Akt Inhibitor MK2206 in Treating Patients With Advanced Gastric or Gastroesophageal Junction Cancer

NCT ID: NCT01260701

Last Updated: 2016-01-18

Study Results

Results available

Outcome measurements, participant flow, baseline characteristics, and adverse events have been published for this study.

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE2

Total Enrollment

75 participants

Study Classification

INTERVENTIONAL

Study Start Date

2011-01-31

Study Completion Date

2015-07-31

Brief Summary

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This phase II clinical trial studies how well Akt inhibitor MK2206 works in treating patients with advanced gastric or gastroesophageal junction cancer. Akt inhibitor MK2206 may stop the growth of tumor cells by blocking some of the enzymes needed for cell growth.

Detailed Description

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PRIMARY OBJECTIVES:

I. To estimate the overall survival (OS) for patients with advanced gastric and gastroesophageal junction (GEJ) adenocarcinoma treated with MK-2206 (Akt inhibitor MK2206).

SECONDARY OBJECTIVES:

I. To estimate the progression free survival (PFS) in this patient population. II. To estimate the response rate (confirmed and unconfirmed complete response \[CR\] and partial response \[PR\] by Response Evaluation Criteria In Solid Tumors \[RECIST\] 1.1) in this patient population.

III. To assess the frequency and severity of toxicity associated with this regimen.

OUTLINE (CLOSED TO ACCRUAL 05/01/13):

Patients receive Akt inhibitor MK2206 orally (PO) every other day on days 1-28. Courses repeat every 28 days in the absence of disease progression or unacceptable toxicity.

After completion of study therapy, patients are followed up every 3 months for 2 years.

Conditions

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Adenocarcinoma of the Gastroesophageal Junction Diffuse Gastric Adenocarcinoma Gastric Intestinal Type Adenocarcinoma Gastric Mixed Adenocarcinoma Recurrent Gastric Carcinoma

Study Design

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Allocation Method

NA

Intervention Model

SINGLE_GROUP

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Treatment (CLOSED TO ACCRUAL 05/01/13)

Patients receive Akt inhibitor MK2206 PO every other day on days 1-28. Courses repeat every 28 days in the absence of disease progression or unacceptable toxicity.

Group Type EXPERIMENTAL

Akt Inhibitor MK2206

Intervention Type DRUG

Given PO

Interventions

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Akt Inhibitor MK2206

Given PO

Intervention Type DRUG

Other Intervention Names

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MK2206

Eligibility Criteria

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Inclusion Criteria

* Patients must have histologically or cytologically confirmed adenocarcinoma of the stomach or gastroesophageal (GE) junction that has progressed after first-line treatment, or is recurrent within 6 months after receiving adjuvant therapy; patients must have had exactly one prior systemic treatment regimen; previous adjuvant (chemotherapy \[chemo\]) radiotherapy is permitted; prior chemotherapy given concurrently with radiation for radiosensitization is not considered one prior systemic regimen
* Patients must have measurable disease; computed tomography (CT) scans or magnetic resonance imaging (MRIs) used to assess measurable disease must have been completed within 28 days prior to registration; CT scans or MRIs used to assess non-measurable disease must have been completed within 42 days prior to registration; all disease must be assessed and documented on the Baseline Tumor Assessment Form (RECIST 1.1)
* Patients must not have known brain metastases
* Patients must not have received chemotherapy or radiotherapy within 3 weeks (6 weeks for nitrosoureas or mitomycin C) prior to registration
* Patient must not have received prior treatment with a phosphatidylinositol 3 (PI3), v-akt murine thymoma viral oncogene homolog 1 (AKT) or mechanistic target of rapamycin (Mtor) inhibitor for any reason
* All toxicities from prior therapy must have resolved to =\< grade 1 (Common Terminology Criteria for Adverse Events \[CTCAE\] version 4.0) prior to registration
* Patients must not be receiving or planning to receive any other investigational agents
* Patients must be able to tolerate oral medications and must not have malabsorption or chronic diarrhea (CTCAE version 4.0 grade 2 or higher); administration through a feeding tube is not permitted
* Hemoglobin \>= 9 g/dL
* Absolute neutrophil count (ANC) \>= 1,500/mcL
* Platelets \>= 100,000/mcL
* Total bilirubin =\< institutional upper limit of normal (IULN)
* Aspartate aminotransferase (AST) and alanine aminotransferase (ALT) both =\< 2.5 x IULN; patients with liver metastases must have AST and ALT =\< 5 x IULN
* Patients must have adequate kidney function as evidenced by at least ONE of the following:

* Serum creatinine (mg/dL) =\< IULN obtained within 14 days prior to registration
* Calculated creatinine clearance \> 50 ml/min; the serum creatinine value used in the calculation must have been obtained within 14 days prior to registration
* Patients must have international normalized ratio (INR) =\< 1.2 unless taking therapeutic doses of warfarin; this result must be obtained within 14 days prior to registration
* Patients must have fasting blood sugar =\< 150 mg/dL within 28 days prior to registration
* Patients must have hemoglobin A1C \< 7% within 28 days prior to registration
* Patients must have an electrocardiogram (ECG) within 28 days prior to registration; patients must have corrected QT interval (QTcF) (by Fridericia's calculation) \< 450 msec (male) or \< 470 msec (female)
* Patients must have a Zubrod performance status of 0-1
* Patient must not have any of the following: a history of congenital long QT syndrome; use of concomitant medications that could prolong the QTc interval; New York Heart Association class III or IV heart failure; history of myocardial infarction within 6 months prior to registration; uncontrolled dysrhythmias; poorly controlled angina; resting heart rate =\< 50 bpm (bradycardia)
* Patients must not be receiving concurrent treatment with drugs that are strong inducers or inhibitors of cytochrome P450 family 3, subfamily A, polypeptide 4 (CYP3A4); patients must be able to safely discontinue treatment with these agents for \>= 2 weeks prior to beginning protocol therapy
* Patient must not have uncontrolled intercurrent illness including, but not limited to, ongoing or active infection, symptomatic congestive heart failure, unstable angina pectoris, cardiac arrhythmia, or psychiatric illness/social situations that would limit compliance with study requirements
* Human immunodeficiency virus (HIV)-positive patients on combination antiretroviral therapy are ineligible
* Patient must not be pregnant or nursing; women/men of reproductive potential must have agreed to use two forms of contraception for the duration of protocol treatment and for one month after discontinuation of MK-2206; a woman is considered to be of "reproductive potential" if she has had menses at any time in the preceding 12 consecutive months; in addition to routine contraceptive methods, "effective contraception" also includes heterosexual celibacy and surgery intended to prevent pregnancy (or with a side effect of pregnancy prevention) defined as a hysterectomy, bilateral oophorectomy or bilateral tubal ligation; however, if at any time a previously celibate patient chooses to become heterosexually active during the time period for use of contraceptive measures outlined in the protocol, he/she is responsible for beginning contraceptive measures
* No other prior malignancy is allowed except for the following: adequately treated basal cell or squamous cell skin cancer, in situ cervical cancer, adequately treated stage I or II cancer from which the patient is currently in complete remission, or any other cancer from which the patient has been disease free for five years
* All patients must be informed of the investigational nature of this study and must sign and give written informed consent in accordance with institutional and federal guidelines
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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National Cancer Institute (NCI)

NIH

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Ramesh Ramanathan

Role: PRINCIPAL_INVESTIGATOR

SWOG Cancer Research Network

Locations

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Providence Hospital

Mobile, Alabama, United States

Site Status

Fairbanks Memorial Hospital

Fairbanks, Alaska, United States

Site Status

The University of Arizona Cancer Center-Orange Grove Campus

Tucson, Arizona, United States

Site Status

The University of Arizona Cancer Center-North Campus

Tucson, Arizona, United States

Site Status

The University of Arizona Medical Center-University Campus

Tucson, Arizona, United States

Site Status

Fowler Family Center for Cancer Care

Jonesboro, Arkansas, United States

Site Status

NEA Baptist Memorial Hospital

Jonesboro, Arkansas, United States

Site Status

University of Arkansas for Medical Sciences

Little Rock, Arkansas, United States

Site Status

USC / Norris Comprehensive Cancer Center

Los Angeles, California, United States

Site Status

UC Irvine Health/Chao Family Comprehensive Cancer Center

Orange, California, United States

Site Status

Poudre Valley Hospital

Fort Collins, Colorado, United States

Site Status

Front Range Cancer Specialists

Fort Collins, Colorado, United States

Site Status

Saint Francis Hospital and Medical Center

Hartford, Connecticut, United States

Site Status

UF Cancer Center at Orlando Health

Orlando, Florida, United States

Site Status

Memorial University Medical Center

Savannah, Georgia, United States

Site Status

Oncare Hawaii Inc-POB II

Honolulu, Hawaii, United States

Site Status

Queen's Medical Center

Honolulu, Hawaii, United States

Site Status

Straub Clinic and Hospital

Honolulu, Hawaii, United States

Site Status

University of Hawaii Cancer Center

Honolulu, Hawaii, United States

Site Status

OnCare Hawaii-Liliha

Honolulu, Hawaii, United States

Site Status

Kuakini Medical Center

Honolulu, Hawaii, United States

Site Status

Oncare Hawaii Inc-Kuakini

Honolulu, Hawaii, United States

Site Status

Kapiolani Medical Center for Women and Children

Honolulu, Hawaii, United States

Site Status

Castle Medical Center

Kailua, Hawaii, United States

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Wilcox Memorial Hospital and Kauai Medical Clinic

Lihue, Hawaii, United States

Site Status

Oncare Hawaii Inc-Pali Momi

‘Aiea, Hawaii, United States

Site Status

Pali Momi Medical Center

‘Aiea, Hawaii, United States

Site Status

Saint Alphonsus Cancer Care Center-Boise

Boise, Idaho, United States

Site Status

Cadence Cancer Center at Delnor

Geneva, Illinois, United States

Site Status

Loyola University Medical Center

Maywood, Illinois, United States

Site Status

Cadence Cancer Center in Warrenville

Warrenville, Illinois, United States

Site Status

Franciscan St. Francis Health-Beech Grove

Beech Grove, Indiana, United States

Site Status

Franciscan Saint Francis Health-Indianapolis

Indianapolis, Indiana, United States

Site Status

Reid Hospital and Health Care Services

Richmond, Indiana, United States

Site Status

Cancer Center of Kansas - Chanute

Chanute, Kansas, United States

Site Status

Cancer Center of Kansas - Dodge City

Dodge City, Kansas, United States

Site Status

Cancer Center of Kansas - Fort Scott

Fort Scott, Kansas, United States

Site Status

Saint Rose Ambulatory and Surgery Center

Great Bend, Kansas, United States

Site Status

Hays Medical Center

Hays, Kansas, United States

Site Status

Hutchinson Regional Medical Center

Hutchinson, Kansas, United States

Site Status

Cancer Center of Kansas-Independence

Independence, Kansas, United States

Site Status

The University of Kansas Cancer Center-West

Kansas City, Kansas, United States

Site Status

University of Kansas Cancer Center

Kansas City, Kansas, United States

Site Status

Cancer Center of Kansas-Kingman

Kingman, Kansas, United States

Site Status

Lawrence Memorial Hospital

Lawrence, Kansas, United States

Site Status

Cancer Center of Kansas-Liberal

Liberal, Kansas, United States

Site Status

Cancer Center of Kansas - Newton

Newton, Kansas, United States

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Kansas City Cancer Centers-Southwest

Overland Park, Kansas, United States

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Cancer Center of Kansas - Parsons

Parsons, Kansas, United States

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Via Christi Hospital-Pittsburg

Pittsburg, Kansas, United States

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Cancer Center of Kansas - Pratt

Pratt, Kansas, United States

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Cancer Center of Kansas - Salina

Salina, Kansas, United States

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Salina Regional Health Center

Salina, Kansas, United States

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Kansas City Cancer Center-Shawnee Mission

Shawnee Mission, Kansas, United States

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Saint Francis Hospital and Medical Center - Topeka

Topeka, Kansas, United States

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Cancer Center of Kansas - Wellington

Wellington, Kansas, United States

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Associates In Womens Health

Wichita, Kansas, United States

Site Status

Cancer Center of Kansas-Wichita Medical Arts Tower

Wichita, Kansas, United States

Site Status

Cancer Center of Kansas - Main Office

Wichita, Kansas, United States

Site Status

Via Christi Regional Medical Center

Wichita, Kansas, United States

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Wichita CCOP

Wichita, Kansas, United States

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Cancer Center of Kansas - Winfield

Winfield, Kansas, United States

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Sinai Hospital of Baltimore

Baltimore, Maryland, United States

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Saint Joseph Mercy Hospital

Ann Arbor, Michigan, United States

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Michigan Cancer Research Consortium CCOP

Ann Arbor, Michigan, United States

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Bronson Battle Creek

Battle Creek, Michigan, United States

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Spectrum Health Big Rapids Hospital

Big Rapids, Michigan, United States

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Oakwood Hospital and Medical Center

Dearborn, Michigan, United States

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Saint John Hospital and Medical Center

Detroit, Michigan, United States

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Hurley Medical Center

Flint, Michigan, United States

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Genesys Hurley Cancer Institute

Flint, Michigan, United States

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Genesys Regional Medical Center-West Flint Campus

Flint, Michigan, United States

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Grand Rapids Clinical Oncology Program

Grand Rapids, Michigan, United States

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Mercy Health Saint Mary's

Grand Rapids, Michigan, United States

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Spectrum Health at Butterworth Campus

Grand Rapids, Michigan, United States

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Allegiance Health

Jackson, Michigan, United States

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Sparrow Hospital

Lansing, Michigan, United States

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Saint Mary Mercy Hospital

Livonia, Michigan, United States

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Mercy Health Mercy Campus

Muskegon, Michigan, United States

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Saint Joseph Mercy Oakland

Pontiac, Michigan, United States

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Saint Joseph Mercy Port Huron

Port Huron, Michigan, United States

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Spectrum Health Reed City Hospital

Reed City, Michigan, United States

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Saint Mary's of Michigan

Saginaw, Michigan, United States

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Munson Medical Center

Traverse City, Michigan, United States

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Saint John Macomb-Oakland Hospital

Warren, Michigan, United States

Site Status

Metro Health Hospital

Wyoming, Michigan, United States

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Truman Medical Center

Kansas City, Missouri, United States

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Kansas City Cancer Center - South

Kansas City, Missouri, United States

Site Status

Kansas City Cancer Centers - North

Kansas City, Missouri, United States

Site Status

Kansas City Cancer Center-Lee's Summit

Lee's Summit, Missouri, United States

Site Status

Saint John's Clinic-Rolla-Cancer and Hematology

Rolla, Missouri, United States

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Cancer Research for the Ozarks NCORP

Springfield, Missouri, United States

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Mercy Hospital Springfield

Springfield, Missouri, United States

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CoxHealth South Hospital

Springfield, Missouri, United States

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Saint Louis University Hospital

St Louis, Missouri, United States

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Montana Cancer Consortium NCORP

Billings, Montana, United States

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Saint Vincent Healthcare

Billings, Montana, United States

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Frontier Cancer Center and Blood Institute-Billings

Billings, Montana, United States

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Billings Clinic Cancer Center

Billings, Montana, United States

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Bozeman Deaconess Cancer Center

Bozeman, Montana, United States

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Bozeman Deaconess Hospital

Bozeman, Montana, United States

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Saint James Community Hospital and Cancer Treatment Center

Butte, Montana, United States

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Benefis Healthcare- Sletten Cancer Institute

Great Falls, Montana, United States

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Great Falls Clinic

Great Falls, Montana, United States

Site Status

Saint Peter's Community Hospital

Helena, Montana, United States

Site Status

Glacier Oncology PLLC

Kalispell, Montana, United States

Site Status

Kalispell Regional Medical Center

Kalispell, Montana, United States

Site Status

Montana Cancer Specialists

Missoula, Montana, United States

Site Status

Saint Patrick Hospital - Community Hospital

Missoula, Montana, United States

Site Status

Winthrop University Hospital

Mineola, New York, United States

Site Status

Interlakes Foundation Inc-Rochester

Rochester, New York, United States

Site Status

University of Rochester

Rochester, New York, United States

Site Status

Randolph Hospital

Asheboro, North Carolina, United States

Site Status

Novant Health Presbyterian Medical Center

Charlotte, North Carolina, United States

Site Status

Wayne Memorial Hospital

Goldsboro, North Carolina, United States

Site Status

Cone Health Cancer Center

Greensboro, North Carolina, United States

Site Status

Iredell Memorial Hospital

Statesville, North Carolina, United States

Site Status

Southeast Cancer Control Consortium CCOP

Winston-Salem, North Carolina, United States

Site Status

Akron General Medical Center

Akron, Ohio, United States

Site Status

Mary Rutan Hospital

Bellefontaine, Ohio, United States

Site Status

Adena Regional Medical Center

Chillicothe, Ohio, United States

Site Status

Good Samaritan Hospital - Cincinnati

Cincinnati, Ohio, United States

Site Status

University of Cincinnati

Cincinnati, Ohio, United States

Site Status

Riverside Methodist Hospital

Columbus, Ohio, United States

Site Status

Columbus CCOP

Columbus, Ohio, United States

Site Status

Grant Medical Center

Columbus, Ohio, United States

Site Status

Mount Carmel Health Center West

Columbus, Ohio, United States

Site Status

Doctors Hospital

Columbus, Ohio, United States

Site Status

Grandview Hospital

Dayton, Ohio, United States

Site Status

Good Samaritan Hospital - Dayton

Dayton, Ohio, United States

Site Status

Miami Valley Hospital

Dayton, Ohio, United States

Site Status

Samaritan North Health Center

Dayton, Ohio, United States

Site Status

Dayton CCOP

Dayton, Ohio, United States

Site Status

Grady Memorial Hospital

Delaware, Ohio, United States

Site Status

Blanchard Valley Hospital

Findlay, Ohio, United States

Site Status

Atrium Medical Center-Middletown Regional Hospital

Franklin, Ohio, United States

Site Status

Wayne Hospital

Greenville, Ohio, United States

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Kettering Medical Center

Kettering, Ohio, United States

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Fairfield Medical Center

Lancaster, Ohio, United States

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Marietta Memorial Hospital

Marietta, Ohio, United States

Site Status

Knox Community Hospital

Mount Vernon, Ohio, United States

Site Status

Licking Memorial Hospital

Newark, Ohio, United States

Site Status

Southern Ohio Medical Center

Portsmouth, Ohio, United States

Site Status

Springfield Regional Medical Center

Springfield, Ohio, United States

Site Status

Upper Valley Medical Center

Troy, Ohio, United States

Site Status

Saint Ann's Hospital

Westerville, Ohio, United States

Site Status

Clinton Memorial Hospital

Wilmington, Ohio, United States

Site Status

Greene Memorial Hospital

Xenia, Ohio, United States

Site Status

Genesis HealthCare System

Zanesville, Ohio, United States

Site Status

University of Oklahoma Health Sciences Center

Oklahoma City, Oklahoma, United States

Site Status

Oregon Health and Science University

Portland, Oregon, United States

Site Status

McLeod Regional Medical Center

Florence, South Carolina, United States

Site Status

University of Tennessee - Knoxville

Knoxville, Tennessee, United States

Site Status

Baylor College of Medicine

Houston, Texas, United States

Site Status

Baylor Saint Luke's Medical Center

Houston, Texas, United States

Site Status

Ben Taub General Hospital

Houston, Texas, United States

Site Status

Michael E DeBakey VA Medical Center

Houston, Texas, United States

Site Status

Danville Regional Medical Center

Danville, Virginia, United States

Site Status

Memorial Hospital Of Martinsville

Martinsville, Virginia, United States

Site Status

Cancer Care Center at Island Hospital

Anacortes, Washington, United States

Site Status

PeaceHealth Saint Joseph Medical Center

Bellingham, Washington, United States

Site Status

Harrison HealthPartners Hematology and Oncology-Bremerton

Bremerton, Washington, United States

Site Status

Highline Medical Center-Main Campus

Burien, Washington, United States

Site Status

Swedish Cancer Institute-Issaquah

Issaquah, Washington, United States

Site Status

Kadlec Clinic Hematology and Oncology

Kennewick, Washington, United States

Site Status

EvergreenHealth Medical Center

Kirkland, Washington, United States

Site Status

Seattle Cancer Care Alliance at EvergreenHealth

Kirkland, Washington, United States

Site Status

Skagit Valley Hospital

Mount Vernon, Washington, United States

Site Status

Harrison HealthPartners Hematology and Oncology-Poulsbo

Poulsbo, Washington, United States

Site Status

Virginia Mason CCOP

Seattle, Washington, United States

Site Status

Harborview Medical Center

Seattle, Washington, United States

Site Status

Minor and James Medical PLLC

Seattle, Washington, United States

Site Status

Pacific Medical Center-First Hill

Seattle, Washington, United States

Site Status

Fred Hutchinson Cancer Research Center

Seattle, Washington, United States

Site Status

Group Health Cooperative of Puget Sound Oncology Consortium

Seattle, Washington, United States

Site Status

Group Health Cooperative-Seattle

Seattle, Washington, United States

Site Status

Swedish Medical Center-First Hill

Seattle, Washington, United States

Site Status

The Polyclinic

Seattle, Washington, United States

Site Status

University of Washington Medical Center

Seattle, Washington, United States

Site Status

United General Hospital

Sedro-Woolley, Washington, United States

Site Status

Cancer Care Northwest - Spokane South

Spokane, Washington, United States

Site Status

Evergreen Hematology and Oncology PS

Spokane, Washington, United States

Site Status

Rockwood Clinic

Spokane, Washington, United States

Site Status

Wenatchee Valley Hospital and Clinics

Wenatchee, Washington, United States

Site Status

Rocky Mountain Oncology

Casper, Wyoming, United States

Site Status

Welch Cancer Center

Sheridan, Wyoming, United States

Site Status

BCCA-Vancouver Cancer Centre

Vancouver, British Columbia, Canada

Site Status

Countries

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United States Canada

References

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Ramanathan RK, McDonough SL, Kennecke HF, Iqbal S, Baranda JC, Seery TE, Lim HJ, Hezel AF, Vaccaro GM, Blanke CD. Phase 2 study of MK-2206, an allosteric inhibitor of AKT, as second-line therapy for advanced gastric and gastroesophageal junction cancer: A SWOG cooperative group trial (S1005). Cancer. 2015 Jul 1;121(13):2193-7. doi: 10.1002/cncr.29363. Epub 2015 Mar 30.

Reference Type DERIVED
PMID: 25827820 (View on PubMed)

Other Identifiers

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NCI-2011-02619

Identifier Type: REGISTRY

Identifier Source: secondary_id

SWOG-S1005

Identifier Type: -

Identifier Source: secondary_id

S1005

Identifier Type: -

Identifier Source: secondary_id

CDR0000689602

Identifier Type: -

Identifier Source: secondary_id

S1005

Identifier Type: OTHER

Identifier Source: secondary_id

S1005

Identifier Type: OTHER

Identifier Source: secondary_id

U10CA180888

Identifier Type: NIH

Identifier Source: secondary_id

View Link

U10CA032102

Identifier Type: NIH

Identifier Source: secondary_id

View Link

NCI-2011-02619

Identifier Type: -

Identifier Source: org_study_id

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