Trial Outcomes & Findings for The Pharmacokinetics of LEO 90105 (Calcipotriol Hydrate Plus Betamethasone Dipropionate) in Japanese Subjects With Extensive Psoriasis Vulgaris (NCT NCT01768013)

NCT ID: NCT01768013

Last Updated: 2025-03-12

Results Overview

The mean Cmax(Maximum Observed Plasma Concentration) of betamethasone dipropionate was determined.

Recruitment status

COMPLETED

Study phase

PHASE1/PHASE2

Target enrollment

13 participants

Primary outcome timeframe

Day 1

Results posted on

2025-03-12

Participant Flow

First subject first visit: 09-Jul-2012 Last subject last visit: 30-Oct-2012

Prior to treatment at Visit 1, a washout period was completed if the subject was treated or had recently been treated with anti-psoriatic treatments or other relevant medication, as defined by the exclusion criteria. The washout period could last up to a maximum of 4 weeks.

Participant milestones

Participant milestones
Measure
LEO 90105 Ointment
Subjects received once daily topical treatment with LEO 90105 (calcipotriol hydrate plus betamethasone dipropionate ointment) on all lesions on the trunk and/or limbs (excluding psoriasis on the genitals and skin folds) for 4 weeks. Subjects were supplied with an amount of medication at day 1, day 7 and day 14 such that the maximum usage of LEO 90105 could be 90 g per week.
Overall Study
STARTED
13
Overall Study
COMPLETED
13
Overall Study
NOT COMPLETED
0

Reasons for withdrawal

Withdrawal data not reported

Baseline Characteristics

The Pharmacokinetics of LEO 90105 (Calcipotriol Hydrate Plus Betamethasone Dipropionate) in Japanese Subjects With Extensive Psoriasis Vulgaris

Baseline characteristics by cohort

Baseline characteristics by cohort
Measure
LEO 90105 Ointment
n=13 Participants
Subjects received once daily topical treatment with LEO 90105 (calcipotriol hydrate plus betamethasone dipropionate ointment) on all lesions on the trunk and/or limbs (excluding psoriasis on the genitals and skin folds) for 4 weeks. Subjects were supplied with an amount of medication at day 1, day 7 and day 14 such that the maximum usage of LEO 90105 could be 90 g per week.
Age, Categorical
<=18 years
0 Participants
n=5 Participants
Age, Categorical
Between 18 and 65 years
8 Participants
n=5 Participants
Age, Categorical
>=65 years
5 Participants
n=5 Participants
Age, Continuous
54.2 years
STANDARD_DEVIATION 15.4 • n=5 Participants
Sex: Female, Male
Female
3 Participants
n=5 Participants
Sex: Female, Male
Male
10 Participants
n=5 Participants
Region of Enrollment
Japan
13 participants
n=5 Participants

PRIMARY outcome

Timeframe: Day 1

The mean Cmax(Maximum Observed Plasma Concentration) of betamethasone dipropionate was determined.

Outcome measures

Outcome measures
Measure
LEO 90105 Ointment
n=13 Participants
Subjects received once daily topical treatment with LEO 90105 (calcipotriol hydrate plus betamethasone dipropionate ointment) on all lesions on the trunk and/or limbs (excluding psoriasis on the genitals and skin folds) for 4 weeks. Subjects were supplied with an amount of medication at day 1, day 7 and day 14 such that the maximum usage of LEO 90105 could be 90 g per week.
Pharmacokinetic: Cmax of Betamethasone Dipropionate
NA pg/mL
Standard Deviation NA
The pharmacokinetic parameter could not be reliably estimated

PRIMARY outcome

Timeframe: Day 7

The mean Cmax (Maximum Observed Plasma Concentration) of betamethasone dipropionate was determined

Outcome measures

Outcome measures
Measure
LEO 90105 Ointment
n=13 Participants
Subjects received once daily topical treatment with LEO 90105 (calcipotriol hydrate plus betamethasone dipropionate ointment) on all lesions on the trunk and/or limbs (excluding psoriasis on the genitals and skin folds) for 4 weeks. Subjects were supplied with an amount of medication at day 1, day 7 and day 14 such that the maximum usage of LEO 90105 could be 90 g per week.
Pharmacokinetic: Cmax of Betamethasone Dipropionate
NA pg/mL
Standard Deviation NA
The pharmacokinetic parameter could not be reliably estimated

PRIMARY outcome

Timeframe: Day 14

The mean Cmax (Maximum Observed Plasma Concentration) of betamethasone dipropionate was determined

Outcome measures

Outcome measures
Measure
LEO 90105 Ointment
n=13 Participants
Subjects received once daily topical treatment with LEO 90105 (calcipotriol hydrate plus betamethasone dipropionate ointment) on all lesions on the trunk and/or limbs (excluding psoriasis on the genitals and skin folds) for 4 weeks. Subjects were supplied with an amount of medication at day 1, day 7 and day 14 such that the maximum usage of LEO 90105 could be 90 g per week.
Pharmacokinetic: Cmax of Betamethasone Dipropionate
NA pg/mL
Standard Deviation NA
The pharmacokinetic parameter could not be reliably estimated

PRIMARY outcome

Timeframe: Day 1

The mean AUClast (Area under the Plasma Concentration-Time Curve from Time 0 to the Last Observed Measurable Concentration) for betamethasone dipropionate was determined

Outcome measures

Outcome measures
Measure
LEO 90105 Ointment
n=13 Participants
Subjects received once daily topical treatment with LEO 90105 (calcipotriol hydrate plus betamethasone dipropionate ointment) on all lesions on the trunk and/or limbs (excluding psoriasis on the genitals and skin folds) for 4 weeks. Subjects were supplied with an amount of medication at day 1, day 7 and day 14 such that the maximum usage of LEO 90105 could be 90 g per week.
Pharmacokinetic: AUClast of Betamethasone Dipropionate
NA h*pg/mL
Standard Deviation NA
The pharmacokinetic parameter could not be reliably estimated

PRIMARY outcome

Timeframe: Day 7

The mean AUClast (Area under the Plasma Concentration-Time Curve from Time 0 to the Last Observed Measurable Concentration) for betamethasone dipropionate was determined

Outcome measures

Outcome measures
Measure
LEO 90105 Ointment
n=13 Participants
Subjects received once daily topical treatment with LEO 90105 (calcipotriol hydrate plus betamethasone dipropionate ointment) on all lesions on the trunk and/or limbs (excluding psoriasis on the genitals and skin folds) for 4 weeks. Subjects were supplied with an amount of medication at day 1, day 7 and day 14 such that the maximum usage of LEO 90105 could be 90 g per week.
Pharmacokinetic: AUClast of Betamethasone Dipropionate
NA h*pg/mL
Standard Deviation NA
The pharmacokinetic parameter could not be reliably estimated

PRIMARY outcome

Timeframe: Day 14

The mean AUClast (Area under the Plasma Concentration-Time Curve from Time 0 to the Last Observed Measurable Concentration) for betamethasone dipropionate was determined

Outcome measures

Outcome measures
Measure
LEO 90105 Ointment
n=13 Participants
Subjects received once daily topical treatment with LEO 90105 (calcipotriol hydrate plus betamethasone dipropionate ointment) on all lesions on the trunk and/or limbs (excluding psoriasis on the genitals and skin folds) for 4 weeks. Subjects were supplied with an amount of medication at day 1, day 7 and day 14 such that the maximum usage of LEO 90105 could be 90 g per week.
Pharmacokinetic: AUClast of Betamethasone Dipropionate
NA h*pg/mL
Standard Deviation NA
The pharmacokinetic parameter could not be reliably estimated

PRIMARY outcome

Timeframe: Day 1

The mean Cmax(Maximum Observed Plasma Concentration) of betamethasone 17- propionate was determined

Outcome measures

Outcome measures
Measure
LEO 90105 Ointment
n=13 Participants
Subjects received once daily topical treatment with LEO 90105 (calcipotriol hydrate plus betamethasone dipropionate ointment) on all lesions on the trunk and/or limbs (excluding psoriasis on the genitals and skin folds) for 4 weeks. Subjects were supplied with an amount of medication at day 1, day 7 and day 14 such that the maximum usage of LEO 90105 could be 90 g per week.
Pharmacokinetic: Cmax of Betamethasone 17-propionate
218.8 pg/mL
Standard Deviation 351.01

PRIMARY outcome

Timeframe: Day 7

The mean Cmax (Maximum Observed Plasma Concentration) of betamethasone 17- propionate was determined

Outcome measures

Outcome measures
Measure
LEO 90105 Ointment
n=13 Participants
Subjects received once daily topical treatment with LEO 90105 (calcipotriol hydrate plus betamethasone dipropionate ointment) on all lesions on the trunk and/or limbs (excluding psoriasis on the genitals and skin folds) for 4 weeks. Subjects were supplied with an amount of medication at day 1, day 7 and day 14 such that the maximum usage of LEO 90105 could be 90 g per week.
Pharmacokinetic: Cmax of Betamethasone 17-propionate
101.5 pg/mL
Standard Deviation 77.551

PRIMARY outcome

Timeframe: Day 14

The mean Cmax (Maximum Observed Plasma Concentration) of betamethasone 17- propionate was determined

Outcome measures

Outcome measures
Measure
LEO 90105 Ointment
n=13 Participants
Subjects received once daily topical treatment with LEO 90105 (calcipotriol hydrate plus betamethasone dipropionate ointment) on all lesions on the trunk and/or limbs (excluding psoriasis on the genitals and skin folds) for 4 weeks. Subjects were supplied with an amount of medication at day 1, day 7 and day 14 such that the maximum usage of LEO 90105 could be 90 g per week.
Pharmacokinetic: Cmax of Betamethasone 17-propionate
116 pg/mL
Standard Deviation 64.826

PRIMARY outcome

Timeframe: Day 1

The mean AUClast (Area under the Plasma Concentration-Time Curve from Time 0 to the Last Observed Measurable Concentration) for betamethasone 17-propionate was determined

Outcome measures

Outcome measures
Measure
LEO 90105 Ointment
n=13 Participants
Subjects received once daily topical treatment with LEO 90105 (calcipotriol hydrate plus betamethasone dipropionate ointment) on all lesions on the trunk and/or limbs (excluding psoriasis on the genitals and skin folds) for 4 weeks. Subjects were supplied with an amount of medication at day 1, day 7 and day 14 such that the maximum usage of LEO 90105 could be 90 g per week.
Pharmacokinetic: AUClast of Betamethasone 17-propionate
1036.7 h*pg/mL
Standard Deviation 1885.01

PRIMARY outcome

Timeframe: Day 7

The mean AUClast (Area under the Plasma Concentration-Time Curve from Time 0 to the Last Observed Measurable Concentration) for betamethasone 17-propionate was determined

Outcome measures

Outcome measures
Measure
LEO 90105 Ointment
n=13 Participants
Subjects received once daily topical treatment with LEO 90105 (calcipotriol hydrate plus betamethasone dipropionate ointment) on all lesions on the trunk and/or limbs (excluding psoriasis on the genitals and skin folds) for 4 weeks. Subjects were supplied with an amount of medication at day 1, day 7 and day 14 such that the maximum usage of LEO 90105 could be 90 g per week.
Pharmacokinetic: AUClast of Betamethasone 17-propionate
570.92 h*pg/mL
Standard Deviation 517.107

PRIMARY outcome

Timeframe: Day 14

The mean AUClast (Area under the Plasma Concentration-Time Curve from Time 0 to the Last Observed Measurable Concentration) for betamethasone 17-propionate was determined

Outcome measures

Outcome measures
Measure
LEO 90105 Ointment
n=13 Participants
Subjects received once daily topical treatment with LEO 90105 (calcipotriol hydrate plus betamethasone dipropionate ointment) on all lesions on the trunk and/or limbs (excluding psoriasis on the genitals and skin folds) for 4 weeks. Subjects were supplied with an amount of medication at day 1, day 7 and day 14 such that the maximum usage of LEO 90105 could be 90 g per week.
Pharmacokinetic: AUClast of Betamethasone 17-propionate
634.65 h*pg/mL
Standard Deviation 467.426

PRIMARY outcome

Timeframe: Day 1

The mean Cmax (Maximum Observed Plasma Concentration) of calcipotriol was determined

Outcome measures

Outcome measures
Measure
LEO 90105 Ointment
n=13 Participants
Subjects received once daily topical treatment with LEO 90105 (calcipotriol hydrate plus betamethasone dipropionate ointment) on all lesions on the trunk and/or limbs (excluding psoriasis on the genitals and skin folds) for 4 weeks. Subjects were supplied with an amount of medication at day 1, day 7 and day 14 such that the maximum usage of LEO 90105 could be 90 g per week.
Pharmacokinetic: Cmax of Calcipotriol
107.6 pg/mL
Standard Deviation NA
The pharmacokinetic parameter could not be reliably estimated

PRIMARY outcome

Timeframe: Day 7

The mean Cmax (Maximum Observed Plasma Concentration) of calcipotriol was determined

Outcome measures

Outcome measures
Measure
LEO 90105 Ointment
n=13 Participants
Subjects received once daily topical treatment with LEO 90105 (calcipotriol hydrate plus betamethasone dipropionate ointment) on all lesions on the trunk and/or limbs (excluding psoriasis on the genitals and skin folds) for 4 weeks. Subjects were supplied with an amount of medication at day 1, day 7 and day 14 such that the maximum usage of LEO 90105 could be 90 g per week.
Pharmacokinetic: Cmax of Calcipotriol
NA pg/mL
Standard Deviation NA
The pharmacokinetic parameter could not be reliably estimated

PRIMARY outcome

Timeframe: Day 14

The mean Cmax (Maximum Observed Plasma Concentration) of calcipotriol was determined

Outcome measures

Outcome measures
Measure
LEO 90105 Ointment
n=13 Participants
Subjects received once daily topical treatment with LEO 90105 (calcipotriol hydrate plus betamethasone dipropionate ointment) on all lesions on the trunk and/or limbs (excluding psoriasis on the genitals and skin folds) for 4 weeks. Subjects were supplied with an amount of medication at day 1, day 7 and day 14 such that the maximum usage of LEO 90105 could be 90 g per week.
Pharmacokinetic: Cmax of Calcipotriol
NA pg/mL
Standard Deviation NA
The pharmacokinetic parameter could not be reliably estimated

PRIMARY outcome

Timeframe: Day 1

The mean AUClast (Area under the Plasma Concentration-Time Curve from Time 0 to the Last Observed Measurable Concentration) for calcipotriol was determined

Outcome measures

Outcome measures
Measure
LEO 90105 Ointment
n=13 Participants
Subjects received once daily topical treatment with LEO 90105 (calcipotriol hydrate plus betamethasone dipropionate ointment) on all lesions on the trunk and/or limbs (excluding psoriasis on the genitals and skin folds) for 4 weeks. Subjects were supplied with an amount of medication at day 1, day 7 and day 14 such that the maximum usage of LEO 90105 could be 90 g per week.
Pharmacokinetic: AUClast of Calcipotriol
169.6 h*pg/mL
Standard Deviation NA
The pharmacokinetic parameter could not be reliably estimated

PRIMARY outcome

Timeframe: Day 7

The mean AUClast (Area under the Plasma Concentration-Time Curve from Time 0 to the Last Observed Measurable Concentration) for calcipotriol was determined

Outcome measures

Outcome measures
Measure
LEO 90105 Ointment
n=13 Participants
Subjects received once daily topical treatment with LEO 90105 (calcipotriol hydrate plus betamethasone dipropionate ointment) on all lesions on the trunk and/or limbs (excluding psoriasis on the genitals and skin folds) for 4 weeks. Subjects were supplied with an amount of medication at day 1, day 7 and day 14 such that the maximum usage of LEO 90105 could be 90 g per week.
Pharmacokinetic: AUClast of Calcipotriol
NA h*pg/mL
Standard Deviation NA
The pharmacokinetic parameter could not be reliably estimated

PRIMARY outcome

Timeframe: Day 14

The mean AUClast (Area under the Plasma Concentration-Time Curve from Time 0 to the Last Observed Measurable Concentration) for calcipotriol was determined

Outcome measures

Outcome measures
Measure
LEO 90105 Ointment
n=13 Participants
Subjects received once daily topical treatment with LEO 90105 (calcipotriol hydrate plus betamethasone dipropionate ointment) on all lesions on the trunk and/or limbs (excluding psoriasis on the genitals and skin folds) for 4 weeks. Subjects were supplied with an amount of medication at day 1, day 7 and day 14 such that the maximum usage of LEO 90105 could be 90 g per week.
Pharmacokinetic: AUClast of Calcipotriol
NA h*pg/mL
Standard Deviation NA
The pharmacokinetic parameter could not be reliably estimated

PRIMARY outcome

Timeframe: Day 1

The mean Cmax (Maximum Observed Plasma Concentration) of MC1080 was determined

Outcome measures

Outcome measures
Measure
LEO 90105 Ointment
n=13 Participants
Subjects received once daily topical treatment with LEO 90105 (calcipotriol hydrate plus betamethasone dipropionate ointment) on all lesions on the trunk and/or limbs (excluding psoriasis on the genitals and skin folds) for 4 weeks. Subjects were supplied with an amount of medication at day 1, day 7 and day 14 such that the maximum usage of LEO 90105 could be 90 g per week.
Pharmacokinetic: Cmax of MC1080
95.35 pg/mL
Standard Deviation NA
The pharmacokinetic parameter could not be reliably estimated

PRIMARY outcome

Timeframe: Day 7

The mean Cmax (Maximum Observed Plasma Concentration) of MC1080 was determined

Outcome measures

Outcome measures
Measure
LEO 90105 Ointment
n=13 Participants
Subjects received once daily topical treatment with LEO 90105 (calcipotriol hydrate plus betamethasone dipropionate ointment) on all lesions on the trunk and/or limbs (excluding psoriasis on the genitals and skin folds) for 4 weeks. Subjects were supplied with an amount of medication at day 1, day 7 and day 14 such that the maximum usage of LEO 90105 could be 90 g per week.
Pharmacokinetic: Cmax of MC1080
57.57 pg/mL
Standard Deviation 36.218

PRIMARY outcome

Timeframe: Day 14

The mean Cmax (Maximum Observed Plasma Concentration) of MC1080 was determined

Outcome measures

Outcome measures
Measure
LEO 90105 Ointment
n=13 Participants
Subjects received once daily topical treatment with LEO 90105 (calcipotriol hydrate plus betamethasone dipropionate ointment) on all lesions on the trunk and/or limbs (excluding psoriasis on the genitals and skin folds) for 4 weeks. Subjects were supplied with an amount of medication at day 1, day 7 and day 14 such that the maximum usage of LEO 90105 could be 90 g per week.
Pharmacokinetic: Cmax of MC1080
NA pg/mL
Standard Deviation NA
The pharmacokinetic parameter could not be reliably estimated

PRIMARY outcome

Timeframe: Day 1

The mean AUClast (Area under the Plasma Concentration-Time Curve from Time 0 to the Last Observed Measurable Concentration) for MC 1080 was determined

Outcome measures

Outcome measures
Measure
LEO 90105 Ointment
n=13 Participants
Subjects received once daily topical treatment with LEO 90105 (calcipotriol hydrate plus betamethasone dipropionate ointment) on all lesions on the trunk and/or limbs (excluding psoriasis on the genitals and skin folds) for 4 weeks. Subjects were supplied with an amount of medication at day 1, day 7 and day 14 such that the maximum usage of LEO 90105 could be 90 g per week.
Pharmacokinetic: AUClast of MC1080
430.9 h*pg/mL
Standard Deviation NA
The pharmacokinetic parameter could not be reliably estimated

PRIMARY outcome

Timeframe: Day 7

To assess the The mean AUClast (Area under the Plasma Concentration-Time Curve from Time 0 to the Last Observed Measurable Concentration) for MC 1080 was determined

Outcome measures

Outcome measures
Measure
LEO 90105 Ointment
n=13 Participants
Subjects received once daily topical treatment with LEO 90105 (calcipotriol hydrate plus betamethasone dipropionate ointment) on all lesions on the trunk and/or limbs (excluding psoriasis on the genitals and skin folds) for 4 weeks. Subjects were supplied with an amount of medication at day 1, day 7 and day 14 such that the maximum usage of LEO 90105 could be 90 g per week.
Pharmacokinetic: AUClast of MC1080.
221.2 h*pg/mL
Standard Deviation 175.16

PRIMARY outcome

Timeframe: Day 14

The mean AUClast (Area under the Plasma Concentration-Time Curve from Time 0 to the Last Observed Measurable Concentration) for MC 1080 was determined

Outcome measures

Outcome measures
Measure
LEO 90105 Ointment
n=13 Participants
Subjects received once daily topical treatment with LEO 90105 (calcipotriol hydrate plus betamethasone dipropionate ointment) on all lesions on the trunk and/or limbs (excluding psoriasis on the genitals and skin folds) for 4 weeks. Subjects were supplied with an amount of medication at day 1, day 7 and day 14 such that the maximum usage of LEO 90105 could be 90 g per week.
Pharmacokinetic: AUClast of MC1080.
NA h*pg/mL
Standard Deviation NA
The pharmacokinetic parameter could not be reliably estimated

SECONDARY outcome

Timeframe: Baseline to Day 28

Psoriasis Area and Severity Index (PASI) is based on the investigator's assessment of the disease. The extent and severity of redness, thickness and scaliness of psoriasis are recorded for three regions (arms, trunk and legs) and these are used to calculate PASI. The PASI can range between 0 (best) to 64.8 (worst). m-PASI indicate that the scale is modified.

Outcome measures

Outcome measures
Measure
LEO 90105 Ointment
n=13 Participants
Subjects received once daily topical treatment with LEO 90105 (calcipotriol hydrate plus betamethasone dipropionate ointment) on all lesions on the trunk and/or limbs (excluding psoriasis on the genitals and skin folds) for 4 weeks. Subjects were supplied with an amount of medication at day 1, day 7 and day 14 such that the maximum usage of LEO 90105 could be 90 g per week.
Efficacy: Percentage Change in m-PASI From Baseline to Day 28
-72.4 percentage of change
Standard Deviation 24.5

SECONDARY outcome

Timeframe: Day 28

Subjects with 'clear' or 'almost clear' disease by investigator's globala ssessment at day 28. Investigator global assessment (IGA) is based on the investigator's assessment of the disease severity (Plaque thickening, Scaling and Erythema) using a 6-point scale (Clear,Almost clear, Mild,Moderate, Severe, and Very severe). The assessment represents the average lesion severity on the trunk and limbs. IGA can range between 1 (best) and 6 (worst). The assessment is based on the condition of the disease at the time of evaluation, and not in relation to the condition at a previous visit.

Outcome measures

Outcome measures
Measure
LEO 90105 Ointment
n=13 Participants
Subjects received once daily topical treatment with LEO 90105 (calcipotriol hydrate plus betamethasone dipropionate ointment) on all lesions on the trunk and/or limbs (excluding psoriasis on the genitals and skin folds) for 4 weeks. Subjects were supplied with an amount of medication at day 1, day 7 and day 14 such that the maximum usage of LEO 90105 could be 90 g per week.
Efficacy: Subjects With 'Clear' or 'Almost Clear' Disease by Investigator's Global Assessment at Day 28.
6 participants

Adverse Events

LEO 90105 Ointment

Serious events: 0 serious events
Other events: 4 other events
Deaths: 0 deaths

Serious adverse events

Adverse event data not reported

Other adverse events

Other adverse events
Measure
LEO 90105 Ointment
n=13 participants at risk
Subjects received once daily topical treatment with LEO 90105 (calcipotriol hydrate plus betamethasone dipropionate ointment) on all lesions on the trunk and/or limbs (excluding psoriasis on the genitals and skin folds) for 4 weeks. Subjects were supplied with an amount of medication at day 1, day 7 and day 14 such that the maximum usage of LEO 90105 could be 90 g per week.
Gastrointestinal disorders
Abdominal discomfort
7.7%
1/13
Infections and infestations
Folliculitis
7.7%
1/13
Injury, poisoning and procedural complications
Skin injury
7.7%
1/13
Musculoskeletal and connective tissue disorders
Arthralgia
7.7%
1/13
Vascular disorders
Orthostatic hypotension
7.7%
1/13

Additional Information

Clinical trial disclosure manager

LEO Pharma A/S

Phone: 00 45 44 94 58 88

Results disclosure agreements

  • Principal investigator is a sponsor employee LEO acknowledges the investigators right to publish the entire results of the study, irrespective of outcome. LEO retains the right to have any publication submitted to LEO for review. Investigators must undertake not to submit any part of their individual data for publication without the prior consent of LEO.
  • Publication restrictions are in place

Restriction type: OTHER