Study to Evaluate the Safety and Tolerability of Tirabrutinib (ONO/GS-4059) Given as Monotherapy in Participants With Relapsed/Refractory NHL and CLL

NCT ID: NCT01659255

Last Updated: 2021-03-16

Study Results

Results available

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

90 participants

Study Classification

INTERVENTIONAL

Study Start Date

2012-08-17

Study Completion Date

2016-01-11

Brief Summary

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The primary objective of the study is to evaluate the safety and tolerability of tirabrutinib (formerly ONO/GS-4059) given as monotherapy to participants with relapsed/refractory non-Hodgkin's lymphoma (NHL) and chronic lymphocytic leukemia (CLL).

Detailed Description

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Conditions

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Non Hodgkins Lymphoma Chronic Lymphocytic Leukaemia

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Tirabrutinib 20 mg Once Daily (CLL)

Participants with relapsed/refractory chronic lymphocytic leukaemia (CLL) received tirabrutinib 20 mg once daily.

Group Type EXPERIMENTAL

Tirabrutinib

Intervention Type DRUG

Capsules administered orally

Tirabrutinib 40 mg Once Daily (CLL)

Participants with relapsed/refractory CLL received tirabrutinib 40 mg once daily.

Group Type EXPERIMENTAL

Tirabrutinib

Intervention Type DRUG

Capsules administered orally

Tirabrutinib 80 mg Once Daily (CLL)

Participants with relapsed/refractory CLL received tirabrutinib 80 mg once daily.

Group Type EXPERIMENTAL

Tirabrutinib

Intervention Type DRUG

Capsules administered orally

Tirabrutinib 160 mg Once Daily (CLL)

Participants with relapsed/refractory CLL received tirabrutinib 160 mg once daily.

Group Type EXPERIMENTAL

Tirabrutinib

Intervention Type DRUG

Capsules administered orally

Tirabrutinib 320 mg Once Daily (CLL)

Participants with relapsed/refractory CLL received tirabrutinib 320 mg once daily.

Group Type EXPERIMENTAL

Tirabrutinib

Intervention Type DRUG

Capsules administered orally

Tirabrutinib 400 mg Once Daily (CLL)

Participants with relapsed/refractory CLL received tirabrutinib 400 mg once daily.

Group Type EXPERIMENTAL

Tirabrutinib

Intervention Type DRUG

Capsules administered orally

Tirabrutinib 500 mg Once Daily (CLL)

Participants with relapsed/refractory CLL received tirabrutinib 500 mg once daily.

Group Type EXPERIMENTAL

Tirabrutinib

Intervention Type DRUG

Capsules administered orally

Tirabrutinib 600 mg Once Daily (CLL)

Participants with relapsed/refractory CLL received tirabrutinib 600 mg once daily.

Group Type EXPERIMENTAL

Tirabrutinib

Intervention Type DRUG

Capsules administered orally

Tirabrutinib 300 mg Twice Daily (CLL)

Participants with relapsed/refractory CLL received tirabrutinib 300 mg twice daily.

Group Type EXPERIMENTAL

Tirabrutinib

Intervention Type DRUG

Capsules administered orally

Tirabrutinib 20 mg Once Daily (NHL)

Participants with relapsed/refractory non-Hodgkin's lymphoma (NHL) received tirabrutinib 20 mg once daily.

Group Type EXPERIMENTAL

Tirabrutinib

Intervention Type DRUG

Capsules administered orally

Tirabrutinib 40 mg Once Daily (NHL)

Participants with relapsed/refractory NHL received tirabrutinib 40 mg once daily.

Group Type EXPERIMENTAL

Tirabrutinib

Intervention Type DRUG

Capsules administered orally

Tirabrutinib 80 mg Once Daily (NHL)

Participants with relapsed/refractory NHL received tirabrutinib 80 mg once daily.

Group Type EXPERIMENTAL

Tirabrutinib

Intervention Type DRUG

Capsules administered orally

Tirabrutinib 160 mg Once Daily (NHL)

Participants with relapsed/refractory NHL received tirabrutinib 160 mg once daily.

Group Type EXPERIMENTAL

Tirabrutinib

Intervention Type DRUG

Capsules administered orally

Tirabrutinib 320 mg Once Daily (NHL)

Participants with relapsed/refractory NHL received tirabrutinib 320 mg once daily.

Group Type EXPERIMENTAL

Tirabrutinib

Intervention Type DRUG

Capsules administered orally

Tirabrutinib 480 mg Once Daily (NHL)

Participants with relapsed/refractory NHL received tirabrutinib 480 mg once daily.

Group Type EXPERIMENTAL

Tirabrutinib

Intervention Type DRUG

Capsules administered orally

Tirabrutinib 600 mg Once Daily (NHL)

Participants with relapsed/refractory NHL received tirabrutinib 600 mg once daily.

Group Type EXPERIMENTAL

Tirabrutinib

Intervention Type DRUG

Capsules administered orally

Tirabrutinib 240 mg Twice Daily (NHL)

Participants with relapsed/refractory NHL received tirabrutinib 240 mg twice daily.

Group Type EXPERIMENTAL

Tirabrutinib

Intervention Type DRUG

Capsules administered orally

Interventions

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Tirabrutinib

Capsules administered orally

Intervention Type DRUG

Other Intervention Names

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ONO/GS-4059

Eligibility Criteria

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Inclusion Criteria

1. Males or females with a confirmed diagnosis of and documented history of relapsed or refractory malignant disease (B-cell lymphoma and/or CLL) for which no therapy of curative or high priority exists and for whom treatment with a Btk inhibitor may be deemed appropriate.
2. Age ≥ 18 years.
3. Eastern Cooperative Oncology Group (ECOG) performance status of ≤ 2.

Exclusion Criteria

1. Central nervous system (CNS) lymphoma.
2. Women who are pregnant or lactating.
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Ono Pharmaceutical Co. Ltd

INDUSTRY

Sponsor Role collaborator

Gilead Sciences

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Gilead Study Director

Role: STUDY_DIRECTOR

Gilead Sciences

Locations

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CHRU - Hopital Claude HURIEZ

Lille, , France

Site Status

Centre hospitalier Lyon Sud

Lyon, , France

Site Status

CHU St Eloi

Montpellier, , France

Site Status

University Hospital of Wales

Cardiff, , United Kingdom

Site Status

Leicester Royal Infirmary

Leicester, , United Kingdom

Site Status

Derriford Hospital

Plymouth, , United Kingdom

Site Status

Countries

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France United Kingdom

References

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Walter HS, Salles GA, Dyer MJ. New Agents to Treat Chronic Lymphocytic Leukemia. N Engl J Med. 2016 Jun 2;374(22):2185-6. doi: 10.1056/NEJMc1602674. No abstract available.

Reference Type RESULT
PMID: 27248633 (View on PubMed)

Walter HS, Rule SA, Dyer MJ, Karlin L, Jones C, Cazin B, Quittet P, Shah N, Hutchinson CV, Honda H, Duffy K, Birkett J, Jamieson V, Courtenay-Luck N, Yoshizawa T, Sharpe J, Ohno T, Abe S, Nishimura A, Cartron G, Morschhauser F, Fegan C, Salles G. A phase 1 clinical trial of the selective BTK inhibitor ONO/GS-4059 in relapsed and refractory mature B-cell malignancies. Blood. 2016 Jan 28;127(4):411-9. doi: 10.1182/blood-2015-08-664086. Epub 2015 Nov 5.

Reference Type RESULT
PMID: 26542378 (View on PubMed)

Fegan, C, Bagshawe J, Salles G, et al. The Bruton's tyrosine kinase (BTK) inhibitor ONO-4059: promising single agent activity and well tolerated in patients with high risk chronic lymphocytic leukaemia (CLL). Paper presented at: 56th American Society of Hematology Annual Meeting and Exposition; December 6-9, 2014; San Franscisco, CA.

Reference Type RESULT

Morschhauser F, Terriou L, Dyer M, et al. The Bruton's tyrosine kinase (BTK) inhibitor ONO-4059: promising single agent activity in patients with relapsed and refractory NHL. Haematologica. 2014 Jun; 99: 150.

Reference Type RESULT

Other Identifiers

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2011-005033-39

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

ONO-4059POE001

Identifier Type: -

Identifier Source: org_study_id

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