Trial Outcomes & Findings for Effect of GTx-758 on Total and Free Testosterone Levels in Men With Prostate Cancer (NCT NCT01326312)

NCT ID: NCT01326312

Last Updated: 2023-06-22

Results Overview

Recruitment status

TERMINATED

Study phase

PHASE2

Target enrollment

159 participants

Primary outcome timeframe

60 days

Results posted on

2023-06-22

Participant Flow

Participant milestones

Participant milestones
Measure
GTx 758 1000mg
GTx-758/Experimental/ nonsteroidal selective ER alpha agonist GTx-758: comparison of different dosages of GTx-758 with leuprolide acetate for depot suspension
GTx-758 2000mg
GTx-758/Experimental/ nonsteroidal selective ER alpha agonist GTx-758: comparison of different dosages of GTx-758 with leuprolide acetate for depot suspension
Lupron Depot
Luteinizing Hormone Releasing Hormone Agonist Lupron Depot: comparison of different dosages of GTx-758 with leuprolide acetate for depot suspension
Overall Study
STARTED
53
55
51
Overall Study
COMPLETED
0
0
0
Overall Study
NOT COMPLETED
53
55
51

Reasons for withdrawal

Reasons for withdrawal
Measure
GTx 758 1000mg
GTx-758/Experimental/ nonsteroidal selective ER alpha agonist GTx-758: comparison of different dosages of GTx-758 with leuprolide acetate for depot suspension
GTx-758 2000mg
GTx-758/Experimental/ nonsteroidal selective ER alpha agonist GTx-758: comparison of different dosages of GTx-758 with leuprolide acetate for depot suspension
Lupron Depot
Luteinizing Hormone Releasing Hormone Agonist Lupron Depot: comparison of different dosages of GTx-758 with leuprolide acetate for depot suspension
Overall Study
Adverse Event
11
11
1
Overall Study
Withdrawal by Subject
1
2
1
Overall Study
Protocol Violation
0
1
0
Overall Study
Lack of Efficacy
13
7
1
Overall Study
Death
1
0
1
Overall Study
progressive disease
0
1
1
Overall Study
Study terminated by Sponsor
8
32
46
Overall Study
Treatment arm terminated
19
0
0
Overall Study
QTc > 500
0
1
0

Baseline Characteristics

Effect of GTx-758 on Total and Free Testosterone Levels in Men With Prostate Cancer

Baseline characteristics by cohort

Baseline characteristics by cohort
Measure
GTx-758 1000mg
n=53 Participants
GTx-758/Experimental/ nonsteroidal selective ER alpha agonist GTx-758: comparison of different dosages of GTx-758 with leuprolide acetate for depot suspension
GTx-758 2000mg
n=55 Participants
GTx-758/Experimental/ nonsteroidal selective ER alpha agonist GTx-758: comparison of different dosages of GTx-758 with leuprolide acetate for depot suspension
Lupron Depot
n=51 Participants
Luteinizing Hormone Releasing Hormone Agonist Lupron Depot: comparison of different dosages of GTx-758 with leuprolide acetate for depot suspension
Total
n=159 Participants
Total of all reporting groups
Age, Continuous
68 years
n=5 Participants
68 years
n=7 Participants
69 years
n=5 Participants
68 years
n=4 Participants
Sex: Female, Male
Female
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
0 Participants
n=4 Participants
Sex: Female, Male
Male
53 Participants
n=5 Participants
55 Participants
n=7 Participants
51 Participants
n=5 Participants
159 Participants
n=4 Participants
Ethnicity (NIH/OMB)
Hispanic or Latino
6 Participants
n=5 Participants
4 Participants
n=7 Participants
5 Participants
n=5 Participants
15 Participants
n=4 Participants
Ethnicity (NIH/OMB)
Not Hispanic or Latino
47 Participants
n=5 Participants
51 Participants
n=7 Participants
46 Participants
n=5 Participants
144 Participants
n=4 Participants
Ethnicity (NIH/OMB)
Unknown or Not Reported
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
0 Participants
n=4 Participants
Race (NIH/OMB)
American Indian or Alaska Native
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
0 Participants
n=4 Participants
Race (NIH/OMB)
Asian
1 Participants
n=5 Participants
1 Participants
n=7 Participants
0 Participants
n=5 Participants
2 Participants
n=4 Participants
Race (NIH/OMB)
Native Hawaiian or Other Pacific Islander
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
0 Participants
n=4 Participants
Race (NIH/OMB)
Black or African American
11 Participants
n=5 Participants
12 Participants
n=7 Participants
10 Participants
n=5 Participants
33 Participants
n=4 Participants
Race (NIH/OMB)
White
41 Participants
n=5 Participants
42 Participants
n=7 Participants
41 Participants
n=5 Participants
124 Participants
n=4 Participants
Race (NIH/OMB)
More than one race
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
0 Participants
n=4 Participants
Race (NIH/OMB)
Unknown or Not Reported
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
0 Participants
n=4 Participants
Region of Enrollment
United States
53 participants
n=5 Participants
55 participants
n=7 Participants
51 participants
n=5 Participants
159 participants
n=4 Participants

PRIMARY outcome

Timeframe: 60 days

Population: Per-Protocol Population

Outcome measures

Outcome measures
Measure
GTx- 758 1000mg
n=32 Participants
GTx-758/Experimental/ nonsteroidal selective ER alpha agonist GTx-758: comparison of different dosages of GTx-758 with leuprolide acetate for depot suspension
GTx-758 2000mg
n=40 Participants
GTx-758/Experimental/ nonsteroidal selective ER alpha agonist GTx-758: comparison of different dosages of GTx-758 with leuprolide acetate for depot suspension
Lupron Depot
n=45 Participants
Luteinizing Hormone Releasing Hormone Agonist Lupron Depot: comparison of different dosages of GTx-758 with leuprolide acetate for depot suspension
Number of Participants Who Are Castrate by Day 60
19 participants
34 participants
43 participants

SECONDARY outcome

Timeframe: 12 months

Population: Castrate Population

Outcome measures

Outcome measures
Measure
GTx- 758 1000mg
n=19 Participants
GTx-758/Experimental/ nonsteroidal selective ER alpha agonist GTx-758: comparison of different dosages of GTx-758 with leuprolide acetate for depot suspension
GTx-758 2000mg
n=34 Participants
GTx-758/Experimental/ nonsteroidal selective ER alpha agonist GTx-758: comparison of different dosages of GTx-758 with leuprolide acetate for depot suspension
Lupron Depot
n=43 Participants
Luteinizing Hormone Releasing Hormone Agonist Lupron Depot: comparison of different dosages of GTx-758 with leuprolide acetate for depot suspension
Number of Participants Who Are Castrate by Day 60 and Maintained Castrate Range From Day 60 to Day 360/End of Study.
0 Participants
3 Participants
9 Participants

SECONDARY outcome

Timeframe: 60 days

Population: Per-Protocol Population

Median time to castration was summarized using the Kaplan-Meier method.

Outcome measures

Outcome measures
Measure
GTx- 758 1000mg
n=32 Participants
GTx-758/Experimental/ nonsteroidal selective ER alpha agonist GTx-758: comparison of different dosages of GTx-758 with leuprolide acetate for depot suspension
GTx-758 2000mg
n=40 Participants
GTx-758/Experimental/ nonsteroidal selective ER alpha agonist GTx-758: comparison of different dosages of GTx-758 with leuprolide acetate for depot suspension
Lupron Depot
n=45 Participants
Luteinizing Hormone Releasing Hormone Agonist Lupron Depot: comparison of different dosages of GTx-758 with leuprolide acetate for depot suspension
Time to Castration in Participants With Prostate Cancer
29 days
Interval 14.0 to 62.0
21 days
Interval 7.0 to 68.0
21 days
Interval 13.0 to 42.0

Adverse Events

GTx- 758 1000mg

Serious events: 11 serious events
Other events: 46 other events
Deaths: 1 deaths

GTx-758 2000mg

Serious events: 6 serious events
Other events: 49 other events
Deaths: 0 deaths

Lupron Depot

Serious events: 4 serious events
Other events: 48 other events
Deaths: 1 deaths

Serious adverse events

Serious adverse events
Measure
GTx- 758 1000mg
n=53 participants at risk
GTx-758/Experimental/ nonsteroidal selective ER alpha agonist GTx-758 2000mg: comparison of different dosages of GTx-758 with leuprolide acetate for depot suspension
GTx-758 2000mg
n=55 participants at risk
GTx-758/Experimental/ nonsteroidal selective ER alpha agonist GTx-758 1000mg: comparison of different dosages of GTx-758 with leuprolide acetate for depot suspension
Lupron Depot
n=51 participants at risk
Luteinizing Hormone Releasing Hormone Agonist Lupron Depot: comparison of different dosages of GTx-758 with leuprolide acetate for depot suspension
Cardiac disorders
Acute Coronary Syndrome
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Blood and lymphatic system disorders
Anaemia
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Psychiatric disorders
Anxiety
0.00%
0/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
Cardiac disorders
Atrial Fibrillation
3.8%
2/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Musculoskeletal and connective tissue disorders
Back Pain
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Cardiac disorders
Cardiac Arrest
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Vascular disorders
Deep Vein Thrombosis
5.7%
3/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Metabolism and nutrition disorders
Dehydration
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Musculoskeletal and connective tissue disorders
Flank Pain
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Injury, poisoning and procedural complications
Hip Fracture
0.00%
0/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
Immune system disorders
Hypersensitivity
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Metabolism and nutrition disorders
Hypnonatraemia
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Infections and infestations
Lung Infection
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Neoplasms benign, malignant and unspecified (incl cysts and polyps)
Metastases to Bone
0.00%
0/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
Cardiac disorders
Myocardial Infarction
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Vascular disorders
Orthostatic Hypotension
0.00%
0/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
Musculoskeletal and connective tissue disorders
Pain in Extremity
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Musculoskeletal and connective tissue disorders
Pathological Fracture
0.00%
0/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
Respiratory, thoracic and mediastinal disorders
Pulmonary Embolism
3.8%
2/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Respiratory, thoracic and mediastinal disorders
Respiratory Failure
0.00%
0/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
Cardiac disorders
Sinus Bradycardia
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Infections and infestations
Urosepsis
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year

Other adverse events

Other adverse events
Measure
GTx- 758 1000mg
n=53 participants at risk
GTx-758/Experimental/ nonsteroidal selective ER alpha agonist GTx-758 2000mg: comparison of different dosages of GTx-758 with leuprolide acetate for depot suspension
GTx-758 2000mg
n=55 participants at risk
GTx-758/Experimental/ nonsteroidal selective ER alpha agonist GTx-758 1000mg: comparison of different dosages of GTx-758 with leuprolide acetate for depot suspension
Lupron Depot
n=51 participants at risk
Luteinizing Hormone Releasing Hormone Agonist Lupron Depot: comparison of different dosages of GTx-758 with leuprolide acetate for depot suspension
Blood and lymphatic system disorders
anemia
1.9%
1/53 • 1 year
5.5%
3/55 • 1 year
0.00%
0/51 • 1 year
Blood and lymphatic system disorders
lymphadenopathy
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Cardiac disorders
acute coronary syndrome
7.5%
4/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Cardiac disorders
angina
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Cardiac disorders
right bundle branch block
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Cardiac disorders
cardiac arrest
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Cardiac disorders
conduction disorder
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Cardiac disorders
coronary artery occlusion
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Cardiac disorders
left ventricular dysfunction
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Cardiac disorders
mitral valve disease
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Cardiac disorders
myocardial infarction
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Cardiac disorders
sinus bradycardia
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Cardiac disorders
sinus tachycardia
0.00%
0/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
Cardiac disorders
ventricular arrhythmia
0.00%
0/53 • 1 year
3.6%
2/55 • 1 year
0.00%
0/51 • 1 year
Ear and labyrinth disorders
vertigo
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Endocrine disorders
hypothyroidism
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Eye disorders
conjunctival hemorrhage
0.00%
0/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
Eye disorders
conjuntivitis
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Eye disorders
visual acuity reduced
0.00%
0/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
Eye disorders
vitreous floaters
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Gastrointestinal disorders
abdominal distension
1.9%
1/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Gastrointestinal disorders
abdominal pain
1.9%
1/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Gastrointestinal disorders
abdominal pain, upper
0.00%
0/53 • 1 year
3.6%
2/55 • 1 year
0.00%
0/51 • 1 year
Gastrointestinal disorders
colitis
0.00%
0/53 • 1 year
3.6%
2/55 • 1 year
0.00%
0/51 • 1 year
Gastrointestinal disorders
colonic polyp
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
2.0%
1/51 • 1 year
Gastrointestinal disorders
constipation
1.9%
1/53 • 1 year
7.3%
4/55 • 1 year
3.9%
2/51 • 1 year
Gastrointestinal disorders
diarrhea
13.2%
7/53 • 1 year
16.4%
9/55 • 1 year
7.8%
4/51 • 1 year
Gastrointestinal disorders
diverticulum
0.00%
0/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
Gastrointestinal disorders
dry mouth
0.00%
0/53 • 1 year
5.5%
3/55 • 1 year
0.00%
0/51 • 1 year
Gastrointestinal disorders
dyspepsia
11.3%
6/53 • 1 year
9.1%
5/55 • 1 year
2.0%
1/51 • 1 year
Gastrointestinal disorders
gastritis
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Gastrointestinal disorders
GI pain
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Gastrointestinal disorders
gastroesophageal reflux disease
1.9%
1/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Gastrointestinal disorders
hemmorhoidal hemmorhage
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Gastrointestinal disorders
hemorrhoids
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
2.0%
1/51 • 1 year
Gastrointestinal disorders
impaired gastric emptying
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Gastrointestinal disorders
large intestinal ulcer
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Gastrointestinal disorders
lip swelling
0.00%
0/53 • 1 year
3.6%
2/55 • 1 year
0.00%
0/51 • 1 year
Gastrointestinal disorders
nausea
13.2%
7/53 • 1 year
5.5%
3/55 • 1 year
7.8%
4/51 • 1 year
Gastrointestinal disorders
oral pain
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Gastrointestinal disorders
rectal discharge
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Gastrointestinal disorders
swollen tongue
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Gastrointestinal disorders
tooth ache
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Gastrointestinal disorders
vomiting
5.7%
3/53 • 1 year
5.5%
3/55 • 1 year
0.00%
0/51 • 1 year
General disorders
chest pain
0.00%
0/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
General disorders
chills
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
3.9%
2/51 • 1 year
General disorders
fatigue
11.3%
6/53 • 1 year
14.5%
8/55 • 1 year
17.6%
9/51 • 1 year
General disorders
influenza like illness
0.00%
0/53 • 1 year
7.3%
4/55 • 1 year
7.8%
4/51 • 1 year
General disorders
infusion site pain
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
General disorders
injection site reaction
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
3.9%
2/51 • 1 year
General disorders
irritability
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
General disorders
localized edema
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
General disorders
non cardiac chest pain
3.8%
2/53 • 1 year
1.8%
1/55 • 1 year
2.0%
1/51 • 1 year
General disorders
edema, peripheral
3.8%
2/53 • 1 year
5.5%
3/55 • 1 year
0.00%
0/51 • 1 year
General disorders
pyrexia
7.5%
4/53 • 1 year
3.6%
2/55 • 1 year
0.00%
0/51 • 1 year
General disorders
vessel puncture site hematoma
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Hepatobiliary disorders
hepatobiliary disease
0.00%
0/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
Immune system disorders
hypersensitivity
3.8%
2/53 • 1 year
3.6%
2/55 • 1 year
0.00%
0/51 • 1 year
Infections and infestations
bronchitis
3.8%
2/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Infections and infestations
cellulitis
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Infections and infestations
eye infection
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Infections and infestations
gingival infection
0.00%
0/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
Infections and infestations
laryngitis
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Infections and infestations
lung infection
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Infections and infestations
nail infection
0.00%
0/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
Infections and infestations
nasopharyngitis
3.8%
2/53 • 1 year
1.8%
1/55 • 1 year
2.0%
1/51 • 1 year
Infections and infestations
oral herpes
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
2.0%
1/51 • 1 year
Infections and infestations
otitis externa
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Infections and infestations
pharyngitis
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
3.9%
2/51 • 1 year
Infections and infestations
pneumonia
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Infections and infestations
sinusitis
0.00%
0/53 • 1 year
0.00%
0/55 • 1 year
3.9%
2/51 • 1 year
Infections and infestations
skin infections
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
Infections and infestations
tooth infections
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Infections and infestations
upper respiratory tract infections
5.7%
3/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
Infections and infestations
urinary tract infections
7.5%
4/53 • 1 year
9.1%
5/55 • 1 year
5.9%
3/51 • 1 year
Infections and infestations
urosepsis
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Injury, poisoning and procedural complications
contusion
3.8%
2/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Injury, poisoning and procedural complications
excoriation
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Injury, poisoning and procedural complications
fall
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Injury, poisoning and procedural complications
hip fracture
0.00%
0/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
Injury, poisoning and procedural complications
procedural pain
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Injury, poisoning and procedural complications
radiation associated pain
0.00%
0/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
Injury, poisoning and procedural complications
recall phenomenon
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Injury, poisoning and procedural complications
rib fracture
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Injury, poisoning and procedural complications
spinal column injury
0.00%
0/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
Investigations
alanine aminotransferase increase
1.9%
1/53 • 1 year
1.8%
1/55 • 1 year
3.9%
2/51 • 1 year
Investigations
aspartate aminotransferase increase
1.9%
1/53 • 1 year
1.8%
1/55 • 1 year
2.0%
1/51 • 1 year
Investigations
blood alkaline phosphatase increase
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Investigations
blood bilirubin increase
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Investigations
blood creatinine increase
0.00%
0/53 • 1 year
3.6%
2/55 • 1 year
0.00%
0/51 • 1 year
Investigations
gamma-glutamyltransferase increase
0.00%
0/53 • 1 year
3.6%
2/55 • 1 year
0.00%
0/51 • 1 year
Investigations
troponin-I increase
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Investigations
weight decreased
1.9%
1/53 • 1 year
5.5%
3/55 • 1 year
0.00%
0/51 • 1 year
Investigations
weight increased
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
9.8%
5/51 • 1 year
Metabolism and nutrition disorders
decreased appetite
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
2.0%
1/51 • 1 year
Investigations
dehydration
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Metabolism and nutrition disorders
hyperlipidemia
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Metabolism and nutrition disorders
hypokalemia
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Metabolism and nutrition disorders
hyponatremia
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Metabolism and nutrition disorders
hypophosphatemia
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Metabolism and nutrition disorders
increased appetite
0.00%
0/53 • 1 year
0.00%
0/55 • 1 year
3.9%
2/51 • 1 year
Metabolism and nutrition disorders
iron overload
0.00%
0/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
Metabolism and nutrition disorders
vitamin D deficiency
1.9%
1/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Musculoskeletal and connective tissue disorders
arthralgia
3.8%
2/53 • 1 year
1.8%
1/55 • 1 year
7.8%
4/51 • 1 year
Musculoskeletal and connective tissue disorders
arthritis
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
3.9%
2/51 • 1 year
Musculoskeletal and connective tissue disorders
back pain
1.9%
1/53 • 1 year
5.5%
3/55 • 1 year
9.8%
5/51 • 1 year
Musculoskeletal and connective tissue disorders
exostosis
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Musculoskeletal and connective tissue disorders
flank pain
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Musculoskeletal and connective tissue disorders
groin pain
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Musculoskeletal and connective tissue disorders
joint effusion
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Musculoskeletal and connective tissue disorders
joint range of motion decreased
1.9%
1/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Musculoskeletal and connective tissue disorders
muscle spasms
5.7%
3/53 • 1 year
7.3%
4/55 • 1 year
0.00%
0/51 • 1 year
Musculoskeletal and connective tissue disorders
musculoskeletal chest pain
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Musculoskeletal and connective tissue disorders
musculoskeletal pain
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
2.0%
1/51 • 1 year
Musculoskeletal and connective tissue disorders
myalgia
0.00%
0/53 • 1 year
3.6%
2/55 • 1 year
2.0%
1/51 • 1 year
Musculoskeletal and connective tissue disorders
neck mass
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Musculoskeletal and connective tissue disorders
neck pain
3.8%
2/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Musculoskeletal and connective tissue disorders
pain in extremity
7.5%
4/53 • 1 year
3.6%
2/55 • 1 year
2.0%
1/51 • 1 year
Musculoskeletal and connective tissue disorders
pathological fracture
0.00%
0/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
Neoplasms benign, malignant and unspecified (incl cysts and polyps)
basal cell carcinoma
0.00%
0/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
Neoplasms benign, malignant and unspecified (incl cysts and polyps)
breast cancer
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Neoplasms benign, malignant and unspecified (incl cysts and polyps)
hepatic cancer, metastatic
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Neoplasms benign, malignant and unspecified (incl cysts and polyps)
lipoma
0.00%
0/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
Neoplasms benign, malignant and unspecified (incl cysts and polyps)
metastases to bone
0.00%
0/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
Neoplasms benign, malignant and unspecified (incl cysts and polyps)
seborrheic keratosis
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
2.0%
1/51 • 1 year
Nervous system disorders
amnesia
0.00%
0/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
Nervous system disorders
cerebrovascular accident
0.00%
0/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
Nervous system disorders
dizziness
3.8%
2/53 • 1 year
10.9%
6/55 • 1 year
9.8%
5/51 • 1 year
Nervous system disorders
dysgeusia
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Nervous system disorders
headache
3.8%
2/53 • 1 year
9.1%
5/55 • 1 year
2.0%
1/51 • 1 year
Nervous system disorders
lethargy
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
3.9%
2/51 • 1 year
Nervous system disorders
neuralgia
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Nervous system disorders
paraesthesia
5.7%
3/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
Nervous system disorders
parosmia
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Nervous system disorders
radiculitis
0.00%
0/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
Nervous system disorders
sinus headache
0.00%
0/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
Nervous system disorders
somnolence
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Nervous system disorders
syncope
0.00%
0/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
Nervous system disorders
tremor
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Psychiatric disorders
anxiety
3.8%
2/53 • 1 year
0.00%
0/55 • 1 year
3.9%
2/51 • 1 year
Psychiatric disorders
confusional state
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Psychiatric disorders
depression
1.9%
1/53 • 1 year
3.6%
2/55 • 1 year
0.00%
0/51 • 1 year
Psychiatric disorders
hallucination
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Psychiatric disorders
insomnia
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
3.9%
2/51 • 1 year
Psychiatric disorders
libido decreased
0.00%
0/53 • 1 year
5.5%
3/55 • 1 year
3.9%
2/51 • 1 year
Psychiatric disorders
mood swings
0.00%
0/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
Renal and urinary disorders
azotemia
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Renal and urinary disorders
bladder spasm
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Renal and urinary disorders
calculus ureteric
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Renal and urinary disorders
cystitis noninfective
0.00%
0/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
Renal and urinary disorders
hematuria
1.9%
1/53 • 1 year
1.8%
1/55 • 1 year
3.9%
2/51 • 1 year
Renal and urinary disorders
lower urinary tract symptoms
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Renal and urinary disorders
micturition urgency
0.00%
0/53 • 1 year
3.6%
2/55 • 1 year
2.0%
1/51 • 1 year
Renal and urinary disorders
nocturia
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
Renal and urinary disorders
pollakiuria
3.8%
2/53 • 1 year
10.9%
6/55 • 1 year
7.8%
4/51 • 1 year
Renal and urinary disorders
renal failure
1.9%
1/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Renal and urinary disorders
renal pain
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Renal and urinary disorders
terminal dribbling
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Renal and urinary disorders
urinary hesitation
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Renal and urinary disorders
urinary incontinence
3.8%
2/53 • 1 year
1.8%
1/55 • 1 year
5.9%
3/51 • 1 year
Renal and urinary disorders
urinary retention
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Renal and urinary disorders
urinary tract pain
3.8%
2/53 • 1 year
1.8%
1/55 • 1 year
2.0%
1/51 • 1 year
Renal and urinary disorders
urinary flow decreased
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Reproductive system and breast disorders
breast discharge
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Reproductive system and breast disorders
breast discomfort
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Reproductive system and breast disorders
breast pain
28.3%
15/53 • 1 year
38.2%
21/55 • 1 year
0.00%
0/51 • 1 year
Reproductive system and breast disorders
breast tenderness
1.9%
1/53 • 1 year
7.3%
4/55 • 1 year
0.00%
0/51 • 1 year
Reproductive system and breast disorders
ejaculation disorder
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Reproductive system and breast disorders
erectile dysfunction
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
2.0%
1/51 • 1 year
Reproductive system and breast disorders
gynecomastia
9.4%
5/53 • 1 year
7.3%
4/55 • 1 year
2.0%
1/51 • 1 year
Reproductive system and breast disorders
nipple pain
1.9%
1/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Reproductive system and breast disorders
edema, genital
1.9%
1/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Reproductive system and breast disorders
pelvic pain
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Reproductive system and breast disorders
perineal erythema
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Reproductive system and breast disorders
prostatic obstruction
0.00%
0/53 • 1 year
3.6%
2/55 • 1 year
0.00%
0/51 • 1 year
Reproductive system and breast disorders
testicular atrophy
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Reproductive system and breast disorders
testicular pain
1.9%
1/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Respiratory, thoracic and mediastinal disorders
asthma
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Respiratory, thoracic and mediastinal disorders
cough
1.9%
1/53 • 1 year
9.1%
5/55 • 1 year
0.00%
0/51 • 1 year
Respiratory, thoracic and mediastinal disorders
dyspnea
3.8%
2/53 • 1 year
9.1%
5/55 • 1 year
2.0%
1/51 • 1 year
Respiratory, thoracic and mediastinal disorders
hiccups
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Respiratory, thoracic and mediastinal disorders
nasal congestion
1.9%
1/53 • 1 year
3.6%
2/55 • 1 year
2.0%
1/51 • 1 year
Respiratory, thoracic and mediastinal disorders
pleuritic pain
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Respiratory, thoracic and mediastinal disorders
pneumonitis
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Respiratory, thoracic and mediastinal disorders
pulmonary embolism
5.7%
3/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Respiratory, thoracic and mediastinal disorders
pulmonary infarction
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Respiratory, thoracic and mediastinal disorders
respiratory failure
0.00%
0/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
Respiratory, thoracic and mediastinal disorders
rhinitis, allergic
1.9%
1/53 • 1 year
3.6%
2/55 • 1 year
0.00%
0/51 • 1 year
Respiratory, thoracic and mediastinal disorders
upper airway cough syndrome
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Skin and subcutaneous tissue disorders
actinic keratosis
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Skin and subcutaneous tissue disorders
alopecia
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Skin and subcutaneous tissue disorders
angioedema
0.00%
0/53 • 1 year
3.6%
2/55 • 1 year
0.00%
0/51 • 1 year
Skin and subcutaneous tissue disorders
dermatitis
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Skin and subcutaneous tissue disorders
dermatitis, allergic
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Skin and subcutaneous tissue disorders
dermatitis, atopic
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Skin and subcutaneous tissue disorders
dry skin
0.00%
0/53 • 1 year
5.5%
3/55 • 1 year
0.00%
0/51 • 1 year
Skin and subcutaneous tissue disorders
erythema multiforme
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Skin and subcutaneous tissue disorders
lentigo
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Skin and subcutaneous tissue disorders
night sweats
0.00%
0/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
Skin and subcutaneous tissue disorders
onychoclasis
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Skin and subcutaneous tissue disorders
photosensitivity reaction
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Skin and subcutaneous tissue disorders
pruritus
3.8%
2/53 • 1 year
0.00%
0/55 • 1 year
3.9%
2/51 • 1 year
Skin and subcutaneous tissue disorders
rash
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Skin and subcutaneous tissue disorders
rash, maculo-papular
5.7%
3/53 • 1 year
5.5%
3/55 • 1 year
0.00%
0/51 • 1 year
Skin and subcutaneous tissue disorders
skin ulcer
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Skin and subcutaneous tissue disorders
swelling face
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Skin and subcutaneous tissue disorders
urticaria
1.9%
1/53 • 1 year
3.6%
2/55 • 1 year
0.00%
0/51 • 1 year
Vascular disorders
deep vein thrombosis
15.1%
8/53 • 1 year
3.6%
2/55 • 1 year
0.00%
0/51 • 1 year
Vascular disorders
hot flush
28.3%
15/53 • 1 year
20.0%
11/55 • 1 year
76.5%
39/51 • 1 year
Vascular disorders
hypotension
0.00%
0/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year
Vascular disorders
lymphedema
0.00%
0/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
Vascular disorders
orthostatic hypotension
0.00%
0/53 • 1 year
0.00%
0/55 • 1 year
2.0%
1/51 • 1 year
Vascular disorders
thrombophlebitis
1.9%
1/53 • 1 year
0.00%
0/55 • 1 year
0.00%
0/51 • 1 year
Vascular disorders
thrombophlebitis, superficial
1.9%
1/53 • 1 year
1.8%
1/55 • 1 year
0.00%
0/51 • 1 year

Additional Information

Mary Breitmeyer

Oncternal

Phone: 858-434-1113

Results disclosure agreements

  • Principal investigator is a sponsor employee
  • Publication restrictions are in place