
8
Overall Study
Clinical laboratory value is ineligible on day 1
4
Overall Study
Platelet count < LLN in Laboratory test
7
Overall Study
QT interval >-450 ms on measurement of an ECG
5

Baseline Characteristics

Open-label Study of ASP2151 in Herpes Simplex Patients

Baseline characteristics by cohort

Baseline characteristics by cohort
Measure
ASP2151
n=265 Participants
200mg once daily
Age, Categorical
<=18 years
4 Participants
n=5 Participants
Age, Categorical
Between 18 and 65 years
247 Participants
n=5 Participants
Age, Categorical
>=65 years
14 Participants
n=5 Participants
Age, Continuous
39.2 year
STANDARD_DEVIATION 12.7 • n=5 Participants
Sex: Female, Male
Female
161 Participants
n=5 Participants
Sex: Female, Male
Male
104 Participants
n=5 Participants
Ethnicity (NIH/OMB)
Hispanic or Latino
0 Participants
n=5 Participants
Ethnicity (NIH/OMB)
Not Hispanic or Latino
0 Participants
n=5 Participants
Ethnicity (NIH/OMB)
Unknown or Not Reported
265 Participants
n=5 Participants
Race (NIH/OMB)
American Indian or Alaska Native
0 Participants
n=5 Participants
Race (NIH/OMB)
Asian
0 Participants
n=5 Participants
Race (NIH/OMB)
Native Hawaiian or Other Pacific Islander
0 Participants
n=5 Participants
Race (NIH/OMB)
Black or African American
0 Participants
n=5 Participants
Race (NIH/OMB)
White
0 Participants
n=5 Participants
Race (NIH/OMB)
More than one race
0 Participants
n=5 Participants
Race (NIH/OMB)
Unknown or Not Reported
265 Participants
n=5 Participants
Region of Enrollment
Japan
265 participants
n=5 Participants
Disease type
Recurrent labial / facial herpes
191 Participants
n=5 Participants
Disease type
Recurrent genital herpes
39 Participants
n=5 Participants
Disease type
Kaposi varicelliform eruption
35 Participants
n=5 Participants

PRIMARY outcome

Timeframe: 8 days

Population: Efficacy analysis set was defined as patients who were diagnosed with labial/facial herpes or recurrent genital herpes at the time of case registration, subsequently received the study drug at least once, and had any efficacy variable measured, except for those found not to have herpes simplex after study drug administration.

The percentage of participants achieving lesion healing by Day 8 of study treatment

Outcome measures

Outcome measures
Measure
ASP2151
n=265 Participants
200mg once daily
Percentage of Participants With Healing by Day 8
194 Participants

SECONDARY outcome

Timeframe: 29 days

Population: Efficacy analysis set was defined as patients who were diagnosed with labial/facial herpes or recurrent genital herpes at the time of case registration, subsequently received the study drug at least once, and had any efficacy variable measured, except for those found not to have herpes simplex after study drug administration.

The criteria for determining healing are as follows: 1. A condition where all erythematous and papular lesions, vesicular and pustular lesions, and erosive and ulcerative lesions have been resolved, and either the complete resolution of crusts or the complete epithelialization beneath any remaining crusts has been achieved. 2. In participants where no crust has formed, a condition characterized by the epithelialization of erosions/ulcers formation in mucosal lesions and potentially other affected areas. 3. In participants where no vesicles or pustules have formed, a condition characterized by the complete resolution of all erythematous and papular lesions.

Outcome measures

Outcome measures
Measure
ASP2151
n=265 Participants
200mg once daily
Time to Healing
7 day
Interval 5.0 to 8.0

SECONDARY outcome

Timeframe: 29 days

Population: Efficacy analysis set was defined as patients who were diagnosed with labial/facial herpes or recurrent genital herpes at the time of case registration, subsequently received the study drug at least once, and had any efficacy variable measured, except for those found not to have herpes simplex after study drug administration.

The criteria for complete crust formation are outlined as follows: 1. A condition where all erythematous and papular lesions, vesicular and pustular lesions, and erosive and ulcerative lesions have been resolved, and all rashes are crusted (epithelialization beneath is not required). 2. In participants where no crust has formed, a condition characterized by the epithelialization of erosions/ulcers formation in mucosal lesions and potentially other affected areas. 3. In participants where no vesicles or pustules have formed, a condition characterized by the complete resolution of all erythematous and papular lesions.

Outcome measures

Outcome measures
Measure
ASP2151
n=265 Participants
200mg once daily
Time to Complete Crusting
6 day
Interval 5.0 to 8.0

SECONDARY outcome

Timeframe: 29 days

Population: Efficacy analysis set was defined as patients who were diagnosed with labial/facial herpes or recurrent genital herpes at the time of case registration, subsequently received the study drug at least once, and had any efficacy variable measured, except for those found not to have herpes simplex after study drug administration.

The day of viral disappearance is the first day on which the results of viral isolation continuously show 'HSV negative' until the final implementation day. The negative means that the results of the isolation and culture are negative, or the isolation and culture has not been performed due to complete crusting or healing of the lesion site.

Outcome measures

Outcome measures
Measure
ASP2151
n=265 Participants
200mg once daily
Time to Virus Disappearance
5 day
Interval 3.0 to 6.0

Adverse Events

ASP2151

Serious events: 2 serious events
Other events: 53 other events
Deaths: 0 deaths

Serious adverse events

Serious adverse events
Measure
ASP2151
n=271 participants at risk
200mg once daily
Infections and infestations
Cellulitis of male external genitalorgan
0.37%
1/271 • 29 days
The safety analysis population consisted of 271 participants, excluding four participants who were registered but never received the investigational drug.
Reproductive system and breast disorders
Cervical dysplasia
0.37%
1/271 • 29 days
The safety analysis population consisted of 271 participants, excluding four participants who were registered but never received the investigational drug.

Other adverse events

Other adverse events
Measure
ASP2151
n=271 participants at risk
200mg once daily
Gastrointestinal disorders
Stomatitis
2.2%
6/271 • 29 days
The safety analysis population consisted of 271 participants, excluding four participants who were registered but never received the investigational drug.
Infections and infestations
Nasopharyngitis
4.1%
11/271 • 29 days
The safety analysis population consisted of 271 participants, excluding four participants who were registered but never received the investigational drug.
Infections and infestations
Folliculitis
2.2%
6/271 • 29 days
The safety analysis population consisted of 271 participants, excluding four participants who were registered but never received the investigational drug.
Investigations
Fibrin degradation products increased
7.7%
21/271 • 29 days
The safety analysis population consisted of 271 participants, excluding four participants who were registered but never received the investigational drug.
Investigations
Alpha 1 microglobulin increased
4.8%
13/271 • 29 days
The safety analysis population consisted of 271 participants, excluding four participants who were registered but never received the investigational drug.

Additional Information

Maruho Co.,Ltd. Kyoto R&D Center

Clinical Development Dept.

Phone: +81-75-325-3255

Results disclosure agreements

  • Principal investigator is a sponsor employee
  • Publication restrictions are in place