Long Term Safety of Naldemedine

NCT ID: NCT01965652

Last Updated: 2018-04-18

Study Results

Results available

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE3

Total Enrollment

1246 participants

Study Classification

INTERVENTIONAL

Study Start Date

2013-09-24

Study Completion Date

2016-01-12

Brief Summary

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The purpose of this study is to evaluate the long-term safety of naldemedine for the treatment of constipation due to opioid therapy.

Detailed Description

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Conditions

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Opioid-induced Constipation

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

QUADRUPLE

Participants Caregivers Investigators Outcome Assessors

Study Groups

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Naldemedine

Participants received 0.2 mg naldemedine tablets orally once daily for 52 weeks.

Group Type EXPERIMENTAL

Naldemedine

Intervention Type DRUG

Naldemedine 0.2 mg tablet taken orally once a day

Placebo

Participants received matching placebo tablets orally once daily for 52 weeks.

Group Type PLACEBO_COMPARATOR

Placebo

Intervention Type DRUG

Placebo tablet taken orally once a day

Interventions

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Naldemedine

Naldemedine 0.2 mg tablet taken orally once a day

Intervention Type DRUG

Placebo

Placebo tablet taken orally once a day

Intervention Type DRUG

Other Intervention Names

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S-297995 Symproic®

Eligibility Criteria

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Inclusion Criteria

1. Subjects aged 18 to 80 years inclusive at the time of informed consent
2. Subjects must have non-malignant chronic pain treated and must have opioid induced constipation (OIC)
3. Subjects must be treated with a stable opioid regimen at a total daily dose on average of ≥ 30 mg equivalents of oral morphine sulfate
4. Subjects may or may not be on a routine laxative regimen at the time of Screening

Exclusion Criteria

1. Evidence of significant structural abnormalities of the gastrointestinal (GI) tract
2. Evidence of active medical diseases affecting bowel transit
3. History of pelvic disorders that may be a cause of constipation
4. Surgery (except for minor procedures) within 60 days of Screening
5. History of chronic constipation prior to starting analgesic medication or any potential non-opioid cause of bowel dysfunction that may be a major contributor to the constipation (e.g. mechanical GI obstruction)
6. Subjects who have never taken laxatives for the treatment of OIC
7. Current use of any prohibited medication including opioid antagonists, partial or mixed agonists/antagonists
Minimum Eligible Age

18 Years

Maximum Eligible Age

80 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Shionogi

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Shionogi Clinical Trials Administrator Clinical Support Help Line

Role: STUDY_DIRECTOR

Shionogi

Locations

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Birmingham, Alabama, United States

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Mobile, Alabama, United States

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Chandler, Arizona, United States

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Glendale, Arizona, United States

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Goodyear, Arizona, United States

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Mesa, Arizona, United States

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Phoenix, Arizona, United States

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Tucson, Arizona, United States

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Fountain Valley, California, United States

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Garden Grove, California, United States

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Glendale, California, United States

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Long Beach, California, United States

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Los Angeles, California, United States

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Oceanside, California, United States

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Sacramento, California, United States

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Santa Ana, California, United States

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Upland, California, United States

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Colorado Springs, Colorado, United States

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Boynton Beach, Florida, United States

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Brandon, Florida, United States

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Brooksville, Florida, United States

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Clearwater, Florida, United States

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Fort Myers, Florida, United States

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Jacksonville, Florida, United States

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Lake City, Florida, United States

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Lakeland, Florida, United States

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Orlando, Florida, United States

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South Miami, Florida, United States

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St. Petersburg, Florida, United States

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Tampa, Florida, United States

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Atlanta, Georgia, United States

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Blue Ridge, Georgia, United States

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Decatur, Georgia, United States

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Savannah, Georgia, United States

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Boise, Idaho, United States

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Aurora, Illinois, United States

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Bloomington, Illinois, United States

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Decatur, Illinois, United States

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Rockford, Illinois, United States

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Schaumburg, Illinois, United States

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Evansville, Indiana, United States

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Lafayette, Indiana, United States

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Valparaiso, Indiana, United States

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Augusta, Kansas, United States

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Newton, Kansas, United States

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Wichita, Kansas, United States

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Hartford, Kentucky, United States

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Eunice, Louisiana, United States

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Lake Charles, Louisiana, United States

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Mandeville, Louisiana, United States

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Brockton, Massachusetts, United States

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Fall River, Massachusetts, United States

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New Bedford, Massachusetts, United States

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Rochester, Michigan, United States

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Saginaw, Michigan, United States

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Traverse City, Michigan, United States

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Biloxi, Mississippi, United States

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Fremont, Nebraska, United States

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Omaha, Nebraska, United States

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Henderson, Nevada, United States

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Las Vegas, Nevada, United States

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Trenton, New Jersey, United States

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Albuquerque, New Mexico, United States

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New York, New York, United States

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Greensboro, North Carolina, United States

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Wilmington, North Carolina, United States

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Winston-Salem, North Carolina, United States

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Akron, Ohio, United States

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Canton, Ohio, United States

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Columbus, Ohio, United States

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Groveport, Ohio, United States

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Kettering, Ohio, United States

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Lebanon, Ohio, United States

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Marion, Ohio, United States

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Munroe Falls, Ohio, United States

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Oklahoma City, Oklahoma, United States

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Tulsa, Oklahoma, United States

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Portland, Oregon, United States

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Huntingdon Valley, Pennsylvania, United States

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Jenkintown, Pennsylvania, United States

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Lansdale, Pennsylvania, United States

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Charleston, South Carolina, United States

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Greer, South Carolina, United States

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Myrtle Beach, South Carolina, United States

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Summerville, South Carolina, United States

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Bristol, Tennessee, United States

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Milan, Tennessee, United States

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Nashville, Tennessee, United States

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Austin, Texas, United States

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Dallas, Texas, United States

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Houston, Texas, United States

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Hurst, Texas, United States

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Sugar Land, Texas, United States

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Bountiful, Utah, United States

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Salt Lake City, Utah, United States

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South Ogden, Utah, United States

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Richmond, Virginia, United States

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Bellevue, Washington, United States

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Edmonds, Washington, United States

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Adelaide, , Australia

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Bedford Park, , Australia

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Camperdown, , Australia

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Carina Heights, , Australia

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Caulfield South, , Australia

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Malvern East, , Australia

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Nambour, , Australia

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Sherwood, , Australia

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St Leonards, , Australia

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Linz, , Austria

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Vienna, , Austria

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Zams, , Austria

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London, , Canada

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Mirabel, , Canada

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Sarnia, , Canada

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Sherbrooke, , Canada

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Toronto, , Canada

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Vancouver, , Canada

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Benešov, , Czechia

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Olomouc, , Czechia

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Ostrava, , Czechia

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Pardubice, , Czechia

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Pribram V- Zdabor, , Czechia

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Glostrup Municipality, , Denmark

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Hellerup, , Denmark

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Odense, , Denmark

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Soulaine Sur Aubance, , France

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Berlin, , Germany

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Dresden, , Germany

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Halle, , Germany

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Hamburg, , Germany

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Hanover, , Germany

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Kassel, , Germany

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Leipzig, , Germany

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Lünen, , Germany

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Mainz, , Germany

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Münster, , Germany

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Stadtroda, , Germany

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Balatonfüred, , Hungary

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Budapest, , Hungary

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Debrecen, , Hungary

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Hatvan, , Hungary

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Szikszó, , Hungary

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Beersheba, , Israel

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Haifa, , Israel

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Tel Aviv, , Israel

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Tel Litwinsky, , Israel

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Asti, , Italy

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Catania, , Italy

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Chieti, , Italy

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Florence, , Italy

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Napoli, , Italy

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Rionero in Vulture, , Italy

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Roma, , Italy

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Rome, , Italy

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Chorzów, , Poland

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Gdansk, , Poland

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Katowice, , Poland

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Lublin, , Poland

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Alberton, , South Africa

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Lyttelton Centurion, , South Africa

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Muckleneuk Pretoria, , South Africa

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Pretoria West Pretoria, , South Africa

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Worcester, , South Africa

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Barcelona, , Spain

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Girona, , Spain

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Seville, , Spain

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Skene, , Sweden

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Stockholm, , Sweden

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Bath, , United Kingdom

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Belfast, , United Kingdom

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Bexhill on Sea East Sussex, , United Kingdom

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Chesterfield, , United Kingdom

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Chestfield Kent, , United Kingdom

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Daventry Northants, , United Kingdom

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Devon, , United Kingdom

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Epworth Doncaster, , United Kingdom

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Harrogate, , United Kingdom

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Hinckley, , United Kingdom

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Liverpool, , United Kingdom

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Norwich, , United Kingdom

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Oldham, , United Kingdom

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Peterborough, , United Kingdom

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Randalstown, County Antrim, , United Kingdom

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Spiro Close, Pulborough West Sussex, , United Kingdom

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Wellingborough Northamptonshire, , United Kingdom

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York, , United Kingdom

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Countries

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United States Australia Austria Canada Czechia Denmark France Germany Hungary Israel Italy Poland South Africa Spain Sweden United Kingdom

References

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Camilleri M, Hale M, Morlion B, Tack J, Webster L, Wild J. Naldemedine Improves Patient-Reported Outcomes of Opioid-Induced Constipation in Patients with Chronic Non-Cancer Pain in the COMPOSE Phase 3 Studies. J Pain Res. 2021 Jul 16;14:2179-2189. doi: 10.2147/JPR.S282738. eCollection 2021.

Reference Type DERIVED
PMID: 34295186 (View on PubMed)

Webster LR, Hale ME, Yamada T, Wild JE. A Renal Impairment Subgroup Analysis of the Safety and Efficacy of Naldemedine for the Treatment of Opioid-Induced Constipation in Patients with Chronic Non-Cancer Pain Receiving Opioid Therapy. J Pain Res. 2020 Mar 24;13:605-612. doi: 10.2147/JPR.S237833. eCollection 2020.

Reference Type DERIVED
PMID: 32280263 (View on PubMed)

Wild J, Webster L, Yamada T, Hale M. Safety and Efficacy of Naldemedine for the Treatment of Opioid-Induced Constipation in Patients with Chronic Non-Cancer Pain Receiving Opioid Therapy: A Subgroup Analysis of Patients >/= 65 Years of Age. Drugs Aging. 2020 Apr;37(4):271-279. doi: 10.1007/s40266-020-00753-2.

Reference Type DERIVED
PMID: 32086791 (View on PubMed)

Other Identifiers

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1326V9235

Identifier Type: -

Identifier Source: org_study_id

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