Study to Evaluate Switching From Regimens Consisting of a Ritonavir-boosted Protease Inhibitor Plus Emtricitabine/Tenofovir Fixed-Dose Combination to the Elvitegravir/Cobicistat/Emtricitabine/Tenofovir DF Single-Tablet Regimen in Virologically Suppressed, HIV-1 Infected Patients

NCT ID: NCT01475838

Last Updated: 2016-06-08

Study Results

Results available

Outcome measurements, participant flow, baseline characteristics, and adverse events have been published for this study.

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE3

Total Enrollment

438 participants

Study Classification

INTERVENTIONAL

Study Start Date

2011-11-30

Study Completion Date

2014-12-31

Brief Summary

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This study will evaluate the non-inferiority of Stribild® (elvitegravir/cobicistat/ emtricitabine/tenofovir disoproxil fumarate (E/C/F/TDF)) single-tablet regimen (STR) relative to regimens consisting of a protease inhibitor (PI) boosted with ritonavir (RTV) plus Truvada® (FTC/TDF) fixed-dose combination in maintaining HIV-1 RNA \< 50 copies/mL at Week 48 in virologically suppressed, HIV-1 infected adults. This study will also evaluate the safety, tolerability, and efficacy of the two regimens through 96 weeks of treatment.

Detailed Description

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Conditions

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Acquired Immunodeficiency Syndrome HIV Infections

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Stribild

Participants will switch from their baseline treatment regimen to Stribild for up to 96 weeks, and may continue to receive Stribild in the extension phase.

Group Type EXPERIMENTAL

Stribild

Intervention Type DRUG

Stribild (E/C/F/TDF) (150/150/200/300 mg) STR administered orally once daily with food

PI+RTV+FTC/TDF

Participants will stay on their baseline treatment regimen antiretroviral regimen consisting of a PI boosted with RTV plus FTC/TDF for up to 96 weeks, and may switch to Stribild in the extension phase.

Group Type ACTIVE_COMPARATOR

PI

Intervention Type DRUG

PI administered according to prescribing information; allowed PIs include atazanavir (ATV), darunavir (DRV), fosamprenavir (FPV), lopinavir (LPV), or saquinavir (SQV)

RTV

Intervention Type DRUG

RTV administered according to prescribing information FTC/TDF administered according to prescribing information

FTC/TDF

Intervention Type DRUG

FTC/TDF (200/300 mg) administered according to prescribing information

Stribild

Intervention Type DRUG

Stribild (E/C/F/TDF) (150/150/200/300 mg) STR administered orally once daily with food

Interventions

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PI

PI administered according to prescribing information; allowed PIs include atazanavir (ATV), darunavir (DRV), fosamprenavir (FPV), lopinavir (LPV), or saquinavir (SQV)

Intervention Type DRUG

RTV

RTV administered according to prescribing information FTC/TDF administered according to prescribing information

Intervention Type DRUG

FTC/TDF

FTC/TDF (200/300 mg) administered according to prescribing information

Intervention Type DRUG

Stribild

Stribild (E/C/F/TDF) (150/150/200/300 mg) STR administered orally once daily with food

Intervention Type DRUG

Other Intervention Names

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Truvada

Eligibility Criteria

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Inclusion Criteria

* Ability to understand and sign a written informed consent form
* Be on a stable antiretroviral regimen consisting of a ritonavir boosted PI plus FTC/TDF continuously for ≥ 6 consecutive months preceding the screening visit
* Be on the first or second antiretroviral drug regimen documented undetectable plasma HIV 1 RNA levels for ≥ 6 months preceding the screening visit
* No previous use of any approved or experimental integrase strand transfer inhibitor (INSTI) for any length of time
* Documented historical genotype prior to starting initial antiretroviral therapy showing no known resistance to TDF or FTC
* HIV RNA \< 50 copies/mL at screening
* Normal ECG
* Hepatic transaminases ≤ 5 × the upper limit of the normal range (ULN)
* Total bilirubin ≤ 1.5 mg/dL, or normal direct bilirubin
* Adequate hematologic function
* Serum amylase ≤ 5 × ULN
* Estimated glomerular filtration rate ≥ 70 mL/min
* Females of childbearing potential must agree to utilize highly effective contraception methods, or be nonheterosexually active, practice sexual abstinence from screening throughout the duration of the study period and for 30 days following the last dose of study drug
* Female participants who utilize hormonal contraceptive as one of their birth control methods must have used the same method for at least three months prior to study dosing
* Male participants must agree to utilize a highly effective method of contraception during heterosexual intercourse from the screening visit, throughout the duration of the study and for 30 days following discontinuation of investigational medicinal product, or must be nonheterosexually active, or practice sexual abstinence
* Age ≥ 18 years

Exclusion Criteria

* A new AIDS-defining condition diagnosed within the 30 days prior to screening
* Females who are breastfeeding
* Positive serum pregnancy test (female of childbearing potential)
* Receiving drug treatment for hepatitis C, or participants who are anticipated to receive treatment for hepatitis C during the course of the study
* Experiencing decompensated cirrhosis
* Have an implanted defibrillator or pacemaker
* Current alcohol or substance abuse that would interfere with compliance
* A history of malignancy within the past 5 years or ongoing malignancy other than cutaneous Kaposi's sarcoma, basal cell carcinoma, or resected, noninvasive cutaneous squamous carcinoma
* Active, serious infections requiring parenteral antibiotic or antifungal therapy within 30 days prior to Baseline, except for intramuscular penicillin for the treatment of syphilis
* Have been treated with immunosuppressant therapies or chemotherapeutic agents within 3 months of study screening, or expected to receive these agents or systemic steroids during the study
* Receiving ongoing therapy with any of the medications, including drugs not to be used with elvitegravir, cobicistat, FTC, or TDF; or those with any known allergies to the excipients of E/C/F/TDF tablets, or FTC/TDF tablets
* No anticipated need to initiate drugs during the study that are contraindicated
* Receiving other investigational drugs
* Participation in any other clinical trial
* Any other clinical condition or prior therapy that would make the participant unsuitable for the study or unable to comply with the dosing requirements
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Gilead Sciences

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Thai Nguyen-Cleary

Role: STUDY_DIRECTOR

Gilead Sciences

Locations

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Hospital Universitari Bellvitge HIV Unit. Infectious Disease Service.

Barcelona, , Spain

Site Status

Hospital Germans Trias I Pujol

Barcelona, , Spain

Site Status

Spectrum Medical Group

Phoenix, Arizona, United States

Site Status

Pueblo Family Physicians

Phoenix, Arizona, United States

Site Status

AIDS Healthcare Foundation

Beverly Hills, California, United States

Site Status

Pacific Oaks Medical Group

Beverly Hills, California, United States

Site Status

Kaiser Permanente

Hayward, California, United States

Site Status

Kaiser Permanente

Los Angeles, California, United States

Site Status

Peter J. Ruane, M.D., Inc.

Los Angeles, California, United States

Site Status

OASIS Clinic

Los Angeles, California, United States

Site Status

Anthony Mills MD Inc

Los Angeles, California, United States

Site Status

Stanford University

Palo Alto, California, United States

Site Status

University of California, Davis

Sacramento, California, United States

Site Status

Kaiser Permanente

Sacramento, California, United States

Site Status

La Playa Medical Group and Clinical Research

San Diego, California, United States

Site Status

Metropolis Medical

San Francisco, California, United States

Site Status

Kaiser Permanente San Francisco

San Francisco, California, United States

Site Status

Dupont Circle Physicians Group, P.C

Washington D.C., District of Columbia, United States

Site Status

Capital Medical Associates, PC

Washington D.C., District of Columbia, United States

Site Status

Gary Richmond, MD

Fort Lauderdale, Florida, United States

Site Status

Midway Immunology & Research Center, LLC

Ft. Pierce, Florida, United States

Site Status

The Kinder Medical Group

Miami, Florida, United States

Site Status

Orlando Immunology Center

Orlando, Florida, United States

Site Status

Idocf/Valuhealthmd, Llc

Orlando, Florida, United States

Site Status

Infectious Diseases Associates of NW FL, P.A.

Pensacola, Florida, United States

Site Status

AHF Health Positive Tampa Bay

Safety Harbor, Florida, United States

Site Status

St. Joseph's Comprehensive Research Institute

Tampa, Florida, United States

Site Status

Atlanta ID Group

Atlanta, Georgia, United States

Site Status

Northwestern University Division of Infectious Diseases

Chicago, Illinois, United States

Site Status

John H. Stroger, Jr. Hospital of Cook County/Ruth M. Rothstein CORE Center

Chicago, Illinois, United States

Site Status

Be Well Medical Center

Berkley, Michigan, United States

Site Status

Hennepin County Medical Center

Minneapolis, Minnesota, United States

Site Status

The Kansas City Free Health Clinic

Kansas City, Missouri, United States

Site Status

I.D. Care Associates PA

Hillsborough, New Jersey, United States

Site Status

Saint Michael's Medical Center

Newark, New Jersey, United States

Site Status

South Jersey Infectious Disease

Somers Point, New Jersey, United States

Site Status

Greiger Clinic

Mount Vernon, New York, United States

Site Status

ID Consultants, P.A.

Charlotte, North Carolina, United States

Site Status

Wake Forest University Health Sciences

Winston-Salem, North Carolina, United States

Site Status

University of Pennsylvania

Philadelphia, Pennsylvania, United States

Site Status

Philadelphia FIGHT

Philadelphia, Pennsylvania, United States

Site Status

Uptown Physicians Group

Dallas, Texas, United States

Site Status

Southwest Infectious Disease Clinical Research, Inc

Dallas, Texas, United States

Site Status

Tarrant County Infectious Disease Associates

Fort Worth, Texas, United States

Site Status

Therapeutic Concepts, PA

Houston, Texas, United States

Site Status

Gordon Crofoot Md, Pa

Houston, Texas, United States

Site Status

St. Hope Foundation Inc

Houston, Texas, United States

Site Status

Innsbruck Medical University

Innsbruck, , Austria

Site Status

Univ.-Kklinik fuer Innere Medizin III

Salzburg, , Austria

Site Status

Medical University of Vienna

Vienna, , Austria

Site Status

Otto-Wagner-Spital

Vienna, , Austria

Site Status

UCL Saint Luc

Brussels, , Belgium

Site Status

University Hospital Ghent

Ghent, , Belgium

Site Status

CHU Sart Tilman

Liège, , Belgium

Site Status

Sunnybrook Health Sciences Centre

Toronto, Ontario, Canada

Site Status

Clinique Medicale Du Quartier Latin

Montreal, Quebec, Canada

Site Status

CHU de Besancon, Hopital Saint-Jacques

Besançon, , France

Site Status

Hôpital de la Croix-Rousse

Lyon, , France

Site Status

CHU Hôpital Gui de Chauliac

Montpellier, , France

Site Status

Archet 1 Chu Nice Department of Infectology

Nice, , France

Site Status

Saint-Louis Hospital

Paris, , France

Site Status

Hopital Saint Antoine

Paris, , France

Site Status

Hôpital Bichat-Claude Bernard

Paris, , France

Site Status

hôpital Tenon

Paris, , France

Site Status

Maladies Infectieuses Dpt

Paris, , France

Site Status

Hôpital Haut Lévêque

Pessac, , France

Site Status

Epimed GmbH

Berlin, , Germany

Site Status

University of Bonn

Bonn, , Germany

Site Status

Infektlonsambulanz Unlkllnik Koln

Cologne, , Germany

Site Status

Universitätsklinikum Essen, Dermatologie, HIV Ambulanz

Essen, , Germany

Site Status

Johann Wolfgang Goethe-University Hospital / Infectious Diseases Hs 68

Frankfurt, , Germany

Site Status

ICH Study Center

Hamburg, , Germany

Site Status

Universitätsklinikum Hamburg-Eppendorf, Ambulanzzentrum des UKE GmbH, Bereich Infektiologie

Hamburg, , Germany

Site Status

Medizinische Hochschule Hannover

Hanover, , Germany

Site Status

Infektionsambulanz, Med Poliklink, Klinikum der Universitat Munchnen

Munich, , Germany

Site Status

Ospedali Riuniti

Bergamo, , Italy

Site Status

Hospital General Universitario de Elche

Elche, Alicante, , Spain

Site Status

Fondazione Centro San Raffaele

Milan, , Italy

Site Status

Clinic of Infectious Diseases, University of Milan-San Paolo Hospital

Milan, , Italy

Site Status

Ospedale Luigi Sacco

Milan, , Italy

Site Status

National Institute for Infectious Diseases "L. Spallanzani"

Rome, , Italy

Site Status

University of Torino, Dept of Infectious Disease

Torino, , Italy

Site Status

HHP Hospital de Cascais

Alcabideche, , Portugal

Site Status

Hospital de Santa Maria-CHLN, EPE

Lisbon, , Portugal

Site Status

Hospital Santo Antonio Dos Capuchos, Centro Hospitalar de Lisboa

Lisbon, , Portugal

Site Status

Clinical Research Puert Rico

San Juan, , Puerto Rico

Site Status

University of Puerto Rico School of Medicine

San Juan, , Puerto Rico

Site Status

Hospital General Universitario Alicante

Alicante, , Spain

Site Status

Hospital clinic

Barcelona, , Spain

Site Status

Infectious Diseases Department, Hospital Carlos III

Madrid, , Spain

Site Status

Hospital Ramon y Cajal

Madrid, , Spain

Site Status

Hospital La Paz

Madrid, , Spain

Site Status

Hospital Virgen del Rocio

Seville, , Spain

Site Status

Geneva University Hospital

Geneva, , Switzerland

Site Status

University Hospital of Zurich; Division of Infectious Diseases and Hospital Epidemiology

Zurich, , Switzerland

Site Status

Zentrum fur Infektionskrankheiten

Zurich, , Switzerland

Site Status

Brighton and Sussex University Hospitals NHS Trust

Brighton, , United Kingdom

Site Status

Royal Free Hampstead NHS Trust

London, , United Kingdom

Site Status

Chelsea and Westminster

London, , United Kingdom

Site Status

Countries

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United States Austria Belgium Canada France Germany Italy Portugal Puerto Rico Spain Switzerland United Kingdom

References

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Arribas JR, Pialoux G, Gathe J, Di Perri G, Reynes J, Tebas P, Nguyen T, Ebrahimi R, White K, Piontkowsky D. Simplification to coformulated elvitegravir, cobicistat, emtricitabine, and tenofovir versus continuation of ritonavir-boosted protease inhibitor with emtricitabine and tenofovir in adults with virologically suppressed HIV (STRATEGY-PI): 48 week results of a randomised, open-label, phase 3b, non-inferiority trial. Lancet Infect Dis. 2014 Jul;14(7):581-9. doi: 10.1016/S1473-3099(14)70782-0. Epub 2014 Jun 5.

Reference Type RESULT
PMID: 24908551 (View on PubMed)

Pozniak A, Markowitz M, Mills A, Stellbrink HJ, Antela A, Domingo P, Girard PM, Henry K, Nguyen T, Piontkowsky D, Garner W, White K, Guyer B. Switching to coformulated elvitegravir, cobicistat, emtricitabine, and tenofovir versus continuation of non-nucleoside reverse transcriptase inhibitor with emtricitabine and tenofovir in virologically suppressed adults with HIV (STRATEGY-NNRTI): 48 week results of a randomised, open-label, phase 3b non-inferiority trial. Lancet Infect Dis. 2014 Jul;14(7):590-9. doi: 10.1016/S1473-3099(14)70796-0. Epub 2014 Jun 5.

Reference Type RESULT
PMID: 24908550 (View on PubMed)

Arribas JR, DeJesus E, van Lunzen J, Zurawski C, Doroana M, Towner W, Lazzarin A, Nelson M, McColl D, Andreatta K, Swamy R, Szwarcberg J, Nguyen T. Simplification to single-tablet regimen of elvitegravir, cobicistat, emtricitabine, tenofovir DF from multi-tablet ritonavir-boosted protease inhibitor plus coformulated emtricitabine and tenofovir DF regimens: week 96 results of STRATEGY-PI. HIV Clin Trials. 2017 May;18(3):118-125. doi: 10.1080/15284336.2017.1330440. Epub 2017 May 30.

Reference Type DERIVED
PMID: 28555519 (View on PubMed)

Gathe J, Arribas JR, Van Lunzen J, Garner W, Speck RM, Bender R, Shreay S, Nguyen T. Patient-Reported Symptoms over 48 Weeks in a Randomized, Open-Label, Phase 3b Non-inferiority Trial of Adults with HIV Switching to Coformulated Elvitegravir, Cobicistat, Emtricitabine, and Tenofovir DF Versus Continuation of Ritonavir-Boosted Protease Inhibitor with Emtricitabine and Tenofovir DF. Patient. 2015 Oct;8(5):445-54. doi: 10.1007/s40271-015-0137-9.

Reference Type DERIVED
PMID: 26286337 (View on PubMed)

Other Identifiers

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2011-004483-30

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

GS-US-236-0115

Identifier Type: -

Identifier Source: org_study_id

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