Trial Outcomes & Findings for Safety and Efficacy of EXC 001 in Subjects Who Have Participated in Prior Studies of EXC 001 (NCT NCT01494922)

NCT ID: NCT01494922

Last Updated: 2021-08-13

Results Overview

Physical examination included the assessment of skin, head, ears, eyes, nose, throat, respiratory system, cardiovascular system, abdomen (including liver and kidneys), musculoskeletal system, neurological system, gastrointestinal system, genitourinary system, endocrine system and lymph nodes. Abnormality in physical examination were based on investigator's discretion.

Recruitment status

COMPLETED

Study phase

PHASE2

Target enrollment

14 participants

Primary outcome timeframe

Day 1 up to Week 24

Results posted on

2021-08-13

Participant Flow

Participants who participated in any of the previous studies (EXC 001-202 \[NCT01037985\], EXC 001-203 \[NCT01037413\] and EXC 001-204 \[NCT01346969\]), had scars at a minimum of 1 year after surgery in previous study which qualified for scar revision and chose scar revision treatment with EXC 001 (PF-06473871) were eligible for this study.

Participant milestones

Participant milestones
Measure
EXC 001 (PF-06473871)
Participants who underwent scar revision surgery on Day 1 and received 4 intradermal injections of EXC 001 (PF-06473871) at a dose of 5 milligram per centimeter (mg/cm) at Week 2, 5, 8 and 11 after the surgical incision was closed, to both sides of the incision/scar. Participants received treatment for total scar length of up to 14 centimeter (cm).
Overall Study
STARTED
14
Overall Study
COMPLETED
13
Overall Study
NOT COMPLETED
1

Reasons for withdrawal

Reasons for withdrawal
Measure
EXC 001 (PF-06473871)
Participants who underwent scar revision surgery on Day 1 and received 4 intradermal injections of EXC 001 (PF-06473871) at a dose of 5 milligram per centimeter (mg/cm) at Week 2, 5, 8 and 11 after the surgical incision was closed, to both sides of the incision/scar. Participants received treatment for total scar length of up to 14 centimeter (cm).
Overall Study
Adverse Event
1

Baseline Characteristics

Safety and Efficacy of EXC 001 in Subjects Who Have Participated in Prior Studies of EXC 001

Baseline characteristics by cohort

Baseline characteristics by cohort
Measure
EXC 001 (PF-06473871)
n=14 Participants
Participants who underwent scar revision surgery on Day 1 and received 4 intradermal injections of EXC 001 (PF-06473871) at a dose of 5 mg/cm at Week 2, 5, 8 and 11 after the surgical incision was closed, to both sides of the incision/scar. Participants received treatment for total scar length of up to 14 cm.
Age, Continuous
44.0 years
STANDARD_DEVIATION 7.51 • n=5 Participants
Sex: Female, Male
Female
14 Participants
n=5 Participants
Sex: Female, Male
Male
0 Participants
n=5 Participants

PRIMARY outcome

Timeframe: Week 2 to Week 24

Population: Safety population included all participants who completed the scar revision surgery (Day 1 visit).

An AE was any untoward medical occurrence in a participant who received study drug without regard to possibility of causal relationship. An SAE was an AE resulting in any of the following outcomes or deemed significant for any other reason: death; initial or prolonged inpatient hospitalization; life-threatening experience (immediate risk of dying); persistent or significant disability/incapacity; congenital anomaly. AEs included SAEs and all non-SAEs that occurred during the study.

Outcome measures

Outcome measures
Measure
EXC 001 (PF-06473871)
n=14 Participants
Participants who underwent scar revision surgery on Day 1 and received 4 intradermal injections of EXC 001 (PF-06473871) at a dose of 5 mg/cm at Week 2, 5, 8 and 11 after the surgical incision was closed, to both sides of the incision/scar. Participants received treatment for total scar length of up to 14 cm.
Number of Participants With Adverse Events (AEs) and Serious Adverse Events (SAEs)
AEs
8 Participants
Number of Participants With Adverse Events (AEs) and Serious Adverse Events (SAEs)
SAEs
0 Participants

PRIMARY outcome

Timeframe: Day 1 up to Week 24

Population: Safety population included all participants who completed the scar revision surgery (Day 1 visit).

Participants were instructed to inform the investigator in case of any itching, redness, pain or any other symptom that appeared to be a rash at the injection sites. Erythematous, raised (indurated) and edematous reactions were considered as positive skin sensitivity reactions. In this outcome measure number of participants with any positive skin sensitivity reaction were reported.

Outcome measures

Outcome measures
Measure
EXC 001 (PF-06473871)
n=14 Participants
Participants who underwent scar revision surgery on Day 1 and received 4 intradermal injections of EXC 001 (PF-06473871) at a dose of 5 mg/cm at Week 2, 5, 8 and 11 after the surgical incision was closed, to both sides of the incision/scar. Participants received treatment for total scar length of up to 14 cm.
Number of Participants With Positive Skin Sensitivity Reaction
2 Participants

PRIMARY outcome

Timeframe: Day 1 up to Week 24

Population: Safety population included all participants who completed the scar revision surgery (Day 1 visit).

Following parameters were analyzed for laboratory examination: hematology (hemoglobin, hematocrit, red blood cell count, platelet count, white blood cell count, total neutrophils, eosinophils, monocytes, basophils, lymphocytes); Hepatobiliary biochemistry: Alanine Aminotransferase (ALT), Aspartate Aminotransferase (AST), Albumin, Alkaline Phosphatase, Total Bilirubin ; Renal Function Tests: Blood Urea Nitrogen (BUN), Creatinine, Creatinine Kinase, Uric Acid ; Electrolytes: Sodium, Potassium; Glucose; Urine analysis: (decimal logarithm of reciprocal of hydrogen ion activity )\[pH\], Specific gravity. Clinically significant laboratory abnormality findings were based on investigator discretion.

Outcome measures

Outcome measures
Measure
EXC 001 (PF-06473871)
n=14 Participants
Participants who underwent scar revision surgery on Day 1 and received 4 intradermal injections of EXC 001 (PF-06473871) at a dose of 5 mg/cm at Week 2, 5, 8 and 11 after the surgical incision was closed, to both sides of the incision/scar. Participants received treatment for total scar length of up to 14 cm.
Number of Participants With Clinically Significant Findings in Laboratory Examinations
0 Participants

PRIMARY outcome

Timeframe: Day 1 up to Week 24

Population: Safety population included all participants who completed the scar revision surgery (Day 1 visit).

Following vital sign parameters were assessed: diastolic blood pressure, systolic blood pressure, respiration rate, pulse rate, temperature and body weight. Number of participants with clinically significant change in any vital sign parameter compared to baseline were reported. Clinically significant change in vital signs criteria were based on investigator's discretion.

Outcome measures

Outcome measures
Measure
EXC 001 (PF-06473871)
n=14 Participants
Participants who underwent scar revision surgery on Day 1 and received 4 intradermal injections of EXC 001 (PF-06473871) at a dose of 5 mg/cm at Week 2, 5, 8 and 11 after the surgical incision was closed, to both sides of the incision/scar. Participants received treatment for total scar length of up to 14 cm.
Number of Participants With Clinically Significant Change in Vital Signs
0 Participants

PRIMARY outcome

Timeframe: Day 1 up to Week 24

Population: Safety population included all participants who completed the scar revision surgery (Day 1 visit).

Following parameters were analyzed: heart rate, PR interval, QT interval, QRS interval and QT interval corrected using Fridericia's formula (QTcF). Clinically significant findings in ECG were based on investigator's discretion.

Outcome measures

Outcome measures
Measure
EXC 001 (PF-06473871)
n=14 Participants
Participants who underwent scar revision surgery on Day 1 and received 4 intradermal injections of EXC 001 (PF-06473871) at a dose of 5 mg/cm at Week 2, 5, 8 and 11 after the surgical incision was closed, to both sides of the incision/scar. Participants received treatment for total scar length of up to 14 cm.
Number of Participants With Clinically Significant Findings in Electrocardiogram (ECG) Abnormalities
0 Participants

PRIMARY outcome

Timeframe: Day 1 up to Week 24

Population: Safety population included all participants who completed the scar revision surgery (Day 1 visit).

Physical examination included the assessment of skin, head, ears, eyes, nose, throat, respiratory system, cardiovascular system, abdomen (including liver and kidneys), musculoskeletal system, neurological system, gastrointestinal system, genitourinary system, endocrine system and lymph nodes. Abnormality in physical examination were based on investigator's discretion.

Outcome measures

Outcome measures
Measure
EXC 001 (PF-06473871)
n=14 Participants
Participants who underwent scar revision surgery on Day 1 and received 4 intradermal injections of EXC 001 (PF-06473871) at a dose of 5 mg/cm at Week 2, 5, 8 and 11 after the surgical incision was closed, to both sides of the incision/scar. Participants received treatment for total scar length of up to 14 cm.
Number of Participants With Abnormalities in Physical Examinations
3 Participants

SECONDARY outcome

Timeframe: Week 24

Population: Analysis population included all participants who completed Week 24 efficacy assessments.

Physician assessment of scar was done using a valid published 10-point rating scale. Assessment included following sub scores: vascularity, pigmentation, thickness, relief, pliability, surface area and overall opinion for scar, on a score of 1 = normal skin to 10 = worst scar imaginable. Composite score was the sum of all the sub scores except the overall opinion score and range from 6 (best score) to 60 (worst score).

Outcome measures

Outcome measures
Measure
EXC 001 (PF-06473871)
n=13 Participants
Participants who underwent scar revision surgery on Day 1 and received 4 intradermal injections of EXC 001 (PF-06473871) at a dose of 5 mg/cm at Week 2, 5, 8 and 11 after the surgical incision was closed, to both sides of the incision/scar. Participants received treatment for total scar length of up to 14 cm.
Physician Observer Scar Assessment Score: Individual Sub Scores and Composite Score
Overall opinion
4.63 units on a scale
Standard Deviation 2.033
Physician Observer Scar Assessment Score: Individual Sub Scores and Composite Score
Vascularity
4.02 units on a scale
Standard Deviation 1.838
Physician Observer Scar Assessment Score: Individual Sub Scores and Composite Score
Pigmentation
3.83 units on a scale
Standard Deviation 1.848
Physician Observer Scar Assessment Score: Individual Sub Scores and Composite Score
Thickness
4.55 units on a scale
Standard Deviation 2.022
Physician Observer Scar Assessment Score: Individual Sub Scores and Composite Score
Relief
4.06 units on a scale
Standard Deviation 2.112
Physician Observer Scar Assessment Score: Individual Sub Scores and Composite Score
Pliability
3.97 units on a scale
Standard Deviation 1.932
Physician Observer Scar Assessment Score: Individual Sub Scores and Composite Score
Surface area
4.71 units on a scale
Standard Deviation 1.534
Physician Observer Scar Assessment Score: Individual Sub Scores and Composite Score
Composite Score
25.15 units on a scale
Standard Deviation 8.744

SECONDARY outcome

Timeframe: Week 24

Population: Analysis population included all participants who completed Week 24 efficacy assessments.

Participants rated pain, itching, color, stiffness, thickness, irregularity and overall opinion of scar on 10-point scale. For pain and itching associated with scar: range = 1 (no, not at all) to 10 (yes, worst imaginable) and for other parameters associated with scar compared to normal skin: range = 1 (no, same as normal skin) to 10 (yes, very different). Composite score is the sum of all sub scores except overall opinion, range 6 (best) to 60 (worst). Scar appearance composite score is the sum of all sub scores except overall opinion, pain and itching, range 4 (best) to 40 (worst).

Outcome measures

Outcome measures
Measure
EXC 001 (PF-06473871)
n=13 Participants
Participants who underwent scar revision surgery on Day 1 and received 4 intradermal injections of EXC 001 (PF-06473871) at a dose of 5 mg/cm at Week 2, 5, 8 and 11 after the surgical incision was closed, to both sides of the incision/scar. Participants received treatment for total scar length of up to 14 cm.
Participant Observer Scar Assessment Score: Individual Sub Scores, Composite Score, Scar Appearance Composite Score
Overall opinion
6.21 units on a scale
Standard Deviation 2.660
Participant Observer Scar Assessment Score: Individual Sub Scores, Composite Score, Scar Appearance Composite Score
Pain
2.46 units on a scale
Standard Deviation 1.620
Participant Observer Scar Assessment Score: Individual Sub Scores, Composite Score, Scar Appearance Composite Score
Itching
2.03 units on a scale
Standard Deviation 1.234
Participant Observer Scar Assessment Score: Individual Sub Scores, Composite Score, Scar Appearance Composite Score
Color
6.72 units on a scale
Standard Deviation 2.323
Participant Observer Scar Assessment Score: Individual Sub Scores, Composite Score, Scar Appearance Composite Score
Stiffness
5.76 units on a scale
Standard Deviation 2.487
Participant Observer Scar Assessment Score: Individual Sub Scores, Composite Score, Scar Appearance Composite Score
Thickness
5.56 units on a scale
Standard Deviation 2.508
Participant Observer Scar Assessment Score: Individual Sub Scores, Composite Score, Scar Appearance Composite Score
Irregular
5.62 units on a scale
Standard Deviation 2.494
Participant Observer Scar Assessment Score: Individual Sub Scores, Composite Score, Scar Appearance Composite Score
Composite Score
28.15 units on a scale
Standard Deviation 10.457
Participant Observer Scar Assessment Score: Individual Sub Scores, Composite Score, Scar Appearance Composite Score
Scar Appearance composite Score
23.67 units on a scale
Standard Deviation 9.110

SECONDARY outcome

Timeframe: Week 24

Population: Analysis population included all participants who completed Week 24 efficacy assessments. Here, "type of unit analyzed" signifies number of scars evaluable.

Physician rated severity of each scar using a photonumeric guide on a scale range from 1 to 5 (where 1 = minimal, 2 = mild, 3 = moderate, 4 = severe, 5 = very severe). Number of scars with different ratings of scar severity were reported. Participants may have received treatment for multiple scars (up to 5 scars), results are reported for all scars (individual scar) and most severe scar for all the participants.

Outcome measures

Outcome measures
Measure
EXC 001 (PF-06473871)
n=28 scars
Participants who underwent scar revision surgery on Day 1 and received 4 intradermal injections of EXC 001 (PF-06473871) at a dose of 5 mg/cm at Week 2, 5, 8 and 11 after the surgical incision was closed, to both sides of the incision/scar. Participants received treatment for total scar length of up to 14 cm.
Number of Scars Classified According to Physician Photonumeric Guide Score Severity Category
Individual Scar: Minimal
5 scars
Number of Scars Classified According to Physician Photonumeric Guide Score Severity Category
Individual Scar: Mild
12 scars
Number of Scars Classified According to Physician Photonumeric Guide Score Severity Category
Individual Scar: Moderate
4 scars
Number of Scars Classified According to Physician Photonumeric Guide Score Severity Category
Individual Scar: Severe
1 scars
Number of Scars Classified According to Physician Photonumeric Guide Score Severity Category
Individual Scar: Very Severe
6 scars
Number of Scars Classified According to Physician Photonumeric Guide Score Severity Category
Most Severe Scar: Minimal
2 scars
Number of Scars Classified According to Physician Photonumeric Guide Score Severity Category
Most Severe Scar: Mild
4 scars
Number of Scars Classified According to Physician Photonumeric Guide Score Severity Category
Most Severe Scar: Moderate
2 scars
Number of Scars Classified According to Physician Photonumeric Guide Score Severity Category
Most Severe Scar: Severe
1 scars
Number of Scars Classified According to Physician Photonumeric Guide Score Severity Category
Most Severe Scar: Very Severe
4 scars

SECONDARY outcome

Timeframe: Week 24

Population: Analysis population included all participants who completed Week 24 efficacy assessments. Here, "type of unit analyzed" signifies number of scars evaluable.

Participants rated severity of each scar using a photonumeric guide on a scale range from 1 to 5 (where 1 = minimal, 2 = mild, 3 = moderate, 4 = severe, 5 = very severe). Number of scars with different ratings of scar severity were reported. Participants may have received treatment for multiple scars (up to 5 scars), results are reported for all scars (individual scar) and most severe scar for all the participants.

Outcome measures

Outcome measures
Measure
EXC 001 (PF-06473871)
n=28 scars
Participants who underwent scar revision surgery on Day 1 and received 4 intradermal injections of EXC 001 (PF-06473871) at a dose of 5 mg/cm at Week 2, 5, 8 and 11 after the surgical incision was closed, to both sides of the incision/scar. Participants received treatment for total scar length of up to 14 cm.
Number of Scars Classified According to Subject Participant Photonumeric Guide Score Severity Category
Individual Scar: Minimal
6 scars
Number of Scars Classified According to Subject Participant Photonumeric Guide Score Severity Category
Individual Scar: Mild
7 scars
Number of Scars Classified According to Subject Participant Photonumeric Guide Score Severity Category
Individual Scar: Moderate
6 scars
Number of Scars Classified According to Subject Participant Photonumeric Guide Score Severity Category
Individual Scar: Severe
3 scars
Number of Scars Classified According to Subject Participant Photonumeric Guide Score Severity Category
Individual Scar: Very Severe
6 scars
Number of Scars Classified According to Subject Participant Photonumeric Guide Score Severity Category
Most Severe Scar: Minimal
2 scars
Number of Scars Classified According to Subject Participant Photonumeric Guide Score Severity Category
Most Severe Scar: Mild
1 scars
Number of Scars Classified According to Subject Participant Photonumeric Guide Score Severity Category
Most Severe Scar: Moderate
4 scars
Number of Scars Classified According to Subject Participant Photonumeric Guide Score Severity Category
Most Severe Scar: Severe
1 scars
Number of Scars Classified According to Subject Participant Photonumeric Guide Score Severity Category
Most Severe Scar: Very Severe
5 scars

Adverse Events

EXC 001 (PF-06473871)

Serious events: 0 serious events
Other events: 8 other events
Deaths: 0 deaths

Serious adverse events

Adverse event data not reported

Other adverse events

Other adverse events
Measure
EXC 001 (PF-06473871)
n=14 participants at risk
Participants who underwent scar revision surgery on Day 1 and received 4 intradermal injections of EXC 001 (PF-06473871) at a dose of 5 mg/cm at Week 2, 5, 8 and 11 after the surgical incision was closed, to both sides of the incision/scar. Participants received treatment for total scar length of up to 14 cm.
Infections and infestations
Sinusitis
7.1%
1/14 • Week 2 to Week 24
Infections and infestations
Fungal Infection
7.1%
1/14 • Week 2 to Week 24
Injury, poisoning and procedural complications
Procedural Pain
7.1%
1/14 • Week 2 to Week 24
Injury, poisoning and procedural complications
Excoriation
7.1%
1/14 • Week 2 to Week 24
General disorders
Injection site erythema
14.3%
2/14 • Week 2 to Week 24
General disorders
Injection site induration
7.1%
1/14 • Week 2 to Week 24
General disorders
Injection site pain
7.1%
1/14 • Week 2 to Week 24
General disorders
Injection site pruritus
7.1%
1/14 • Week 2 to Week 24
Skin and subcutaneous tissue disorders
Acne
7.1%
1/14 • Week 2 to Week 24
Gastrointestinal disorders
Lip swelling
7.1%
1/14 • Week 2 to Week 24
Gastrointestinal disorders
Vomiting
7.1%
1/14 • Week 2 to Week 24
Psychiatric disorders
Anxiety
7.1%
1/14 • Week 2 to Week 24
Psychiatric disorders
Depression
7.1%
1/14 • Week 2 to Week 24
Skin and subcutaneous tissue disorders
Pruritus
7.1%
1/14 • Week 2 to Week 24
Nervous system disorders
Headache
7.1%
1/14 • Week 2 to Week 24

Additional Information

Pfizer ClinicalTrials.gov Call Center

Pfizer Inc.

Phone: 1-800-718-1021

Results disclosure agreements

  • Principal investigator is a sponsor employee Pfizer has the right to review disclosures, requesting a delay of less than 60 days. Investigator will postpone single center publications until after disclosure of pooled data (all sites), less than 12 months from study completion/termination at all participating sites. Investigator may not disclose previously undisclosed confidential information other than study results.
  • Publication restrictions are in place

Restriction type: OTHER