Dose Escalation Study of LEE011 in Combination With Buparlisib and Letrozole in HR+, HER2-negative Post-menopausal Women With Advanced Breast Cancer.

NCT ID: NCT02154776

Last Updated: 2020-12-19

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

13 participants

Study Classification

INTERVENTIONAL

Study Start Date

2014-06-27

Study Completion Date

2016-10-26

Brief Summary

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This is a multi-center, open-label, non-randomized, phase I study

Detailed Description

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Conditions

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Advanced or Metastatic Breast Cancer

Keywords

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LEE011, buparlisib, letrozole, HR +, HER2 - negative, post-menopausal, breast cancer, CDK 4/6, PI3K, MTD

Study Design

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Allocation Method

NA

Intervention Model

SINGLE_GROUP

Primary Study Purpose

OTHER

Blinding Strategy

NONE

Study Groups

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LEE011 + buparlisib + letrozole

open label, dose escalation evaluating max tolerated dose of the triple combination

Group Type EXPERIMENTAL

LEE011

Intervention Type DRUG

3 weeks on and 1 week off

Buparlisib

Intervention Type DRUG

daily

Letrozole

Intervention Type DRUG

2.5 mg daily;

Interventions

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LEE011

3 weeks on and 1 week off

Intervention Type DRUG

Buparlisib

daily

Intervention Type DRUG

Letrozole

2.5 mg daily;

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

1. Women with advanced (recurrent or metastatic) breast cancer who received no prior therapy for advanced disease.
2. Patient is postmenopausal.
3. Patient may have received ≤ 2 lines of chemotherapy for metastatic or recurrent breast cancer in the dose-escalation phase.
4. Patient has a histologically and/or cytologically confirmed diagnosis of estrogen-receptor positive and/or progesterone receptor positive breast cancer by local laboratory.
5. Patient has HER2-negative breast cancer defined as a negative in situ hybridization test or an IHC status of 0, 1+ or 2+. If IHC is 2+, a negative in situ hybridization (FISH, CISH, or SISH) test is required by local laboratory testing.
6. Patient must have either:

* Measurable disease, i.e., at least one measurable lesion as per RECIST 1.1 criteria or at least one predominantly lytic bone lesion

Exclusion Criteria

1. Patient who received any CDK4/6 or PI3K inhibitor.
2. Patient has active cardiac disease or a history of cardiac dysfunction including any of the following:

* History of angina pectoris, symptomatic pericarditis, or myocardial infarction within 12 months prior to study entry
* History of documented congestive heart failure (New York Heart Association functional classification III-IV)
* Documented cardiomyopathy
* Patient has a Left Ventricular Ejection Fraction (LVEF) \< 50% as determined by Multiple Gated acquisition (MUGA) scan or echocardiogram (ECHO)
* History of any cardiac arrhythmias, e.g., ventricular, supraventricular, nodal arrhythmias, or conduction abnormality in the previous 12 months.
* On screening, any of the following cardiac parameters: bradycardia (heart rate \< 50 at rest), tachycardia (heart rate \> 90 at rest), PR interval \> 220 msec, QRS interval \>109 msec, or QTcF \>450 msec.

Systolic blood pressure \>160 or \<90 mmHg
3. Patient is currently receiving any of the following medications:

* That are known strong inducers or inhibitors of CYP3A4.
* That have a known risk to prolong the QT interval or induce Torsades de Pointes.
* That have a narrow therapeutic window and are predominantly metabolized through CYP3A4.
4. Certain scores on an anxiety and depression mood questionnaires
Minimum Eligible Age

18 Years

Eligible Sex

FEMALE

Accepts Healthy Volunteers

No

Sponsors

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Novartis Pharmaceuticals

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Novartis Pharmaceuticals

Role: STUDY_DIRECTOR

Novartis Pharmaceuticals

Locations

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University of California at Los Angeles UCLA SC

Los Angeles, California, United States

Site Status

Horizon Oncology Center SC

Lafayette, Indiana, United States

Site Status

Medical University of South Carolina SC

Charleston, South Carolina, United States

Site Status

South Texas Accelerated Research Therapeutics SC

San Antonio, Texas, United States

Site Status

University of Utah / Huntsman Cancer Institute SC-3

Salt Lake City, Utah, United States

Site Status

Novartis Investigative Site

Madrid, , Spain

Site Status

Countries

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United States Spain

Related Links

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https://www.novctrd.com/ctrdweb/trialresult/trialresults/pdf?trialResultId=16810

Results for CLEE011A2112C can be found on the Novartis Clinical Trial Results Website

Other Identifiers

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CLEE011A2112C

Identifier Type: -

Identifier Source: org_study_id