Trial Outcomes & Findings for Open-label Study to Evaluate the Safety and Tolerability of iv Lacosamide in Japanese Adults With Partial-onset Seizures (NCT NCT02192814)

NCT ID: NCT02192814

Last Updated: 2017-08-25

Results Overview

An Adverse Event (AE) is any untoward medical occurrence in a patient or clinical investigation subject administered a pharmaceutical product that does not necessarily have a causal relationship with this treatment. An AE can therefore be any unfavorable and unintended sign (including an abnormal laboratory finding), symptom, or disease temporally associated with the use of a medicinal (investigational) product, whether or not related to the medicinal (investigational) product.

Recruitment status

COMPLETED

Study phase

PHASE3

Target enrollment

9 participants

Primary outcome timeframe

During the study (Screening through End of Study (Day -1 through Day 6))

Results posted on

2017-08-25

Participant Flow

This multicenter, open-label study started recruiting in June 2014.

Participant Flow refers to the Safety Set (SS), consisting of all enrolled subjects who received at least 1 infusion of iv LCM.

Participant milestones

Participant milestones
Measure
Lacosamide (LCM)
On Day - 1, Lacosamide (LCM) oral tablets were administered in accordance with each subject's LCM dosage regimen in EP0009 (NCT01832038). The oral tablets were taken from EP0009 supply. During the Treatment Period, subjects received a 30-minute infusion of intravenous (iv) LCM twice daily, once in the morning and once in the evening, for 5 days. The daily dose of iv LCM was the same as the subject's daily dose of oral LCM in EP0009 (200 - 400 mg/day).
Overall Study
STARTED
9
Overall Study
COMPLETED
9
Overall Study
NOT COMPLETED
0

Reasons for withdrawal

Withdrawal data not reported

Baseline Characteristics

Open-label Study to Evaluate the Safety and Tolerability of iv Lacosamide in Japanese Adults With Partial-onset Seizures

Baseline characteristics by cohort

Baseline characteristics by cohort
Measure
Lacosamide (LCM)
n=9 Participants
On Day - 1, Lacosamide (LCM) oral tablets were administered in accordance with each subject's LCM dosage regimen in EP0009 (NCT01832038). The oral tablets were taken from EP0009 supply. During the Treatment Period, subjects received a 30-minute infusion of intravenous (iv) LCM twice daily, once in the morning and once in the evening, for 5 days. The daily dose of iv LCM was the same as the subject's daily dose of oral LCM in EP0009 (200 - 400 mg/day).
Age, Categorical
<=18 years
0 Participants
n=5 Participants
Age, Categorical
Between 18 and 65 years
9 Participants
n=5 Participants
Age, Categorical
>=65 years
0 Participants
n=5 Participants
Age, Continuous
26.9 years
STANDARD_DEVIATION 10.0 • n=5 Participants
Sex: Female, Male
Female
5 Participants
n=5 Participants
Sex: Female, Male
Male
4 Participants
n=5 Participants
Weight
55.99 kilogram (kg)
STANDARD_DEVIATION 13.13 • n=5 Participants
Height
159.07 centimeter (cm)
STANDARD_DEVIATION 8.63 • n=5 Participants

PRIMARY outcome

Timeframe: During the study (Screening through End of Study (Day -1 through Day 6))

Population: The Safety Set (SS) consisted of all enrolled subjects who received at least 1 infusion of iv LCM.

An Adverse Event (AE) is any untoward medical occurrence in a patient or clinical investigation subject administered a pharmaceutical product that does not necessarily have a causal relationship with this treatment. An AE can therefore be any unfavorable and unintended sign (including an abnormal laboratory finding), symptom, or disease temporally associated with the use of a medicinal (investigational) product, whether or not related to the medicinal (investigational) product.

Outcome measures

Outcome measures
Measure
Lacosamide (LCM)
n=9 Participants
On Day - 1, Lacosamide (LCM) oral tablets were administered in accordance with each subject's LCM dosage regimen in EP0009 (NCT01832038). The oral tablets were taken from EP0009 supply. During the Treatment Period, subjects received a 30-minute infusion of intravenous (iv) LCM twice daily, once in the morning and once in the evening, for 5 days. The daily dose of iv LCM was the same as the subject's daily dose of oral LCM in EP0009 (200 - 400 mg/day).
The Total Number of Subjects Experiencing at Least One Adverse Event During the Study
4 participants

PRIMARY outcome

Timeframe: During the study (Screening through End of Study (Day -1 through Day 6))

Population: The Safety Set (SS) consisted of all enrolled subjects who received at least 1 infusion of iv LCM.

An Adverse Event (AE) is any untoward medical occurrence in a patient or clinical investigation subject administered a pharmaceutical product that does not necessarily have a causal relationship with this treatment. An AE can therefore be any unfavorable and unintended sign (including an abnormal laboratory finding), symptom, or disease temporally associated with the use of a medicinal (investigational) product, whether or not related to the medicinal (investigational) product.

Outcome measures

Outcome measures
Measure
Lacosamide (LCM)
n=9 Participants
On Day - 1, Lacosamide (LCM) oral tablets were administered in accordance with each subject's LCM dosage regimen in EP0009 (NCT01832038). The oral tablets were taken from EP0009 supply. During the Treatment Period, subjects received a 30-minute infusion of intravenous (iv) LCM twice daily, once in the morning and once in the evening, for 5 days. The daily dose of iv LCM was the same as the subject's daily dose of oral LCM in EP0009 (200 - 400 mg/day).
The Total Number of Subject Withdrawal Due to Adverse Events During the Study
0 participants

SECONDARY outcome

Timeframe: 20 minutes prior infusion at Day 1

Population: The Safety Set (SS) consisted of all enrolled subjects who received at least 1 infusion of iv LCM.

Outcome measures

Outcome measures
Measure
Lacosamide (LCM)
n=9 Participants
On Day - 1, Lacosamide (LCM) oral tablets were administered in accordance with each subject's LCM dosage regimen in EP0009 (NCT01832038). The oral tablets were taken from EP0009 supply. During the Treatment Period, subjects received a 30-minute infusion of intravenous (iv) LCM twice daily, once in the morning and once in the evening, for 5 days. The daily dose of iv LCM was the same as the subject's daily dose of oral LCM in EP0009 (200 - 400 mg/day).
Plasma Trough Concentration (Ctrough) for Lacosamide (LCM) on Day 1
4.738 µg/mL
Geometric Coefficient of Variation 50.5

SECONDARY outcome

Timeframe: 20 minutes prior infusion at Day 2

Population: The Safety Set (SS) consisted of all enrolled subjects who received at least 1 infusion of iv LCM.

Outcome measures

Outcome measures
Measure
Lacosamide (LCM)
n=9 Participants
On Day - 1, Lacosamide (LCM) oral tablets were administered in accordance with each subject's LCM dosage regimen in EP0009 (NCT01832038). The oral tablets were taken from EP0009 supply. During the Treatment Period, subjects received a 30-minute infusion of intravenous (iv) LCM twice daily, once in the morning and once in the evening, for 5 days. The daily dose of iv LCM was the same as the subject's daily dose of oral LCM in EP0009 (200 - 400 mg/day).
Plasma Trough Concentration (Ctrough) for Lacosamide (LCM) on Day 2
4.004 µg/mL
Geometric Coefficient of Variation 55.4

SECONDARY outcome

Timeframe: 20 minutes prior infusion at Day 5

Population: The Safety Set (SS) consisted of all enrolled subjects who received at least 1 infusion of iv LCM.

Outcome measures

Outcome measures
Measure
Lacosamide (LCM)
n=9 Participants
On Day - 1, Lacosamide (LCM) oral tablets were administered in accordance with each subject's LCM dosage regimen in EP0009 (NCT01832038). The oral tablets were taken from EP0009 supply. During the Treatment Period, subjects received a 30-minute infusion of intravenous (iv) LCM twice daily, once in the morning and once in the evening, for 5 days. The daily dose of iv LCM was the same as the subject's daily dose of oral LCM in EP0009 (200 - 400 mg/day).
Plasma Trough Concentration (Ctrough) for Lacosamide (LCM) on Day 5
3.615 µg/mL
Geometric Coefficient of Variation 60.0

SECONDARY outcome

Timeframe: 20 minutes prior infusion at Day 1

Population: The Safety Set (SS) consisted of all enrolled subjects who received at least 1 infusion of iv LCM.

Outcome measures

Outcome measures
Measure
Lacosamide (LCM)
n=9 Participants
On Day - 1, Lacosamide (LCM) oral tablets were administered in accordance with each subject's LCM dosage regimen in EP0009 (NCT01832038). The oral tablets were taken from EP0009 supply. During the Treatment Period, subjects received a 30-minute infusion of intravenous (iv) LCM twice daily, once in the morning and once in the evening, for 5 days. The daily dose of iv LCM was the same as the subject's daily dose of oral LCM in EP0009 (200 - 400 mg/day).
Maximum Plasma Concentration (Cmax) for Lacosamide (LCM) (End of Infusion) on Day 1
10.838 µg/mL
Geometric Coefficient of Variation 46.6

SECONDARY outcome

Timeframe: 20 minutes prior infusion at Day 2

Population: The Safety Set (SS) consisted of all enrolled subjects who received at least 1 infusion of iv LCM.

Outcome measures

Outcome measures
Measure
Lacosamide (LCM)
n=9 Participants
On Day - 1, Lacosamide (LCM) oral tablets were administered in accordance with each subject's LCM dosage regimen in EP0009 (NCT01832038). The oral tablets were taken from EP0009 supply. During the Treatment Period, subjects received a 30-minute infusion of intravenous (iv) LCM twice daily, once in the morning and once in the evening, for 5 days. The daily dose of iv LCM was the same as the subject's daily dose of oral LCM in EP0009 (200 - 400 mg/day).
Maximum Plasma Concentration (Cmax) for Lacosamide (LCM) (End of Infusion) on Day 2
10.330 µg/mL
Geometric Coefficient of Variation 50.0

SECONDARY outcome

Timeframe: 20 minutes prior infusion at Day 5

Population: The Safety Set (SS) consisted of all enrolled subjects who received at least 1 infusion of iv LCM.

Outcome measures

Outcome measures
Measure
Lacosamide (LCM)
n=9 Participants
On Day - 1, Lacosamide (LCM) oral tablets were administered in accordance with each subject's LCM dosage regimen in EP0009 (NCT01832038). The oral tablets were taken from EP0009 supply. During the Treatment Period, subjects received a 30-minute infusion of intravenous (iv) LCM twice daily, once in the morning and once in the evening, for 5 days. The daily dose of iv LCM was the same as the subject's daily dose of oral LCM in EP0009 (200 - 400 mg/day).
Maximum Plasma Concentration (Cmax) for Lacosamide (LCM) (End of Infusion) on Day 5
9.621 µg/mL
Geometric Coefficient of Variation 38.8

OTHER_PRE_SPECIFIED outcome

Timeframe: From Day -1 to Day 5

No descriptive statistics have been calculated for this exploratory Outcome Measure.

Outcome measures

Outcome data not reported

Adverse Events

Lacosamide (LCM)

Serious events: 0 serious events
Other events: 4 other events
Deaths: 0 deaths

Serious adverse events

Adverse event data not reported

Other adverse events

Other adverse events
Measure
Lacosamide (LCM)
n=9 participants at risk
On Day - 1, Lacosamide (LCM) oral tablets were administered in accordance with each subject's LCM dosage regimen in EP0009 (NCT01832038). The oral tablets were taken from EP0009 supply. During the Treatment Period, subjects received a 30-minute infusion of intravenous (iv) LCM twice daily, once in the morning and once in the evening, for 5 days. The daily dose of iv LCM was be the same as the subject's current daily dose of oral LCM in EP0009 (200 - 400 mg/day).
Infections and infestations
Nasopharyngitis
11.1%
1/9 • Number of events 1 • Adverse Events (AEs) were collected from Screening Period (Day -1) until End-of-Study Period (Day 6).
Adverse Events refer to the Safety Set (SS) which constisted of all all enrolled subjects who received at least 1 infusion of iv LCM.
Gastrointestinal disorders
Abdominal pain upper
11.1%
1/9 • Number of events 1 • Adverse Events (AEs) were collected from Screening Period (Day -1) until End-of-Study Period (Day 6).
Adverse Events refer to the Safety Set (SS) which constisted of all all enrolled subjects who received at least 1 infusion of iv LCM.
Gastrointestinal disorders
Toothache
11.1%
1/9 • Number of events 1 • Adverse Events (AEs) were collected from Screening Period (Day -1) until End-of-Study Period (Day 6).
Adverse Events refer to the Safety Set (SS) which constisted of all all enrolled subjects who received at least 1 infusion of iv LCM.
Gastrointestinal disorders
Vomiting
11.1%
1/9 • Number of events 1 • Adverse Events (AEs) were collected from Screening Period (Day -1) until End-of-Study Period (Day 6).
Adverse Events refer to the Safety Set (SS) which constisted of all all enrolled subjects who received at least 1 infusion of iv LCM.
General disorders
Injection site erythema
11.1%
1/9 • Number of events 1 • Adverse Events (AEs) were collected from Screening Period (Day -1) until End-of-Study Period (Day 6).
Adverse Events refer to the Safety Set (SS) which constisted of all all enrolled subjects who received at least 1 infusion of iv LCM.
General disorders
Injection site pain
11.1%
1/9 • Number of events 1 • Adverse Events (AEs) were collected from Screening Period (Day -1) until End-of-Study Period (Day 6).
Adverse Events refer to the Safety Set (SS) which constisted of all all enrolled subjects who received at least 1 infusion of iv LCM.
Injury, poisoning and procedural complications
Procedural headache
11.1%
1/9 • Number of events 1 • Adverse Events (AEs) were collected from Screening Period (Day -1) until End-of-Study Period (Day 6).
Adverse Events refer to the Safety Set (SS) which constisted of all all enrolled subjects who received at least 1 infusion of iv LCM.
Injury, poisoning and procedural complications
Thermal burn
11.1%
1/9 • Number of events 1 • Adverse Events (AEs) were collected from Screening Period (Day -1) until End-of-Study Period (Day 6).
Adverse Events refer to the Safety Set (SS) which constisted of all all enrolled subjects who received at least 1 infusion of iv LCM.

Additional Information

UCB Clinical Trial Call Center

UCB Pharma

Phone: +1877 822

Results disclosure agreements

  • Principal investigator is a sponsor employee
  • Publication restrictions are in place

Restriction type: GT60