Pharmacokinetics of RLX030 in Subjects With Mild, Moderate and Severe Hepatic Impairment Compared to Healthy Subjects

NCT ID: NCT01433458

Last Updated: 2020-12-21

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

55 participants

Study Classification

INTERVENTIONAL

Study Start Date

2011-07-31

Study Completion Date

2011-12-31

Brief Summary

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This study will assess the pharmacokinetics of RLX030 during and after administration in subjects with mild to severe hepatic impairment and matched healthy control subjects.

20 to 24 patients and 20 to 24 healthy subjects will be enrolled.

Detailed Description

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Conditions

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Hepatic Impairment

Keywords

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Hepatic impairment healthy volunteers RLX030 pharmacokinetics

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

OTHER

Blinding Strategy

NONE

Study Groups

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RLX030: Group 1 mild hepatic impairment

Patients with mild hepatic impairment will receive a single IV 24 hour infusion of RLX030

Group Type EXPERIMENTAL

RLX030A

Intervention Type DRUG

RLX030 is administered as a continuous 24 hour infusion

RLX030: Group 2 moderate hepatic impairment

Patients with moderate hepatic impairment will receive a single IV 24 hour infusion of RLX030

Group Type EXPERIMENTAL

RLX030A

Intervention Type DRUG

RLX030 is administered as a continuous 24 hour infusion

RLX030: Group 3 severe hepatic impairment

Patients with severe hepatic impairment will receive a single IV 24 hour infusion of RLX030

Group Type EXPERIMENTAL

RLX030A

Intervention Type DRUG

RLX030 is administered as a continuous 24 hour infusion

RLX030: Group 4 - healthy volunteers

Participants will receive a single IV 24 hour infusion of RLX030. This group will consist of 3 sub-groups to match patients of groups 1, 2and 3.

Group Type ACTIVE_COMPARATOR

RLX030A

Intervention Type DRUG

RLX030 is administered as a continuous 24 hour infusion

Interventions

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RLX030A

RLX030 is administered as a continuous 24 hour infusion

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* All subjects:

• Female subjects must be of non-child bearing potential OR use an effective method of contraception and sexually active males must use a condom during intercourse while taking the drug and for 5 half-lives after stopping treatment
* Subjects with hepatic impairment:

* Subjects must have either mild, moderate or severe hepatic impairment

Exclusion Criteria

* All subjects

* Hepatic impairment due to non-liver disease
* Use of other investigational drugs at time of enrollment
* History of malignancy of any organ system
* Donation or loss of 400 mL or more of blood or plasma within 8 weeks prior to initial dosing
* Hemoglobin levels below 10.0 g/dL at screening or baseline
* Subjects with hepatic impairment:

* Presence of any non-controlled and clinically significant disease that could affect the study outcome or that would place the patient at undue risk
* Treatment with any cytostatic drug, vasodilator, autonomic alpha blocker or B2 agonist
* Any surgical or medical condition other than hepatic impairment which might significantly alter the distribution or excretion of drugs
Minimum Eligible Age

18 Years

Maximum Eligible Age

70 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

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Novartis Pharmaceuticals

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Novartis Pharmaceuticals

Role: STUDY_DIRECTOR

Novartis Pharmaceuticals

Locations

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Novartis Investigative Site

Grünstadt, , Germany

Site Status

Novartis Investigative Site

Moscow, , Russia

Site Status

Countries

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Germany Russia

References

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Kobalava Z, Villevalde S, Kotovskaya Y, Hinrichsen H, Petersen-Sylla M, Zaehringer A, Pang Y, Rajman I, Canadi J, Dahlke M, Lloyd P, Halabi A. Pharmacokinetics of serelaxin in patients with hepatic impairment: a single-dose, open-label, parallel group study. Br J Clin Pharmacol. 2015 Jun;79(6):937-45. doi: 10.1111/bcp.12572.

Reference Type DERIVED
PMID: 25511105 (View on PubMed)

Related Links

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https://www.novctrd.com/ctrdweb/trialresult/trialresults/pdf?trialResultId=7565

Results for CRLX030A2101 can be found on the Novartis Clinical Trial Results Website

Other Identifiers

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2011-001596-39

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

CRLX030A2101

Identifier Type: -

Identifier Source: org_study_id