Pharmacokinetic Study of Single and Repeated Dose of Roflumilast 500 µg , in Healthy Chinese Subjects

NCT ID: NCT01354782

Last Updated: 2016-10-26

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

32 participants

Study Classification

INTERVENTIONAL

Study Start Date

2011-05-31

Study Completion Date

2011-09-30

Brief Summary

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The primary objective is to assess the pharmacokinetics (PK) of roflumilast and its metabolite roflumilast N-oxide after single and repeated oral administrations of roflumilast 500 μg in healthy Chinese subjects.

Detailed Description

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Conditions

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Chronic Obstructive Pulmonary Disease

Keywords

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Pharmacokinetic Roflumilast

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

SINGLE_GROUP

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Roflumilast

(This is a pharmacokinetic study)

Group Type EXPERIMENTAL

Roflumilast

Intervention Type DRUG

Period I: single dose of roflumilast 500 μg orally in the morning.

Period II: repeated dose of roflumilast 500 μg orally in the morning for 14 days.

Interventions

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Roflumilast

Period I: single dose of roflumilast 500 μg orally in the morning.

Period II: repeated dose of roflumilast 500 μg orally in the morning for 14 days.

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Healthy male and female (24 male and 8 female) subjects of Chinese ethnic origin, age 40 years and older.
* Assessed as healthy based on a screening examination including medical history, physical examination, blood pressure, pulse rate, ECG assessment, and clinical laboratory results.
* Body weight according to a Body Mass Index (BMI) between 19 and 28 kg/\[m²\], (both inclusive) and a body weight ≥ 50 kg.
* Females with childbearing potential who are using medically acceptable and reliable method of contraception for the entire study duration, such as tubal ligation, hysterectomy, intrauterine device without hormones or post-menopausal females, the latter is defined as females who have had no menstrual period for at least 2 years.

Exclusion Criteria

* History or current evidence of clinically relevant allergies or idiosyncrasy to drugs or food
* History of allergic reactions to roflumilast or any inactive ingredients of the trial medication
* History or current evidence of any clinically relevant cardiovascular, pulmonary, hepatic, renal, gastrointestinal, hematological, endocrinological, metabolic, neurological, psychiatric, or other disease (within the last 2 years)
* History of malignancy within the past 5 years
* Electrocardiogram (ECG) abnormalities of clinical relevance (e.g. QTc according to Bazett's formula: QTc \> 450 msec (male), QTc \> 470 msec (female), PQ ≥ 220 msec)
* Blood pressure ≥ 140 mm HG systolic or ≥ 90 mm HG diastolic
* Elevated transaminases \> 2 x upper Limit of normal range and or increased of the total bilirubin \> 1.5 upper Limit of normal range
* Clinically relevant abnormalities in clinical chemical, hematological or any other laboratory variables
* Chronic or clinically relevant acute infections
* Proneness to orthostatic dysregulation, faintings, or blackouts
* Positive results in any of the virology tests of acute or chronic infectious HIV and hepatitis A, B, and C virus infections
* Positive drug screen
* Abuse of alcohol or drugs
* Positive β-HCG pregnancy test (female)
* Pregnant or lactating females
Minimum Eligible Age

40 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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AstraZeneca

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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AstraZeneca AstraZeneca

Role: STUDY_DIRECTOR

AstraZeneca

Locations

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Nycomed Investigational Site

Beijing, , China

Site Status

Countries

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China

Related Links

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Other Identifiers

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RO-2455-101-EC

Identifier Type: -

Identifier Source: org_study_id