Open-label Study of the Safety and Activity of Oprozomib in Patients With Hematologic Malignancies

NCT ID: NCT01416428

Last Updated: 2022-11-08

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

TERMINATED

Clinical Phase

PHASE1/PHASE2

Total Enrollment

210 participants

Study Classification

INTERVENTIONAL

Study Start Date

2011-10-15

Study Completion Date

2019-08-12

Brief Summary

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The purpose of this study is to determine the maximum tolerated dose (MTD), activity, and safety of oprozomib in patients with hematologic malignancies.

Detailed Description

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Conditions

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Multiple Myeloma Waldenstrom Macroglobulinemia

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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QDx2 Dosing Schedule

QDx2 is defined as patients receiving Oprozomib Tablets once daily on Days 1, 2, 8, and 9 of the 14-day cycle.

The schedule will be evaluated in Phase 1 for MTD in patients with hematologic malignancies, and will also be evaluated in Phase 2 for ORR in patients with MM and WM.

Group Type EXPERIMENTAL

oprozomib

Intervention Type DRUG

Patients enrolled will receive Oprozomib Tablets once daily either on Days 1-5 (QDx5 schedule) or on Days 1, 2, 8, and 9 (QDx2 weekly schedule) of the 14-day treatment cycle.

QDx5 Dosing Schedule

QDx5 is defined as patients receiving Oprozomib Tablets once daily on Days 1 to 5 of the 14-day cycle.

The schedule will be evaluated in Phase 1 for MTD in patients with hematologic malignancies, and will also be evaluated in Phase 2 for ORR in patients with MM and WM.

Group Type EXPERIMENTAL

oprozomib

Intervention Type DRUG

Patients enrolled will receive Oprozomib Tablets once daily either on Days 1-5 (QDx5 schedule) or on Days 1, 2, 8, and 9 (QDx2 weekly schedule) of the 14-day treatment cycle.

Interventions

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oprozomib

Patients enrolled will receive Oprozomib Tablets once daily either on Days 1-5 (QDx5 schedule) or on Days 1, 2, 8, and 9 (QDx2 weekly schedule) of the 14-day treatment cycle.

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

Phase 1b

* Histologically confirmed diagnosis of a hematologic malignancy, excluding patients with acute leukemia or MDS.
* Relapsed after standard therapy for their malignancy and considered to be an appropriate candidate for a Phase 1 clinical study by their treating physician.

Phase 2

* Multiple myeloma with measurable disease
* Waldenström macroglobulinemia with symptomatic relapse
* Eastern Cooperative Oncology Group (ECOG) Performance Status 0-2.

Ethical/Other

* Patients must sign a written informed consent form in accordance with federal, local, and institutional guidelines.
* Female patients of childbearing potential must have a negative serum or urine pregnancy test and agree to use effective contraception. Male patients must use an effective barrier method of contraception.

Exclusion Criteria

* Chemotherapy with approved or investigational anticancer therapeutics, including steroid therapy intended to treat underlying malignancy, within 3 weeks prior to first dose or 6 weeks for antibody therapy.
* Radiation therapy within 3 weeks prior to first dose. Radioimmunotherapy within 8 weeks prior to first dose. Localized radiation therapy within 1 week prior to first dose.
* Immunotherapy within 3 weeks prior to first dose (except for antibody therapy, where 6 weeks is required).
* Prior stem cell transplant (SCT) therapy (autologous SCT within the prior 8 weeks; allogeneic SCT within the prior 16 weeks). Patients with prior allogeneic SCT should not have evidence of moderate-to-severe graft-vs-host disease (GvHD; as defined in Filipovich 2005).
* Evidence of central nervous system (CNS) lymphoma.
* Prior treatment with carfilzomib unless in the phase 2.
* Major surgery within 3 weeks prior to first dose.
* Symptomatic Congestive heart failure, ischemia, conduction abnormalities, or myocardial infarction within 6 months.
* Acute active infection requiring systemic antibiotics, antivirals, or antifungals.
* Known or suspected human immunodeficiency virus (HIV) infection or patients who are HIV seropositive.
* Active hepatitis A, B, or C infection.
* Significant neuropathy (Grade 3, Grade 4, or Grade 2 with pain) at the time of the first dose.
* Patients with pleural effusions requiring routine thoracentesis or ascites requiring routine paracentesis.
* History of previous clinically significant GI bleed in the last 6 months prior to first dose.
* Female patients who are pregnant or lactating.
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Amgen

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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MD

Role: STUDY_DIRECTOR

Amgen

Locations

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Mayo Clinic Scottsdale

Scottsdale, Arizona, United States

Site Status

Pacific Cancer Care

Salinas, California, United States

Site Status

Colorado Blood Cancer Institute

Denver, Colorado, United States

Site Status

Mayo Clinic

Jacksonville, Florida, United States

Site Status

Winship Cancer Institute, Emory University

Atlanta, Georgia, United States

Site Status

Rush University Medical Center

Chicago, Illinois, United States

Site Status

University of Chicago Medical Center

Chicago, Illinois, United States

Site Status

University of Maryland, Greenebaum Cancer Center

Baltimore, Maryland, United States

Site Status

Dana Farber Cancer Institute

Boston, Massachusetts, United States

Site Status

Mass General Hospital

Boston, Massachusetts, United States

Site Status

Virginia Piper Cancer Institute

Minneapolis, Minnesota, United States

Site Status

Mayo Clinic

Rochester, Minnesota, United States

Site Status

Washington University School of Medicine Division of Oncology

St Louis, Missouri, United States

Site Status

John Theurer Cancer Center at Hackensack University

Hackensack, New Jersey, United States

Site Status

Hematology Oncology of Northern New Jersey

Morristown, New Jersey, United States

Site Status

New York Oncology Hematology

Albany, New York, United States

Site Status

Mount Sinai Medical Center

New York, New York, United States

Site Status

Sarah Cannon Research Institute / Tennessee Oncology, PLLC

Nashville, Tennessee, United States

Site Status

Columbia Basin Hematology and Oncology

Kennewick, Washington, United States

Site Status

Countries

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United States

Related Links

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http://www.amgentrials.com

AmgenTrials clinical trials website

Other Identifiers

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2011-001

Identifier Type: -

Identifier Source: org_study_id

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