A Study to Evaluate The Pharmacokinetics Of Crizotinib (PF-02341066) In Subjects With Impaired Renal Function

NCT ID: NCT01419041

Last Updated: 2012-10-01

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

16 participants

Study Classification

INTERVENTIONAL

Study Start Date

2011-11-30

Study Completion Date

2012-08-31

Brief Summary

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The present study is being conducted to evaluate whether or not severe renal impairment has an effect on crizotinib Pharmacokinetics.

Detailed Description

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Conditions

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Renal Impairment

Keywords

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renal impairment crizotinib pharmacokinetics

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

BASIC_SCIENCE

Blinding Strategy

NONE

Study Groups

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Arm A

CLCR: Creatinine clearance

Group Type OTHER

crizotinib

Intervention Type DRUG

Single-dose oral 250 mg crizotinib in subjects with normal renal function (CLcr =\>90 mL/min)

Arm B

CLCR: Creatinine clearance

Group Type OTHER

crizotinib

Intervention Type DRUG

Single-dose oral 250 mg crizotinib in subjects with severe renal impairment (CLcr \<30 mL/min)

Interventions

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crizotinib

Single-dose oral 250 mg crizotinib in subjects with normal renal function (CLcr =\>90 mL/min)

Intervention Type DRUG

crizotinib

Single-dose oral 250 mg crizotinib in subjects with severe renal impairment (CLcr \<30 mL/min)

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

All Subjects

* Healthy male and/or female of non childbearing potential subjects between the ages of 18 and 65 years, inclusive ('healthy' is defined as no clinically relevant abnormalities identified by a detailed medical history, full physical examination, including blood pressure and pulse rate measurement, 12 lead ECG, and clinical laboratory tests).
* Body Mass Index (BMI) of 18 to 40 kg/m2 inclusive; and a total body weight \>50 kg (\>110 lbs).

Subjects with Normal Renal Function (Group 1)

* Normal renal function (CLcr =\>90 mL/min) during the screening period.
* Matched 1-to-1 to subjects in Group 2 with respect to age (+/-5 years), weight (+/-10 kg), gender, and race according to protocol.

Subjects with Severe Renal Impairment (Groups 2)

* Good general health commensurate with the population with chronic kidney disease.
* Severe renal impairment (CLcr\<30 mL/min) during the screening period.

Exclusion Criteria

All Subjects

* Renal allograft recipients.
* Any condition possibly affecting drug absorption.
* 12 lead ECG demonstrating QTc \>470 msec at screening.
* Urinary incontinence without catheterization.
* A positive urine drug screen.
* History of regular alcohol consumption.
* Treatment with an investigational drug within 30 days (or as determined by the local requirement, whichever is longer) or 5 half lives preceding the first dose of study medication.
* Pregnant or nursing females; females of childbearing potential, including those with tubal ligation.
* Blood donation of approximately 1 pint (500 mL) within 56 days prior to dosing.

Subjects with Severe Renal Impairment (Groups 2)

* Subjects with any significant hepatic, cardiac or pulmonary disease (apart from stable ischemic heart disease), or subjects who are clinically nephrotic.
* Subjects requiring hemodialysis.
* Subjects with strict fluid restriction (ie, \<1500 mL/24 hours).
* Significant bleeding diathesis which could preclude multiple venipuncture.
* Use of food or drugs that are CYP3A4 inhibitors and inducers.
* Herbal supplements and hormone replacement therapy must be discontinued 28 days prior to the first dose of trial medication
* Concurrent use of drugs that are CYP3A4 substrates with narrow therapeutic indices.
Minimum Eligible Age

18 Years

Maximum Eligible Age

75 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

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Pfizer

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Pfizer CT.gov Call Center

Role: STUDY_DIRECTOR

Pfizer

Locations

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Pfizer Investigational Site

Anaheim, California, United States

Site Status

Pfizer Investigational Site

DeLand, Florida, United States

Site Status

Pfizer Investigational Site

Saint Paul, Minnesota, United States

Site Status

Countries

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United States

Related Links

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Other Identifiers

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A8081020

Identifier Type: -

Identifier Source: org_study_id