Phase 2 Healthy Volunteer Study to Evaluate the Ability of PRT064445 to Reverse the Effects of Several Blood Thinner Drugs on Laboratory Tests (Module 1 of 4)

NCT ID: NCT01758432

Last Updated: 2023-08-07

Study Results

Results available

Outcome measurements, participant flow, baseline characteristics, and adverse events have been published for this study.

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE2

Total Enrollment

54 participants

Study Classification

INTERVENTIONAL

Study Start Date

2012-12-31

Study Completion Date

2015-09-30

Brief Summary

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The purpose of this study is to evaluate the ability of PRT064445 to reverse the effects of several blood thinner drugs on laboratory tests. The study also is evaluating the blood levels of PRT064445 given at different doses.

Detailed Description

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A randomized, double-blind, vehicle-controlled study to assess the safety, tolerability, pharmacokinetics, and pharmacodynamics of intravenously administered PRT064445 after dosing to steady state with one of four direct/indirect fXa inhibitors in healthy volunteers

Conditions

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Healthy Volunteers

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

This study has four modules with a total of 21 cohorts, each module was reported and submitted separately.

Module 1, NCT01758432 (54 subjects with 7cohorts including placebo); Module 2, NCT03578146 (48 subjects with 6 cohorts including placebo); Module 3, NCT03551730 (27 subjects with 4 cohorts including placebo); Module 4, NCT03551743 (28 subjects with 4 cohorts including placebo)
Primary Study Purpose

TREATMENT

Blinding Strategy

QUADRUPLE

Participants Caregivers Investigators Outcome Assessors

Study Groups

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Module 1 (90 mg bolus)

90 mg PRT064445 given as a single IV

Group Type EXPERIMENTAL

PRT064445/Apixaban

Intervention Type COMBINATION_PRODUCT

Placebo/Apixaban

Intervention Type COMBINATION_PRODUCT

Module 1 (210 mg bolus)

210 mg PRT064445 given as a single IV bolus

Group Type EXPERIMENTAL

PRT064445/Apixaban

Intervention Type COMBINATION_PRODUCT

Placebo/Apixaban

Intervention Type COMBINATION_PRODUCT

Module 1 (420 mg bolus)

420 mg PRT064445 given as a single IV bolus

Group Type EXPERIMENTAL

PRT064445/Apixaban

Intervention Type COMBINATION_PRODUCT

Placebo/Apixaban

Intervention Type COMBINATION_PRODUCT

Module 1 (420 mg bolus + 180 mg infusion) 4 mg/min

600 mg PRT064445 given as follows: 420 mg IV over \~14 minutes (\~30 mg/min), followed by a continuous infusion of 180 mg (4 mg/min over 45 minutes)

Group Type EXPERIMENTAL

PRT064445/Apixaban

Intervention Type COMBINATION_PRODUCT

Placebo/Apixaban

Intervention Type COMBINATION_PRODUCT

Module 1 (420 mg bolus + 180 mg bolus) 30mg/min

600 mg PRT064445 given as follows: up to 420 mg IV over \~14 minutes (\~30 mg/min), followed by a second bolus of 180 mg IV over \~6 minutes (\~30 mg/min), 45 minutes after completion of the bolus

Group Type EXPERIMENTAL

PRT064445/Apixaban

Intervention Type COMBINATION_PRODUCT

Placebo/Apixaban

Intervention Type COMBINATION_PRODUCT

Module 1 (420 mg bolus + 480 mg infusion) 4mg/min

900 mg PRT064445 given as follows: 420 mg IV, followed by a continuous infusion of 480 mg (4 mg/min over 120 minutes

Group Type EXPERIMENTAL

PRT064445/Apixaban

Intervention Type COMBINATION_PRODUCT

Placebo/Apixaban

Intervention Type COMBINATION_PRODUCT

Module 1 Placebo

Placebo administered intravenously (IV) as a bolus, two bolus doses or a bolus followed by continuous infusion.

Group Type PLACEBO_COMPARATOR

Placebo

Intervention Type DRUG

Interventions

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PRT064445/Apixaban

Intervention Type COMBINATION_PRODUCT

Placebo/Apixaban

Intervention Type COMBINATION_PRODUCT

Placebo

Intervention Type DRUG

Other Intervention Names

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Andexanet

Eligibility Criteria

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Inclusion Criteria

* Healthy men or women between the ages of 18 and 45 years old

Exclusion Criteria

* History (including family history) or symptoms of, or risk factors for bleeding
* History (including family history) of or risk factors for a hypercoagulable or thrombotic condition
* Absolute/relative contraindication to anticoagulation or treatment with specific anticoagulants
* History of major surgery, severe trauma or bone fracture within 3 months prior to dosing; or planned surgery within 1 month after dosing.
Minimum Eligible Age

18 Years

Maximum Eligible Age

45 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

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Portola Pharmaceuticals

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Locations

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Tempe, Arizona, United States

Site Status

Countries

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United States

References

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Siegal D, Lu G, Leeds JM, Karbarz M, Castillo J, Mathur V, Hutchaleelaha A, Sinha U, Kitt M, McClure M, Hollenbach SJ, Curnutte JT, Conley PB, Crowther M. Safety, pharmacokinetics, and reversal of apixaban anticoagulation with andexanet alfa. Blood Adv. 2017 Sep 22;1(21):1827-1838. doi: 10.1182/bloodadvances.2017007112. eCollection 2017 Sep 26.

Reference Type DERIVED
PMID: 29296829 (View on PubMed)

Other Identifiers

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12-502 Module 1

Identifier Type: -

Identifier Source: org_study_id

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