Study of Ipatasertib or Apitolisib With Abiraterone Acetate Versus Abiraterone Acetate in Participants With Castration-Resistant Prostate Cancer Previously Treated With Docetaxel Chemotherapy

NCT ID: NCT01485861

Last Updated: 2023-09-14

Study Results

Results available

Outcome measurements, participant flow, baseline characteristics, and adverse events have been published for this study.

View full results

Basic Information

Get a concise snapshot of the trial, including recruitment status, study phase, enrollment targets, and key timeline milestones.

Recruitment Status

COMPLETED

Clinical Phase

PHASE1/PHASE2

Total Enrollment

298 participants

Study Classification

INTERVENTIONAL

Study Start Date

2012-01-11

Study Completion Date

2022-08-31

Brief Summary

Review the sponsor-provided synopsis that highlights what the study is about and why it is being conducted.

This multicenter, international, Phase Ib/II trial consists of three stages: a Phase Ib, open-label stage in which the recommended Phase II dose was determined for ipataseritib administrated in combination with abiraterone and of apitolisib administrated in combination with abiraterone (this phase is no longer active), a Phase II, 3-arm, double-blind, randomized comparison of ipatasertib with abiraterone and prednisone/prednisolone versus placebo with abiraterone and prednisone/prednisolone and a safety single-arm, open-label cohort of ipatasertib 400 mg daily alone or in combination with prednisone/prednisolone or prednisone/prednisolone plus abiraterone.

Detailed Description

Dive into the extended narrative that explains the scientific background, objectives, and procedures in greater depth.

Conditions

See the medical conditions and disease areas that this research is targeting or investigating.

Prostate Cancer

Study Design

Understand how the trial is structured, including allocation methods, masking strategies, primary purpose, and other design elements.

Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

DOUBLE

Participants Investigators
In Phase II participants and investigators were blinded with regard to treatment status (i.e., ipatasertib vs. placebo). Phase Ib and the safety cohort were open-label.

Study Groups

Review each arm or cohort in the study, along with the interventions and objectives associated with them.

Phase Ib: Ipatasertib 400 mg + abiraterone

Participants will receive ipatasertib 400 mg once daily, abiraterone 1000 mg once daily, and prednisone/prednisolone 5 mg twice daily (bid) continuously in 28-day treatment cycles until disease progression or intolerable toxicity.

Group Type EXPERIMENTAL

Abiraterone

Intervention Type DRUG

Orally once daily

Ipatasertib

Intervention Type DRUG

Orally once daily

Prednisone

Intervention Type DRUG

Orally bid

Prednisolone

Intervention Type DRUG

Orally bid

Phase Ib: Apitolisib 30 mg + abiraterone

Participants will receive apitolisib 30 mg once daily, abiraterone 1000 mg once daily, and prednisone/prednisolone 5 mg twice daily (bid) continuously in 28-day treatment cycles until disease progression or intolerable toxicity.

Group Type EXPERIMENTAL

Abiraterone

Intervention Type DRUG

Orally once daily

Apitolisib

Intervention Type DRUG

Orally once daily

Prednisone

Intervention Type DRUG

Orally bid

Prednisolone

Intervention Type DRUG

Orally bid

Phase II: Ipatasertib 400 mg + abiraterone

Participants will receive Ipatasertib 400 mg once daily, abiraterone 1000 mg once daily, and prednisone/prednisolone 5 mg bid continuously in 28-day treatment cycles until disease progression or intolerable toxicity.

Group Type EXPERIMENTAL

Abiraterone

Intervention Type DRUG

Orally once daily

Ipatasertib

Intervention Type DRUG

Orally once daily

Prednisone

Intervention Type DRUG

Orally bid

Prednisolone

Intervention Type DRUG

Orally bid

Phase II: Ipatasertib 200 mg + abiraterone

Participants will receive Ipatasertib 200 mg once daily, abiraterone 1000 mg once daily, and prednisone/prednisolone 5 mg bid continuously in 28-day treatment cycles until disease progression or intolerable toxicity.

Group Type EXPERIMENTAL

Abiraterone

Intervention Type DRUG

Orally once daily

Ipatasertib

Intervention Type DRUG

Orally once daily

Prednisone

Intervention Type DRUG

Orally bid

Prednisolone

Intervention Type DRUG

Orally bid

Phase II: Placebo + abiraterone

Participants will receive placebo (for Ipatasertib) once daily, abiraterone 1000 mg once daily, and prednisone/prednisolone 5 mg bid continuously in 28-day treatment cycles until disease progression or intolerable toxicity.

Group Type PLACEBO_COMPARATOR

Abiraterone

Intervention Type DRUG

Orally once daily

Placebo

Intervention Type DRUG

Orally once daily

Prednisone

Intervention Type DRUG

Orally bid

Prednisolone

Intervention Type DRUG

Orally bid

Safety Cohort: Ipataseritib 400 mg + Abiraterone + Prednisone

Participants will receive ipatasertib 400 mg orally once daily and/or prednisone/prednisolone 5 mg orally once daily or bid and/or abiraterone 1000 mg orally once daily according to the following schedule: ipatasertib in the morning during Cycle 1, Days 1-7; ipatasertib in the morning plus prednisone/prednisolone once at night during Cycle 1, Day 8; ipatasertib in the morning plus prednisone/prednisolone bid (morning and night) during Cycle 1, Days 9-11; ipatasertib in the morning plus prednisone/prednisolone bid (morning and night) and abiraterone in the morning during Cycle 1, Days 12-18; ipatasertib in the evening plus prednisone/prednisolone bid (morning and night) and abiraterone at the same time as ipatasertib during Cycle 1, Days 19-25; Cycle 2 and beyond ipatasertib once daily in the morning or evening, abiraterone at the same time as ipatasertib, and prednisone/prednisolone bid.

Group Type EXPERIMENTAL

Abiraterone

Intervention Type DRUG

Orally once daily

Ipatasertib

Intervention Type DRUG

Orally once daily

Prednisone

Intervention Type DRUG

Orally bid

Prednisolone

Intervention Type DRUG

Orally bid

Interventions

Learn about the drugs, procedures, or behavioral strategies being tested and how they are applied within this trial.

Abiraterone

Orally once daily

Intervention Type DRUG

Apitolisib

Orally once daily

Intervention Type DRUG

Ipatasertib

Orally once daily

Intervention Type DRUG

Placebo

Orally once daily

Intervention Type DRUG

Prednisone

Orally bid

Intervention Type DRUG

Prednisolone

Orally bid

Intervention Type DRUG

Eligibility Criteria

Check the participation requirements, including inclusion and exclusion rules, age limits, and whether healthy volunteers are accepted.

Inclusion Criteria

* Histologically confirmed metastatic or advanced prostate adenocarcinoma that has been previously treated with docetaxel-based therapy and has progressed during treatment of at least one hormonal therapy(prior docetaxel is not required for the safety cohort)
* Two rising PSA levels greater than or equal to (\>/=) 2 ng/mL measured \>/= 1 week apart or radiographic evidence of disease progression in soft tissue or bone
* Eastern Cooperative Oncology Group (ECOG) performance status of 0 or 1 at screening
* Adequate hematologic and organ function
* Documented willingness to use an effective means of contraception
* Safety cohort only: agreement to use CGM for first cycle of treatment

Exclusion Criteria

* History of Type I or Type II diabetes mellitus requiring insulin; safety cohort: patients who are receiving any pharmacologic treatment for diabetes are not eligible
* New York Heart Association Class III or IV heart failure or Left ventricular ejection fraction \< 50% or ventricular arrhythmia requiring medication
* Significant atherosclerotic disease, as evidenced by: unstable angina, history of myocardial infarction within 6 months prior to Day 1, or cerebrovascular accident within 6 months prior to Day 1
* Active autoimmune disease that is not controlled by nonsteroidal anti-inflammatory drugs or active inflammatory disease which requires immunosuppressive therapy
* Clinically significant history of liver disease
* History of adrenal insufficiency or hyperaldosteronism
* Phase II only: Previous therapy for prostate cancer with 17 alpha-hydroxylase/C17,20-lyase inhibitors, including abiraterone
* Phase II only: Previous treatment for prostate cancer with Protein kinase B phosphatidylinositol 3 kinase and/or mammalian target of rapamycin inhibitors
* Need for chronic corticosteroid therapy of \>/= 20 mg of prednisone per day or an equivalent dose of other anti inflammatory corticosteroids or immunosuppressant
Minimum Eligible Age

18 Years

Eligible Sex

MALE

Accepts Healthy Volunteers

No

Sponsors

Meet the organizations funding or collaborating on the study and learn about their roles.

Genentech, Inc.

INDUSTRY

Sponsor Role lead

Responsible Party

Identify the individual or organization who holds primary responsibility for the study information submitted to regulators.

Responsibility Role SPONSOR

Principal Investigators

Learn about the lead researchers overseeing the trial and their institutional affiliations.

Clinical Trials

Role: STUDY_DIRECTOR

Genentech, Inc.

Locations

Explore where the study is taking place and check the recruitment status at each participating site.

HonorHealth Research Institute ? Bisgrove

Scottsdale, Arizona, United States

Site Status

Pacific Hematology Oncology Associates

San Francisco, California, United States

Site Status

Florida Cancer Specialists - Fort Myers (New Hampshire Ct)

Fort Myers, Florida, United States

Site Status

Florida Cancer Specialists; Sarasota

Sarasota, Florida, United States

Site Status

Kaiser Permanente Medical Ctr

Honolulu, Hawaii, United States

Site Status

Johns Hopkins Univ; Bunting Blaustein Cancer Center

Baltimore, Maryland, United States

Site Status

Karmanos Cancer Institute

Detroit, Michigan, United States

Site Status

Urology Cancer Center & GU Research Network

Omaha, Nebraska, United States

Site Status

New York Cancer and Blood Specialists - Setauket Medical Oncology

East Setauket, New York, United States

Site Status

Weill Cornell Medical College

New York, New York, United States

Site Status

Carolina Urologic Research Center

Myrtle Beach, South Carolina, United States

Site Status

Sarah Cannon Cancer Center - Tennessee Oncology, Pllc

Nashville, Tennessee, United States

Site Status

Masarykuv onkologicky ustav

Brno, , Czechia

Site Status

Fakultni nemocnice Hradec Kralove; I. interni klinika,Oddeleni invazivni kardiologie

Hradec Králové, , Czechia

Site Status

Urocentrum Praha s.r.o.

Prague, , Czechia

Site Status

Vseobecna fakultni nemocnice v Praze

Prague, , Czechia

Site Status

Fakultni Thomayerova Nemocnice; Revmatologicke Oddeleni

Prague, , Czechia

Site Status

ICO Paul Papin; Oncologie Medicale.

Angers, , France

Site Status

Centre Léon Bérard - Centre régional de lutte contre le cancer Rhône-Alpes

Lyon, , France

Site Status

Hia Du Val De Grace

Paris, , France

Site Status

Institut Curie; Oncologie Medicale

Paris, , France

Site Status

GH Paris Saint Joseph; Hopital De Jour Oncologie

Paris, , France

Site Status

Hopital d'Instruction des Armees de Begin

Saint-Mandé, , France

Site Status

Institut Gustave Roussy; Departement Oncologie Medicale

Villejuif, , France

Site Status

Alexandras Hospital; Dept. of Clin. Therapeutics, Athens Uni School of Medicine

Athens, , Greece

Site Status

Univ General Hosp Heraklion; Medical Oncology

Heraklion, , Greece

Site Status

University Hospital of Larissa; Oncology

Larissa, , Greece

Site Status

University Hospital of Patras Medical Oncology

Pátrai, , Greece

Site Status

Metropolitan Hospital; 2Nd Oncology Clinic

Piraeus, , Greece

Site Status

IRST Istituto Scientifico Romagnolo Per Lo Studio E Cura Dei Tumori, Sede Meldola; Oncologia Medica

Meldola, Emilia-Romagna, Italy

Site Status

Azienda Ospedaliera Istituti Ospitalieri

Cremona, Lombardy, Italy

Site Status

Irccs Ospedale San Raffaele;Oncologia Medica

Milan, Lombardy, Italy

Site Status

Irccs Istituto Nazionale Dei Tumori (Int);S.C. Medicina Oncologica 2

Milan, Lombardy, Italy

Site Status

Ospedale S. Donato; Divisione Di Reumatologia

Arezzo, Tuscany, Italy

Site Status

Het Nederlands Kanker Inst

Amsterdam, , Netherlands

Site Status

Vu Medisch Centrum; Afdeling Longziekten

Amsterdam, , Netherlands

Site Status

UMC St Radboud

Nijmegen, , Netherlands

Site Status

Sint Franciscus Gasthuis; Inwendige Geneeskunde

Rotterdam, , Netherlands

Site Status

MC Haaglanden; Oncologie

The Hague, , Netherlands

Site Status

Sf. Constantin Hospital; Oncology

Brasov, , Romania

Site Status

Prof. Dr. Th. Burghele Clin Urology Hosp

Bucharest, , Romania

Site Status

Prof. Dr. I. Chiricuta Institute of Oncology

Cluj-Napoca, , Romania

Site Status

ONCOMED - Medical Centre

Timișoara, , Romania

Site Status

Municipal Hosp Turdal; Oncology

Turda, , Romania

Site Status

Hospital General Universitario de Elche; Servicio de Oncologia

Elche, Alicante, Spain

Site Status

Hospital Universitari Germans Trias i Pujol; Servicio de Oncologia

Badalona, Barcelona, Spain

Site Status

Corporacio Sanitaria Parc Tauli; Servicio de Oncologia

Sabadell, Barcelona, Spain

Site Status

Hospital Univ Vall d'Hebron; Servicio de Oncologia

Sant Andreu de la Barca, Barcelona, Spain

Site Status

Clinica Universitaria de Navarra

Pamplona, Navarre, Spain

Site Status

Hospital General Universitario Gregorio Marañon

Madrid, , Spain

Site Status

Hospital Universitario 12 de Octubre; Servicio de Oncologia

Madrid, , Spain

Site Status

Hospital Madrid Norte Sanchinarro

Madrid, , Spain

Site Status

Hospital Clinico Universitario Virgen de la Victoria

Málaga, , Spain

Site Status

Queen Elizabeth Hospital; Centre for Clinical Haematology

Birmingham, , United Kingdom

Site Status

Gartnavel General Hospital

Glasgow, , United Kingdom

Site Status

St. James University Hospital; Pharmacy Department

Leeds, , United Kingdom

Site Status

The Clatterbridge Cancer Centre NHS Foundation Trust

Liverpool, , United Kingdom

Site Status

Sarah Cannon Research Institute

London, , United Kingdom

Site Status

The Royal Marsden Hospital

Sutton, , United Kingdom

Site Status

Countries

Review the countries where the study has at least one active or historical site.

United States Czechia France Greece Italy Netherlands Romania Spain United Kingdom

Other Identifiers

Review additional registry numbers or institutional identifiers associated with this trial.

2011-004126-10

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

GO27983

Identifier Type: -

Identifier Source: org_study_id

More Related Trials

Additional clinical trials that may be relevant based on similarity analysis.