Study of AEB071 (a Protein Kinase C Inhibitor) in Patients With CD79-mutant Diffuse Large B-Cell Lymphoma

NCT ID: NCT01402440

Last Updated: 2020-12-19

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

TERMINATED

Clinical Phase

PHASE1

Total Enrollment

15 participants

Study Classification

INTERVENTIONAL

Study Start Date

2011-11-30

Study Completion Date

2014-04-30

Brief Summary

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This study has two phases, a dose escalation phase and a dose expansion phase. For dose escalation, the primary objective is to estimate the maximum tolerated dose of AEB071 in patients with diffuse large b-cell lymphoma. The endpoint for this objective will be occurrence of Dose Limiting Toxicity. For dose expansion, the primary objective is to characterize the safety and tolerability of the maximum tolerated dose or recommended phase 2 dose of AEB071 in patients with diffuse large b-cell lymphoma. The endpoints for this objective will be occurrence of Adverse Events (AEs), Serious Adverse Events (SAEs), assessment of clinical laboratory values, and vital sign measurements.

Detailed Description

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Conditions

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Diffuse Large B-Cell Lymphoma

Keywords

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Diffuse Large B-Cell Lymphoma, Phase 1, CD79 Mutation

Study Design

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Allocation Method

NA

Intervention Model

SINGLE_GROUP

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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AEB071

Group Type EXPERIMENTAL

AEB071

Intervention Type DRUG

Interventions

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AEB071

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Diffuse large B-cell lymphoma (DLBCL) with activating mutations in CD79 (A or B subunits). DLBCL that arose from transformed indolent lymphoma is allowed.
* Prior treatment and relapse following anthracycline-based chemotherapy and autologous bone marrow or stem cell transplant. Patients who are not transplant eligible may be considered for the study following a single regimen of chemotherapy such as R-CHOP or R-EPOCH alone. There is no limit to prior therapy allowed.

* Patients may be treated with localized radiation to as many as two sites of disease, so long as measurable or evaluable disease remains at untreated sites.
* Patients may be treated with corticosteriods immediately prior to enrollment and during the course of the study treatment as long as steriod treatment is tapered to a toal daily dosage of 10mg or less of prednisone (or it's equivalent) prior to AEB071 administration
* WHO performance status of ≤2

Exclusion Criteria

* Patients at screening who are treated with strong inducers or inhibitors of cytochrome P450 3A4 (CYP3A4) that can not be discontinued.
* Impaired cardiac function or clinically significant cardiac diseases, including any of the following:
* History or presence of ventricular tachyarrhythmia
* Angina pectoris or acute myocardial infarction ≤ 3 months prior to starting study drug
* Other clinically significant heart disease (e.g., symptomatic congestive heart failure; uncontrolled arrhythmia or hypertension; history of labile hypertension or poor compliance with an antihypertensive regimen)
* Patients with another malignancy that was treated within the last three years with the exceptions of localized basal cell carcinoma and cervical carcinoma.
* Patients with impairment of GI function or GI disease that could interfere with the absorption of AEB071.
* Patients with a known history of Human Immunodeficiency Virus (HIV)

* HIV testing is not required as part of this study
* Patients with a known history of active hepatitis B or C infection unless they are on antiviral therapy

* The determination of active hepatitis status should be as per standard of care at each site
* Hepatitis B and C testing is not required as part of this study

Time since the last prior therapy for treatment of underlying malignancy\*\*:

* Cytotoxic chemotherapy: ≤ than the duration of the most recent cycle of the previous regimen (with a minimum of 2 weeks for all)
* Biologic therapy (e.g., antibodies): ≤ 4 weeks
* ≤ 5 x t1/2 of a small molecule therapeutic, not otherwise defined above

\*\*Patients must have recovered or stabilized from all toxicities related to their previous treatment except for alopecia
* Patients with any history of significant coagulopathy or a medical condition requiring long term systemic anticoagulation that would interfere with biopsies.
* Patients having undergone major surgery less than 4 weeks prior to enrollment or that have not fully recovered from prior surgery.
* Pregnant or nursing (lactating) women
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Novartis Pharmaceuticals

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Novartis Pharmaceuticals

Role: STUDY_DIRECTOR

Novartis Pharmaceuticals

Novarts Pharmaceuticals

Role: STUDY_DIRECTOR

Novarts Pharmaceuticals

Locations

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City of Hope National Medical Center

Duarte, California, United States

Site Status

Washington University School of Medicine Div. of Medical Oncology

St Louis, Missouri, United States

Site Status

Hackensack University Medical Center Hackensack (SC)

Hackensack, New Jersey, United States

Site Status

Memorial Sloan Kettering Cancer Center MSK 2

New York, New York, United States

Site Status

Ohio State Comprehensive Cancer Center/James Cancer Hospital Ohio State

Columbus, Ohio, United States

Site Status

University of Texas/MD Anderson Cancer Center SC Location

Houston, Texas, United States

Site Status

Novartis Investigative Site

Créteil, , France

Site Status

Novartis Investigative Site

Lille, , France

Site Status

Novartis Investigative Site

Pierre-Benite Cédex, , France

Site Status

Novartis Investigative Site

Rouen, , France

Site Status

Novartis Investigative Site

Berlin, , Germany

Site Status

Novartis Investigative Site

München, , Germany

Site Status

Novartis Investigative Site

Shatin, New Territories, Hong Kong, Hong Kong

Site Status

Novartis Investigative Site

Milan, MI, Italy

Site Status

Novartis Investigative Site

Torino, TO, Italy

Site Status

Novartis Investigative Site

Amsterdam, , Netherlands

Site Status

Novartis Investigative Site

Groningen, , Netherlands

Site Status

Novartis Investigative Site

Rotterdam, , Netherlands

Site Status

Novartis Investigative Site

Rotterdam, , Netherlands

Site Status

Novartis Investigative Site

Seoul, Korea, South Korea

Site Status

Novartis Investigative Site

Barcelona, Catalonia, Spain

Site Status

Novartis Investigative Site

Barcelona, , Spain

Site Status

Novartis Investigative Site

Taipei, , Taiwan

Site Status

Novartis Investigative Site

Manchester, , United Kingdom

Site Status

Countries

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United States France Germany Hong Kong Italy Netherlands South Korea Spain Taiwan United Kingdom

Related Links

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https://www.novctrd.com/ctrdweb/trialresult/trialresults/pdf?trialResultId=13343

Results for OEB071X2101 can be found on the Novartis Clinical Trial Results Website

Other Identifiers

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2010-024367-41

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

COEB071X2101

Identifier Type: -

Identifier Source: org_study_id