To Assess the Pharmacokinetics, Safety and Tolerability of Selumetinib in Renal Impaired Subjects and Healthy Subjects

NCT ID: NCT02063204

Last Updated: 2015-06-30

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

24 participants

Study Classification

INTERVENTIONAL

Study Start Date

2014-03-31

Study Completion Date

2014-07-31

Brief Summary

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A study to assess the pharmacokinetics, safety and tolerability of Selumetinib (AZD6244, ARRY-142886) in subjects with renal impairment and healthy subjects

Detailed Description

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An open label study to assess the pharmacokinetics, safety and tolerability of 50 mg single oral dose of Selumetinib (AZD6244, ARRY-142886) in subjects with renal impairment and healthy subjects

Conditions

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Solid Tumours

Keywords

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Phase I, healthy, pharmacokinetics, renal impairment

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

BASIC_SCIENCE

Blinding Strategy

NONE

Study Groups

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HV selumetinib Stage 1

Healthy volunteer (HV)group to receive selumetinib 50mg (2x25mg) orally

Group Type EXPERIMENTAL

selumetinib

Intervention Type DRUG

selumetinib 50 mg (2x25mg) administered by mouth as capsules

ESRD selumetinib Stage 1

End stage renal disease (ESRD)patients to recieve selumetinib 50mg (2x25mg) orally

Group Type EXPERIMENTAL

selumetinib

Intervention Type DRUG

selumetinib 50 mg (2x25mg) administered by mouth as capsules

Selumetinib stage 2

If deemed necessary patients with mild and/or moderate and/or severe renal impairment will recieve selumetinib 50mg(2x25mg) orally

Group Type EXPERIMENTAL

selumetinib

Intervention Type DRUG

selumetinib 50 mg (2x25mg) administered by mouth as capsules

Interventions

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selumetinib

selumetinib 50 mg (2x25mg) administered by mouth as capsules

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

1. Male and female (non childbearing potential) subjects aged 18 years or more with suitable veins for cannulation or repeated venipuncture.
2. Have a weight of at least 50 kg (110 lbs) and body mass index (BMI) between 18 and 40 kg/m2, inclusive.

Inclusion healthy volunteers only:
3. Must be in good health as determined by a medical history, physical examination, 12 lead ECG, clinical laboratory evaluations, and an ophthalmic examination performed before the administration of the investigational product.

Inclusion renal impaired patients only:
4. Stable renal function

Exclusion Criteria

1. Subjects of Japanese or non Japanese Asian ethnicity.
2. Any one parent or grandparent (maternal or paternal) is Japanese or non-Japanese Asian (e.g. China, Taiwan, Korea, Philippines, Thailand, Vietnam and Malaysia). Asian Indians are acceptable.
3. Subjects who smoke more than 10 cigarettes or the equivalent in tobacco per day
4. In the opinion of the investigator, any evidence of additional severe or uncontrolled systemic disease (eg, currently unstable or uncompensated hepatic, cardiovascular, or respiratory disease) or laboratory finding, physical examination, hematology, clinical chemistry, urinalysis, vital signs, or 12-lead ECG that makes it undesirable for the subject to participate in the study.

Exclusion renal impaired patients only:
5. Subjects with an active renal transplant (subjects who have previously received a renal transplant and are currently undergoing dialysis due to transplant failure may be enrolled).
6. Acute coronary syndrome within 6 months prior to administration of the investigational product.
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

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AstraZeneca

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Thomas C Marbury, MD

Role: PRINCIPAL_INVESTIGATOR

Orlando Clinical Research Centre, US

Ian Smith, MD

Role: STUDY_DIRECTOR

Astrazeneca United kingdom

Locations

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Research Site

Orlando, Florida, United States

Site Status

Countries

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United States

Related Links

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Other Identifiers

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D1532C00081

Identifier Type: -

Identifier Source: org_study_id