Drug Drug Interaction Study Between BI 201335 and BI 207127 in Chronic Hepatitis C Infected Patients

NCT ID: NCT01525628

Last Updated: 2016-06-10

Study Results

Results available

Outcome measurements, participant flow, baseline characteristics, and adverse events have been published for this study.

View full results

Basic Information

Get a concise snapshot of the trial, including recruitment status, study phase, enrollment targets, and key timeline milestones.

Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

72 participants

Study Classification

INTERVENTIONAL

Study Start Date

2012-04-30

Study Completion Date

2014-10-31

Brief Summary

Review the sponsor-provided synopsis that highlights what the study is about and why it is being conducted.

To evaluate the drug-drug interactions between BI 201335 and BI 207127 as well as their combined effect on CYP probe drug substrates and on tenofovir and raltegravir in treatment naive or prior treatment relapse patients with chronic hepatitis C infection.

Detailed Description

Dive into the extended narrative that explains the scientific background, objectives, and procedures in greater depth.

Conditions

See the medical conditions and disease areas that this research is targeting or investigating.

Hepatitis C, Chronic

Study Design

Understand how the trial is structured, including allocation methods, masking strategies, primary purpose, and other design elements.

Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

Review each arm or cohort in the study, along with the interventions and objectives associated with them.

Group A

Effect of BI 207127 on BI 201335, the effect of BI 201335 and dual oral direct acting antiviral (DAAs) on caffeine, tolbutamide and midazolam

Group Type EXPERIMENTAL

tolbutamide

Intervention Type DRUG

CYP2C9 probe drug

midazolam

Intervention Type DRUG

CYP3A probe drug

caffeine

Intervention Type DRUG

CYP1A2 probe drug

BI 201335

Intervention Type DRUG

HCV protease inhibitor

pegylated interferon

Intervention Type DRUG

HCV treatment

BI 207127

Intervention Type DRUG

HCV polymerase inhibitor

ribavirin

Intervention Type DRUG

HCV treatment

Group B

Effect of BI 201335 on BI 207127, the effect of BI 207127 and metabolites and dual oral DAAs on caffeine, tolbutamide and midazolam

Group Type EXPERIMENTAL

BI 201335

Intervention Type DRUG

HCV protease inhibitor

caffeine

Intervention Type DRUG

CYP1A2 probe drug

tolbutamide

Intervention Type DRUG

CYP2C9 probe drug

pegylated interferon

Intervention Type DRUG

HCV treatment

BI 207127

Intervention Type DRUG

HCV polymerase inhibitor

ribavirin

Intervention Type DRUG

HCV treatment

midazolam

Intervention Type DRUG

CYP3A probe drug

Group C

Effect of Dual oral DAAs on tenofovir

Group Type EXPERIMENTAL

tenofovir

Intervention Type DRUG

nucleoside analogue

BI 207127

Intervention Type DRUG

HCV polymerase inhibitor

ribavirin

Intervention Type DRUG

HCV treatment

BI 201335

Intervention Type DRUG

HCV protease inhibitor

Group D

Effect of BI 201335 and BI 207127 at 600 mg b.i.d. on caffeine, tolbutamide and midazolam

Group Type EXPERIMENTAL

midazolam

Intervention Type DRUG

CYP3A probe drug

BI 201335

Intervention Type DRUG

HCV protease inhibitor

BI 207127

Intervention Type DRUG

HCV polymerase inhibitor

ribavirin

Intervention Type DRUG

HCV treatment

caffeine

Intervention Type DRUG

CYP1A2 probe drug

tolbutamide

Intervention Type DRUG

CYP2C9 probe drug

Group E

Effect of BI 201335 and BI 207127 on raltegravir

Group Type EXPERIMENTAL

BI 201335

Intervention Type DRUG

HCV protease inhibitor

ribavirin

Intervention Type DRUG

HCV treatment

BI 207127

Intervention Type DRUG

HCV polymerase inhibitor

Interventions

Learn about the drugs, procedures, or behavioral strategies being tested and how they are applied within this trial.

midazolam

CYP3A probe drug

Intervention Type DRUG

BI 201335

HCV protease inhibitor

Intervention Type DRUG

tenofovir

nucleoside analogue

Intervention Type DRUG

caffeine

CYP1A2 probe drug

Intervention Type DRUG

tolbutamide

CYP2C9 probe drug

Intervention Type DRUG

tolbutamide

CYP2C9 probe drug

Intervention Type DRUG

midazolam

CYP3A probe drug

Intervention Type DRUG

caffeine

CYP1A2 probe drug

Intervention Type DRUG

pegylated interferon

HCV treatment

Intervention Type DRUG

BI 201335

HCV protease inhibitor

Intervention Type DRUG

BI 201335

HCV protease inhibitor

Intervention Type DRUG

BI 207127

HCV polymerase inhibitor

Intervention Type DRUG

BI 207127

HCV polymerase inhibitor

Intervention Type DRUG

BI 201335

HCV protease inhibitor

Intervention Type DRUG

BI 207127

HCV polymerase inhibitor

Intervention Type DRUG

ribavirin

HCV treatment

Intervention Type DRUG

ribavirin

HCV treatment

Intervention Type DRUG

ribavirin

HCV treatment

Intervention Type DRUG

pegylated interferon

HCV treatment

Intervention Type DRUG

ribavirin

HCV treatment

Intervention Type DRUG

caffeine

CYP1A2 probe drug

Intervention Type DRUG

tolbutamide

CYP2C9 probe drug

Intervention Type DRUG

BI 207127

HCV polymerase inhibitor

Intervention Type DRUG

midazolam

CYP3A probe drug

Intervention Type DRUG

BI 201335

HCV protease inhibitor

Intervention Type DRUG

BI 207127

HCV polymerase inhibitor

Intervention Type DRUG

ribavirin

HCV treatment

Intervention Type DRUG

Eligibility Criteria

Check the participation requirements, including inclusion and exclusion rules, age limits, and whether healthy volunteers are accepted.

Inclusion Criteria

1. Chronic hepatitis C genotype 1 infection, diagnosed at least 6 months prior to screening
2. Treatment naive or confirmed prior treatment relapse or partial response following treatment with interferon and ribavirin
3. Age 18 to 70 years
4. HCV RNA (Hepatitis C Virus RiboNucleic Acid) = 1,000 IU/mL at screening
5. Liver biopsy or fibroscan to exclude cirrhosis

Exclusion Criteria

1. Hepatitis C Virus (HCV) infection of mixed genotype; Hepatitis B Virus (HBV) or Human Immunodeficiency Virus (HIV) co-infection
2. Evidence of acute or chronic liver disease due to causes other than chronic HCV infection,
3. Decompensated liver disease, or history of decompensated liver disease,
4. Body weight \< 40 or \> 125 kg,
5. Clinical evidence of significant or unstable cardiovascular disease, chronic pulmonary disease, history or evidence of retinopathy or clinically significant ophthalmological disorder
6. Pre-existing psychiatric condition that could interfere with the subject's participation in and completion of the study
7. Laboratory parameters disorders (thalassemia major, sickle cell anemia or glucose 6 phosphate dehydrogenase deficit)
8. Hemoglobin \< 12 g/dL for women and \< 13 g/dL for men
9. Patients who have been previously treated with at least one dose of any antiviral or immunomodulatory drug other than interferon alfa or ribavirin for acute or chronic HCV infection
Minimum Eligible Age

18 Years

Maximum Eligible Age

70 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

Meet the organizations funding or collaborating on the study and learn about their roles.

Boehringer Ingelheim

INDUSTRY

Sponsor Role lead

Responsible Party

Identify the individual or organization who holds primary responsibility for the study information submitted to regulators.

Responsibility Role SPONSOR

Principal Investigators

Learn about the lead researchers overseeing the trial and their institutional affiliations.

Boehringer Ingelheim

Role: STUDY_CHAIR

Boehringer Ingelheim

Locations

Explore where the study is taking place and check the recruitment status at each participating site.

1241.27.0006 Boehringer Ingelheim Investigational Site

La Mesa, California, United States

Site Status

1241.27.0005 Boehringer Ingelheim Investigational Site

Rockville, Maryland, United States

Site Status

1241.27.0004 Boehringer Ingelheim Investigational Site

Marlton, New Jersey, United States

Site Status

1241.27.0003 Boehringer Ingelheim Investigational Site

Philadelphia, Pennsylvania, United States

Site Status

1241.27.0001 Boehringer Ingelheim Investigational Site

Salt Lake City, Utah, United States

Site Status

1241.27.0200 Boehringer Ingelheim Investigational Site

Vancouver, British Columbia, Canada

Site Status

1241.27.0600 Boehringer Ingelheim Investigational Site

Vancouver, British Columbia, Canada

Site Status

1241.27.0700 Boehringer Ingelheim Investigational Site

Vancouver, British Columbia, Canada

Site Status

1241.27.0400 Boehringer Ingelheim Investigational Site

Victoria, British Columbia, Canada

Site Status

1241.27.0100 Boehringer Ingelheim Investigational Site

London, Ontario, Canada

Site Status

1241.27.0300 Boehringer Ingelheim Investigational Site

Ottawa, Ontario, Canada

Site Status

1241.27.0500 Boehringer Ingelheim Investigational Site

Montreal, Quebec, Canada

Site Status

1241.27.4907 Boehringer Ingelheim Investigational Site

Cologne, , Germany

Site Status

1241.27.4901 Boehringer Ingelheim Investigational Site

Frankfurt am Main, , Germany

Site Status

1241.27.4903 Boehringer Ingelheim Investigational Site

Leipzig, , Germany

Site Status

1241.27.4906 Boehringer Ingelheim Investigational Site

Mainz, , Germany

Site Status

Countries

Review the countries where the study has at least one active or historical site.

United States Canada Germany

Other Identifiers

Review additional registry numbers or institutional identifiers associated with this trial.

2012-004102-10

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

1241.27

Identifier Type: -

Identifier Source: org_study_id

More Related Trials

Additional clinical trials that may be relevant based on similarity analysis.