A Clinical Trial to Compare the Pharmacokinetics of Imatinib Mesylate Tablet 400mg (1 Tablet) and Glivec Film-coated Tablet 100mg (4 Tablets)(Phase I)

NCT ID: NCT01751919

Last Updated: 2014-10-01

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

Get a concise snapshot of the trial, including recruitment status, study phase, enrollment targets, and key timeline milestones.

Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

37 participants

Study Classification

INTERVENTIONAL

Study Start Date

2012-05-31

Study Completion Date

2012-08-31

Brief Summary

Review the sponsor-provided synopsis that highlights what the study is about and why it is being conducted.

1. Investigational Product

1. Imatinib mesylate tablet 400 mg
2. Glivec film-coated tablet 100 mg (Comparator)
2. Expected target disease

1. chronic myeloid leukemia
2. Gastrointestinal stromal tumors
3. Study design : Randomized, open-label, single dose, two-period, two-way, crossover study

1. 36 healthy subjects, 2 groups (18 subjects/group)
2. 2 Period (either 1-a(1 tablet) or 1-b(4 tablet))
3. wash-out period : 14 days
4. Evaluation on pharmacokinetics(PKs) and safety

1. PKs : Cmax, AUClast, Tmax, AUCinf, t1/2
2. safety : adverse events, physical examination, vital sign, ECG, Laboratory test
5. Statistical method

1. Demography Characteristics
2. Pharmacokinetic parameters
3. Safety data

Detailed Description

Dive into the extended narrative that explains the scientific background, objectives, and procedures in greater depth.

Conditions

See the medical conditions and disease areas that this research is targeting or investigating.

Chronic Myeloid Leukemia Gastrointestinal Stromal Tumor

Study Design

Understand how the trial is structured, including allocation methods, masking strategies, primary purpose, and other design elements.

Allocation Method

RANDOMIZED

Intervention Model

CROSSOVER

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

Review each arm or cohort in the study, along with the interventions and objectives associated with them.

Group 1 (RT)

* Period 1: Glivec film-coated tablet 100 mg, 4 tablets (Active comparator)
* Period 2: Imatinib mesylate tablet 400 mg, 1 tablet (experimental)

Group Type OTHER

Imatinib mesylate tablet 400 mg, 1 Tablet

Intervention Type DRUG

Glivec film-coated tablet 100 mg, 4 Tablets

Intervention Type DRUG

Group 2 (TR)

* Period 1: Imatinib mesylate tablet 400 mg, 1 tablet (experimental)
* Period 2: Glivec film-coated tablet 100 mg, 4 tablets (Active comparator)

Group Type OTHER

Imatinib mesylate tablet 400 mg, 1 Tablet

Intervention Type DRUG

Glivec film-coated tablet 100 mg, 4 Tablets

Intervention Type DRUG

Interventions

Learn about the drugs, procedures, or behavioral strategies being tested and how they are applied within this trial.

Imatinib mesylate tablet 400 mg, 1 Tablet

Intervention Type DRUG

Glivec film-coated tablet 100 mg, 4 Tablets

Intervention Type DRUG

Eligibility Criteria

Check the participation requirements, including inclusion and exclusion rules, age limits, and whether healthy volunteers are accepted.

Inclusion Criteria

* healthy male volunteers between the ages of 20 to 50 years old
* weight more than 55kg and within the range of ±20% of ideal body weight (IBW)
* having neither congenital/chronic diseases nor pathological symptoms/findings as results of medical examination
* doctor determines to be suitable as subjects within 3 weeks ago before administration

Exclusion Criteria

* Hypersensitivity(or history of hypersensitivity) to medicines including imatinib mesylate
* Active Liver Diseases or exceed 1.5 times the normal range of AST, ALT, total bilirubin
* Creatinine clearance \< 80 mL/min
* Gastrointestinal diseases or surgeries that affect absorption of drug
* Excessive drinking(exceed 21units/week)
* Smoking over 10 cigarettes per day
Minimum Eligible Age

20 Years

Maximum Eligible Age

50 Years

Eligible Sex

MALE

Accepts Healthy Volunteers

Yes

Sponsors

Meet the organizations funding or collaborating on the study and learn about their roles.

Dong-A ST Co., Ltd.

INDUSTRY

Sponsor Role lead

Responsible Party

Identify the individual or organization who holds primary responsibility for the study information submitted to regulators.

Responsibility Role SPONSOR

Locations

Explore where the study is taking place and check the recruitment status at each participating site.

Kyungpook National University

Daegu, , South Korea

Site Status

Countries

Review the countries where the study has at least one active or historical site.

South Korea

References

Explore related publications, articles, or registry entries linked to this study.

Parrillo-Campiglia S, Ercoli MC, Umpierrez O, Rodriguez P, Marquez S, Guarneri C, Estevez-Parrillo FT, Laurenz M, Estevez-Carrizo FE. Bioequivalence of two film-coated tablets of imatinib mesylate 400 mg: a randomized, open-label, single-dose, fasting, two-period, two-sequence crossover comparison in healthy male South American volunteers. Clin Ther. 2009 Oct;31(10):2224-32. doi: 10.1016/j.clinthera.2009.10.009.

Reference Type BACKGROUND
PMID: 19922893 (View on PubMed)

Nikolova Z, Peng B, Hubert M, Sieberling M, Keller U, Ho YY, Schran H, Capdeville R. Bioequivalence, safety, and tolerability of imatinib tablets compared with capsules. Cancer Chemother Pharmacol. 2004 May;53(5):433-8. doi: 10.1007/s00280-003-0756-z.

Reference Type BACKGROUND
PMID: 15132131 (View on PubMed)

Other Identifiers

Review additional registry numbers or institutional identifiers associated with this trial.

Imatinib_CML_I

Identifier Type: -

Identifier Source: org_study_id

More Related Trials

Additional clinical trials that may be relevant based on similarity analysis.