A Study in Cancer Patients With Hepatic Impairment to Evaluate the Pharmacokinetics and Safety of NKTR-102 (Etirinotecan Pegol)

NCT ID: NCT01991678

Last Updated: 2017-10-06

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

25 participants

Study Classification

INTERVENTIONAL

Study Start Date

2013-11-30

Study Completion Date

2017-09-30

Brief Summary

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The purpose of this study is to investigate the PK and safety of NKTR-102 in patients with mild, moderate, or severe hepatic impairment.

Detailed Description

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Safety and PK data from patients with mild, moderate, or severe hepatic impairment will be compared with a control group consisting of patients with normal hepatic function.

Conditions

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Advanced or Metastatic Solid Tumors in Patients With Hepatic Impairment

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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normal hepatic function

12 Patients will receive a 90-minute IV infusion

Group Type EXPERIMENTAL

145 mg/m2 NKTR 102

Intervention Type DRUG

mild hepatic dysfunction

6 Patients will receive a 90-minute IV infusion

Group Type EXPERIMENTAL

120 mg/m2 NKTR 102

Intervention Type DRUG

severe hepatic dysfunction

6 Patients will receive a 90-minute IV infusion

Group Type EXPERIMENTAL

50 mg/m2 NKTR 102

Intervention Type DRUG

Interventions

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145 mg/m2 NKTR 102

Intervention Type DRUG

120 mg/m2 NKTR 102

Intervention Type DRUG

50 mg/m2 NKTR 102

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Relapsed or progressive advanced solid tumor malignancies
* Measurable or non-measurable disease
* Eastern Cooperative Oncology Group (ECOG) performance status of 0-2
* Life expectancy greater than 3 months
* Resolution of all acute toxic effects of prior chemotherapy, and other cancer treatments
* Adequate bone morrow and kidney function
* No signs of decompensated liver cirrhosis or ascites requiring therapeutic paracentesis
* Agree to use adequate contraception

Exclusion Criteria

* Previous chemotherapy, immunotherapy, chemo-embolization, targeted therapy or investigational agent for malignancy within 4 weeks prior to day 1
* Cytochrome P450 CYP3A4 inducers and inhibitors within 4 weeks prior to day 1
* Intake of grapefruit, grapefruit juice, Seville oranges, or other products containing grapefruit or Seville oranges within 14 days prior to day 1
* UGT1A1 genotype of TA 7 in both alleles (homozygous UGT1A1\*28) or TA 8 in either one or both alleles (hetero- or homozygous for UGT1A1\*37)
* Major surgery within 4 weeks prior to day 1
* Undergone a liver or other organ transplant
* Concurrent treatment with other anti-cancer therapy
* Untreated central nervous system metastases
* Ongoing or active infection
* Chronic or acute GI disorders resulting in diarrhea
* Pregnancy or lactation
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Nektar Therapeutics

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Ivan Gergel, MD

Role: STUDY_DIRECTOR

Nektar Therapeutics

Locations

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USC/LA County

Los Angeles, California, United States

Site Status

UCSF Helen Diller Family Comprehensive Cancer Center

San Francisco, California, United States

Site Status

University Hospitals Case-Medical Center Seidman Cancer Center

Cleveland, Ohio, United States

Site Status

Countries

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United States

Other Identifiers

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12-102-13

Identifier Type: -

Identifier Source: org_study_id