Multiple Ascending-Dose Study to Evaluate the Safety, Tolerability and Pharmacokinetics of BMS-933043 in Healthy Subjects

NCT ID: NCT01605994

Last Updated: 2014-06-27

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

115 participants

Study Classification

INTERVENTIONAL

Study Start Date

2012-07-31

Study Completion Date

2013-12-31

Brief Summary

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Includes a placebo-controlled sequential, ascending multiple-dose panels (10 panels, 8 ascending doses, and 2 fixed Japanese Panels exploring safety, tolerability, and Pharmacokinetic (PK) measures

Detailed Description

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Conditions

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Healthy Adult Normals

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

BASIC_SCIENCE

Blinding Strategy

QUADRUPLE

Participants Caregivers Investigators Outcome Assessors

Study Groups

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Panel 1:BMS-933043(2mg)/Placebo+Antacid Buffer Solution

BMS-933043 2 mg solution by mouth twice daily for 10 days

OR

Placebo matching with BMS-933043 0 mg solution by mouth twice daily for 10 days

Antacid Buffer Predose 150 mL solution by mouth twice daily for 10 days

Group Type EXPERIMENTAL

BMS-933043

Intervention Type DRUG

Placebo matching with BMS-933043

Intervention Type DRUG

Antacid Buffer Predose Solution

Intervention Type DRUG

Panel 2:BMS-933043(5mg)/Placebo+Antacid Buffer Solution

BMS-933043 5 mg solution by mouth twice daily for 10 days

OR

Placebo matching with BMS-933043 0 mg solution by mouth twice daily for 10 days

Antacid Buffer Predose 150 mL solution by mouth twice daily for 10 days

Group Type EXPERIMENTAL

BMS-933043

Intervention Type DRUG

Placebo matching with BMS-933043

Intervention Type DRUG

Antacid Buffer Predose Solution

Intervention Type DRUG

Panel 3:BMS-933043(10mg)/Placebo+Antacid Buffer Solution

BMS-933043 10 mg solution by mouth twice daily for 10 days

OR

Placebo matching with BMS-933043 0 mg solution by mouth twice daily for 10 days

Antacid Buffer Predose 150 mL solution by mouth twice daily for 10 days

Group Type EXPERIMENTAL

BMS-933043

Intervention Type DRUG

Placebo matching with BMS-933043

Intervention Type DRUG

Antacid Buffer Predose Solution

Intervention Type DRUG

Panel 4:BMS-933043(25mg)/Placebo+Antacid Buffer Solution

BMS-933043 25 mg solution by mouth twice daily for 10 days

OR

Placebo matching with BMS-933043 0 mg solution by mouth twice daily for 10 days

Antacid Buffer Predose 150 mL solution by mouth twice daily for 10 days

Group Type EXPERIMENTAL

BMS-933043

Intervention Type DRUG

Placebo matching with BMS-933043

Intervention Type DRUG

Antacid Buffer Predose Solution

Intervention Type DRUG

Panel 5:BMS-933043(50mg)/Placebo+Antacid Buffer Solution

BMS-933043 50 mg solution by mouth twice daily for 10 days

OR

Placebo matching with BMS-933043 0 mg solution by mouth twice daily for 10 days

Antacid Buffer Predose 150 mL solution by mouth twice daily for 10 days

CSF sampling required

Group Type EXPERIMENTAL

BMS-933043

Intervention Type DRUG

Placebo matching with BMS-933043

Intervention Type DRUG

Antacid Buffer Predose Solution

Intervention Type DRUG

Panel 6:BMS-933043(100mg)/Placebo+Antacid Buffer Solution

BMS-933043 100 mg solution by mouth twice daily for 10 days

OR

Placebo matching with BMS-933043 0 mg solution by mouth twice daily for 10 days

Antacid Buffer Predose 150 mL solution by mouth twice daily for 10 days

Group Type EXPERIMENTAL

BMS-933043

Intervention Type DRUG

Placebo matching with BMS-933043

Intervention Type DRUG

Antacid Buffer Predose Solution

Intervention Type DRUG

Panel 7:BMS-933043(200mg)/Placebo+Antacid Buffer Solution

BMS-933043 200 mg solution by mouth twice daily for 10 days

OR

Placebo matching with BMS-933043 0 mg solution by mouth twice daily for 10 days

Antacid Buffer Predose 150 mL solution by mouth twice daily for 10 days

Group Type EXPERIMENTAL

BMS-933043

Intervention Type DRUG

Placebo matching with BMS-933043

Intervention Type DRUG

Antacid Buffer Predose Solution

Intervention Type DRUG

Panel 8:BMS-933043(25mg)/Placebo+Antacid Buffer Predose

MAD Phase: Japanese Subjects. Cerebrospinal fluid (CSF) sampling not required

BMS-933043 25 mg solution by mouth twice daily for 10 days

OR

Placebo matching with BMS-933043 0 mg solution by mouth twice daily for 10 days

Antacid Buffer Predose 150 mL solution by mouth twice daily for 10 days

Group Type EXPERIMENTAL

BMS-933043

Intervention Type DRUG

Placebo matching with BMS-933043

Intervention Type DRUG

Antacid Buffer Predose Solution

Intervention Type DRUG

Panel 9:BMS-933043(200mg)/Placebo+Antacid Buffer Predose

Japanese Subjects. CSF sampling not required.

BMS-933043 200 mg solution by mouth twice daily for 10 days

OR

Placebo matching with BMS-933043 0 mg solution by mouth twice daily for 10 days

Antacid Buffer Predose 150 mL solution by mouth twice daily for 10 days

Group Type EXPERIMENTAL

BMS-933043

Intervention Type DRUG

Placebo matching with BMS-933043

Intervention Type DRUG

Antacid Buffer Predose Solution

Intervention Type DRUG

Panel 10:BMS-933043(350mg)/Placebo+Antacid Buffer Predose

BMS-933043 350 mg solution by mouth twice daily for 10 days

OR

Placebo matching with BMS-933043 0 mg solution by mouth twice daily for 10 days

Antacid Buffer Predose 150 mL solution by mouth twice daily for 10 days

Group Type EXPERIMENTAL

BMS-933043

Intervention Type DRUG

Placebo matching with BMS-933043

Intervention Type DRUG

Antacid Buffer Predose Solution

Intervention Type DRUG

CSF Panel:BMS-933043(MTD)/Placebo+Antacid Buffer Predose

If Panel 5 does not run. CSF Sampling at steady state

BMS-933043 maximum tolerated dose (MTD), solution by mouth twice daily for 10 days

OR

Placebo matching with BMS-933043 0 mg solution by mouth twice daily for 10 days

Antacid Buffer Predose 150 mL solution by mouth twice daily for 10 days

Group Type EXPERIMENTAL

BMS-933043

Intervention Type DRUG

Placebo matching with BMS-933043

Intervention Type DRUG

Antacid Buffer Predose Solution

Intervention Type DRUG

Interventions

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BMS-933043

Intervention Type DRUG

Placebo matching with BMS-933043

Intervention Type DRUG

Antacid Buffer Predose Solution

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Healthy subjects as determined by no clinically significant deviation from normal medical history, physical examination, ECGs and clinical laboratory determinations
* Body Mass Index (BMI) of 18 to 30 kg/m2, inclusive. BMI = weight (kg)/ \[height (m)\]2
* Normal Neurological Exam (LP subjects only: to rule out focal CNS lesions that would render LP unsafe)
* Men and women, ages 18 to 55 years, inclusive.
* Women who are not of childbearing potential (WOCBP) \[ie, who are postmenopausal or surgically sterile\] and men
* Women must have a negative serum or urine pregnancy test (minimum sensitivity 25 IU/L or equivalent units of HCG) within 24 hours prior to the start of investigational product.
* Women must not be breastfeeding
* Sexually active fertile men must use effective birth control if their partners are WOCBP throughout the study and for 90 days after last dose

Exclusion Criteria

* Any significant acute or chronic medical illness
* Current or recent (within 3 months of study drug administration) gastrointestinal disease
* Any major surgery within 4 weeks of study drug administration
* Any gastrointestinal surgery that could impact upon the absorption of study drug
* Donation of blood or plasma to a blood bank or in a clinical study (except a screening visit) within 4 weeks of study drug administration
* Blood transfusion within 4 weeks of study drug administration
* Inability to tolerate oral medication
* Inability to be venipunctured and/or tolerate venous access
* Smoking more than 1 cigarette/cigar per week, within 3 months prior to screening
* Regular daily use of nicotine products or Varenicline (Chantix® or Champix®) within 3 months prior to screening
* Recent (within 6 months of study drug administration) drug or alcohol abuse as defined in Diagnostic and Statistical Manual of Mental Disorders (4th Edition) \[DSM IV\], Diagnostic Criteria for Drug and Alcohol Abuse
* History of cardiac arrhythmias, or palpitations associated with presyncope or syncope or history of unexplained syncope
Minimum Eligible Age

18 Years

Maximum Eligible Age

55 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

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Bristol-Myers Squibb

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Bristol-Myers Squibb

Role: STUDY_DIRECTOR

Bristol-Myers Squibb

Locations

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Clinilabs, Inc.

New York, New York, United States

Site Status

Countries

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United States

Related Links

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Other Identifiers

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CN171-002

Identifier Type: -

Identifier Source: org_study_id

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